Cc1c(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)cnn1C1CCC1 REAL300012003001
Cc1cc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)n(C2CCCC2)n1 REAL300012003002
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccnn2CC(F)F)C[C@@H]1C(=O)O REAL300012003003
CC(C)(C)OC(=O)N1C[C@@H](NCc2c(F)ccnc2Cl)C[C@@H]1C(=O)O REAL300012003004
CN(C)c1cncc(F)c1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003005
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccn(C3CCC3)n2)C[C@@H]1C(=O)O REAL300012003006
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccn(CC(F)F)n2)C[C@@H]1C(=O)O REAL300012003007
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccn(C3CC3(F)F)n2)C[C@@H]1C(=O)O REAL300012003008
CC(C)(C)OC(=O)N1C[C@@H](NCc2cnn(C3CCOCC3)c2)C[C@@H]1C(=O)O REAL300012003009
Cc1cn(C)c(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)n1 REAL300012003010
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccn(C3CCCC3)n2)C[C@@H]1C(=O)O REAL300012003011
CC(C)(C)OC(=O)N1C[C@@H](NCc2ncc(Cl)cc2Cl)C[C@@H]1C(=O)O REAL300012003012
Cc1nscc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003013
Cc1nn(C2CCCC2)cc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003014
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccccc2C(F)F)C[C@@H]1C(=O)O REAL300012003015
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccc3[nH]ncc3c2)C[C@@H]1C(=O)O REAL300012003016
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccc(Cl)c(F)c2F)C[C@@H]1C(=O)O REAL300012003017
Cc1c(F)cccc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003018
COc1c(C#N)cccc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003019
Cc1nc(Cl)ccc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003020
COc1cc(Cl)cc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c1 REAL300012003021
COc1cc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)cc(F)c1F REAL300012003022
COc1cc(C)ncc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003023
CC(C)n1cnc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c1 REAL300012003024
Cn1nccc1-c1n[nH]cc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003025
Cc1onc(C2CC2)c1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003026
COC(=O)c1c(C)[nH]c(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c1C REAL300012003027
CC(C)Oc1ccc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)o1 REAL300012003028
CC(C)(C)OC(=O)N1C[C@@H](NCc2c(Cl)ccc3c2OCO3)C[C@@H]1C(=O)O REAL300012003029
CC(C)(C)OC(=O)N1C[C@@H](NCc2cc(F)cc(C#N)c2)C[C@@H]1C(=O)O REAL300012003030
COc1ccccc1C=CCN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003031
Cc1nn(C2CCC2)cc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003032
Cc1c(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)cnn1CC(F)F REAL300012003033
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccc(-c3ccccn3)nc2)C[C@@H]1C(=O)O REAL300012003034
Cn1nc(-c2ccco2)cc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003035
COc1ccc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c(C)n1 REAL300012003036
CCN(C)c1ccc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c(C)c1 REAL300012003037
CC(C)(C)OC(=O)N1C[C@@H](NCc2scc(Cl)c2Cl)C[C@@H]1C(=O)O REAL300012003038
Cc1sncc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003039
COc1cc(C)cc(OC)c1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003040
Cc1oncc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003041
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccc(CF)cc2)C[C@@H]1C(=O)O REAL300012003042
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccc3sccc3c2)C[C@@H]1C(=O)O REAL300012003043
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccc(-c3ccncc3)cc2)C[C@@H]1C(=O)O REAL300012003044
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccccc2CO)C[C@@H]1C(=O)O REAL300012003045
Cc1nsc(C)c1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003046
CC(C)(C)OC(=O)N1C[C@@H](NCc2cnoc2C(C)(C)C)C[C@@H]1C(=O)O REAL300012003047
C=CCn1cc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)cn1 REAL300012003048
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccc3cn[nH]c3c2)C[C@@H]1C(=O)O REAL300012003049
CCC(C)c1ccc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)cc1 REAL300012003050
CC(C)(C)OC(=O)N1C[C@@H](NCc2cccc(C(C)(F)F)n2)C[C@@H]1C(=O)O REAL300012003051
CC(C)(C)OC(=O)N1C[C@@H](NCc2cccc3c2CCCC3)C[C@@H]1C(=O)O REAL300012003052
CC(=Cc1cc(F)cc(F)c1)CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003053
CC(C)(C)OC(=O)N1C[C@@H](NCc2ccc(-n3ccnn3)cc2)C[C@@H]1C(=O)O REAL300012003054
Cc1c(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)ccc2ccccc12 REAL300012003055
COc1c(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)ccc2[nH]ccc12 REAL300012003056
Cc1nc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c(C)s1 REAL300012003057
CCCn1ncc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c1C REAL300012003058
Cc1ccc2cccnc2c1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003059
COC(=O)c1cc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)n(C)c1 REAL300012003060
CCCn1nc(C)cc1CN[C@H]1C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C1 REAL300012003061
Cn1cc(CN[C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c(C2CCC2)n1 REAL300012003062
CC(C)(C)OC(=O)N1C[C@@H](NCc2cnc(C(C)(C)C)o2)C[C@@H]1C(=O)O REAL300012003063
Cc1ccc(-n2cc(CNC(Cc3cscn3)C(=O)O)c(C(C)(C)C)n2)cc1 REAL300012003064
O=C(O)C(Cc1cscn1)NCc1ccc2ncccc2c1 REAL300012003065
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCc1ccccc1 REAL300012003066
Cc1nn(-c2ccc(F)cc2)c(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003067
CC(C)(C)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003068
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccccc1 REAL300012003069
O=C(O)C(Cc1cscn1)NCc1ccc(Br)o1 REAL300012003070
Cc1nn(-c2ccccc2)cc1CNC(Cc1cscn1)C(=O)O REAL300012003071
N#CCCn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2ccccc2)n1 REAL300012003072
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC(F)F REAL300012003073
CCCOc1ccc(Br)cc1CNC(Cc1cscn1)C(=O)O REAL300012003074
CCOc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC REAL300012003075
O=C(O)C(Cc1cscn1)NCc1ccccc1OCc1ccccc1 REAL300012003076
CCCCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003077
O=C(O)C(Cc1cscn1)NCc1ccc(-c2cccc([N+](=O)[O-])c2)o1 REAL300012003078
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccc([N+](=O)[O-])cc2)o1 REAL300012003079
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1Br REAL300012003080
CC(C)Oc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003081
CCCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003082
CCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003083
C=CCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003084
CCCCCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003085
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccc(Cl)cc2)o1 REAL300012003086
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2Cl)o1 REAL300012003087
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccc(Cl)cc2)s1 REAL300012003088
O=C(O)C(Cc1cscn1)NCc1cnn(Cc2ccccc2)c1 REAL300012003089
CCc1oc2ccccc2c1CNC(Cc1cscn1)C(=O)O REAL300012003090
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2[N+](=O)[O-])o1 REAL300012003091
O=C(O)C(Cc1cscn1)NCc1csc(-c2ccc(F)cc2)n1 REAL300012003092
O=C(O)C(Cc1cscn1)NCc1ccccc1OC(F)(F)F REAL300012003093
O=C(O)C(Cc1cscn1)NCc1ccc(SC(F)(F)F)cc1 REAL300012003094
COc1cc(CNC(Cc2cscn2)C(=O)O)c([N+](=O)[O-])cc1O REAL300012003095
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(Cl)c1 REAL300012003096
O=C(O)C(Cc1cscn1)NCc1ccc(OC(F)(F)F)cc1 REAL300012003097
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccc([N+](=O)[O-])cc2)s1 REAL300012003098
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2[N+](=O)[O-])s1 REAL300012003099
