CSc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)o1 REAL300018133001
O=C(O)[C@@H]1CN(Cc2cnc(-c3ccccc3F)s2)C[C@H]1C(F)(F)F REAL300018133002
Cn1cc(-c2nc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cs2)cn1 REAL300018133003
COc1ccc(-c2ccccc2C)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133004
O=C(O)[C@@H]1CN(Cc2cc(Cl)ccc2OCC2CC2)C[C@H]1C(F)(F)F REAL300018133005
O=C(O)[C@@H]1CN(Cc2cccc(C3CC3)c2)C[C@H]1C(F)(F)F REAL300018133006
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ncc1Br REAL300018133007
CC(C)(C)c1csc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)n1 REAL300018133008
O=C(O)[C@@H]1CN(Cc2ncc(Br)cc2F)C[C@H]1C(F)(F)F REAL300018133009
O=C(O)[C@@H]1CN(Cc2cnc(C3CCCC3)s2)C[C@H]1C(F)(F)F REAL300018133010
O=C(O)[C@@H]1CN(Cc2cnc(-c3c(F)cccc3F)s2)C[C@H]1C(F)(F)F REAL300018133011
O=C(O)[C@@H]1CN(Cc2cnc(C3CCCCC3)s2)C[C@H]1C(F)(F)F REAL300018133012
O=C(O)[C@@H]1CN(Cc2cnc(C3CC3)s2)C[C@H]1C(F)(F)F REAL300018133013
CC(C)Cc1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133014
CC(C)c1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133015
O=C(O)[C@@H]1CN(Cc2cnc(-c3cccs3)s2)C[C@H]1C(F)(F)F REAL300018133016
O=C(O)[C@@H]1CN(Cc2cnc(-c3cccc(Cl)c3)s2)C[C@H]1C(F)(F)F REAL300018133017
O=C(O)[C@@H]1CN(Cc2cnc(-c3ccsc3)s2)C[C@H]1C(F)(F)F REAL300018133018
Cc1ccc(-c2ncc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)s2)cc1C REAL300018133019
Cc1ccc(-c2ncc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)s2)o1 REAL300018133020
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(Br)cc1F REAL300018133021
Cc1cc(Br)ccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133022
O=C(O)[C@@H]1CN(Cc2cnc(CCc3ccccc3)s2)C[C@H]1C(F)(F)F REAL300018133023
COCCc1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133024
O=C(O)[C@@H]1CN(Cc2cnn(CC(F)(F)F)c2)C[C@H]1C(F)(F)F REAL300018133025
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2ccccc2F)C[C@H]1C(F)(F)F REAL300018133026
O=C(O)[C@@H]1CN(Cc2nc3cc(Br)ccc3o2)C[C@H]1C(F)(F)F REAL300018133027
O=C(O)[C@@H]1CN(CCCc2c(Cl)cccc2Cl)C[C@H]1C(F)(F)F REAL300018133028
COCCOc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133029
O=C(O)[C@@H]1CN(Cc2ccc(Cl)cc2Br)C[C@H]1C(F)(F)F REAL300018133030
Cc1c(Br)cncc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133031
O=C(O)[C@@H]1CN(Cc2cn3ccc(Br)cc3n2)C[C@H]1C(F)(F)F REAL300018133032
C#CCOc1cccc(Cl)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133033
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2c(F)cccc2F)C[C@H]1C(F)(F)F REAL300018133034
COc1ccc(Cn2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)nn2)cc1 REAL300018133035
O=C(O)[C@@H]1CN(Cc2nc3c(s2)CCC3)C[C@H]1C(F)(F)F REAL300018133036
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2ccc(F)cc2)n1 REAL300018133037
Cc1nn(-c2ccccc2F)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133038
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2cccs2)n1 REAL300018133039
O=C(O)[C@@H]1CN(Cc2cc(Cl)ccc2OC2CCCC2)C[C@H]1C(F)(F)F REAL300018133040
O=C(O)[C@@H]1CN(Cc2c(Cl)cccc2N2CCCC2)C[C@H]1C(F)(F)F REAL300018133041
O=C(O)[C@@H]1CN(Cc2c(Cl)cccc2Oc2ccccc2)C[C@H]1C(F)(F)F REAL300018133042
Cc1ccc(-n2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c(C)n2)cc1 REAL300018133043
CC(C)(C)c1nn(-c2ccccc2)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133044
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C(C)(C)C)n1 REAL300018133045
Cc1ccc(-c2nn(C)cc2CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)o1 REAL300018133046
CN(C)c1ccc(F)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133047
O=C(O)[C@@H]1CN(Cc2cnc(-c3cccnc3)s2)C[C@H]1C(F)(F)F REAL300018133048
CC(C)(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)c1ccccc1 REAL300018133049
CC(CCc1ccccc1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133050
Cc1ccc(CCCN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cn1 REAL300018133051
COc1ccc(CC(C)CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1F REAL300018133052
CC(CC1CCCCC1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133053
Cc1cc2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)oc2cc1C REAL300018133054
CCc1nn(C)c(CC)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133055
O=C(O)[C@@H]1CN(Cc2cnc(C3CCC3)s2)C[C@H]1C(F)(F)F REAL300018133056
CCc1cccc2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)oc12 REAL300018133057
CCCC1CCC(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)CC1 REAL300018133058
CC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)c1ccc(S(C)(=O)=O)cc1 REAL300018133059
CC(C)C1CCC(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)CC1 REAL300018133060
COCc1c(C)cc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133061
CC(C)Cn1nccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133062
O=C(O)[C@@H]1CN(Cc2cn(CC3CCCO3)nn2)C[C@H]1C(F)(F)F REAL300018133063
CCCn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)nn1 REAL300018133064
O=C(O)[C@@H]1CN(Cc2cn(-c3ccc(F)cc3Cl)nn2)C[C@H]1C(F)(F)F REAL300018133065
Cc1cc(C)c(C=CCN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1C REAL300018133066
CC(=Cc1cccc([N+](=O)[O-])c1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133067
CC(=Cc1ccccc1OC(F)F)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133068
CC(=Cc1ccccc1C(F)(F)F)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133069
COCc1ccccc1C=C(C)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133070
Cn1nc(Br)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133071
O=C(O)[C@@H]1CN(Cc2ccc(CC(F)(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133072
O=C(O)[C@@H]1CN(Cc2cc(C3CC3)no2)C[C@H]1C(F)(F)F REAL300018133073
O=C(O)[C@@H]1CN(Cc2c(C3CC3)nc3sccn23)C[C@H]1C(F)(F)F REAL300018133074
CC(C)n1ncnc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133075
O=C(O)[C@@H]1CN(CC2CCN(c3ccccc3)C2)C[C@H]1C(F)(F)F REAL300018133076
Cn1nc(C(F)(F)F)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133077
NS(=O)(=O)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133078
Cc1nn2c(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c(C(C)C)nc2s1 REAL300018133079
O=C(O)[C@@H]1CN(CC2C3CC4CC(C3)CC2C4)C[C@H]1C(F)(F)F REAL300018133080
CCOP(=O)(CCCN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)OCC REAL300018133081
O=C(O)[C@@H]1CN(CC2CC2(Cl)Cl)C[C@H]1C(F)(F)F REAL300018133082
O=C(O)[C@@H]1CN(Cc2cccc(C3CCCC3)c2)C[C@H]1C(F)(F)F REAL300018133083
O=C(O)[C@@H]1CN(Cc2ccc3c(c2)OCCCCO3)C[C@H]1C(F)(F)F REAL300018133084
Cc1scc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133085
CC(C)(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)Oc1ccccc1 REAL300018133086
O=C(O)[C@@H]1CN(Cc2ccccc2CC(F)(F)F)C[C@H]1C(F)(F)F REAL300018133087
COc1cc(OC)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1F REAL300018133088
COC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)C1CCCCC1 REAL300018133089
CC(C)OC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)c1ccccc1 REAL300018133090
CCCCCCCCCC(C)CCN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133091
COC(Cc1ccccc1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133092
COC1(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)CCCCC1 REAL300018133093
O=C(O)[C@@H]1CN(Cc2conc2Cc2ccccc2)C[C@H]1C(F)(F)F REAL300018133094
O=C(O)[C@@H]1CN(Cc2ccccc2Cl)C[C@H]1C(F)(F)F REAL300018133095
O=C(O)[C@@H]1CN(Cc2cccc([N+](=O)[O-])c2)C[C@H]1C(F)(F)F REAL300018133096
O=C(O)[C@@H]1CN(Cc2ccc([N+](=O)[O-])cc2)C[C@H]1C(F)(F)F REAL300018133097
O=C(O)[C@@H]1CN(Cc2cccc3ccccc23)C[C@H]1C(F)(F)F REAL300018133098
CN(C)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133099
CCN(CC)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133100
O=C(O)[C@@H]1CN(Cc2ccc(Br)cc2)C[C@H]1C(F)(F)F REAL300018133101
O=C(O)[C@@H]1CN(Cc2ccc(Cl)cc2)C[C@H]1C(F)(F)F REAL300018133102
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc(OC)c1OC REAL300018133103
O=C(O)[C@@H]1CN(Cc2ccccc2OC(F)F)C[C@H]1C(F)(F)F REAL300018133104
O=C(O)[C@@H]1CN(Cc2ccccc2[N+](=O)[O-])C[C@H]1C(F)(F)F REAL300018133105
O=C(O)[C@@H]1CN(Cc2ccc(Cl)cc2Cl)C[C@H]1C(F)(F)F REAL300018133106
O=C(O)[C@@H]1CN(Cc2ccc(N3CCOCC3)cc2)C[C@H]1C(F)(F)F REAL300018133107
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)c1Br REAL300018133108
CC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)c1cc(F)cc(F)c1 REAL300018133109
O=C(O)[C@@H]1CN(Cc2ccnn2-c2ccncc2)C[C@H]1C(F)(F)F REAL300018133110
Cc1ccnc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1Br REAL300018133111
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2cnn(C)c2)c1 REAL300018133112
O=C(O)[C@@H]1CN(Cc2cccc(F)c2OCC(F)(F)F)C[C@H]1C(F)(F)F REAL300018133113
Cn1ncc(C(F)(F)F)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133114
Cn1nc2c(c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)CCCC2 REAL300018133115
O=C(O)[C@@H]1CN(Cc2scnc2C2CC2)C[C@H]1C(F)(F)F REAL300018133116
O=C(O)[C@@H]1CN(Cc2ccc(Cl)cc2-n2cncn2)C[C@H]1C(F)(F)F REAL300018133117
COCCCn1nccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133118
NS(=O)(=O)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1Cl REAL300018133119
CSCc1cnc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133120
O=C(O)[C@@H]1CN(Cc2cscc2C(F)(F)F)C[C@H]1C(F)(F)F REAL300018133121
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3)c(Cl)c2)C[C@H]1C(F)(F)F REAL300018133122
Cc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)sc2c(Cl)cccc12 REAL300018133123
COC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)C1CCOCC1 REAL300018133124
O=C(O)[C@@H]1CN(Cc2nc3cc([N+](=O)[O-])ccc3o2)C[C@H]1C(F)(F)F REAL300018133125
O=C(O)[C@@H]1CN(Cc2ccsc2C(F)(F)F)C[C@H]1C(F)(F)F REAL300018133126
COC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)C1CCOC1 REAL300018133127
O=C(O)[C@@H]1CN(Cc2ccnn2C2CCOCC2)C[C@H]1C(F)(F)F REAL300018133128
C[C@]1(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)C[C@@H]1c1ccccc1 REAL300018133129
O=C(O)[C@@H]1CN(C[C@@H]2C[C@H]2c2ccccc2)C[C@H]1C(F)(F)F REAL300018133130
Cc1cccc(-n2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c(C)n2)c1 REAL300018133131
O=C(O)[C@@H]1CN(Cc2ccnn2CC2CCC2)C[C@H]1C(F)(F)F REAL300018133132
COC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)C1CCCC1 REAL300018133133
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133134
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(OC)c1 REAL300018133135
O=C(O)[C@@H]1CN(Cc2ccc(C(F)(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133136
O=C(O)[C@@H]1CN(Cc2ccc(OC(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133137
O=C(O)[C@@H]1CN(Cc2cccc(Oc3ccccc3)c2)C[C@H]1C(F)(F)F REAL300018133138
O=C(O)[C@@H]1CN(Cc2cccc(Cl)c2)C[C@H]1C(F)(F)F REAL300018133139
COc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133140
CC(=Cc1ccccc1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133141
CC(C)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133142
O=C(O)[C@@H]1CN(CC=Cc2ccccc2[N+](=O)[O-])C[C@H]1C(F)(F)F REAL300018133143
O=C(O)[C@@H]1CN(Cc2cccc(C(F)(F)F)c2)C[C@H]1C(F)(F)F REAL300018133144
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(OC)c1OC REAL300018133145
CCOc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133146
CCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133147
COc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133148
O=C(O)[C@@H]1CN(Cc2ccc(OCc3ccccc3)cc2)C[C@H]1C(F)(F)F REAL300018133149
COc1ccc(Br)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133150
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3)cc2)C[C@H]1C(F)(F)F REAL300018133151
COc1ccc2ccccc2c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133152
CSc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133153
O=C(O)[C@@H]1CN(Cc2c(Cl)cccc2Cl)C[C@H]1C(F)(F)F REAL300018133154
COc1cc(OC)c(OC)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133155
O=C(O)[C@@H]1CN(CC(c2ccccc2)c2ccccc2)C[C@H]1C(F)(F)F REAL300018133156
Cc1cc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)c1 REAL300018133157
O=C(O)[C@@H]1CN(Cc2cccc(OCc3ccccc3)c2)C[C@H]1C(F)(F)F REAL300018133158
O=C(O)[C@@H]1CN(Cc2ccccc2Br)C[C@H]1C(F)(F)F REAL300018133159
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)c1 REAL300018133160
Cc1ccc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133161
O=C(O)[C@@H]1CN(Cc2ccc3ncccc3c2)C[C@H]1C(F)(F)F REAL300018133162
CC(C)(C)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133163
COc1cc(OC)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(OC)c1 REAL300018133164
CCCCCCC(=Cc1ccccc1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133165
CCCCCC(=Cc1ccccc1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133166
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2ccccc2)C[C@H]1C(F)(F)F REAL300018133167
Cc1nn(-c2ccccc2)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133168
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC(F)F REAL300018133169
O=C(O)[C@@H]1CN(Cc2cccc(F)c2OC(F)(F)F)C[C@H]1C(F)(F)F REAL300018133170
O=C(O)[C@@H]1CN(Cc2c(C(F)(F)F)nc3n2CCCC3)C[C@H]1C(F)(F)F REAL300018133171
Cn1ncc(C2CC2)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133172
Cn1ncc(C2CCC2)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133173
O=C(O)[C@@H]1CN(Cc2cn(C3CCC3)nn2)C[C@H]1C(F)(F)F REAL300018133174
CC(C)(C)n1nnc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)n1 REAL300018133175
C=CCCn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)nn1 REAL300018133176
O=C(O)[C@@H]1CN(CC[C@@H]2C[C@H]2c2ccccc2)C[C@H]1C(F)(F)F REAL300018133177
Cc1cc(C)c(C=CCN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)c1 REAL300018133178
O=C(O)[C@@H]1CN(Cc2cccc(CC3CCC3)c2)C[C@H]1C(F)(F)F REAL300018133179
Cn1nc2c(c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)CSCC2 REAL300018133180
CCOc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC REAL300018133181
O=C(O)[C@@H]1CN(Cc2ccccc2OCc2ccccc2)C[C@H]1C(F)(F)F REAL300018133182
CCCCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133183
O=C(O)[C@@H]1CN(Cc2ccc(-c3cccc([N+](=O)[O-])c3)o2)C[C@H]1C(F)(F)F REAL300018133184
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccc([N+](=O)[O-])cc3)o2)C[C@H]1C(F)(F)F REAL300018133185
CCCc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133186
Cc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133187
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1Br REAL300018133188
CC(C)Oc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133189
CCCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133190
CCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133191
C=CCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133192
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccc(Cl)cc3)o2)C[C@H]1C(F)(F)F REAL300018133193
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3Cl)o2)C[C@H]1C(F)(F)F REAL300018133194
CCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133195
O=C(O)[C@@H]1CN(Cc2cc3ccccc3o2)C[C@H]1C(F)(F)F REAL300018133196
O=C(O)[C@@H]1CN(Cc2c(OC(F)F)ccc3ccccc23)C[C@H]1C(F)(F)F REAL300018133197
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3)o2)C[C@H]1C(F)(F)F REAL300018133198
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC(C)C REAL300018133199
CCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OCC REAL300018133200
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1[N+](=O)[O-] REAL300018133201
CCn1c2ccccc2c2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)ccc21 REAL300018133202
O=C(O)[C@@H]1CN(Cc2ccc3ccccc3c2)C[C@H]1C(F)(F)F REAL300018133203
CC(C)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1[N+](=O)[O-] REAL300018133204
O=C(O)[C@@H]1CN(Cc2cc(Br)c3c(c2)OCO3)C[C@H]1C(F)(F)F REAL300018133205
Cc1nn(Cc2ccccc2)c(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133206
CCOc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OCC(C)C REAL300018133207
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c([N+](=O)[O-])cc1OC REAL300018133208
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc(OC)c1 REAL300018133209
O=C(O)[C@@H]1CN(Cc2cc3c(cc2Br)OCO3)C[C@H]1C(F)(F)F REAL300018133210
COc1ccc2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)ccc2c1 REAL300018133211
CCCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OCC REAL300018133212
Cc1nn(-c2ccccc2)c(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133213
COc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1OC(F)F REAL300018133214
O=C(O)[C@@H]1CN(Cc2ccc(CSC(F)F)o2)C[C@H]1C(F)(F)F REAL300018133215
Cc1ccc(Cn2nc(C)c(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c2C)cc1 REAL300018133216
CCN(CC)c1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133217
Cc1ccc(COc2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc2)cc1 REAL300018133218
O=C(O)[C@@H]1CN(Cc2ccc(N3CCCCC3)cc2)C[C@H]1C(F)(F)F REAL300018133219
CN(c1ccccc1)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133220
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc(Cl)c1OC REAL300018133221
Cc1nn(C)c(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133222
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OCC(C)C REAL300018133223
CCCOc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC REAL300018133224
O=C(O)[C@@H]1CN(Cc2ccc(Br)s2)C[C@H]1C(F)(F)F REAL300018133225
CCOc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc(Cl)c1OC REAL300018133226
C=CCOc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133227
COc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1OC(C)C REAL300018133228
C#CCOc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133229
CCOc1c(Cl)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133230