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccc(F)cc1 REAL300012003100
Cc1ccc(-c2n[nH]cc2CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003101
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1cccs1 REAL300012003102
COc1ccc(-c2n[nH]cc2CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003103
O=C(O)C(Cc1cscn1)NCc1csc2ccccc12 REAL300012003104
CCOc1c(CNC(Cc2cscn2)C(=O)O)c(C)nn1CC(C)C REAL300012003105
O=C(O)C(Cc1cscn1)NCC1=Cc2ccccc2OC1 REAL300012003106
Cc1ccc(-c2ccc(CNC(Cc3cscn3)C(=O)O)o2)cc1 REAL300012003107
Cc1ccc(-c2n[nH]cc2CNC(Cc2cscn2)C(=O)O)o1 REAL300012003108
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1cccnc1 REAL300012003109
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccc2c(c1)OCCO2 REAL300012003110
O=C(O)C(Cc1cscn1)NCc1ccc(OCC2CCCO2)cc1 REAL300012003111
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)s1 REAL300012003112
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccc(F)cc2)s1 REAL300012003113
O=C(O)C(Cc1cscn1)NCc1cccc2cccnc12 REAL300012003114
O=C(O)C(Cc1cscn1)NCc1ccccc1OCc1ccccn1 REAL300012003115
COc1nc2ccccc2cc1CNC(Cc1cscn1)C(=O)O REAL300012003116
O=C(O)C(Cc1cscn1)NCc1ccc(-n2cccn2)cc1 REAL300012003117
O=C(O)C(Cc1cscn1)NCc1ccc(-n2cncn2)cc1 REAL300012003118
CC(C)n1ncc2cc(CNC(Cc3cscn3)C(=O)O)c(Cl)nc21 REAL300012003119
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2Cl)s1 REAL300012003120
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OCc1ccncc1 REAL300012003121
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2F)s1 REAL300012003122
O=C(O)C(Cc1cscn1)NCc1cc(C(F)(F)F)ccc1Cl REAL300012003123
O=C(O)C(Cc1cscn1)NCc1ccc(F)cc1Cl REAL300012003124
O=C(O)C(Cc1cscn1)NCc1ccc(F)c(Cl)c1 REAL300012003125
O=C(O)C(Cc1cscn1)NCc1ccc(F)c(C(F)(F)F)c1 REAL300012003126
CCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003127
O=C(O)C(Cc1cscn1)NCc1cc(Cl)ccc1Cl REAL300012003128
O=C(O)C(Cc1cscn1)NCc1ccc(F)cc1C(F)(F)F REAL300012003129
O=C(O)C(Cc1cscn1)NCc1cc(F)c(F)c(F)c1 REAL300012003130
O=C(O)C(Cc1cscn1)NCc1cc(F)cc(C(F)(F)F)c1 REAL300012003131
O=C(O)C(Cc1cscn1)NCc1cc(C(F)(F)F)ccc1F REAL300012003132
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(Cl)c1OC REAL300012003133
O=C(O)C(Cc1cscn1)NCc1cc2ccccc2s1 REAL300012003134
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)c(F)c1 REAL300012003135
O=C(O)C(Cc1cscn1)NCc1cc(Cl)ccc1OC(F)F REAL300012003136
O=C(O)C(Cc1cscn1)NCc1ccc(-c2cccc(Cl)c2)s1 REAL300012003137
N#Cc1cccc(COc2cccc(CNC(Cc3cscn3)C(=O)O)c2)c1 REAL300012003138
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccc2c(c1)OCO2 REAL300012003139
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OCC(F)(F)F REAL300012003140
O=C(O)C(Cc1cscn1)NCc1ccc(OCc2ccncc2)cc1 REAL300012003141
CC(C)c1nn(C)cc1CNC(Cc1cscn1)C(=O)O REAL300012003142
O=C(O)C(Cc1cscn1)NCc1cc(Br)c2c(c1)OCCO2 REAL300012003143
O=C(O)C(Cc1cscn1)NCc1ccc(-n2ccc(C(F)(F)F)n2)cc1 REAL300012003144
CC(C)c1nn(C)c(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003145
COCCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003146
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1Cl REAL300012003147
O=C(O)C(Cc1cscn1)NCc1csc(-c2ccccn2)n1 REAL300012003148
CC(C)n1c(CNC(Cc2cscn2)C(=O)O)nc2ccccc21 REAL300012003149
CC(C)(C)OC(=O)Nc1ccc(CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003150
O=C(O)C(Cc1cscn1)NCc1cccc(OCC(F)(F)F)c1 REAL300012003151
O=C(O)C(Cc1cscn1)NCc1cccc2c1OCCO2 REAL300012003152
O=C(O)C(Cc1cscn1)NCc1cccc2c1OCCCO2 REAL300012003153
CCCn1c(CNC(Cc2cscn2)C(=O)O)nc2ccccc21 REAL300012003154
CCCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003155
O=C(O)C(Cc1cscn1)NCc1cc(-c2ccccc2)cs1 REAL300012003156
O=C(O)C(Cc1cscn1)NCc1cccc(OC2CCCC2)c1 REAL300012003157
CC(C)Oc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003158
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2cc3ccccc3o2)n1 REAL300012003159
Cc1ccc(-c2nc(CNC(Cc3cscn3)C(=O)O)cs2)cc1 REAL300012003160
CC(C)c1nc(CNC(Cc2cscn2)C(=O)O)cs1 REAL300012003161
O=C(O)C(Cc1cscn1)NCc1cccc(OCc2ccccc2F)c1 REAL300012003162
O=C(O)C(Cc1cscn1)NCc1csc(COc2ccccc2)n1 REAL300012003163
Cc1ccc(OCc2nc(CNC(Cc3cscn3)C(=O)O)cs2)cc1 REAL300012003164
CC(C)(C)c1nc(CNC(Cc2cscn2)C(=O)O)cs1 REAL300012003165
O=C(O)C(Cc1cscn1)NCc1csc(-c2ccsc2)n1 REAL300012003166
O=C(O)C(Cc1cscn1)NCc1ccc(-c2cccc(F)c2)s1 REAL300012003167
CN(C)C(=O)COc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003168
O=C(O)C(Cc1cscn1)NCc1ccccc1OC1CCCC1 REAL300012003169
COc1ccc(OCc2ccccn2)c(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003170
Cc1ccc(-c2ccc(CNC(Cc3cscn3)C(=O)O)s2)cc1 REAL300012003171
O=C(O)C(Cc1cscn1)NCc1cc([N+](=O)[O-])ccc1OC(F)F REAL300012003172
COc1c(Cl)cc(Cl)cc1CNC(Cc1cscn1)C(=O)O REAL300012003173
O=C(O)C(Cc1cscn1)NCc1cc(Br)ccc1Cl REAL300012003174
O=C(O)C(Cc1cscn1)NCc1cc(Cl)ccc1Br REAL300012003175
O=C(O)C(Cc1cscn1)NCc1ccc(Oc2cc(F)cc(F)c2)cc1 REAL300012003176
CCOc1c(OC)cc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003177
COCCCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003178
Cc1cc(CNC(Cc2cscn2)C(=O)O)cnc1Cl REAL300012003179
COc1ccc(OC(F)F)c(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003180
O=C(O)C(Cc1cscn1)NCc1c(Cl)cccc1OC(F)F REAL300012003181
O=C(O)C(Cc1cscn1)NCc1cccc(OCCCc2ccccc2)c1 REAL300012003182
Cc1cc(CNC(Cc2cscn2)C(=O)O)ccc1Oc1cccnc1 REAL300012003183
O=C(COc1ccccc1CNC(Cc1cscn1)C(=O)O)NCC1CC1 REAL300012003184
Cc1ccc(-c2ncc(CNC(Cc3cscn3)C(=O)O)s2)cc1 REAL300012003185
O=C(O)C(Cc1cscn1)NCc1cc(Cl)cc2cccnc12 REAL300012003186
O=C(O)C(Cc1cscn1)NCc1ccc(F)c2cccnc12 REAL300012003187
O=C(O)C(Cc1cscn1)NCc1cc(F)cc2cccnc12 REAL300012003188
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)c2cccnc12 REAL300012003189
O=C(O)C(Cc1cscn1)NCc1ccc(-c2c(F)cccc2F)o1 REAL300012003190
Cc1cc(F)ccc1-c1ccc(CNC(Cc2cscn2)C(=O)O)o1 REAL300012003191
CCc1ccc(-c2ccc(CNC(Cc3cscn3)C(=O)O)o2)cc1 REAL300012003192
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(OC(F)F)c1 REAL300012003193
COc1ccc2oc(CNC(Cc3cscn3)C(=O)O)cc2c1 REAL300012003194
O=C(O)C(Cc1cscn1)NCC=Cc1ccc(Cl)cc1 REAL300012003195
Cc1oc2ccccc2c1CNC(Cc1cscn1)C(=O)O REAL300012003196
O=C(O)C(Cc1cscn1)NCc1coc2ccccc12 REAL300012003197
O=C(O)C(Cc1cscn1)NCc1ccc(Oc2ccccc2)o1 REAL300012003198
Cc1ccc(CNC(Cc2cscn2)C(=O)O)cc1Br REAL300012003199
O=C(O)C(Cc1cscn1)NCC=Cc1ccc(F)cc1F REAL300012003200
Cc1cc(CNC(Cc2cscn2)C(=O)O)ccc1Br REAL300012003201
O=C(O)C(Cc1cscn1)NCc1ccn(-c2ccccc2)n1 REAL300012003202
O=C(O)C(Cc1cscn1)NCc1ccsc1Cl REAL300012003203
O=C(O)C(Cc1cscn1)NCc1cc(Cl)cc2c1OCC2 REAL300012003204
O=C(O)C(Cc1cscn1)NCc1cc2c(F)cccc2[nH]1 REAL300012003205
O=C(O)C(Cc1cscn1)NCc1cc2ccc(F)cc2[nH]1 REAL300012003206
CCOc1cccc(CNC(Cc2cscn2)C(=O)O)n1 REAL300012003207
Cc1cc(CNC(Cc2cscn2)C(=O)O)cc2cccnc12 REAL300012003208
Cc1cc(CNC(Cc2cscn2)C(=O)O)ccc1Cl REAL300012003209
O=C(O)C(Cc1cscn1)NCc1cnc2ccsc2c1 REAL300012003210
CC(C)(C)c1ccc(-c2ccc(CNC(Cc3cscn3)C(=O)O)o2)cc1 REAL300012003211
CCC(C)CN(C)c1ccc(F)cc1CNC(Cc1cscn1)C(=O)O REAL300012003212
CCCCCN(C)c1ccc(F)cc1CNC(Cc1cscn1)C(=O)O REAL300012003213
CCCc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003214
CCN(c1ccccc1)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003215
CCN(CC)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1F REAL300012003216
COc1cc(CNC(Cc2cscn2)C(=O)O)c(SC)cc1OC REAL300012003217
COc1ccc2nc(CNC(Cc3cscn3)C(=O)O)sc2c1 REAL300012003218
Cn1c(CNC(Cc2cscn2)C(=O)O)nc2ccc(Cl)cc21 REAL300012003219
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1C#N REAL300012003220
O=C(O)C(Cc1cscn1)NCc1ccc(SC(F)F)cc1 REAL300012003221
Cc1cc(Cl)cc(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003222
O=C(O)C(Cc1cscn1)NCc1ccc(OC(F)F)c(F)c1 REAL300012003223
CCOc1ccc(CNC(Cc2cscn2)C(=O)O)nc1 REAL300012003224
Cc1cc(C(F)(F)F)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003225
COc1cc(CNC(Cc2cscn2)C(=O)O)cc(Cl)c1OC REAL300012003226
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCC(C)C REAL300012003227
CCCOc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC REAL300012003228
O=C(O)C(Cc1cscn1)NCc1ccc(Br)s1 REAL300012003229
CCOc1cc(CNC(Cc2cscn2)C(=O)O)cc(Cl)c1OC REAL300012003230
C=CCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003231
COc1cccc(CNC(Cc2cscn2)C(=O)O)c1OC(C)C REAL300012003232
CCOc1c(Cl)cc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003233
CCCOc1c(CNC(Cc2cscn2)C(=O)O)cccc1OCC REAL300012003234
CCCCOc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC REAL300012003235
CCCOc1c(Cl)cc(CNC(Cc2cscn2)C(=O)O)cc1OCC REAL300012003236
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC(F)F REAL300012003237
CCOc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC(F)F REAL300012003238
Cc1cc(CNC(Cc2cscn2)C(=O)O)cc(C)c1OC(F)F REAL300012003239
CCOc1cc2c(cc1CNC(Cc1cscn1)C(=O)O)OC(C)C2 REAL300012003240
COc1cc(CNC(Cc2cscn2)C(=O)O)cc2c1OCCO2 REAL300012003241
O=C(O)C(Cc1cscn1)NCc1ccc(-c2nc3ccccc3s2)o1 REAL300012003242
CCCCn1nc(C)c(CNC(Cc2cscn2)C(=O)O)c1Cl REAL300012003243
CCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1OC(F)F REAL300012003244
O=C(O)C(Cc1cscn1)NCc1ccccc1OCC(=O)N1CCCC1 REAL300012003245
Cc1cc(C)c(CNC(Cc2cscn2)C(=O)O)cc1C REAL300012003246
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2)s1 REAL300012003247
CCCOc1c(Cl)cc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003248
CC(C)(C)c1nn(Cc2ccccc2)cc1CNC(Cc1cscn1)C(=O)O REAL300012003249
O=C(O)C(Cc1cscn1)NCc1ccc(-c2cccc(F)c2F)o1 REAL300012003250
CC(C)(CNC(Cc1cscn1)C(=O)O)c1ccccc1 REAL300012003251
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(C2CCCCC2)n1 REAL300012003252
CC(CCc1ccccc1)CNC(Cc1cscn1)C(=O)O REAL300012003253
CC1(C)CCc2nc(CNC(Cc3cscn3)C(=O)O)sc2C1 REAL300012003254
CCc1cccc(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003255
Cc1cc2cc(CNC(Cc3cscn3)C(=O)O)oc2cc1C REAL300012003256
CCCC1CCC(CNC(Cc2cscn2)C(=O)O)CC1 REAL300012003257
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccc(Cl)cc1 REAL300012003258
O=C(O)C(Cc1cscn1)NCc1ccc(-n2ccnc2)cc1 REAL300012003259
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2F)o1 REAL300012003260
O=C(O)C(Cc1cscn1)NCc1cc(Cl)c2c(c1)OCCO2 REAL300012003261
CCCCc1oc2ccccc2c1CNC(Cc1cscn1)C(=O)O REAL300012003262
O=C(O)C(Cc1cscn1)NCc1ccc(-n2cnc3ccccc32)cc1 REAL300012003263
Cc1nn(-c2ccc(F)cc2)c(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003264
O=C(O)C(Cc1cscn1)NCc1cc(Cl)c2c(c1)OCCCO2 REAL300012003265
COc1ccc(C)cc1CNC(Cc1cscn1)C(=O)O REAL300012003266
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1F REAL300012003267
O=C(O)C(Cc1cscn1)NCC1CCC(C(F)(F)F)CC1 REAL300012003268
CC(C)C1CC(CNC(Cc2cscn2)C(=O)O)CCO1 REAL300012003269
O=C(O)C(Cc1cscn1)NCc1ccc(OCC(F)(F)F)c(F)c1 REAL300012003270
O=C(O)C(Cc1cscn1)NCc1cn(-c2ccc(F)cc2Cl)nn1 REAL300012003271
O=C(O)C(Cc1cscn1)NCc1cn(-c2ccc(F)c(Cl)c2)nn1 REAL300012003272
CCSc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003273
O=C(O)C(Cc1cscn1)NCc1c(O)ccc(Cl)c1F REAL300012003274
CCn1nc(CNC(Cc2cscn2)C(=O)O)c2ccccc21 REAL300012003275
COCCC1(CNC(Cc2cscn2)C(=O)O)CCCCC1 REAL300012003276
O=C(O)C(Cc1cscn1)NCc1cc(Br)c(Cl)s1 REAL300012003277
CCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003278
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccc(Cl)c(Cl)c2)o1 REAL300012003279
Cc1nn(Cc2ccccc2)c(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003280
O=C(O)C(Cc1cscn1)NCc1cc2ccccc2o1 REAL300012003281
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2)o1 REAL300012003282
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC(C)C REAL300012003283
CCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCC REAL300012003284
Cc1ccc(CNC(Cc2cscn2)C(=O)O)cc1[N+](=O)[O-] REAL300012003285
CC(C)Oc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003286
CCCCCCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003287
CC(CNC(Cc1cscn1)C(=O)O)Cc1ccc(C(C)(C)C)cc1 REAL300012003288
O=C(O)C(Cc1cscn1)NCc1cccc2cc[nH]c12 REAL300012003289
O=C(O)C(Cc1cscn1)NCc1sccc1Br REAL300012003290
O=C(O)C(Cc1cscn1)NCc1ccccc1N1CCOCC1 REAL300012003291
O=C(O)C(Cc1cscn1)NCc1cc(F)ccc1Br REAL300012003292
CC(C)Cc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003293
Cc1ccc(-c2cccc(CNC(Cc3cscn3)C(=O)O)c2)cc1 REAL300012003294
COc1ccc(Br)c(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003295
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1[N+](=O)[O-] REAL300012003296
O=C(O)C(Cc1cscn1)NCc1cc(Cl)cc(Cl)c1 REAL300012003297
O=C(O)C(Cc1cscn1)NCc1cc(F)cc(Cl)c1 REAL300012003298
O=C(O)C(Cc1cscn1)NCc1cc(Br)co1 REAL300012003299
Cc1ccccc1-c1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003300
O=C(O)C(Cc1cscn1)NCc1cc(C(F)(F)F)cc(C(F)(F)F)c1 REAL300012003301
O=C(O)C(Cc1cscn1)NCc1cccc(OC(F)F)c1 REAL300012003302
CCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCC REAL300012003303
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)cc1F REAL300012003304
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)c(C(F)(F)F)c1 REAL300012003305
O=C(O)C(Cc1cscn1)NCc1ccc(F)cc1Br REAL300012003306
O=C(O)C(Cc1cscn1)NCc1cccc(OC(F)(F)F)c1 REAL300012003307
O=C(O)C(Cc1cscn1)NCc1cc(Cl)ccc1F REAL300012003308
COc1ccccc1-c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003309
O=C(O)C(Cc1cscn1)NCc1ccc(-c2cccc(C(F)(F)F)c2)o1 REAL300012003310
O=C(O)C(Cc1cscn1)NCc1cccc(Cl)c1F REAL300012003311
COc1ccc(CNC(Cc2cscn2)C(=O)O)c2ccccc12 REAL300012003312
O=C(O)C(Cc1cscn1)NCc1n[nH]cc1-c1ccccc1 REAL300012003313
Cn1c(CNC(Cc2cscn2)C(=O)O)nc2ccccc21 REAL300012003314
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(Br)c1O REAL300012003315
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)CCO2 REAL300012003316
O=C(O)C(Cc1cscn1)NCc1csc(Br)c1 REAL300012003317
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCc1cccnc1 REAL300012003318
COc1cc(CNC(Cc2cscn2)C(=O)O)c(-c2ccccc2)cc1OC REAL300012003319
O=C(O)C(Cc1cscn1)NCc1cccc(-c2ccccc2)c1 REAL300012003320
O=C(O)C(Cc1cscn1)NCc1ccccc1OCc1cccnc1 REAL300012003321
O=C(O)C(Cc1cscn1)NCc1ccc(N2CCCC2)nc1 REAL300012003322
O=C(O)C(Cc1cscn1)NCc1cccc2[nH]ccc12 REAL300012003323
O=C(O)C(Cc1cscn1)NCc1ccc(Br)c(F)c1 REAL300012003324
O=C(O)C(Cc1cscn1)NCc1cccc(-c2ccccn2)c1 REAL300012003325
O=C(O)C(Cc1cscn1)NCc1cccc(-c2cccnc2)c1 REAL300012003326
O=C(O)C(Cc1cscn1)NCc1cccc(-c2ccncc2)c1 REAL300012003327
Cc1nn(C(C)(C)C)c(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003328
CN1CCN(c2ccc(CNC(Cc3cscn3)C(=O)O)cc2)CC1 REAL300012003329
O=C(O)C(Cc1cscn1)NCc1ccc(Oc2cnccn2)cc1 REAL300012003330
CNC(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003331
O=C(O)C(Cc1cscn1)NCc1cnn(-c2ccc(F)cc2)c1 REAL300012003332
Cc1nn(-c2ccc(Cl)cc2)c(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003333
O=C(O)C(Cc1cscn1)NCc1cnn(-c2ccc(Cl)cc2)c1 REAL300012003334
Cc1nn(-c2ccc(F)cc2F)c(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003335
Cc1cc(CNC(Cc2cscn2)C(=O)O)cc(C)c1OCc1ccccn1 REAL300012003336
O=C(O)C(Cc1cscn1)NCc1ccc(OCC(F)(F)F)cc1 REAL300012003337
O=C(O)C(Cc1cscn1)NCc1ccc2ccccc2c1 REAL300012003338
COc1cccc2cc(CNC(Cc3cscn3)C(=O)O)oc12 REAL300012003339
CC(C)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1[N+](=O)[O-] REAL300012003340
O=C(O)C(Cc1cscn1)NCc1cc(Br)c2c(c1)OCO2 REAL300012003341
Cc1nn(Cc2ccccc2)c(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003342
CCOc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OCC(C)C REAL300012003343
O=C(O)C(Cc1cscn1)NCc1cc(Br)ccc1F REAL300012003344
O=C(O)C(Cc1cscn1)NCc1ccc(Br)cc1F REAL300012003345
COc1cc(CNC(Cc2cscn2)C(=O)O)cc(OC)c1 REAL300012003346
COc1ccc2cc(CNC(Cc3cscn3)C(=O)O)ccc2c1 REAL300012003347
O=C(O)C(Cc1cscn1)NCc1cc([N+](=O)[O-])ccc1O REAL300012003348
O=C(O)C(Cc1cscn1)NCc1cc(Br)cs1 REAL300012003349
CCCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCC REAL300012003350