CCCOc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cccc1OCC REAL300018133231
CCCCOc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC REAL300018133232
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC(F)F REAL300018133233
Cc1nc2ccccn2c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133234
O=C(O)[C@@H]1CN(Cc2csc(-c3ccc(Cl)cc3)n2)C[C@H]1C(F)(F)F REAL300018133235
CCOc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC(F)F REAL300018133236
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc(C)c1OC(F)F REAL300018133237
CCOc1cc2c(cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)OC(C)C2 REAL300018133238
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc2c1OCCO2 REAL300018133239
O=C(O)[C@@H]1CN(Cc2ccc(-c3nc4ccccc4s3)o2)C[C@H]1C(F)(F)F REAL300018133240
CCOc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1OC(F)F REAL300018133241
Cc1cc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1C REAL300018133242
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc2c1OCO2 REAL300018133243
O=C(O)[C@@H]1CN(Cc2cnn(-c3ccccc3)n2)C[C@H]1C(F)(F)F REAL300018133244
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3)s2)C[C@H]1C(F)(F)F REAL300018133245
CCCOc1c(Cl)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133246
COc1cc2c(cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)OC(C)C2 REAL300018133247
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2ccc(Cl)cc2)C[C@H]1C(F)(F)F REAL300018133248
O=C(O)[C@@H]1CN(Cc2ccc(-n3ccnc3)cc2)C[C@H]1C(F)(F)F REAL300018133249
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3F)o2)C[C@H]1C(F)(F)F REAL300018133250
O=C(O)[C@@H]1CN(Cc2cc(Cl)c3c(c2)OCCO3)C[C@H]1C(F)(F)F REAL300018133251
CCCCc1oc2ccccc2c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133252
O=C(O)[C@@H]1CN(Cc2ccc(-n3cnc4ccccc43)cc2)C[C@H]1C(F)(F)F REAL300018133253
Cc1nn(-c2ccc(F)cc2)c(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133254
O=C(O)[C@@H]1CN(Cc2cc(Cl)c3c(c2)OCCCO3)C[C@H]1C(F)(F)F REAL300018133255
COc1ccc(C)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133256
O=C(O)[C@@H]1CN(Cc2cnc3ccccc3n2)C[C@H]1C(F)(F)F REAL300018133257
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1F REAL300018133258
O=C(O)[C@@H]1CN(Cc2cnn(-c3ccccc3)c2)C[C@H]1C(F)(F)F REAL300018133259
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccc(Cl)cc3)s2)C[C@H]1C(F)(F)F REAL300018133260
O=C(O)[C@@H]1CN(Cc2cnn(Cc3ccccc3)c2)C[C@H]1C(F)(F)F REAL300018133261
CCc1oc2ccccc2c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133262
CC1CC1c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)o1 REAL300018133263
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3[N+](=O)[O-])o2)C[C@H]1C(F)(F)F REAL300018133264
COc1ccc(-c2nc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cs2)cc1 REAL300018133265
O=C(O)[C@@H]1CN(Cc2ccccc2OC(F)(F)F)C[C@H]1C(F)(F)F REAL300018133266
O=C(O)[C@@H]1CN(Cc2ccc(SC(F)(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133267
O=C(O)[C@@H]1CN(Cc2ccc(OCc3cccc(F)c3)cc2)C[C@H]1C(F)(F)F REAL300018133268
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1C REAL300018133269
O=C(O)[C@@H]1CN(Cc2cnn(Cc3ccccc3Cl)c2)C[C@H]1C(F)(F)F REAL300018133270
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(Cl)c1 REAL300018133271
O=C(O)[C@@H]1CN(Cc2ccc(OC(F)(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133272
CC(C)(C)c1n[nH]cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133273
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2ccc(F)cc2)C[C@H]1C(F)(F)F REAL300018133274
Cc1ccc(-c2n[nH]cc2CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133275
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2cccs2)C[C@H]1C(F)(F)F REAL300018133276
COc1ccc(-c2n[nH]cc2CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133277
O=C(O)[C@@H]1CN(Cc2csc3ccccc23)C[C@H]1C(F)(F)F REAL300018133278
CCOc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)nn1CC(C)C REAL300018133279
O=C(O)[C@@H]1CN(CC2=Cc3ccccc3OC2)C[C@H]1C(F)(F)F REAL300018133280
Cc1ccc(-c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)o2)cc1 REAL300018133281
Cc1ccc(-c2n[nH]cc2CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)o1 REAL300018133282
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2ccc3c(c2)OCCO3)C[C@H]1C(F)(F)F REAL300018133283
O=C(O)[C@@H]1CN(Cc2ccc(OCC3CCCO3)cc2)C[C@H]1C(F)(F)F REAL300018133284
O=C(O)[C@@H]1CN(Cc2ccc(Cl)s2)C[C@H]1C(F)(F)F REAL300018133285
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccc(F)cc3)s2)C[C@H]1C(F)(F)F REAL300018133286
O=C(O)[C@@H]1CN(Cc2cccc3cccnc23)C[C@H]1C(F)(F)F REAL300018133287
O=C(O)[C@@H]1CN(Cc2ccccc2OCc2ccccn2)C[C@H]1C(F)(F)F REAL300018133288
O=C(O)[C@@H]1CN(Cc2ccc(-n3cncn3)c(F)c2)C[C@H]1C(F)(F)F REAL300018133289
O=C(O)[C@@H]1CN(Cc2ccc(-n3cncn3)cc2)C[C@H]1C(F)(F)F REAL300018133290
O=C(O)[C@@H]1CN(Cc2ccc3[nH]ccc3c2)C[C@H]1C(F)(F)F REAL300018133291
Cc1nc(C)c2c(C)c(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)sc2n1 REAL300018133292
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3Cl)s2)C[C@H]1C(F)(F)F REAL300018133293
O=C(O)[C@@H]1CN(CC23C4=C5C6=C2[Fe]56432789C3=C2C7C8=C39)C[C@H]1C(F)(F)F REAL300018133294
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccc3F)s2)C[C@H]1C(F)(F)F REAL300018133295
O=C(O)[C@@H]1CN(Cc2ccc(F)cc2Cl)C[C@H]1C(F)(F)F REAL300018133296
COc1cccc(OC)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133297
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1F REAL300018133298
O=C(O)[C@@H]1CN(Cc2cc(Cl)ccc2[N+](=O)[O-])C[C@H]1C(F)(F)F REAL300018133299
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(Cl)c1OC REAL300018133300
O=C(O)[C@@H]1CN(Cc2ccc(-c3cccs3)cc2)C[C@H]1C(F)(F)F REAL300018133301
O=C(O)[C@@H]1CN(Cc2cc3ccccc3s2)C[C@H]1C(F)(F)F REAL300018133302
CC(C)Oc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133303
CCCCCCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133304
CC(Cc1ccc(C(C)(C)C)cc1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133305
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1F REAL300018133306
O=C(O)[C@@H]1CN(Cc2cccc3cc[nH]c23)C[C@H]1C(F)(F)F REAL300018133307
O=C(O)[C@@H]1CN(Cc2csc([N+](=O)[O-])c2)C[C@H]1C(F)(F)F REAL300018133308
O=C(O)[C@@H]1CN(Cc2ccccc2N2CCOCC2)C[C@H]1C(F)(F)F REAL300018133309
CC(C)Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133310
Cc1ccc(-c2cccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c2)cc1 REAL300018133311
Cc1cc(C)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133312
COc1ccc(Br)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133313
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1[N+](=O)[O-] REAL300018133314
O=C(O)[C@@H]1CN(Cc2cc(Cl)cc(Cl)c2)C[C@H]1C(F)(F)F REAL300018133315
Cc1cccc(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133316
Cc1ccccc1-c1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133317
O=C(O)[C@@H]1CN(Cc2cccc(OC(F)F)c2)C[C@H]1C(F)(F)F REAL300018133318
CCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OCC REAL300018133319
O=C(O)[C@@H]1CN(Cc2ccc(Cl)c(C(F)(F)F)c2)C[C@H]1C(F)(F)F REAL300018133320
O=C(O)[C@@H]1CN(Cc2ccc(F)cc2Br)C[C@H]1C(F)(F)F REAL300018133321
O=C(O)[C@@H]1CN(Cc2ccc3c(c2)OC(F)(F)O3)C[C@H]1C(F)(F)F REAL300018133322
O=C(O)[C@@H]1CN(Cc2ccnc3ccccc23)C[C@H]1C(F)(F)F REAL300018133323
O=C(O)[C@@H]1CN(Cc2cccc(OC(F)(F)F)c2)C[C@H]1C(F)(F)F REAL300018133324
CS(=O)(=O)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133325
COc1ccccc1-c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133326
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccc(Cl)cc3)cc2)C[C@H]1C(F)(F)F REAL300018133327
O=C(O)[C@@H]1CN(Cc2cccc(-c3ccc(Cl)cc3)c2)C[C@H]1C(F)(F)F REAL300018133328
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c2ccccc12 REAL300018133329
CCc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133330
Cn1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)nc2ccccc21 REAL300018133331
O=C(O)[C@@H]1CN(Cc2ccc3c(c2)CCO3)C[C@H]1C(F)(F)F REAL300018133332
O=C(O)[C@@H]1CN(Cc2csc(Br)c2)C[C@H]1C(F)(F)F REAL300018133333
O=C(O)[C@@H]1CN(Cc2ccccc2OCc2ccncc2)C[C@H]1C(F)(F)F REAL300018133334
O=C(O)[C@@H]1CN(Cc2ccccc2OCc2cccnc2)C[C@H]1C(F)(F)F REAL300018133335
O=C(O)[C@@H]1CN(Cc2ccc(N3CCCC3)nc2)C[C@H]1C(F)(F)F REAL300018133336
CS(=O)(=O)Nc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133337
O=C(O)[C@@H]1CN(Cc2cccc3[nH]ccc23)C[C@H]1C(F)(F)F REAL300018133338
O=C(O)[C@@H]1CN(Cc2ccc3cc[nH]c3c2)C[C@H]1C(F)(F)F REAL300018133339
O=C(O)[C@@H]1CN(Cc2cccc3c2OC(F)(F)O3)C[C@H]1C(F)(F)F REAL300018133340
Cc1cc(F)ccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133341
CC1(C)CCc2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)ccc2O1 REAL300018133342
CN(C)c1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133343
O=C(O)[C@@H]1CN(Cc2cccc(-c3cccnc3)c2)C[C@H]1C(F)(F)F REAL300018133344
O=C(O)[C@@H]1CN(Cc2cccc(-c3ccncc3)c2)C[C@H]1C(F)(F)F REAL300018133345
CN1CCN(c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc2)CC1 REAL300018133346
Cc1nn(C)c(N2CCOCC2)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133347
O=C(O)[C@@H]1CN(Cc2ccc(Oc3cnccn3)cc2)C[C@H]1C(F)(F)F REAL300018133348
O=C(O)[C@@H]1CN(Cc2cnn(-c3ccc(F)cc3)c2)C[C@H]1C(F)(F)F REAL300018133349
O=C(O)[C@@H]1CN(Cc2cnn(-c3ccc(Cl)cc3)c2)C[C@H]1C(F)(F)F REAL300018133350
CC(C)(C)n1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cn1 REAL300018133351
CN1CCC(N(C)c2ccccc2CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)CC1 REAL300018133352
O=C(O)[C@@H]1CN(Cc2ccc(OCC(F)(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133353
O=C(O)[C@@H]1CN(Cc2ccc(OCCN3CCCC3)cc2)C[C@H]1C(F)(F)F REAL300018133354
O=C(O)[C@@H]1CN(Cc2cc(Cl)ccc2OC(F)F)C[C@H]1C(F)(F)F REAL300018133355
O=C(O)[C@@H]1CN(Cc2ccc(-c3cccc(Cl)c3)s2)C[C@H]1C(F)(F)F REAL300018133356
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2ccc3c(c2)OCO3)C[C@H]1C(F)(F)F REAL300018133357
COc1cccc(-c2n[nH]cc2CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133358
O=C(O)[C@@H]1CN(Cc2cnc(N3CCCC3)nc2)C[C@H]1C(F)(F)F REAL300018133359
O=C(O)[C@@H]1CN(Cc2ccc(OCc3ccncc3)cc2)C[C@H]1C(F)(F)F REAL300018133360
O=C(O)[C@@H]1CN(Cc2cccc(OCc3ccccn3)c2)C[C@H]1C(F)(F)F REAL300018133361
CN(C)CCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133362
CC(C)c1nn(C)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133363
COCCOc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133364
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1Cl REAL300018133365
O=C(O)[C@@H]1CN(CC2=Cc3cc(Cl)cc(Cl)c3OC2)C[C@H]1C(F)(F)F REAL300018133366
O=C(O)[C@@H]1CN(Cc2csc(-c3ccccn3)n2)C[C@H]1C(F)(F)F REAL300018133367
O=C(O)[C@@H]1CN(Cc2cc3c(cc2[N+](=O)[O-])OCCO3)C[C@H]1C(F)(F)F REAL300018133368
CC(C)n1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)nc2ccccc21 REAL300018133369
COc1ncc(Br)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133370
COc1ncccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133371
O=C(O)[C@@H]1CN(Cc2ccc(Br)cn2)C[C@H]1C(F)(F)F REAL300018133372
O=C(O)[C@@H]1CN(Cc2cnc(N3CCOCC3)s2)C[C@H]1C(F)(F)F REAL300018133373
O=C(O)[C@@H]1CN(Cc2cccc3ncccc23)C[C@H]1C(F)(F)F REAL300018133374
O=C(O)[C@@H]1CN(Cc2cccc(OCC(F)(F)F)c2)C[C@H]1C(F)(F)F REAL300018133375
O=C(O)[C@@H]1CN(Cc2cccc3c2OCCO3)C[C@H]1C(F)(F)F REAL300018133376
O=C(O)[C@@H]1CN(Cc2cccc3c2OCCCO3)C[C@H]1C(F)(F)F REAL300018133377
O=C(O)[C@@H]1CN(Cc2cnc(-c3ccccc3)nc2)C[C@H]1C(F)(F)F REAL300018133378
O=C(O)[C@@H]1CN(Cc2cnc(N3CCOCC3)nc2)C[C@H]1C(F)(F)F REAL300018133379
CCCn1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)nc2ccccc21 REAL300018133380
CCCOc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133381
C#CCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133382
O=C(O)[C@@H]1CN(Cc2cc(-c3ccccc3)cs2)C[C@H]1C(F)(F)F REAL300018133383
O=C(O)[C@@H]1CN(Cc2ccc(F)c(-c3cccs3)c2)C[C@H]1C(F)(F)F REAL300018133384
Cc1n[nH]c2ncc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc12 REAL300018133385
O=C(O)[C@@H]1CN(Cc2cccc(OC3CCCC3)c2)C[C@H]1C(F)(F)F REAL300018133386
CCc1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133387
O=C(O)[C@@H]1CN(Cc2ccccc2-n2cncn2)C[C@H]1C(F)(F)F REAL300018133388
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2cccnc2)n1 REAL300018133389
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2ccncc2)n1 REAL300018133390
O=C(O)[C@@H]1CN(Cc2cnc3ccccn23)C[C@H]1C(F)(F)F REAL300018133391
CN(C)c1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133392
CC(C)Oc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133393
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2cc3ccccc3o2)n1 REAL300018133394
Cc1ccc(-c2nc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cs2)cc1 REAL300018133395
CC(C)c1nc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cs1 REAL300018133396
O=C(O)[C@@H]1CN(Cc2csc(C3CC3)n2)C[C@H]1C(F)(F)F REAL300018133397
O=C(O)[C@@H]1CN(Cc2cccc(OCc3ccccc3F)c2)C[C@H]1C(F)(F)F REAL300018133398
O=C(O)[C@@H]1CN(Cc2csc(COc3ccccc3)n2)C[C@H]1C(F)(F)F REAL300018133399
CCc1nc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cs1 REAL300018133400
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2ccc([N+](=O)[O-])cc2)n1 REAL300018133401
CC(C)(C)c1nc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cs1 REAL300018133402
O=C(O)[C@@H]1CN(Cc2csc(-c3ccsc3)n2)C[C@H]1C(F)(F)F REAL300018133403
O=C(O)[C@@H]1CN(Cc2ccc(-c3cccc(F)c3)s2)C[C@H]1C(F)(F)F REAL300018133404
O=C(O)[C@@H]1CN(Cc2ccc3nccnc3c2)C[C@H]1C(F)(F)F REAL300018133405
O=C(O)[C@@H]1CN(Cc2ccccc2OC2CCCC2)C[C@H]1C(F)(F)F REAL300018133406
O=C(O)[C@@H]1CN(Cc2cn3cc(Cl)ccc3n2)C[C@H]1C(F)(F)F REAL300018133407
CC(C)(C)c1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133408
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)s1 REAL300018133409
Cc1ccc(-c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)s2)cc1 REAL300018133410
O=C(O)[C@@H]1CN(Cc2cc([N+](=O)[O-])ccc2OC(F)F)C[C@H]1C(F)(F)F REAL300018133411
COc1c(Cl)cc(Cl)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133412
C#CCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133413
CCOc1c(OC)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133414
COCCCOc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133415
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1SC REAL300018133416
CCC(C)Oc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC REAL300018133417
C=C(C)COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC REAL300018133418
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OCCC(C)C REAL300018133419
CCOCc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1OC REAL300018133420
O=C(O)[C@@H]1CN(Cc2cc(-c3ccccc3)[nH]n2)C[C@H]1C(F)(F)F REAL300018133421
CCOc1ccc([N+](=O)[O-])cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133422
Cc1nn(C)c(OCC(F)(F)F)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133423
O=C(O)[C@@H]1CN(Cc2cn(-c3ccccc3)nn2)C[C@H]1C(F)(F)F REAL300018133424
O=C(O)[C@@H]1CN(Cc2nc(-c3ccccc3)cs2)C[C@H]1C(F)(F)F REAL300018133425
CCn1nc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133426
C=CCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1Cl REAL300018133427
O=C(O)[C@@H]1CN(Cc2cnc(-c3ccccc3)s2)C[C@H]1C(F)(F)F REAL300018133428
COc1cc2c(c(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c1)OC(C)C2 REAL300018133429
Cn1nc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c2ccccc21 REAL300018133430
O=C(O)[C@@H]1CN(Cc2n[nH]c3ccccc23)C[C@H]1C(F)(F)F REAL300018133431
CN(C)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1F REAL300018133432
O=C(O)[C@@H]1CN(Cc2nccn2CC(F)(F)F)C[C@H]1C(F)(F)F REAL300018133433
CC1(C)Cc2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)ccc2O1 REAL300018133434
O=C(O)[C@@H]1CN(Cc2coc(-c3ccccc3)n2)C[C@H]1C(F)(F)F REAL300018133435
O=C(O)[C@@H]1CN(Cc2csc(-c3cccs3)n2)C[C@H]1C(F)(F)F REAL300018133436
O=C(O)[C@@H]1CN(CC2CCCCCCC2)C[C@H]1C(F)(F)F REAL300018133437
Cc1cccc(-c2[nH]ncc2CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133438
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc(C(F)(F)F)c1 REAL300018133439
O=C(O)[C@@H]1CN(Cc2ccc(Br)cc2Cl)C[C@H]1C(F)(F)F REAL300018133440
CN(C)c1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)n1C REAL300018133441
O=C(O)[C@@H]1CN(Cc2nc(-c3ccccc3)c[nH]2)C[C@H]1C(F)(F)F REAL300018133442
CC(C)COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133443
COCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133444
CC1(C)CCCC(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)C1 REAL300018133445
O=C(O)[C@@H]1CN(Cc2ccc(OC(F)F)c(Cl)c2)C[C@H]1C(F)(F)F REAL300018133446
Cc1cc(N(C)C)ccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133447
O=C(O)[C@@H]1CN(Cc2ccc3c(c2)CCC3)C[C@H]1C(F)(F)F REAL300018133448
COc1cc2c(cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)OCO2 REAL300018133449
COc1cc(Cl)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133450
COc1ccsc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133451
CC(C)COc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133452
O=C(O)[C@@H]1CN(Cc2ccc(F)c3ccccc23)C[C@H]1C(F)(F)F REAL300018133453
C=CCOc1c(Cl)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133454
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1Cn1cccn1 REAL300018133455
CC(C)COc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133456
CC1(C)Cc2cccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c2O1 REAL300018133457
O=C(O)[C@@H]1CN(Cc2c(Cl)cncc2Cl)C[C@H]1C(F)(F)F REAL300018133458
O=C(O)[C@@H]1CN(Cc2nc3c(s2)CCCC3)C[C@H]1C(F)(F)F REAL300018133459
O=C(O)[C@@H]1CN(Cc2ccncc2Br)C[C@H]1C(F)(F)F REAL300018133460
O=C(O)[C@@H]1CN(Cc2ccncc2Cl)C[C@H]1C(F)(F)F REAL300018133461