Cc1nn(-c2ccccc2)c(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003351
COc1cccc(CNC(Cc2cscn2)C(=O)O)c1OC(F)F REAL300012003352
O=C(O)C(Cc1cscn1)NCc1ccc(CSC(F)F)o1 REAL300012003353
O=C(O)C(Cc1cscn1)NCc1cc2ccccc2nc1N1CCCCC1 REAL300012003354
O=C(O)C(Cc1cscn1)NCc1cc2ccccc2nc1O REAL300012003355
O=C(O)C(Cc1cscn1)NCc1cc(Cl)cc(Cl)c1O REAL300012003356
O=C(O)C(Cc1cscn1)NCc1ccc(F)c(Br)c1 REAL300012003357
Cc1ccc(COc2ccc(CNC(Cc3cscn3)C(=O)O)cc2)cc1 REAL300012003358
O=C(O)C(Cc1cscn1)NCc1ccc(N2CCCCC2)cc1 REAL300012003359
CCCCCCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003360
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1SC REAL300012003361
N#CCCCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003362
CCCCCOc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC REAL300012003363
CCC(C)Oc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC REAL300012003364
CCCCCCCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003365
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCCCC#N REAL300012003366
C=C(C)COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC REAL300012003367
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCCC(C)C REAL300012003368
C=CCc1cc(CNC(Cc2cscn2)C(=O)O)cc(OC)c1O REAL300012003369
O=C(O)C(Cc1cscn1)NCc1cc(-c2ccccc2)[nH]n1 REAL300012003370
CCOc1ccc([N+](=O)[O-])cc1CNC(Cc1cscn1)C(=O)O REAL300012003371
Cc1nn(C)c(OCC(F)(F)F)c1CNC(Cc1cscn1)C(=O)O REAL300012003372
O=C(O)C(Cc1cscn1)NCc1cn(-c2ccccc2)nn1 REAL300012003373
O=C(O)C(Cc1cscn1)NCc1nc(-c2ccccc2)cs1 REAL300012003374
O=C(O)C(Cc1cscn1)NCc1ccc(N2CCOCC2)c(F)c1 REAL300012003375
Cn1cnc2cc(CNC(Cc3cscn3)C(=O)O)ccc21 REAL300012003376
CCn1nc(C)c(CNC(Cc2cscn2)C(=O)O)c1C REAL300012003377
C=CCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1Cl REAL300012003378
O=C(O)C(Cc1cscn1)NCc1cnc(-c2ccccc2)s1 REAL300012003379
COc1cc(CNC(Cc2cscn2)C(=O)O)c2c(c1)CC(C)O2 REAL300012003380
CC1(C)Cc2cc(CNC(Cc3cscn3)C(=O)O)ccc2O1 REAL300012003381
O=C(O)C(Cc1cscn1)NCc1coc(-c2ccccc2)n1 REAL300012003382
O=C(O)C(Cc1cscn1)NCc1csc(-c2cccs2)n1 REAL300012003383
Cc1cccc(-c2[nH]ncc2CNC(Cc2cscn2)C(=O)O)c1 REAL300012003384
O=C(O)C(Cc1cscn1)NCc1cc(Cl)cc(C(F)(F)F)c1 REAL300012003385
O=C(O)C(Cc1cscn1)NCc1ccc(Br)cc1Cl REAL300012003386
Cc1ccc(CNC(Cc2cscn2)C(=O)O)c(Br)c1 REAL300012003387
CC(C)COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003388
COCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003389
N#Cc1ccccc1COc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003390
O=C(O)C(Cc1cscn1)NCc1ccc(OC(F)F)c(Cl)c1 REAL300012003391
O=C(O)C(Cc1cscn1)NCc1csc(-c2cccc([N+](=O)[O-])c2)n1 REAL300012003392
Cn1nc(-c2ccccc2)c(CNC(Cc2cscn2)C(=O)O)c1Cl REAL300012003393
COc1cc2c(cc1CNC(Cc1cscn1)C(=O)O)OCO2 REAL300012003394
O=C(O)C(Cc1cscn1)NCc1cncc2ccccc12 REAL300012003395
CC(C)COc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003396
Cc1cc(Cl)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003397
O=C(O)C(Cc1cscn1)NCC=Cc1ccc(F)cc1 REAL300012003398
O=C(O)C(Cc1cscn1)NCc1cncc(Br)c1 REAL300012003399
Cn1nnc2cc(CNC(Cc3cscn3)C(=O)O)ccc21 REAL300012003400
CC1(C)Cc2cccc(CNC(Cc3cscn3)C(=O)O)c2O1 REAL300012003401
O=C(O)C(Cc1cscn1)NCc1cc(Br)cc2c1OCC2 REAL300012003402
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2ccccc2)n1 REAL300012003403
O=C(O)C(Cc1cscn1)NCc1cccc(-n2cccn2)c1 REAL300012003404
Cc1cc(CNC(Cc2cscn2)C(=O)O)sc1Br REAL300012003405
O=C(O)C(Cc1cscn1)NCc1ccc(Br)c2cccnc12 REAL300012003406
Cc1ccc2cc(CNC(Cc3cscn3)C(=O)O)ccc2n1 REAL300012003407
COc1ccc(Oc2ccc(CNC(Cc3cscn3)C(=O)O)cc2)cc1 REAL300012003408
O=C(O)C(Cc1cscn1)NCc1ncccc1C(F)(F)F REAL300012003409
Cc1cc(C)cc(-c2ccc(CNC(Cc3cscn3)C(=O)O)cc2)c1 REAL300012003410
Cc1cc(CNC(Cc2cscn2)C(=O)O)ccc1-n1cncn1 REAL300012003411
O=C(O)C(Cc1cscn1)NCc1cc2cc(F)ccc2o1 REAL300012003412
O=C(O)C(Cc1cscn1)NCc1ccc(OCC(F)F)cc1 REAL300012003413
COCc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003414
Cc1nn(-c2ccc(Cl)cc2)cc1CNC(Cc1cscn1)C(=O)O REAL300012003415
O=C(O)C(Cc1cscn1)NCc1cccc(OCc2ccc(F)cc2)c1 REAL300012003416
CCCCOc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003417
O=C(O)C(Cc1cscn1)NCc1ccc(Sc2ccccc2)cc1 REAL300012003418
Cc1cc(CNC(Cc2cscn2)C(=O)O)c(OC(F)F)cc1C REAL300012003419
COc1cc(C)c(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003420
Cn1c(CNC(Cc2cscn2)C(=O)O)nc2cc(Cl)ccc21 REAL300012003421
CS(=O)(=O)c1cccc(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003422
CCS(=O)(=O)c1c(Cl)cccc1CNC(Cc1cscn1)C(=O)O REAL300012003423
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccsc1 REAL300012003424
CSc1cc(Br)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003425
O=C(O)C(Cc1cscn1)NCc1cnn(Cc2ccc(F)cc2)c1 REAL300012003426
CC1CCc2nc(CNC(Cc3cscn3)C(=O)O)sc2C1 REAL300012003427
CC(C)(C)C1CCC(CNC(Cc2cscn2)C(=O)O)CC1 REAL300012003428
COc1cc(-c2ccccc2)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003429
COc1ccc(-c2ccccc2)cc1CNC(Cc1cscn1)C(=O)O REAL300012003430
COc1ccc(-c2ccncc2)cc1CNC(Cc1cscn1)C(=O)O REAL300012003431
O=C(O)C(Cc1cscn1)NCc1ccc(OCC2CC2)cc1 REAL300012003432
COc1cc(Cl)c(CNC(Cc2cscn2)C(=O)O)cc1Cl REAL300012003433
CC(C)Cc1ncc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003434
O=C(O)C(Cc1cscn1)NCc1cnc(-c2cccs2)s1 REAL300012003435
O=C(O)C(Cc1cscn1)NCc1cnc(-c2ccsc2)s1 REAL300012003436
Cc1ccc(-c2ncc(CNC(Cc3cscn3)C(=O)O)s2)o1 REAL300012003437
Cc1cc(Br)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003438
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)c(Br)c1 REAL300012003439
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccccc1F REAL300012003440
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccncc2)cc1F REAL300012003441
O=C(O)C(Cc1cscn1)NCc1c(Cl)oc2ccccc12 REAL300012003442
COCCOc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003443
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)cc1Br REAL300012003444
COc1c(Br)cccc1CNC(Cc1cscn1)C(=O)O REAL300012003445
O=C(O)C(Cc1cscn1)NCc1nc2c(s1)CCC2 REAL300012003446
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2cccs2)n1 REAL300012003447
O=C(O)C(Cc1cscn1)NCc1cc(Cl)ccc1OC1CCCC1 REAL300012003448
O=C(O)C(Cc1cscn1)NCc1c(Cl)cccc1Oc1ccccc1 REAL300012003449
O=C(O)C(Cc1cscn1)NCc1cc(Cl)ccc1OCC1CCCO1 REAL300012003450
CC(C)(C)c1nn(-c2ccccc2)cc1CNC(Cc1cscn1)C(=O)O REAL300012003451
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccc(F)cc2)o1 REAL300012003452
CC(C)(C)c1ncc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003453
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)OCCO2 REAL300012003454
O=C(O)C(Cc1cscn1)NCc1cccc(Br)c1 REAL300012003455
O=C(O)C(Cc1cscn1)NCc1cnn(-c2ccccc2)c1 REAL300012003456
O=C(O)C(Cc1cscn1)NCc1cnn(Cc2ccccc2Cl)c1 REAL300012003457
CC(C)(C)n1cc(CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003458
CC(=O)Nc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003459
O=C(O)C(Cc1cscn1)NCc1cccc([N+](=O)[O-])c1 REAL300012003460
O=C(O)C(Cc1cscn1)NCc1ccc([N+](=O)[O-])cc1 REAL300012003461
O=C(O)C(Cc1cscn1)NCc1cccc2ccccc12 REAL300012003462
CN(C)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003463
CCN(CC)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003464
O=C(O)C(Cc1cscn1)NCc1ccc(Br)cc1 REAL300012003465
COc1cc(CNC(Cc2cscn2)C(=O)O)cc(OC)c1OC REAL300012003466
O=C(O)C(Cc1cscn1)NCc1c(F)cccc1Cl REAL300012003467
O=C(O)C(Cc1cscn1)NCc1ccccc1OC(F)F REAL300012003468
COc1cccc(CNC(Cc2cscn2)C(=O)O)c1OC REAL300012003469
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)cc1Cl REAL300012003470
O=C(O)C(Cc1cscn1)NCc1ccc(N2CCOCC2)cc1 REAL300012003471
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003472
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(OC)c1 REAL300012003473
O=C(O)C(Cc1cscn1)NCc1ccc(C(F)(F)F)cc1 REAL300012003474
O=C(O)C(Cc1cscn1)NCc1cccc(Cl)c1Cl REAL300012003475
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)c(Cl)c1 REAL300012003476