CC(C)(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)N1CCOCC1 REAL300018133462
O=C(O)[C@@H]1CN(Cc2cc(F)cc(Br)c2)C[C@H]1C(F)(F)F REAL300018133463
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2ccccc2)n1 REAL300018133464
CCc1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cn1 REAL300018133465
O=C(O)[C@@H]1CN(Cc2cccc(-n3cccn3)c2)C[C@H]1C(F)(F)F REAL300018133466
O=C(O)[C@@H]1CN(Cc2ccc(C(F)(F)F)cc2[N+](=O)[O-])C[C@H]1C(F)(F)F REAL300018133467
O=C(O)[C@@H]1CN(Cc2ccc3cnccc3c2)C[C@H]1C(F)(F)F REAL300018133468
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)sc1Br REAL300018133469
O=C(O)[C@@H]1CN(Cc2cccc3[nH]ncc23)C[C@H]1C(F)(F)F REAL300018133470
O=C(O)[C@@H]1CN(Cc2cccc3cn[nH]c23)C[C@H]1C(F)(F)F REAL300018133471
O=C(O)[C@@H]1CN(Cc2cc3cc(Br)ccc3o2)C[C@H]1C(F)(F)F REAL300018133472
O=C(O)[C@@H]1CN(Cc2cnc3n2CCC3)C[C@H]1C(F)(F)F REAL300018133473
COc1cc(F)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133474
CC(C)(C)c1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cn1 REAL300018133475
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(Cl)c1 REAL300018133476
COc1ccc(OC(F)F)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133477
O=C(O)[C@@H]1CN(Cc2c(Cl)cccc2OC(F)F)C[C@H]1C(F)(F)F REAL300018133478
O=C(O)[C@@H]1CN(Cc2ccc([N+](=O)[O-])c(Cl)c2)C[C@H]1C(F)(F)F REAL300018133479
O=C(O)[C@@H]1CN(CCc2cccc(Cl)c2)C[C@H]1C(F)(F)F REAL300018133480
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1Oc1cccnc1 REAL300018133481
Cc1ccc(-c2ncc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)s2)cc1 REAL300018133482
O=C(O)[C@@H]1CN(Cc2cc(Cl)cc3cccnc23)C[C@H]1C(F)(F)F REAL300018133483
O=C(O)[C@@H]1CN(Cc2c(Cl)ccc3cccnc23)C[C@H]1C(F)(F)F REAL300018133484
O=C(O)[C@@H]1CN(Cc2ccc(F)c3cccnc23)C[C@H]1C(F)(F)F REAL300018133485
O=C(O)[C@@H]1CN(Cc2cc(F)cc3cccnc23)C[C@H]1C(F)(F)F REAL300018133486
O=C(O)[C@@H]1CN(Cc2ccc(Cl)c3cccnc23)C[C@H]1C(F)(F)F REAL300018133487
CS(=O)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133488
O=C(O)[C@@H]1CN(Cc2ccc([N+](=O)[O-])cc2Cl)C[C@H]1C(F)(F)F REAL300018133489
CC(C)CCn1cccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133490
O=C(O)[C@@H]1CN(Cc2ccc(-c3c(F)cccc3F)o2)C[C@H]1C(F)(F)F REAL300018133491
Cc1cc(F)ccc1-c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)o1 REAL300018133492
CCc1ccc(-c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)o2)cc1 REAL300018133493
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(OC(F)F)c1 REAL300018133494
CCn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2ccccc2)n1 REAL300018133495
O=C(O)[C@@H]1CN(Cc2ccc3c(c2)CCCC3)C[C@H]1C(F)(F)F REAL300018133496
Cc1ccc(C(C)CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133497
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1C(C)(C)C REAL300018133498
COCc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)o1 REAL300018133499
CC(C)(C)Oc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133500
CC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)C1CCCCC1 REAL300018133501
NS(=O)(=O)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133502
CCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)c1 REAL300018133503
COc1cc(C)ccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133504
O=C(O)[C@@H]1CN(CC2CCc3ccccc3C2)C[C@H]1C(F)(F)F REAL300018133505
Nc1c(Cl)cc(Cl)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133506
COCc1csc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133507
CCCc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133508
CC(C)n1ccnc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133509
Cc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cccc1[N+](=O)[O-] REAL300018133510
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1Br REAL300018133511
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1Cl REAL300018133512
COc1cccc(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133513
O=C(O)[C@@H]1CN(Cc2cccc3ccoc23)C[C@H]1C(F)(F)F REAL300018133514
O=C(O)[C@@H]1CN(Cc2ccn(-c3ccccc3)n2)C[C@H]1C(F)(F)F REAL300018133515
O=C(O)[C@@H]1CN(Cc2cnc(C(F)(F)F)s2)C[C@H]1C(F)(F)F REAL300018133516
CCc1nn(C)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133517
O=C(O)[C@@H]1CN(Cc2cc3n(n2)CCCC3)C[C@H]1C(F)(F)F REAL300018133518
CCc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133519
COc1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133520
O=C(O)[C@@H]1CN(Cc2cc3c(cn2)OCCO3)C[C@H]1C(F)(F)F REAL300018133521
O=C(O)[C@@H]1CN(Cc2cnc3ccc(Cl)cn23)C[C@H]1C(F)(F)F REAL300018133522
Cc1cccn2c(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cnc12 REAL300018133523
Cn1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cnc1Cl REAL300018133524
Cn1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cnc1Br REAL300018133525
O=C(O)[C@@H]1CN(Cc2cn(-c3ccc(F)cc3)nn2)C[C@H]1C(F)(F)F REAL300018133526
O=C(O)[C@@H]1CN(Cc2cc(C(F)(F)F)[nH]n2)C[C@H]1C(F)(F)F REAL300018133527
O=C(O)[C@@H]1CN(Cc2cc3c(F)cccc3[nH]2)C[C@H]1C(F)(F)F REAL300018133528
O=C(O)[C@@H]1CN(Cc2cc3ccc(F)cc3[nH]2)C[C@H]1C(F)(F)F REAL300018133529
CCOc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)n1 REAL300018133530
Cc1c(Cl)cccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133531
O=C(O)[C@@H]1CN(Cc2cc3ccncc3s2)C[C@H]1C(F)(F)F REAL300018133532
Cc1cccc2ncc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)n12 REAL300018133533
Cc1cc(Cl)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133534
COCc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133535
O=C(O)[C@@H]1CN(Cc2cnc3c(F)cccc3c2)C[C@H]1C(F)(F)F REAL300018133536
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc2cccnc12 REAL300018133537
CCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1C REAL300018133538
COc1c(C)cnc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133539
COc1cc2ccccc2cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133540
CS(=O)(=O)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133541
O=C(O)[C@@H]1CN(Cc2cnn3cc(Br)cnc23)C[C@H]1C(F)(F)F REAL300018133542
CC(C)(C)c1ccc(-c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)o2)cc1 REAL300018133543
Nc1c(F)cccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133544
CCC(C)CN(C)c1ccc(F)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133545
CCCCCN(C)c1ccc(F)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133546
O=C(O)[C@@H]1CN(Cc2ccc(C(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133547
O=C(O)[C@@H]1CN(Cc2cc3cc(Cl)cnc3o2)C[C@H]1C(F)(F)F REAL300018133548
O=C(O)[C@@H]1CN(Cc2cccc3c2CCC3)C[C@H]1C(F)(F)F REAL300018133549
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c([N+](=O)[O-])n1 REAL300018133550
O=C(O)[C@@H]1CN(Cc2nc(Cl)cs2)C[C@H]1C(F)(F)F REAL300018133551
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)sn1 REAL300018133552
O=C(O)[C@@H]1CN(Cc2cnc3ccc(Br)cn23)C[C@H]1C(F)(F)F REAL300018133553
O=C(O)[C@@H]1CN(Cc2nccc3ccccc23)C[C@H]1C(F)(F)F REAL300018133554
COc1cccc(Cl)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133555
Cc1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)n1-c1ccccc1 REAL300018133556
CCN(c1ccccc1)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133557
CCCn1nc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133558
CCN(CC)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1F REAL300018133559
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(SC)cc1OC REAL300018133560
CCCC(CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1)c1ccccc1 REAL300018133561
O=C(O)[C@@H]1CN(Cc2cnc(C3CC3)o2)C[C@H]1C(F)(F)F REAL300018133562
CC(C)Oc1ccc(F)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133563
O=C(O)[C@@H]1CN(Cc2nc3ccc(F)cc3s2)C[C@H]1C(F)(F)F REAL300018133564
O=C(O)[C@@H]1CN(Cc2cc(F)ccc2OC(F)F)C[C@H]1C(F)(F)F REAL300018133565
COc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc2ccccc12 REAL300018133566
CCOc1cncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133567
CCOc1cc(F)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133568
COc1ccc(C(C)CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133569
Cn1nc(C2CC2)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133570
COc1cccc2c(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cccc12 REAL300018133571
O=C(O)[C@@H]1CN(Cc2ccnn2CC2CC2)C[C@H]1C(F)(F)F REAL300018133572
CC(C)c1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133573
NS(=O)(=O)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)o1 REAL300018133574
COc1cncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133575
O=C(O)[C@@H]1CN(CCc2ccc(F)cc2Cl)C[C@H]1C(F)(F)F REAL300018133576
O=C(O)[C@@H]1CN(Cc2cc3cnccc3o2)C[C@H]1C(F)(F)F REAL300018133577
O=C(O)[C@@H]1CN(Cc2ccc(C(F)(F)F)s2)C[C@H]1C(F)(F)F REAL300018133578
Cc1cccc2[nH]c(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc12 REAL300018133579