CCN(Cc1ccccc1)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003477
O=C(O)C(Cc1cscn1)NCc1ccc(OC(F)F)cc1 REAL300012003478
O=C(O)C(Cc1cscn1)NCc1ccccc1C(F)(F)F REAL300012003479
CCCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003480
CC(C)CCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003481
CCCCCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003482
O=C(O)C(Cc1cscn1)NCc1cccc(Oc2ccccc2)c1 REAL300012003483
CCCOc1ccc(CNC(Cc2cscn2)C(=O)O)c(OCCC)c1 REAL300012003484
CC(=Cc1ccccc1)CNC(Cc1cscn1)C(=O)O REAL300012003485
CCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003486
CC(C)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003487
O=C(O)C(Cc1cscn1)NCc1cccc(C(F)(F)F)c1 REAL300012003488
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(OC)c1OC REAL300012003489
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OCc1ccccc1 REAL300012003490
CCOc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003491
CCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003492
COc1ccc(Br)cc1CNC(Cc1cscn1)C(=O)O REAL300012003493
COc1cc(CNC(Cc2cscn2)C(=O)O)cc(Br)c1O REAL300012003494
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2)cc1 REAL300012003495
COc1ccc2ccccc2c1CNC(Cc1cscn1)C(=O)O REAL300012003496
CSc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003497
O=C(O)C(Cc1cscn1)NCc1c(Cl)cccc1Cl REAL300012003498
COc1cc(OC)c(OC)cc1CNC(Cc1cscn1)C(=O)O REAL300012003499
Cc1cc(C)c(CNC(Cc2cscn2)C(=O)O)c(C)c1 REAL300012003500
Cc1nn(-c2ccccc2)c(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003501
O=C(O)C(Cc1cscn1)NCc1cccc(OCc2ccccc2)c1 REAL300012003502
O=C(O)C(Cc1cscn1)NCc1ccccc1Br REAL300012003503
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1O REAL300012003504
Cc1nn(C)c(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003505
O=C(O)C(Cc1cscn1)NCc1cnn(CC(F)(F)F)c1 REAL300012003506
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(C(C)(C)C)n1 REAL300012003507
O=C(O)C(Cc1cscn1)NCc1ccccc1I REAL300012003508
O=C(O)C(Cc1cscn1)NCc1ccc(OC(F)F)cc1OC(F)F REAL300012003509
O=C(O)C(Cc1cscn1)NCc1ccc(N2CCCCC2)c([N+](=O)[O-])c1 REAL300012003510
CN(CCC#N)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003511
O=C(O)C(Cc1cscn1)NCc1c(OC(F)F)ccc2ccccc12 REAL300012003512
CCOc1cccc(CNC(Cc2cscn2)C(=O)O)c1OC REAL300012003513
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OCC(N)=O REAL300012003514
C#CCOc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003515
CCNC(=O)COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003516
COc1cc(CNC(Cc2cscn2)C(=O)O)cc2c1OCO2 REAL300012003517
O=C(O)C(Cc1cscn1)NCc1cnn(-c2ccccc2)n1 REAL300012003518
COc1cc2c(cc1CNC(Cc1cscn1)C(=O)O)OC(C)C2 REAL300012003519
COc1cc(CNC(Cc2cscn2)C(=O)O)cc(OC)c1OCC(N)=O REAL300012003520
COc1cc(CNC(Cc2cscn2)C(=O)O)cc(Cl)c1OCC(N)=O REAL300012003521
CCN(C(C)=O)c1nc(CNC(Cc2cscn2)C(=O)O)cs1 REAL300012003522
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1C REAL300012003523
CC(C)(C)c1n[nH]cc1CNC(Cc1cscn1)C(=O)O REAL300012003524
COc1cccc(OC)c1CNC(Cc1cscn1)C(=O)O REAL300012003525
COc1ccc(F)c(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003526
O=C(O)C(Cc1cscn1)NCc1cccc(I)c1 REAL300012003527
O=C(O)C(Cc1cscn1)NCc1ccc(I)cc1 REAL300012003528
CSc1ccc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003529
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccc(C(F)(F)F)cc1 REAL300012003530
Cc1ccccc1-c1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003531
O=C(O)C(Cc1cscn1)NCc1cccc2c1OCO2 REAL300012003532
O=C(O)C(Cc1cscn1)NCc1sccc1Cl REAL300012003533
CS(=O)(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003534
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccc(Cl)cc2)cc1 REAL300012003535
COc1ccc(F)cc1CNC(Cc1cscn1)C(=O)O REAL300012003536
NC(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003537
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1F REAL300012003538
COc1ccc(Cl)cc1CNC(Cc1cscn1)C(=O)O REAL300012003539
COC(=O)c1cc(CNC(Cc2cscn2)C(=O)O)cn1C REAL300012003540
Cc1ccc(CNC(Cc2cscn2)C(=O)O)cc1Cl REAL300012003541
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1C REAL300012003542
N#Cc1ccc(CNC(Cc2cscn2)C(=O)O)c(F)c1 REAL300012003543
O=C(O)C(Cc1cscn1)NCc1cccc(OCc2ccccn2)c1 REAL300012003544
O=C(O)C(Cc1cscn1)NCc1ccc(Br)cn1 REAL300012003545
O=C(O)C(Cc1cscn1)NCc1cnc(N2CCOCC2)s1 REAL300012003546
C#CCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003547
O=C(O)C(Cc1cscn1)NCc1cn2ccccc2n1 REAL300012003548
Cc1nn(C)c2ncc(CNC(Cc3cscn3)C(=O)O)cc12 REAL300012003549
O=C(O)C(Cc1cscn1)NCc1csc(C2CC2)n1 REAL300012003550
O=C(O)C(Cc1cscn1)NCc1cn2cc(Cl)ccc2n1 REAL300012003551
CCOCc1cc(CNC(Cc2cscn2)C(=O)O)ccc1OC REAL300012003552
NC(=O)c1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003553
O=C(O)C(Cc1cscn1)NCc1nccn1CC(F)(F)F REAL300012003554
O=C(O)C(Cc1cscn1)NCc1csc(-c2ccc3c(c2)OCO3)n1 REAL300012003555
COc1cccc(CNC(Cc2cscn2)C(=O)O)c1F REAL300012003556
O=C(O)C(Cc1cscn1)NCc1c(F)cccc1Br REAL300012003557
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)CCC2 REAL300012003558
O=C(O)C(Cc1cscn1)NCc1cscc1Br REAL300012003559
CC(C)COc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003560
O=C(O)C(Cc1cscn1)NCc1nc2c(s1)CCCC2 REAL300012003561
O=C(O)C(Cc1cscn1)NCc1cc(F)cc(Br)c1 REAL300012003562
O=C(O)C(Cc1cscn1)NCc1ccc2cnccc2c1 REAL300012003563
O=C(O)C(Cc1cscn1)NCc1cccc(F)c1Br REAL300012003564
COc1cc(F)cc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003565
O=C(O)C(Cc1cscn1)NCc1cccc(Br)c1F REAL300012003566
CC(C)(C)c1ncc(CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003567
CS(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003568
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)CCCC2 REAL300012003569
COC(=O)c1cc(CNC(Cc2cscn2)C(=O)O)c[nH]1 REAL300012003570
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(C)c1OC REAL300012003571
O=C(O)C(Cc1cscn1)NCc1csc(Cl)c1Cl REAL300012003572
COc1cc(C)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003573
O=C(O)C(Cc1cscn1)NCc1cnc(C(F)(F)F)s1 REAL300012003574
CS(=O)(=O)c1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003575
O=C(O)C(Cc1cscn1)NCc1cc(Cl)cs1 REAL300012003576
O=C(O)C(Cc1cscn1)NCc1ccc(C2CCCC2)cc1 REAL300012003577
Cc1cc(Cl)cc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003578
COCc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003579
O=C(O)C(Cc1cscn1)NCc1nccn1-c1ccccc1 REAL300012003580
O=C(O)C(Cc1cscn1)NCc1ccc(C2CC2)cc1 REAL300012003581
O=C(O)C(Cc1cscn1)NCc1ncc(Cl)s1 REAL300012003582
O=C(O)C(Cc1cscn1)NCc1ccnn1C1CCCC1 REAL300012003583
COc1cc2ccccc2cc1CNC(Cc1cscn1)C(=O)O REAL300012003584
O=C(O)C(Cc1cscn1)NCc1ccc(C(F)F)cc1 REAL300012003585
COc1cc(C)c(CNC(Cc2cscn2)C(=O)O)c(C)n1 REAL300012003586
COc1cccc(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003587
CCc1cc(OC)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003588
Cc1ncc(CNC(Cc2cscn2)C(=O)O)n1-c1ccccc1 REAL300012003589
CCCn1nc(C)c(CNC(Cc2cscn2)C(=O)O)c1C REAL300012003590
O=C(O)C(Cc1cscn1)NCc1cnc(C2CC2)nc1 REAL300012003591
COCCn1cc(CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003592
O=C(O)C(Cc1cscn1)NCc1ccc(C2CCC2)cc1 REAL300012003593
COc1cc(CNC(Cc2cscn2)C(=O)O)cc2ccccc12 REAL300012003594
CCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1F REAL300012003595
COc1cccc2c(CNC(Cc3cscn3)C(=O)O)cccc12 REAL300012003596
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1C#N REAL300012003597
Cc1ccccc1-n1nccc1CNC(Cc1cscn1)C(=O)O REAL300012003598
O=C(O)C(Cc1cscn1)NCc1ncc(C(F)(F)F)s1 REAL300012003599
Cc1cc(CNC(Cc2cscn2)C(=O)O)ccc1C#N REAL300012003600
O=C(O)C(Cc1cscn1)NCc1cc2c(cc1OC(F)F)OCO2 REAL300012003601
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(Br)c1 REAL300012003602
CC(C)Cn1cc(CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003603
O=C(O)C(Cc1cscn1)NCc1ccccc1C1CC1 REAL300012003604
Cc1cc(Br)c(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003605
CC(C)(C)OC(=O)c1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003606
CC(C)Sc1cccc(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003607
CN1C(=O)CCc2cc(CNC(Cc3cscn3)C(=O)O)ccc21 REAL300012003608
Cc1ccc(OC(F)F)c(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003609
O=C(O)C(Cc1cscn1)NCc1cnc(-c2ccc(Cl)cc2)s1 REAL300012003610
O=C(O)C(Cc1cscn1)NCc1cnc(-c2ccccc2F)s1 REAL300012003611
COc1ccc(-c2ccccc2C)cc1CNC(Cc1cscn1)C(=O)O REAL300012003612
O=C(O)C(Cc1cscn1)NCc1cc(Cl)ccc1OCC1CC1 REAL300012003613
Cc1nn(C(C)C)cc1CNC(Cc1cscn1)C(=O)O REAL300012003614
O=C(O)C(Cc1cscn1)NCc1ccnc2c(Br)cccc12 REAL300012003615
O=C(O)C(Cc1cscn1)NCc1cnc(C2CCCC2)s1 REAL300012003616
O=C(O)C(Cc1cscn1)NCc1cnc(-c2c(F)cccc2F)s1 REAL300012003617
O=C(O)C(Cc1cscn1)NCc1cnc(C2CC2)s1 REAL300012003618
CC(C)c1ncc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003619
O=C(O)C(Cc1cscn1)NCc1cnc(-c2ccco2)s1 REAL300012003620
O=C(O)C(Cc1cscn1)NCc1ccc(Br)c(Cl)c1 REAL300012003621
O=C(O)C(Cc1cscn1)NCc1cnc(CCc2ccccc2)s1 REAL300012003622
Cn1cc(-c2ccc(CNC(Cc3cscn3)C(=O)O)cc2)cn1 REAL300012003623
O=C(O)C(Cc1cscn1)NCc1cnn(CC(F)F)c1 REAL300012003624
O=C(O)C(Cc1cscn1)NCc1ccc(Oc2cccc(F)c2)cc1 REAL300012003625
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2ccc(F)cc2)n1 REAL300012003626
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2ccc(C#N)cc2)n1 REAL300012003627
CN(C)C(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)[nH]1 REAL300012003628
NC(=O)c1csc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003629
CN(c1ccccc1)c1ccc(CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003630
CCc1nn(C)c(CC)c1CNC(Cc1cscn1)C(=O)O REAL300012003631
O=C(O)C(Cc1cscn1)NCc1cnc(C2CCC2)s1 REAL300012003632
O=C(O)C(Cc1cscn1)NCc1cnc(C2CCCO2)s1 REAL300012003633
Cc1ccccc1-n1cc(CNC(Cc2cscn2)C(=O)O)nn1 REAL300012003634
Cn1nc(Br)cc1CNC(Cc1cscn1)C(=O)O REAL300012003635
Cn1cc(-c2ccc(CNC(Cc3cscn3)C(=O)O)s2)cn1 REAL300012003636
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)OCCCCO2 REAL300012003637
CCOc1c(Cl)cccc1CNC(Cc1cscn1)C(=O)O REAL300012003638
CCc1cccc(F)c1CNC(Cc1cscn1)C(=O)O REAL300012003639
O=C(O)C(Cc1cscn1)NCc1ccc(F)c(Cl)c1Cl REAL300012003640
O=C(O)C(Cc1cscn1)NCc1ccn(C(F)F)n1 REAL300012003641
COc1ccccc1-n1nccc1CNC(Cc1cscn1)C(=O)O REAL300012003642
O=C(O)C(Cc1cscn1)NCc1c(F)cccc1OC(F)(F)F REAL300012003643
O=C(O)C(Cc1cscn1)NCc1ccnn1-c1ccc(F)cc1 REAL300012003644
Cc1ccc(CNC(Cc2cscn2)C(=O)O)c(-c2cnn(C)c2)c1 REAL300012003645
Cc1ccc(CNC(Cc2cscn2)C(=O)O)c(-c2ccnn2C)c1 REAL300012003646
CC(C)c1cnc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003647
O=C(O)C(Cc1cscn1)NCc1cnn(-c2ccc(C(F)(F)F)cc2)c1 REAL300012003648
Cc1cc(Br)c(CNC(Cc2cscn2)C(=O)O)cc1Cl REAL300012003649
O=C(O)C(Cc1cscn1)NCc1cnn(Cc2ccccc2)c1Cl REAL300012003650
CC(C)(C)c1cnc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003651
O=C(O)C(Cc1cscn1)NCc1scnc1C1CC1 REAL300012003652
N#CCCn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2ccncc2)n1 REAL300012003653
O=C(O)C(Cc1cscn1)NCc1ccc(Cl)cc1-n1cncn1 REAL300012003654
COC(=O)c1cc(CNC(Cc2cscn2)C(=O)O)n(C)c1C REAL300012003655
COCCCn1nccc1CNC(Cc1cscn1)C(=O)O REAL300012003656
Cc1cc(F)c(CNC(Cc2cscn2)C(=O)O)c(Cl)c1 REAL300012003657
COCCOCc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003658
CSCc1cnc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003659
O=C(O)C(Cc1cscn1)NCc1cscc1C(F)(F)F REAL300012003660
Cc1c(CNC(Cc2cscn2)C(=O)O)sc2c(Cl)cccc12 REAL300012003661
O=C(OCc1ccccc1)c1cc(CNC(Cc2cscn2)C(=O)O)c[nH]1 REAL300012003662
O=C(O)C(Cc1cscn1)NCc1cccc(C2CC2)c1 REAL300012003663
N#Cc1ccc(CNC(Cc2cscn2)C(=O)O)cc1F REAL300012003664
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)OC(F)(F)O2 REAL300012003665
Cc1cc(F)c(CNC(Cc2cscn2)C(=O)O)c(F)c1 REAL300012003666
Cc1ccc(-c2nn(C)cc2CNC(Cc2cscn2)C(=O)O)o1 REAL300012003667
CC(C)Cn1nccc1CNC(Cc1cscn1)C(=O)O REAL300012003668
O=C(O)C(Cc1cscn1)NCc1cc(Br)cnc1Cl REAL300012003669
COC(=O)c1[nH]cc(CNC(Cc2cscn2)C(=O)O)c1C REAL300012003670
Cc1ccc(-c2ncc(CNC(Cc3cscn3)C(=O)O)s2)cc1C REAL300012003671
Cc1nn(-c2ccccc2F)cc1CNC(Cc1cscn1)C(=O)O REAL300012003672
Cc1nn(-c2ccccc2Cl)cc1CNC(Cc1cscn1)C(=O)O REAL300012003673
Cc1ccc(-n2cc(CNC(Cc3cscn3)C(=O)O)c(C)n2)cc1 REAL300012003674
CC(C)(C#N)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003675
CC(C)c1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003676
O=C(O)C(Cc1cscn1)NCc1cc2n(n1)CCCC2 REAL300012003677
O=C(O)C(Cc1cscn1)NCc1cnnn1-c1ccccc1 REAL300012003678
O=C(O)C(Cc1cscn1)NCc1cc2cnccc2o1 REAL300012003679
COc1cc(OC)c(CNC(Cc2cscn2)C(=O)O)cc1F REAL300012003680
COc1cc(F)c(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003681
Cc1ccc(CNC(Cc2cscn2)C(=O)O)c(Cl)c1 REAL300012003682
Cc1cccc(-n2cc(CNC(Cc3cscn3)C(=O)O)c(C)n2)c1 REAL300012003683
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(F)c1 REAL300012003684
O=C(O)C(Cc1cscn1)NCc1cccc2c1CCC2 REAL300012003685
COc1cccc(F)c1CNC(Cc1cscn1)C(=O)O REAL300012003686
CCCOc1ccc(CNC(Cc2cscn2)C(=O)O)c(C)c1 REAL300012003687
O=C(O)C(Cc1cscn1)NCc1cc2ccncc2s1 REAL300012003688
O=C(O)C(Cc1cscn1)NCc1cc2cc(Br)ccc2o1 REAL300012003689
CCc1cccc2cc(CNC(Cc3cscn3)C(=O)O)oc12 REAL300012003690
C=CCCn1cc(CNC(Cc2cscn2)C(=O)O)nn1 REAL300012003691
O=C(O)C(Cc1cscn1)NCc1ccnn1CC1CC1 REAL300012003692
O=C(O)C(Cc1cscn1)NCc1cccc(OC2CC2)c1F REAL300012003693
CCOc1ccc(CNC(Cc2cscn2)C(=O)O)c(C)c1 REAL300012003694
O=C(O)C(Cc1cscn1)NCc1cccc(F)c1OC(F)F REAL300012003695
O=C(O)C(Cc1cscn1)NCc1cc(F)ccc1OC(F)F REAL300012003696
O=C(O)C(Cc1cscn1)NCc1cccc(C2CCCC2)c1 REAL300012003697
Cn1cc(-c2nn(C)cc2CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003698
COCc1csc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003699
O=C(O)C(Cc1cscn1)NCc1cn(C2CCC2)nn1 REAL300012003700
O=C(O)C(Cc1cscn1)NCc1cnc(-c2cccc(Cl)c2)s1 REAL300012003701
O=C(O)C(Cc1cscn1)NCc1csc(C(F)(F)F)c1 REAL300012003702
O=C(O)C(Cc1cscn1)NCc1ccc(C(F)(F)F)o1 REAL300012003703
O=C(O)C(Cc1cscn1)NCc1ccsc1C(F)(F)F REAL300012003704
CN(C)c1c(CNC(Cc2cscn2)C(=O)O)ccc(F)c1F REAL300012003705
O=C(O)C(Cc1cscn1)NCc1c(F)ccc(F)c1Cl REAL300012003706
CC(C)Oc1cc(Cl)c(CNC(Cc2cscn2)C(=O)O)cc1Cl REAL300012003707
O=C(O)C(Cc1cscn1)NCc1ccc(OC2CCOC2)cc1 REAL300012003708
CN(C)c1cc(F)c(CNC(Cc2cscn2)C(=O)O)cc1F REAL300012003709
COC(=O)c1cc(CNC(Cc2cscn2)C(=O)O)n2c1CCCC2 REAL300012003710
O=C(O)C(Cc1cscn1)NCc1ccc(F)c(F)c1F REAL300012003711
COc1cc(CNC(Cc2cscn2)C(=O)O)cc(C(F)(F)F)c1 REAL300012003712
C=CCOc1c(Cl)cc(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003713
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC1CC1 REAL300012003714
Cn1nc(C(F)(F)F)cc1CNC(Cc1cscn1)C(=O)O REAL300012003715
COCC(C)Oc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003716
CCCc1ccc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003717
O=C(O)C(Cc1cscn1)NCc1ccc(-c2cccs2)cc1 REAL300012003718
O=C(O)C(Cc1cscn1)NCc1ccnn1CCc1ccccc1 REAL300012003719
CC(C)c1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003720
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(Cl)n1 REAL300012003721
O=C(O)C(Cc1cscn1)NCc1cccc(F)c1OCC(F)(F)F REAL300012003722
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1C(C)(C)C REAL300012003723
O=C(O)C(Cc1cscn1)NCc1cccc(CC2CCC2)c1 REAL300012003724
COc1cccc(OC(F)(F)F)c1CNC(Cc1cscn1)C(=O)O REAL300012003725
Cc1cc(CNC(Cc2cscn2)C(=O)O)ncc1Br REAL300012003726
Cc1cc(CNC(Cc2cscn2)C(=O)O)c(Br)cc1F REAL300012003727
O=C(O)C(Cc1cscn1)NCc1c(O)cccc1Br REAL300012003728
Cn1cc(-c2nc(CNC(Cc3cscn3)C(=O)O)cs2)cn1 REAL300012003729
COc1cc(CNC(Cc2cscn2)C(=O)O)ccc1Cl REAL300012003730
O=C(O)C(Cc1cscn1)NCc1ccnn1CC1CCC1 REAL300012003731
O=C(O)C(Cc1cscn1)NCc1cn(-c2ccc(F)cc2)nn1 REAL300012003732
O=C(O)C(Cc1cscn1)NCc1ccccc1CC(F)(F)F REAL300012003733
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(Br)n1 REAL300012003734
CC(=O)Nc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003735