O=C(O)[C@@H]1CN(Cc2csc(C(F)(F)F)c2)C[C@H]1C(F)(F)F REAL300018133580
CCCOc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)c1 REAL300018133581
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC1CC1 REAL300018133582
O=C(O)[C@@H]1CN(Cc2ccc(C(F)F)nc2)C[C@H]1C(F)(F)F REAL300018133583
O=C(O)[C@@H]1CN(Cc2ncc(Br)s2)C[C@H]1C(F)(F)F REAL300018133584
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C(F)F)n1 REAL300018133585
O=C(O)[C@@H]1CN(Cc2cccc3c2CCOC3)C[C@H]1C(F)(F)F REAL300018133586
O=C(O)[C@@H]1CN(CC2CC2c2ccc(F)cc2)C[C@H]1C(F)(F)F REAL300018133587
NS(=O)(=O)c1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133588
CCCn1nccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133589
Cc1ccc2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)[nH]c2c1 REAL300018133590
O=C(O)[C@@H]1CN(Cc2cnn3c2CCC3)C[C@H]1C(F)(F)F REAL300018133591
O=C(O)[C@@H]1CN(Cc2cc3n(n2)CCC3)C[C@H]1C(F)(F)F REAL300018133592
O=C(O)[C@@H]1CN(Cc2ncc(C(F)(F)F)s2)C[C@H]1C(F)(F)F REAL300018133593
O=C(O)[C@@H]1CN(Cc2cccc(F)c2OC(F)F)C[C@H]1C(F)(F)F REAL300018133594
Cc1ccc([N+](=O)[O-])c(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133595
O=C(O)[C@@H]1CN(Cc2cc3cccnc3o2)C[C@H]1C(F)(F)F REAL300018133596
Cc1cc(C)cc(-c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc2)c1 REAL300018133597
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1-n1cncn1 REAL300018133598
O=C(O)[C@@H]1CN(Cc2cc3cc(F)ccc3o2)C[C@H]1C(F)(F)F REAL300018133599
O=C(O)[C@@H]1CN(Cc2ccc(OCC(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133600
O=C(O)[C@@H]1CN(Cc2cc3c(cc2OC(F)F)OCO3)C[C@H]1C(F)(F)F REAL300018133601
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(Br)c1 REAL300018133602
COCc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133603
Cc1nn(-c2ccc(Cl)cc2)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133604
CN(C)Cc1nc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cs1 REAL300018133605
O=C(O)[C@@H]1CN(Cc2ccc(Sc3ccccc3)cc2)C[C@H]1C(F)(F)F REAL300018133606
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(OC(F)F)cc1C REAL300018133607
Cc1ccc(CCN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133608
COc1cc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC REAL300018133609
O=C(O)[C@@H]1CN(Cc2ccccc2C2CC2)C[C@H]1C(F)(F)F REAL300018133610
O=C(O)[C@@H]1CN(Cc2cc(Cl)cc(Cl)c2[N+](=O)[O-])C[C@H]1C(F)(F)F REAL300018133611
Cc1sc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1Br REAL300018133612
O=C(O)[C@@H]1CN(CCc2ccc(F)cc2F)C[C@H]1C(F)(F)F REAL300018133613
Cc1cc(C)cc(CCN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133614
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2cccc(Cl)c2)C[C@H]1C(F)(F)F REAL300018133615
COc1ccc(-n2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cn2)cc1 REAL300018133616
Cc1nn(-c2ccccc2Cl)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133617
CN(Cc1cccs1)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133618
O=C(O)[C@@H]1CN(Cc2c(F)cncc2Br)C[C@H]1C(F)(F)F REAL300018133619
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2ccsc2)C[C@H]1C(F)(F)F REAL300018133620
O=C(O)[C@@H]1CN(Cc2cc(-c3ccccn3)n[nH]2)C[C@H]1C(F)(F)F REAL300018133621
Cn1ncc2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cnc21 REAL300018133622
CC(C)Sc1cccc(Cl)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133623
CSc1cc(Br)ccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133624
CN(Cc1ccccc1)CC(C)(C)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133625
Cn1cc(CCCN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cn1 REAL300018133626
CN1CCN(c2ncc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cn2)CC1 REAL300018133627
O=C(O)[C@@H]1CN(Cc2nnn(-c3ccccc3)c2C2CC2)C[C@H]1C(F)(F)F REAL300018133628
Cn1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)nc2cc(C(F)(F)F)ccc21 REAL300018133629
CC1CCc2nc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)sc2C1 REAL300018133630
CCc1cnc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)s1 REAL300018133631
O=C(O)[C@@H]1CN(Cc2ccccc2N2CCCCC2)C[C@H]1C(F)(F)F REAL300018133632
Cn1cnc2cccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c21 REAL300018133633
COc1ccc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133634
O=C(O)[C@@H]1CN(Cc2cc(C3CCC3)on2)C[C@H]1C(F)(F)F REAL300018133635
CC1(c2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)no2)CC1 REAL300018133636
CCc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133637
Cc1cc(F)cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133638
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)c1C REAL300018133639
CC(C)(C)c1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133640
O=C(O)[C@@H]1CN(Cc2cnc3n2CCCCC3)C[C@H]1C(F)(F)F REAL300018133641
COc1ccc2sc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc2c1 REAL300018133642
O=C(O)[C@@H]1CN(Cc2conc2C2CC2)C[C@H]1C(F)(F)F REAL300018133643
O=C(O)[C@@H]1CN(Cc2cc(-c3ccccc3)no2)C[C@H]1C(F)(F)F REAL300018133644
CCN1CCc2cc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)ccc21 REAL300018133645
CSc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1Cl REAL300018133646
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1C1CC1 REAL300018133647
CCOc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccn1 REAL300018133648
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1C1CC1 REAL300018133649
Cc1ccn(-c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c(C)c2)n1 REAL300018133650
O=C(O)[C@@H]1CN(Cc2ccc(C(F)(F)C(F)(F)F)cc2)C[C@H]1C(F)(F)F REAL300018133651
Cc1cc(-n2cc(Cl)cn2)ccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133652
Cc1nn(-c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc2)cc1Cl REAL300018133653
O=C(O)[C@@H]1CN(Cc2cnc(C3CCOCC3)o2)C[C@H]1C(F)(F)F REAL300018133654
O=C(O)[C@@H]1CN(Cc2cc(C3CC3)on2)C[C@H]1C(F)(F)F REAL300018133655
CC1Oc2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc2C1C REAL300018133656
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OC(F)F REAL300018133657
CC(C)c1ccc(O)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133658
Cc1c(C(F)(F)F)n[nH]c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133659
Cc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1O REAL300018133660
O=C(O)[C@@H]1CN(Cc2nc(C3CC3)cs2)C[C@H]1C(F)(F)F REAL300018133661
O=C(O)[C@@H]1CN(Cc2cn(CC3CC3)nn2)C[C@H]1C(F)(F)F REAL300018133662
O=C(O)[C@@H]1CN(Cc2ccc3c(c2)OCC3)C[C@H]1C(F)(F)F REAL300018133663
O=C(O)[C@@H]1CN(Cc2nc3c([nH]2)CCCC3)C[C@H]1C(F)(F)F REAL300018133664
O=C(O)[C@@H]1CN(Cc2ccc3c(c2)CCOC3)C[C@H]1C(F)(F)F REAL300018133665
Cc1cccc(F)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133666
O=C(O)[C@@H]1CN(Cc2ccccc2C2CCC2)C[C@H]1C(F)(F)F REAL300018133667
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C2CCOCC2)n1 REAL300018133668
O=C(O)[C@@H]1CN(Cc2cncc(-c3cccnc3)c2)C[C@H]1C(F)(F)F REAL300018133669
CSc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133670
CC(C)(C)n1nccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133671
CC(C)c1cnn(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133672
O=C(O)[C@@H]1CN(Cc2ccc(CC3CC3)s2)C[C@H]1C(F)(F)F REAL300018133673
O=C(O)[C@@H]1CN(Cc2ccc(OC3CC3)cc2)C[C@H]1C(F)(F)F REAL300018133674
O=C(O)[C@@H]1CN(Cc2ccc(OC(F)(F)F)cc2F)C[C@H]1C(F)(F)F REAL300018133675
O=C(O)[C@@H]1CN(Cc2cccc(C(F)(F)C(F)(F)F)c2)C[C@H]1C(F)(F)F REAL300018133676
Cc1cc(-n2ccnc2C)ccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133677
Cc1ncn(-c2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc2)c1C REAL300018133678
O=C(O)[C@@H]1CN(Cc2ccc(C3CC3)c(C3CC3)c2)C[C@H]1C(F)(F)F REAL300018133679
CN(C)CCc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133680
Cc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)oc2ccc(F)cc12 REAL300018133681
Cn1nc(-c2ccccc2)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133682
CCCn1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)n1 REAL300018133683
CC(C)n1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)n1 REAL300018133684
CC(C)(C)c1cncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133685
O=C(O)[C@@H]1CN(Cc2ccn(CC(F)(F)F)n2)C[C@H]1C(F)(F)F REAL300018133686
Cn1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)nc2c1CCCC2 REAL300018133687
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C(F)(F)F)n1 REAL300018133688
O=C(O)[C@@H]1CN(Cc2cc3ccccc3cn2)C[C@H]1C(F)(F)F REAL300018133689
COc1nc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc1C REAL300018133690
O=C(O)[C@@H]1CN(Cc2cccc(C(F)F)c2F)C[C@H]1C(F)(F)F REAL300018133691
O=C(O)[C@@H]1CN(Cc2cccc3c2COCC3)C[C@H]1C(F)(F)F REAL300018133692
CCOc1ccc(Cl)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133693
O=C(O)[C@@H]1CN(Cc2c[nH]nc2-c2cccc(F)c2)C[C@H]1C(F)(F)F REAL300018133694
O=C(O)[C@@H]1CN(Cc2cc3c(o2)CCCC3)C[C@H]1C(F)(F)F REAL300018133695
CCC(C)n1nccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133696
O=C(O)[C@@H]1CN(Cc2cnn(C3CCCCC3)c2)C[C@H]1C(F)(F)F REAL300018133697
COc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cccc1C(C)(C)C REAL300018133698
Cn1cc(Br)nc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133699
COc1cc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cn1 REAL300018133700
O=C(O)[C@@H]1CN(Cc2nc3ccccc3s2)C[C@H]1C(F)(F)F REAL300018133701
CCCn1cncc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133702
Cc1cc(C)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C)c1Br REAL300018133703
O=C(O)[C@@H]1CN(CC=Cc2ccc3c(c2)OCO3)C[C@H]1C(F)(F)F REAL300018133704
O=C(O)[C@@H]1CN(Cc2ccc(CC3CCC3)cc2)C[C@H]1C(F)(F)F REAL300018133705
CCc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cnn1CC REAL300018133706
Cc1occ(C(F)(F)F)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133707
CC(F)(F)c1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1 REAL300018133708
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccsc3)nc2)C[C@H]1C(F)(F)F REAL300018133709
Cn1cc(-c2n[nH]cc2CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cn1 REAL300018133710
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccsc3)cc2)C[C@H]1C(F)(F)F REAL300018133711
O=C(O)[C@@H]1CN(Cc2cccc3cc(Cl)ccc23)C[C@H]1C(F)(F)F REAL300018133712
COc1c(C)c(C)c(OC)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133713
O=C(O)[C@@H]1CN(Cc2ccccc2OC2CCCCC2)C[C@H]1C(F)(F)F REAL300018133714
O=C(O)[C@@H]1CN(Cc2ccc(Oc3cccc(Cl)c3)cc2)C[C@H]1C(F)(F)F REAL300018133715
C=CCc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133716
O=C(O)[C@@H]1CN(Cc2ccccc2COC2CCCCC2)C[C@H]1C(F)(F)F REAL300018133717
COc1cccc(Oc2ccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)cc2)c1 REAL300018133718
COc1ccccc1Oc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133719
COCc1ccccc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133720
O=C(O)[C@@H]1CN(Cc2ccccc2Cc2ccc(Cl)cc2)C[C@H]1C(F)(F)F REAL300018133721
O=C(O)[C@@H]1CN(Cc2cccc(SC(F)(F)F)c2)C[C@H]1C(F)(F)F REAL300018133722
O=C(O)[C@@H]1CN(Cc2ccc3c(c2)COCC3)C[C@H]1C(F)(F)F REAL300018133723
Cc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)sc2cc(F)ccc12 REAL300018133724
O=C(O)[C@@H]1CN(Cc2cc(-c3ccncc3)n[nH]2)C[C@H]1C(F)(F)F REAL300018133725
COc1ccc(F)c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1OC REAL300018133726
O=C(O)[C@@H]1CN(CC=Cc2ccncc2)C[C@H]1C(F)(F)F REAL300018133727
CCn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C2CC2)n1 REAL300018133728
CCc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)nc1 REAL300018133729
COc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1OCCO REAL300018133730
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(-c2ccnn2C)n1 REAL300018133731
CC(C)(C)c1nocc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133732
O=C(O)[C@@H]1CN(Cc2ccc3ccncc3c2)C[C@H]1C(F)(F)F REAL300018133733
Cc1cc2cccc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)c2o1 REAL300018133734
O=C(O)[C@@H]1CN(Cc2cccc(F)c2C(F)(F)F)C[C@H]1C(F)(F)F REAL300018133735
O=C(O)[C@@H]1CN(Cc2c(F)cccc2OCC(F)(F)F)C[C@H]1C(F)(F)F REAL300018133736
O=C(O)[C@@H]1CN(Cc2conc2C2CCC2)C[C@H]1C(F)(F)F REAL300018133737
O=C(O)[C@@H]1CN(Cc2ccc(C(F)(F)F)cc2F)C[C@H]1C(F)(F)F REAL300018133738
CC(C)Oc1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1F REAL300018133739
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)n(C2CCCC2)n1 REAL300018133740
O=C(O)[C@@H]1CN(Cc2ccnn2CC(F)F)C[C@H]1C(F)(F)F REAL300018133741
O=C(O)[C@@H]1CN(Cc2cc3cnccc3[nH]2)C[C@H]1C(F)(F)F REAL300018133742
O=C(O)[C@@H]1CN(Cc2cnn(-c3cccc(F)c3)c2)C[C@H]1C(F)(F)F REAL300018133743
O=C(O)[C@@H]1CN(Cc2ccn(C3CCC3)n2)C[C@H]1C(F)(F)F REAL300018133744
O=C(O)[C@@H]1CN(Cc2ccn(CC(F)F)n2)C[C@H]1C(F)(F)F REAL300018133745
O=C(O)[C@@H]1CN(Cc2ccn(C3CC3(F)F)n2)C[C@H]1C(F)(F)F REAL300018133746
O=C(O)[C@@H]1CN(Cc2ccn(C3CCCC3)n2)C[C@H]1C(F)(F)F REAL300018133747
O=C(O)[C@@H]1CN(Cc2ccc(F)c3ccoc23)C[C@H]1C(F)(F)F REAL300018133748
O=C(O)[C@@H]1CN(Cc2cc(Cl)cc3ccoc23)C[C@H]1C(F)(F)F REAL300018133749
COc1ccc2sc(CN3C[C@@H](C(=O)O)[C@H](C(F)(F)F)C3)nc2c1 REAL300018133750
O=C(O)[C@@H]1CN(Cc2cnc3cc(Br)ccn23)C[C@H]1C(F)(F)F REAL300018133751
Cc1cc(Br)cc(C)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133752
Cn1nc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1-c1ccco1 REAL300018133753
O=C(O)[C@@H]1CN(Cc2c(Cl)ccc3c2OCO3)C[C@H]1C(F)(F)F REAL300018133754
O=C(O)[C@@H]1CN(Cc2ccc(C3CCCCC3)cc2)C[C@H]1C(F)(F)F REAL300018133755
Cc1nn(C2CCC2)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133756
COc1ccccc1C=CCN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133757
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccccn3)nc2)C[C@H]1C(F)(F)F REAL300018133758
Cn1nc(-c2ccco2)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133759
O=C(O)[C@@H]1CN(Cc2ccc(Cc3ccccc3)cc2)C[C@H]1C(F)(F)F REAL300018133760
O=C(O)[C@@H]1CN(Cc2cc(-c3ccccc3)ccn2)C[C@H]1C(F)(F)F REAL300018133761
CC(C)(C)c1nn(C(C)(C)C)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133762
COc1cc(C)cc(OC)c1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133763
O=C(O)[C@@H]1CN(Cc2ccc(CF)cc2)C[C@H]1C(F)(F)F REAL300018133764
O=C(O)[C@@H]1CN(Cc2ccc(OC(F)(F)F)c(Cl)c2)C[C@H]1C(F)(F)F REAL300018133765
O=C(O)[C@@H]1CN(Cc2cccc(C3CC(F)(F)C3(F)F)c2)C[C@H]1C(F)(F)F REAL300018133766
O=C(O)[C@@H]1CN(Cc2ccc3sccc3c2)C[C@H]1C(F)(F)F REAL300018133767
O=C(O)[C@@H]1CN(Cc2ccc(-c3ccncc3)cc2)C[C@H]1C(F)(F)F REAL300018133768
Cc1cccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C(F)(F)F REAL300018133769
C=CCn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cn1 REAL300018133770
O=C(O)[C@@H]1CN(Cc2ccc3cn[nH]c3c2)C[C@H]1C(F)(F)F REAL300018133771
CCC(C)c1ccc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cc1 REAL300018133772
Cn1c(Cc2ccccc2)cnc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133773
O=C(O)[C@@H]1CN(Cc2cccc3c2CCCC3)C[C@H]1C(F)(F)F REAL300018133774
CC(=Cc1cc(F)cc(F)c1)CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133775
O=C(O)[C@@H]1CN(Cc2ccc(-n3ccnn3)cc2)C[C@H]1C(F)(F)F REAL300018133776
Cc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc2ccccc12 REAL300018133777
CC(C)c1nn(C(C)(C)C)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133778
COc1c(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)ccc2[nH]ccc12 REAL300018133779
O=C(O)[C@@H]1CN(Cc2ccc(N3CCC(O)C3)cc2)C[C@H]1C(F)(F)F REAL300018133780
CCCn1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c1C REAL300018133781
Cc1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)cnc1-n1cccn1 REAL300018133782
CCCn1nc(C)cc1CN1C[C@@H](C(=O)O)[C@H](C(F)(F)F)C1 REAL300018133783
Cn1cc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)c(C2CCC2)n1 REAL300018133784
CC(C)(C)c1ncc(CN2C[C@@H](C(=O)O)[C@H](C(F)(F)F)C2)o1 REAL300018133785
Cc1cc(Br)c(OCC(=O)O)c(CNC(C)C)c1 REAL300018133786
CC(C)NCc1cnc2c(Br)cc(C(=O)O)cn12 REAL300018133787
CC(C)NCc1cnc2c(C(=O)O)cc(Br)cn12 REAL300018133788
CC(C)NC1CC(C(=O)O)(c2cccc(Br)c2)C1 REAL300018133789
O=C(O)c1ccccc1-c1ccc(CNc2ccc3c(c2)OCO3)o1 REAL300018133790
O=C(O)c1ccc(COc2ccccc2CNc2ccc3c(c2)OCO3)cc1 REAL300018133791
O=C(O)c1ccc(-c2ccc(CNc3ccc4c(c3)OCO4)o2)cc1 REAL300018133792
O=C(O)c1ccc(-c2ccc(CNc3ccc4c(c3)OCO4)o2)cc1 REAL300018133793
O=C(O)c1nn(-c2ccccc2)cc1CNc1ccc2c(c1)OCO2 REAL300018133794
Cc1cc(CNc2ccc3c(c2)OCO3)cc(C)c1OCC(=O)O REAL300018133795
O=C(O)CCCN1CCC(Nc2ccc3c(c2)OCO3)CC1 REAL300018133796
Cc1nn(CCC(=O)O)c(C)c1CNc1ccc2c(c1)OCO2 REAL300018133797
O=C(O)COc1ccc(CNc2ccc3c(c2)OCO3)cc1 REAL300018133798
O=C(O)COc1ccc(CNc2ccc3c(c2)OCO3)cc1 REAL300018133799
CC(Oc1ccc(CNc2ccc3c(c2)OCO3)cc1)C(=O)O REAL300018133800
COc1ccc(CNc2ccc3c(c2)OCO3)c2cc(C(=O)O)oc12 REAL300018133801
O=C(O)C(F)(F)C1CCCC(Nc2ccc3c(c2)OCO3)C1 REAL300018133802
O=C(O)c1ccc(CNc2ccc3c(c2)OCO3)cc1Cl REAL300018133803
O=C(O)c1ccc(CNc2ccc3c(c2)OCO3)c(C(F)(F)F)c1 REAL300018133804
Cc1cc(Br)c(OCC(=O)O)c(CNc2ccc3c(c2)OCO3)c1 REAL300018133805
O=C(O)c1ccc(CNc2ccc3c(c2)OCO3)cc1Br REAL300018133806
O=C(O)CCCC1CCCC(Nc2ccc3c(c2)OCO3)C1 REAL300018133807
O=C(O)Cn1cc(CNc2ccc3c(c2)OCO3)c(-c2ccccc2)n1 REAL300018133808
O=C(O)C1(c2ccccc2)CC(Nc2ccc3c(c2)OCO3)C1 REAL300018133809
O=C(O)c1cc2cc(CNc3ccc4c(c3)OCO4)sc2s1 REAL300018133810
O=C(O)c1cnn2cc(CNc3ccc4c(c3)OCO4)cnc12 REAL300018133811
CC(Oc1ccc(Cl)cc1CNc1ccc2c(c1)OCO2)C(=O)O REAL300018133812
O=C(O)c1cc(F)c(CNc2ccc3c(c2)OCO3)c(F)c1 REAL300018133813
O=C(O)c1ccc2ncc(CNc3ccc4c(c3)OCO4)n2c1 REAL300018133814
O=C(O)c1cc(Br)c2ncc(CNc3ccc4c(c3)OCO4)n2c1 REAL300018133815
O=C(O)c1cnc2c(CNc3ccc4c(c3)OCO4)cccn12 REAL300018133816
O=C(O)c1cccc(CNc2ccc3c(c2)OCO3)c1Br REAL300018133817
O=C(O)[C@H]1C[C@H](n2ccc(CNc3ccc4c(c3)OCO4)n2)C1 REAL300018133818