Cn1ncc2cc(CNC(Cc3cscn3)C(=O)O)cnc21 REAL300012003736
O=C(O)C(Cc1cscn1)NCc1ncc(Br)cc1F REAL300012003737
COc1cc(Cl)c(CNC(Cc2cscn2)C(=O)O)cc1OC REAL300012003738
O=C(O)C(Cc1cscn1)NCc1ccc(CC(F)(F)F)cc1 REAL300012003739
CC(C)(C)OC(=O)NCc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003740
Cn1nc2c(c1CNC(Cc1cscn1)C(=O)O)CCCC2 REAL300012003741
CCOC(=O)c1[nH]c(C)c(CNC(Cc2cscn2)C(=O)O)c1C REAL300012003742
O=C(O)C(Cc1cscn1)NCc1cnc(Cl)c(F)c1 REAL300012003743
O=C(O)C(Cc1cscn1)NCc1ccc(-c2ccccc2)c(Cl)c1 REAL300012003744
O=C(O)C(Cc1cscn1)NCc1ccc(Br)c(F)c1F REAL300012003745
O=C(O)C(Cc1cscn1)NCc1ccsc1Br REAL300012003746
CCOc1cc(CNC(Cc2cscn2)C(=O)O)c(F)cc1OC REAL300012003747
COc1ncc(Br)cc1CNC(Cc1cscn1)C(=O)O REAL300012003748
O=C(O)C(Cc1cscn1)NCc1ccc(F)c2ccccc12 REAL300012003749
O=C(O)C(Cc1cscn1)NCc1cccnc1Br REAL300012003750
COc1cc(CNC(Cc2cscn2)C(=O)O)c(F)cc1Br REAL300012003751
O=C(O)C(Cc1cscn1)NCc1cccc(Br)c1Cl REAL300012003752
O=C(O)C(Cc1cscn1)NCc1cccc(F)c1OC(F)(F)F REAL300012003753
CC(C)Oc1ccc(F)cc1CNC(Cc1cscn1)C(=O)O REAL300012003754
CCOc1cc(F)cc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003755
O=C(O)C(Cc1cscn1)NCc1ccc(C(=O)N2CCCC2)cc1 REAL300012003756
O=C(O)C(Cc1cscn1)NCc1ccc(OC(F)F)cc1F REAL300012003757
CC(C)(C)Oc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003758
Cc1c(Cl)cccc1CNC(Cc1cscn1)C(=O)O REAL300012003759
COc1cc(CNC(Cc2cscn2)C(=O)O)c(F)cc1C REAL300012003760
Cc1ccc(CNC(Cc2cscn2)C(=O)O)c(C)c1Br REAL300012003761
Cc1ccnc(CNC(Cc2cscn2)C(=O)O)c1Br REAL300012003762
CC(C)(C)OC(=O)Nc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003763
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2cc(F)ccc2F)n1 REAL300012003764
CC(C)(C)c1csc(CNC(Cc2cscn2)C(=O)O)n1 REAL300012003765
COCCc1ncc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003766
O=C(O)C(Cc1cscn1)NCc1cc(Cl)cc(Br)c1O REAL300012003767
O=C(O)C(Cc1cscn1)NCc1cc(Br)cc(F)c1O REAL300012003768
O=C(O)C(Cc1cscn1)NCc1cc(F)cc(F)c1O REAL300012003769
Cn1nc2c(c1CNC(Cc1cscn1)C(=O)O)CSCC2 REAL300012003770
CCn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2ccccc2)n1 REAL300012003771
O=C(O)C(Cc1cscn1)NCc1cccc2c1CCOC2 REAL300012003772
COCc1c(C)cc(C)c(CNC(Cc2cscn2)C(=O)O)c1C REAL300012003773
O=C(O)C(Cc1cscn1)NCc1ccc2oc(=O)oc2c1 REAL300012003774
Cc1sc(CNC(Cc2cscn2)C(=O)O)cc1Br REAL300012003775
O=C(O)C(Cc1cscn1)NCc1cccc(-c2ccc(Cl)cc2)c1 REAL300012003776
O=C(O)C(Cc1cscn1)NCc1cccc2ncccc12 REAL300012003777
CCCOc1ccc(CNC(Cc2cscn2)C(=O)O)cc1C REAL300012003778
O=C(O)C(Cc1cscn1)NCc1ccc2nccnc2c1 REAL300012003779
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1COc1ccccc1 REAL300012003780
COc1ccc(CNC(Cc2cscn2)C(=O)O)cc1Cn1cccn1 REAL300012003781
CCOc1cccc(F)c1CNC(Cc1cscn1)C(=O)O REAL300012003782
Cc1ccc(Br)c(F)c1CNC(Cc1cscn1)C(=O)O REAL300012003783
Cc1c(CNC(Cc2cscn2)C(=O)O)cccc1[N+](=O)[O-] REAL300012003784
Cc1ccc([N+](=O)[O-])c(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003785
COc1ccc(Cn2cc(CNC(Cc3cscn3)C(=O)O)nn2)cc1 REAL300012003786
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(F)c1OC REAL300012003787
COC(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)c(F)c1 REAL300012003788
O=C(O)C(Cc1cscn1)NCc1cccc(Oc2ccccn2)c1 REAL300012003789
O=C(O)C(Cc1cscn1)NCc1cccc(COc2ccccc2)c1 REAL300012003790
O=C(O)C(Cc1cscn1)NCc1ccccc1OCC(F)F REAL300012003791
COc1cc(C)ccc1Oc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003792
Cc1ccccc1-n1nc(C)c(CNC(Cc2cscn2)C(=O)O)c1C REAL300012003793
Cc1cc(C#N)cc(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003794
CC(C)(C)c1coc(CNC(Cc2cscn2)C(=O)O)n1 REAL300012003795
CCCc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003796
O=C(O)C(Cc1cscn1)NCc1csc(-c2ccc(Cl)cc2)n1 REAL300012003797
COc1ccc(-c2nc(CNC(Cc3cscn3)C(=O)O)cs2)cc1 REAL300012003798
O=C(O)C(Cc1cscn1)NCc1ccc(OCCN2CCCC2)cc1 REAL300012003799
Cc1n[nH]c2ncc(CNC(Cc3cscn3)C(=O)O)cc12 REAL300012003800
CS(=O)(=O)Nc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003801
Cn1nc(CNC(Cc2cscn2)C(=O)O)c2ccccc21 REAL300012003802
O=C(O)C(Cc1cscn1)NCc1n[nH]c2ccccc12 REAL300012003803
Cn1c(Cl)nc(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003804
O=C(O)C(Cc1cscn1)NCc1nccc2ccccc12 REAL300012003805
Cc1nc2ccccn2c1CNC(Cc1cscn1)C(=O)O REAL300012003806
CN(Cc1ccccc1)CC(C)(C)CNC(Cc1cscn1)C(=O)O REAL300012003807
O=C(O)C(Cc1cscn1)NCc1cc(-c2ccccn2)n[nH]1 REAL300012003808
O=C(O)C(Cc1cscn1)NCc1cscc1Cl REAL300012003809
Cc1nn2c(CNC(Cc3cscn3)C(=O)O)c(C)nc2s1 REAL300012003810
Cc1nn2c(CNC(Cc3cscn3)C(=O)O)c(C(C)C)nc2s1 REAL300012003811
CCCC(CNC(Cc1cscn1)C(=O)O)c1ccccc1 REAL300012003812
O=C(O)C(Cc1cscn1)NCc1c(Cl)ccc2cccnc12 REAL300012003813
O=C(O)C(Cc1cscn1)NCc1ccc(C(F)(F)F)s1 REAL300012003814
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(OCc2cccnc2)c1 REAL300012003815
O=C(O)C(Cc1cscn1)NCc1nc2ccc(Br)cc2s1 REAL300012003816
CN(C)c1ccc(CNC(Cc2cscn2)C(=O)O)c(C(F)(F)F)c1 REAL300012003817
CC(=Cc1ccccc1C(F)(F)F)CNC(Cc1cscn1)C(=O)O REAL300012003818
Cc1nn(-c2ccccn2)c(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003819
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)CCN2Cc1ccccc1 REAL300012003820
CC(C)C1CCC(CNC(Cc2cscn2)C(=O)O)CC1 REAL300012003821
O=C(O)C(Cc1cscn1)NCc1c(Cl)nc2cc(Cl)ccn12 REAL300012003822
O=C(O)C(Cc1cscn1)NCc1cn2ccc(Br)cc2n1 REAL300012003823
CC(=Cc1ccccc1OC(F)F)CNC(Cc1cscn1)C(=O)O REAL300012003824
COCc1ccccc1C=C(C)CNC(Cc1cscn1)C(=O)O REAL300012003825
Cn1nccc1-c1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003826
O=C(O)C(Cc1cscn1)NCc1conc1Cc1ccccc1 REAL300012003827
Cn1ncc(CNC(Cc2cscn2)C(=O)O)c1Cl REAL300012003828
O=C(O)C(Cc1cscn1)NCc1cc2cccnc2o1 REAL300012003829
COc1ccc(-n2cc(CNC(Cc3cscn3)C(=O)O)cn2)cc1 REAL300012003830
CN(Cc1cccs1)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003831
O=C(O)C(Cc1cscn1)NCc1cc2cc(Cl)cnc2o1 REAL300012003832
O=C(O)C(Cc1cscn1)NC[C@@H]1C[C@H]1c1ccccc1 REAL300012003833
O=C(O)C(Cc1cscn1)NCc1ccncc1Br REAL300012003834
CS(=O)(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003835
O=C(O)C(Cc1cscn1)NCc1cnn(C2CCCC2)c1-c1ccccc1 REAL300012003836
O=C(O)C(Cc1cscn1)NCc1ccnn1-c1ccccn1 REAL300012003837
NS(=O)(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)c(F)c1 REAL300012003838
CC(C)(C)n1nnc(CNC(Cc2cscn2)C(=O)O)n1 REAL300012003839
Cc1c(Br)cncc1CNC(Cc1cscn1)C(=O)O REAL300012003840
Cn1ncc(C(F)(F)F)c1CNC(Cc1cscn1)C(=O)O REAL300012003841
Cn1ncc(C2CC2)c1CNC(Cc1cscn1)C(=O)O REAL300012003842
Cn1ncc(C2CCC2)c1CNC(Cc1cscn1)C(=O)O REAL300012003843
Cc1cccc2[nH]c(CNC(Cc3cscn3)C(=O)O)cc12 REAL300012003844
O=C(O)C(Cc1cscn1)NCc1ccnn1-c1ccncc1 REAL300012003845
Cc1ccc2cc(CNC(Cc3cscn3)C(=O)O)[nH]c2c1 REAL300012003846
CCOc1cncc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003847
O=C(O)C(Cc1cscn1)NCc1ccnn1C1CCOCC1 REAL300012003848
O=C(O)C(Cc1cscn1)NCc1cccc2[nH]ncc12 REAL300012003849
CCC(F)(F)C(C)(C)CNC(Cc1cscn1)C(=O)O REAL300012003850
O=C(O)C(Cc1cscn1)NCc1ccc2cc[nH]c2c1 REAL300012003851
O=C(O)C(Cc1cscn1)NCc1cc2c(=O)[nH]ccc2o1 REAL300012003852
O=C(O)C(Cc1cscn1)NCc1ccc(C(F)F)nc1 REAL300012003853
CN(C)c1ccc(C#N)cc1CNC(Cc1cscn1)C(=O)O REAL300012003854
O=C(O)C(Cc1cscn1)NCc1cn(CC2CCOC2)nn1 REAL300012003855
COc1cncc(CNC(Cc2cscn2)C(=O)O)c1C REAL300012003856
Cc1cc(C)c(C=CCNC(Cc2cscn2)C(=O)O)c(C)c1 REAL300012003857
O=C(O)C(Cc1cscn1)NCc1ccc(OCCN2CCOCC2)cc1 REAL300012003858
CC(C)(C)OC(=O)NC(CNC(Cc1cscn1)C(=O)O)CC(F)F REAL300012003859
O=C(O)C(Cc1cscn1)NCc1cn(CC2CCCO2)nn1 REAL300012003860
CN(C)c1ccc(F)cc1CNC(Cc1cscn1)C(=O)O REAL300012003861
O=C(O)C(Cc1cscn1)NCc1cnc2c(F)cccc2c1 REAL300012003862
Cc1cc(C)c(C=CCNC(Cc2cscn2)C(=O)O)cc1C REAL300012003863
NS(=O)(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003864
O=C(O)C(Cc1cscn1)NCc1nccc2c1CCCC2 REAL300012003865
Cc1nn(C)c(CNC(Cc2cscn2)C(=O)O)c1Cl REAL300012003866
Cn1ccc(-c2nc(CNC(Cc3cscn3)C(=O)O)cs2)n1 REAL300012003867
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(C2CCCC2)n1 REAL300012003868
Cc1cccc(CNC(Cc2cscn2)C(=O)O)c1Br REAL300012003869
O=C(O)C(Cc1cscn1)NCc1cccc(Oc2ccc(F)cc2)c1 REAL300012003870
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)CCCO2 REAL300012003871
CN(C)C(=O)c1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003872
CCc1n[nH]c(Cl)c1CNC(Cc1cscn1)C(=O)O REAL300012003873
O=C(O)C(Cc1cscn1)NCc1c(C2CC2)n[nH]c1Cl REAL300012003874
Cc1cc(CNC(Cc2cscn2)C(=O)O)c2c(n1)CCCC2 REAL300012003875
O=C(O)C(Cc1cscn1)NCc1ccccc1N1CCCCC1 REAL300012003876
O=C(O)C(Cc1cscn1)NCc1csc(C(F)(F)F)n1 REAL300012003877
O=C(O)C(Cc1cscn1)NCc1ccc(C(F)F)c(F)c1 REAL300012003878
COC(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1C REAL300012003879
COc1ccc(CNC(Cc2cscn2)C(=O)O)c(C)c1 REAL300012003880
Cc1c(Cl)ccc(CNC(Cc2cscn2)C(=O)O)c1Cl REAL300012003881
N#Cc1ccc(Br)c(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003882
CC1Cc2cc(CNC(Cc3cscn3)C(=O)O)ccc2O1 REAL300012003883
O=C(O)C(Cc1cscn1)NCc1cccc2[nH]c(=O)oc12 REAL300012003884
O=C(O)C(Cc1cscn1)NCc1cccc2c1OCC2 REAL300012003885
CSCc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003886
O=C(O)C(Cc1cscn1)NCc1cnn(CC2CCC2)c1 REAL300012003887
Cn1nc2c(c1CNC(Cc1cscn1)C(=O)O)COCC2 REAL300012003888
Cn1nc2c(c1CNC(Cc1cscn1)C(=O)O)CCC2 REAL300012003889
O=C(O)C(Cc1cscn1)NCc1ccnn1C1CCC1 REAL300012003890
O=C(O)C(Cc1cscn1)NCc1cnn(C2CCC2)c1 REAL300012003891
COC(=O)C(C)Oc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003892
COC(=O)COc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003893
COc1ccc(C)c(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003894
Cn1cnc2cccc(CNC(Cc3cscn3)C(=O)O)c21 REAL300012003895
CN(C)C(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003896
Cc1ccc(CNC(Cc2cscn2)C(=O)O)c(C)c1C REAL300012003897
CCNC(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003898
CC(C)(C)c1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003899
O=C(O)C(Cc1cscn1)NCc1cnc2n1CCCCC2 REAL300012003900
COc1ccc2sc(CNC(Cc3cscn3)C(=O)O)cc2c1 REAL300012003901
CCN(CC)C(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003902
CCN1CCc2cc(CNC(Cc3cscn3)C(=O)O)ccc21 REAL300012003903
CCN(C)C(=O)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003904
Cc1c(CNC(Cc2cscn2)C(=O)O)cnn1C(C)C REAL300012003905
CSc1ccc(CNC(Cc2cscn2)C(=O)O)cc1Cl REAL300012003906
Cc1cc(CNC(Cc2cscn2)C(=O)O)ccc1C1CC1 REAL300012003907
CCOc1cc(CNC(Cc2cscn2)C(=O)O)ccn1 REAL300012003908
Cc1ccc(CNC(Cc2cscn2)C(=O)O)cc1C1CC1 REAL300012003909
Cc1ccn(-c2ccc(CNC(Cc3cscn3)C(=O)O)c(C)c2)n1 REAL300012003910
O=C(O)C(Cc1cscn1)NCc1ccc(C(F)(F)C(F)(F)F)cc1 REAL300012003911
Cc1cc(-n2cc(Cl)cn2)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003912
CCc1cc(Br)c(CNC(Cc2cscn2)C(=O)O)s1 REAL300012003913
Cc1nn(-c2ccc(CNC(Cc3cscn3)C(=O)O)cc2)cc1Cl REAL300012003914
COC(=O)c1cc2oc(CNC(Cc3cscn3)C(=O)O)cc2[nH]1 REAL300012003915
COCCOc1ccc(CNC(Cc2cscn2)C(=O)O)o1 REAL300012003916
CC(C)(CNC(Cc1cscn1)C(=O)O)c1ccc(Br)cc1 REAL300012003917
Cc1nn(C(C)C)c(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003918
O=C(O)C(Cc1cscn1)NCc1cc(Cl)cc(Br)c1 REAL300012003919
Cc1ccc(-c2ccccc2CNC(Cc2cscn2)C(=O)O)c(C)c1 REAL300012003920
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(C2CC2)n1 REAL300012003921
COc1cccc(-c2csc(CNC(Cc3cscn3)C(=O)O)n2)c1 REAL300012003922
CC(C)(C)OC(=O)NCc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003923
COC(=O)c1cc(CNC(Cc2cscn2)C(=O)O)n2c1COCC2 REAL300012003924
O=C(O)C(Cc1cscn1)NCc1ccc(C(=O)N2CCCCC2)cc1 REAL300012003925
Cn1nc(C2CC2)cc1CNC(Cc1cscn1)C(=O)O REAL300012003926
Cc1cc(-n2ccnc2)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003927
O=C(O)C(Cc1cscn1)NCc1ccc(C(F)(F)F)c(Cl)c1Cl REAL300012003928
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1ccc(Cl)o1 REAL300012003929
O=C(O)C(Cc1cscn1)NCc1cnc(C2CCOCC2)o1 REAL300012003930
COc1nccc(CNC(Cc2cscn2)C(=O)O)c1F REAL300012003931
O=C(O)C(Cc1cscn1)NCc1c(Cl)cccc1Br REAL300012003932
O=C(O)C(Cc1cscn1)NCc1ccc(F)c(Br)c1F REAL300012003933
O=C(O)C(Cc1cscn1)NCc1cn2ccnc2s1 REAL300012003934
Cc1oc(C(C)(C)C)cc1CNC(Cc1cscn1)C(=O)O REAL300012003935
O=C(O)C(Cc1cscn1)NCc1cn(Cc2ccccc2)nn1 REAL300012003936
CC(C)(C)OC(=O)N1CCC(CNC(Cc2cscn2)C(=O)O)CC1 REAL300012003937
Cc1cc(Br)cnc1CNC(Cc1cscn1)C(=O)O REAL300012003938
O=C(O)C(Cc1cscn1)NCc1cccc(S(=O)(=O)C(F)F)c1 REAL300012003939
CC1Oc2ccc(CNC(Cc3cscn3)C(=O)O)cc2C1C REAL300012003940
Cc1ccc(CNC(Cc2cscn2)C(=O)O)cc1OC(F)F REAL300012003941
Cc1nc(Cl)c(CNC(Cc2cscn2)C(=O)O)cc1Br REAL300012003942
CC(C)Cc1ccccc1CNC(Cc1cscn1)C(=O)O REAL300012003943
Cn1ncc(CNC(Cc2cscn2)C(=O)O)c1S(C)(=O)=O REAL300012003944
Cc1c(C(F)(F)F)n[nH]c1CNC(Cc1cscn1)C(=O)O REAL300012003945
CC(C)Cn1cc(CNC(Cc2cscn2)C(=O)O)nn1 REAL300012003946
O=C(O)C(Cc1cscn1)NCc1nc(C2CC2)cs1 REAL300012003947
O=C(O)C(Cc1cscn1)NCc1cc(C(F)(F)F)[nH]n1 REAL300012003948
O=C(O)C(Cc1cscn1)NCc1ccc2c(c1)OCC2 REAL300012003949
Cn1cc(Cl)c(CNC(Cc2cscn2)C(=O)O)n1 REAL300012003950
CS(=O)(=O)c1sccc1CNC(Cc1cscn1)C(=O)O REAL300012003951
CSc1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003952
CC(C)c1cnn(C)c1CNC(Cc1cscn1)C(=O)O REAL300012003953
Cc1sc(C)c(CNC(Cc2cscn2)C(=O)O)c1Br REAL300012003954
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(-c2cccc(F)c2)n1 REAL300012003955
CCCn1cc(CNC(Cc2cscn2)C(=O)O)c(C)n1 REAL300012003956
O=C(O)C(Cc1cscn1)NCc1cc2ncccc2o1 REAL300012003957
O=C(O)C(Cc1cscn1)NCc1ccc(CC2CC2)s1 REAL300012003958
O=C(O)C(Cc1cscn1)NCc1ccc(OC2CC2)cc1 REAL300012003959
O=C(O)C(Cc1cscn1)NCc1ccc(OC(F)(F)F)cc1F REAL300012003960
O=C(O)C(Cc1cscn1)NCc1cccc(C(F)(F)C(F)(F)F)c1 REAL300012003961
Cc1cc(-n2ccnc2C)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003962
Cc1ncn(-c2ccc(CNC(Cc3cscn3)C(=O)O)cc2)c1C REAL300012003963
CNC(=O)c1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003964
O=C(O)C(Cc1cscn1)NCc1ccc(C2CC2)c(C2CC2)c1 REAL300012003965
CN(C)CCc1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003966
CCNC(=O)c1cccc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003967
Cc1c(CNC(Cc2cscn2)C(=O)O)oc2ccc(F)cc12 REAL300012003968
O=C(O)C(Cc1cscn1)NCc1cc(C2CCC2)[nH]n1 REAL300012003969
Cn1nc(-c2ccccc2)cc1CNC(Cc1cscn1)C(=O)O REAL300012003970
CC(C)(C)c1cncc(CNC(Cc2cscn2)C(=O)O)c1 REAL300012003971
O=C(O)C(Cc1cscn1)NCc1cc2c(Br)cccc2s1 REAL300012003972
O=C(O)C(Cc1cscn1)NCc1ccn(CC(F)(F)F)n1 REAL300012003973
O=C(O)C(Cc1cscn1)NCc1cccc2[nH]c3ccccc3c12 REAL300012003974
Cn1c(CNC(Cc2cscn2)C(=O)O)nc2c1CCCC2 REAL300012003975
COc1nc(Cl)ccc1CNC(Cc1cscn1)C(=O)O REAL300012003976
Cn1cc(CNC(Cc2cscn2)C(=O)O)c(C(F)(F)F)n1 REAL300012003977
O=C(O)C(Cc1cscn1)NCc1cccc(C(F)F)c1F REAL300012003978
O=C(O)C(Cc1cscn1)NCc1cccc2c1COCC2 REAL300012003979
CCOc1ccc(Cl)cc1CNC(Cc1cscn1)C(=O)O REAL300012003980
O=C(O)C(Cc1cscn1)NCc1nc2c(s1)COCC2 REAL300012003981
O=C(O)C(Cc1cscn1)NCc1c[nH]nc1-c1cccc(F)c1 REAL300012003982
O=C(O)C(Cc1cscn1)NCc1cc2c(o1)CCCC2 REAL300012003983
O=C(O)C(Cc1cscn1)NCc1cc(F)cc([N+](=O)[O-])c1 REAL300012003984
O=C(O)C(Cc1cscn1)NCc1cnn(C2CCCCC2)c1 REAL300012003985
O=C(O)C(Cc1cscn1)NCc1cnn(-c2ccccc2)c1Cl REAL300012003986
O=C(O)C(Cc1cscn1)NCc1c(F)cc(Br)cc1F REAL300012003987
CN(CCO)c1ccc(CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003988
COc1c(CNC(Cc2cscn2)C(=O)O)cccc1C(C)(C)C REAL300012003989
Cn1cc(Br)nc1CNC(Cc1cscn1)C(=O)O REAL300012003990
COc1cc(C)c(CNC(Cc2cscn2)C(=O)O)cn1 REAL300012003991
COc1cc(C)c(CNC(Cc2cscn2)C(=O)O)cc1O REAL300012003992
O=C(O)C(Cc1cscn1)NCc1cc2ccc(F)cc2[nH]c1=O REAL300012003993
Cn1c(=O)c(CNC(Cc2cscn2)C(=O)O)cc2ccccc21 REAL300012003994
COc1nc(CNC(Cc2cscn2)C(=O)O)ccc1C REAL300012003995
Cc1cc(C)c(CNC(Cc2cscn2)C(=O)O)c(C)c1Br REAL300012003996
O=C(O)C(Cc1cscn1)NCC=Cc1ccc2c(c1)OCO2 REAL300012003997
O=C(O)C(Cc1cscn1)NCc1ccc(CC2CCC2)cc1 REAL300012003998
COC(F)(F)C(F)(F)c1ccc(CNC(Cc2cscn2)C(=O)O)cc1 REAL300012003999
CCc1c(CNC(Cc2cscn2)C(=O)O)cnn1CC REAL300012004000