O=C(O)[C@H]1C[C@H](n2nccc2CNc2ccc3c(c2)OCO3)C1 REAL300018133819
O=C(O)c1cc(CNc2ccc3c(c2)OCO3)cc(C(F)(F)F)c1 REAL300018133820
O=C(O)c1cc(Br)cn2c(CNc3ccc4c(c3)OCO4)cnc12 REAL300018133821
O=C(O)C1(c2cccc(Br)c2)CC(Nc2ccc3c(c2)OCO3)C1 REAL300018133822
O=C(O)c1cc(Br)cc(CNc2ccc3c(c2)OCO3)c1 REAL300018133823
CC(C)CN(Cc1ccc(-c2ccccc2C(=O)O)o1)CC(C)C REAL300018133824
CC(C)CN(Cc1ccc(-c2ccc(C(=O)O)cc2)o1)CC(C)C REAL300018133825
CC(C)CN(Cc1ccc(-c2ccc(C(=O)O)cc2)o1)CC(C)C REAL300018133826
Cc1cc(CN(CC(C)C)CC(C)C)cc(C)c1OCC(=O)O REAL300018133827
CC(C)CN(Cc1ccc(OC(C)C(=O)O)cc1)CC(C)C REAL300018133828
CC(C)CN(Cc1ccc(C(=O)O)c(Br)c1)CC(C)C REAL300018133829
CC(C)CN(Cc1cc2cc(C(=O)O)sc2s1)CC(C)C REAL300018133830
CC(C)CN(Cc1cnc2c(C(=O)O)cnn2c1)CC(C)C REAL300018133831
CC(C)CN(Cc1cnc2ccc(C(=O)O)cn12)CC(C)C REAL300018133832
CC(C)CN(Cc1cnc2c(Br)cc(C(=O)O)cn12)CC(C)C REAL300018133833
CC(C)CN(Cc1cccn2c(C(=O)O)cnc12)CC(C)C REAL300018133834
CC(C)CN(Cc1cccc(C(=O)O)c1Br)CC(C)C REAL300018133835
CC(C)CN(Cc1ccn([C@H]2C[C@H](C(=O)O)C2)n1)CC(C)C REAL300018133836
CC(C)CN(Cc1ccnn1[C@H]1C[C@H](C(=O)O)C1)CC(C)C REAL300018133837
CC(C)CN(Cc1cc(C(=O)O)cc(C(F)(F)F)c1)CC(C)C REAL300018133838
CC(C)CN(Cc1cnc2c(C(=O)O)cc(Br)cn12)CC(C)C REAL300018133839
CC(C)CN(Cc1cc(Br)cc(C(=O)O)c1)CC(C)C REAL300018133840
O=C(O)c1ccccc1-c1ccc(CNc2ccc3c(c2)OCCO3)o1 REAL300018133841
O=C(O)c1ccc(COc2ccccc2CNc2ccc3c(c2)OCCO3)cc1 REAL300018133842
O=C(O)c1ccc(-c2ccc(CNc3ccc4c(c3)OCCO4)o2)cc1 REAL300018133843
O=C(O)c1ccc(-c2ccc(CNc3ccc4c(c3)OCCO4)o2)cc1 REAL300018133844
O=C(O)c1nn(-c2ccccc2)cc1CNc1ccc2c(c1)OCCO2 REAL300018133845
Cc1cc(CNc2ccc3c(c2)OCCO3)cc(C)c1OCC(=O)O REAL300018133846
O=C(O)CCCN1CCC(Nc2ccc3c(c2)OCCO3)CC1 REAL300018133847
Cc1nn(CCC(=O)O)c(C)c1CNc1ccc2c(c1)OCCO2 REAL300018133848
O=C(O)COc1ccc(CNc2ccc3c(c2)OCCO3)cc1 REAL300018133849
O=C(O)COc1ccc(CNc2ccc3c(c2)OCCO3)cc1 REAL300018133850
CC(Oc1ccc(CNc2ccc3c(c2)OCCO3)cc1)C(=O)O REAL300018133851
COc1ccc(CNc2ccc3c(c2)OCCO3)c2cc(C(=O)O)oc12 REAL300018133852
O=C(O)C=Cc1ccc(CNc2ccc3c(c2)OCCO3)o1 REAL300018133853
O=C(O)C(F)(F)C1CCCC(Nc2ccc3c(c2)OCCO3)C1 REAL300018133854
O=C(O)C(F)(F)C1CCC(Nc2ccc3c(c2)OCCO3)C1 REAL300018133855
O=C(O)c1ccc(CNc2ccc3c(c2)OCCO3)cc1Cl REAL300018133856
O=C(O)c1ccc(CNc2ccc3c(c2)OCCO3)c(C(F)(F)F)c1 REAL300018133857
O=C(O)c1ccc(CNc2ccc3c(c2)OCCO3)cc1Br REAL300018133858
CCc1oc(CNc2ccc3c(c2)OCCO3)cc1C(=O)O REAL300018133859
O=C(O)CCCC1CCCC(Nc2ccc3c(c2)OCCO3)C1 REAL300018133860
CC(CCCC(C)(C)C(=O)O)Nc1ccc2c(c1)OCCO2 REAL300018133861
O=C(O)Cn1cc(CNc2ccc3c(c2)OCCO3)c(-c2ccccc2)n1 REAL300018133862
O=C(O)C1(c2ccccc2)CC(Nc2ccc3c(c2)OCCO3)C1 REAL300018133863
O=C(O)CCc1ccc(CNc2ccc3c(c2)OCCO3)o1 REAL300018133864
O=C(O)c1cc(CNc2ccc3c(c2)OCCO3)ccc1F REAL300018133865
O=C(O)c1cc2cc(CNc3ccc4c(c3)OCCO4)sc2s1 REAL300018133866
O=C(O)c1cnn2cc(CNc3ccc4c(c3)OCCO4)cnc12 REAL300018133867
CC(Oc1ccc(Cl)cc1CNc1ccc2c(c1)OCCO2)C(=O)O REAL300018133868
O=C(O)c1cc(F)c(CNc2ccc3c(c2)OCCO3)c(F)c1 REAL300018133869
O=C(O)c1ccc2ncc(CNc3ccc4c(c3)OCCO4)n2c1 REAL300018133870
Cc1cc(C(=O)O)ncc1CNc1ccc2c(c1)OCCO2 REAL300018133871
O=C(O)c1cnc2c(CNc3ccc4c(c3)OCCO4)cccn12 REAL300018133872
O=C(O)c1cccc(CNc2ccc3c(c2)OCCO3)c1Br REAL300018133873
O=C(O)[C@H]1C[C@H](n2ccc(CNc3ccc4c(c3)OCCO4)n2)C1 REAL300018133874
O=C(O)[C@H]1C[C@H](n2nccc2CNc2ccc3c(c2)OCCO3)C1 REAL300018133875
O=C(O)c1cc(CNc2ccc3c(c2)OCCO3)cc(C(F)(F)F)c1 REAL300018133876
O=C(O)c1ccc(O)c(CNc2ccc3c(c2)OCCO3)c1 REAL300018133877
O=C(O)c1cc(Br)cc(CNc2ccc3c(c2)OCCO3)c1 REAL300018133878
Cc1ccc(C)c(NCc2ccc(-c3ccccc3C(=O)O)o2)c1 REAL300018133879
Cc1ccc(C)c(NCc2ccccc2OCc2ccc(C(=O)O)cc2)c1 REAL300018133880
Cc1ccc(C)c(NCc2ccc(-c3ccc(C(=O)O)cc3)o2)c1 REAL300018133881
Cc1ccc(C)c(NCc2ccc(-c3ccc(C(=O)O)cc3)o2)c1 REAL300018133882
Cc1ccc(C)c(NCc2cn(-c3ccccc3)nc2C(=O)O)c1 REAL300018133883
Cc1ccc(C)c(NCc2cc(C)c(OCC(=O)O)c(C)c2)c1 REAL300018133884
Cc1ccc(C)c(NCc2c(C)nn(CCC(=O)O)c2C)c1 REAL300018133885
COc1ccc(CNc2cc(C)ccc2C)c2cc(C(=O)O)oc12 REAL300018133886
Cc1ccc(C)c(NCc2ccc(C(=O)O)cc2C(F)(F)F)c1 REAL300018133887
Cc1cc(Br)c(OCC(=O)O)c(CNc2cc(C)ccc2C)c1 REAL300018133888
Cc1ccc(C)c(NCc2ccc(C(=O)O)c(Br)c2)c1 REAL300018133889
Cc1ccc(C)c(NCc2cn(CC(=O)O)nc2-c2ccccc2)c1 REAL300018133890
Cc1ccc(C)c(NCc2cc3cc(C(=O)O)sc3s2)c1 REAL300018133891
Cc1ccc(C)c(NCc2cc(Cl)ccc2OC(C)C(=O)O)c1 REAL300018133892
Cc1ccc(C)c(NCc2cnc3c(Br)cc(C(=O)O)cn23)c1 REAL300018133893
Cc1ccc(C)c(NCc2cccc(C(=O)O)c2Br)c1 REAL300018133894
Cc1ccc(C)c(NCc2cc(C(=O)O)cc(C(F)(F)F)c2)c1 REAL300018133895
Cc1ccc(C)c(NCc2cnc3c(C(=O)O)cc(Br)cn23)c1 REAL300018133896
Cc1ccc(C)c(NC2CC(C(=O)O)(c3cccc(Br)c3)C2)c1 REAL300018133897
Cc1ccc(C)c(NCc2cc(Br)cc(C(=O)O)c2)c1 REAL300018133898
O=C(O)c1ccc(COc2ccccc2CNCc2ccco2)cc1 REAL300018133899
COc1ccc(CNCc2ccco2)c2cc(C(=O)O)oc12 REAL300018133900
Cc1cc(Br)c(OCC(=O)O)c(CNCc2ccco2)c1 REAL300018133901
O=C(O)c1ccc(CNCc2ccco2)cc1Br REAL300018133902
O=C(O)Cn1cc(CNCc2ccco2)c(-c2ccccc2)n1 REAL300018133903
CC(Oc1ccc(Cl)cc1CNCc1ccco1)C(=O)O REAL300018133904
O=C(O)c1cc(Br)c2ncc(CNCc3ccco3)n2c1 REAL300018133905
O=C(O)c1cccc(CNCc2ccco2)c1Br REAL300018133906
O=C(O)c1cc(Br)cn2c(CNCc3ccco3)cnc12 REAL300018133907
O=C(O)C1(c2cccc(Br)c2)CC(NCc2ccco2)C1 REAL300018133908
O=C(O)c1cc(Br)cc(CNCc2ccco2)c1 REAL300018133909
O=C(O)c1ccccc1-c1ccc(CNCc2ccc3c(c2)OCO3)o1 REAL300018133910
O=C(O)c1ccc(COc2ccccc2CNCc2ccc3c(c2)OCO3)cc1 REAL300018133911
O=C(O)c1ccc(-c2ccc(CNCc3ccc4c(c3)OCO4)o2)cc1 REAL300018133912
O=C(O)c1ccc(-c2ccc(CNCc3ccc4c(c3)OCO4)o2)cc1 REAL300018133913
O=C(O)c1nn(-c2ccccc2)cc1CNCc1ccc2c(c1)OCO2 REAL300018133914
Cc1cc(CNCc2ccc3c(c2)OCO3)cc(C)c1OCC(=O)O REAL300018133915
O=C(O)CCCN1CCC(NCc2ccc3c(c2)OCO3)CC1 REAL300018133916
Cc1nn(CCC(=O)O)c(C)c1CNCc1ccc2c(c1)OCO2 REAL300018133917
O=C(O)COc1ccc(CNCc2ccc3c(c2)OCO3)cc1 REAL300018133918
O=C(O)COc1ccc(CNCc2ccc3c(c2)OCO3)cc1 REAL300018133919
CC(Oc1ccc(CNCc2ccc3c(c2)OCO3)cc1)C(=O)O REAL300018133920
COc1ccc(CNCc2ccc3c(c2)OCO3)c2cc(C(=O)O)oc12 REAL300018133921
O=C(O)C=Cc1ccc(CNCc2ccc3c(c2)OCO3)o1 REAL300018133922
O=C(O)C(F)(F)C1CCCC(NCc2ccc3c(c2)OCO3)C1 REAL300018133923
O=C(O)C(F)(F)C1CCC(NCc2ccc3c(c2)OCO3)C1 REAL300018133924
O=C(O)c1ccc(CNCc2ccc3c(c2)OCO3)cc1Cl REAL300018133925
O=C(O)c1ccc(CNCc2ccc3c(c2)OCO3)c(C(F)(F)F)c1 REAL300018133926
O=C(O)c1ccc(CNCc2ccc3c(c2)OCO3)cc1Br REAL300018133927
CCc1oc(CNCc2ccc3c(c2)OCO3)cc1C(=O)O REAL300018133928
O=C(O)CCCC1CCCC(NCc2ccc3c(c2)OCO3)C1 REAL300018133929
CC(CCCC(C)(C)C(=O)O)NCc1ccc2c(c1)OCO2 REAL300018133930
O=C(O)Cn1cc(CNCc2ccc3c(c2)OCO3)c(-c2ccccc2)n1 REAL300018133931
O=C(O)C1(c2ccccc2)CC(NCc2ccc3c(c2)OCO3)C1 REAL300018133932
O=C(O)CCc1ccc(CNCc2ccc3c(c2)OCO3)o1 REAL300018133933
O=C(O)c1cc(CNCc2ccc3c(c2)OCO3)ccc1F REAL300018133934
O=C(O)c1cc2cc(CNCc3ccc4c(c3)OCO4)sc2s1 REAL300018133935
O=C(O)c1cnn2cc(CNCc3ccc4c(c3)OCO4)cnc12 REAL300018133936
CC(Oc1ccc(Cl)cc1CNCc1ccc2c(c1)OCO2)C(=O)O REAL300018133937
O=C(O)c1cc(F)c(CNCc2ccc3c(c2)OCO3)c(F)c1 REAL300018133938
O=C(O)c1ccc2ncc(CNCc3ccc4c(c3)OCO4)n2c1 REAL300018133939
Cc1cc(C(=O)O)ncc1CNCc1ccc2c(c1)OCO2 REAL300018133940
O=C(O)c1cnc2c(CNCc3ccc4c(c3)OCO4)cccn12 REAL300018133941
O=C(O)c1cccc(CNCc2ccc3c(c2)OCO3)c1Br REAL300018133942
O=C(O)[C@H]1C[C@H](n2ccc(CNCc3ccc4c(c3)OCO4)n2)C1 REAL300018133943
O=C(O)[C@H]1C[C@H](n2nccc2CNCc2ccc3c(c2)OCO3)C1 REAL300018133944
O=C(O)c1cc(CNCc2ccc3c(c2)OCO3)cc(C(F)(F)F)c1 REAL300018133945
O=C(O)c1ccc(O)c(CNCc2ccc3c(c2)OCO3)c1 REAL300018133946
O=C(O)c1cc(Br)cc(CNCc2ccc3c(c2)OCO3)c1 REAL300018133947
CCCCC(CC)CNCc1ccc(-c2ccccc2C(=O)O)o1 REAL300018133948
CCCCC(CC)CNCc1ccccc1OCc1ccc(C(=O)O)cc1 REAL300018133949
CCCCC(CC)CNCc1ccc(-c2ccc(C(=O)O)cc2)o1 REAL300018133950
CCCCC(CC)CNCc1ccc(-c2ccc(C(=O)O)cc2)o1 REAL300018133951
CCCCC(CC)CNCc1cn(-c2ccccc2)nc1C(=O)O REAL300018133952
CCCCC(CC)CNCc1cc(C)c(OCC(=O)O)c(C)c1 REAL300018133953
CCCCC(CC)CNCc1c(C)nn(CCC(=O)O)c1C REAL300018133954
CCCCC(CC)CNCc1ccc(OC(C)C(=O)O)cc1 REAL300018133955
CCCCC(CC)CNCc1ccc(OC)c2oc(C(=O)O)cc12 REAL300018133956
CCCCC(CC)CNC1CCCC(C(F)(F)C(=O)O)C1 REAL300018133957
CCCCC(CC)CNCc1ccc(C(=O)O)cc1C(F)(F)F REAL300018133958
CCCCC(CC)CNCc1cc(C)cc(Br)c1OCC(=O)O REAL300018133959
CCCCC(CC)CNCc1ccc(C(=O)O)c(Br)c1 REAL300018133960
CCCCC(CC)CNCc1cn(CC(=O)O)nc1-c1ccccc1 REAL300018133961
CCCCC(CC)CNC1CC(C(=O)O)(c2ccccc2)C1 REAL300018133962
CCCCC(CC)CNCc1cc2cc(C(=O)O)sc2s1 REAL300018133963
CCCCC(CC)CNCc1cnc2c(C(=O)O)cnn2c1 REAL300018133964
CCCCC(CC)CNCc1cc(Cl)ccc1OC(C)C(=O)O REAL300018133965
CCCCC(CC)CNCc1cnc2ccc(C(=O)O)cn12 REAL300018133966
CCCCC(CC)CNCc1cnc2c(Br)cc(C(=O)O)cn12 REAL300018133967
CCCCC(CC)CNCc1cccn2c(C(=O)O)cnc12 REAL300018133968
CCCCC(CC)CNCc1cccc(C(=O)O)c1Br REAL300018133969
CCCCC(CC)CNCc1ccn([C@H]2C[C@H](C(=O)O)C2)n1 REAL300018133970
CCCCC(CC)CNCc1ccnn1[C@H]1C[C@H](C(=O)O)C1 REAL300018133971
CCCCC(CC)CNCc1cc(C(=O)O)cc(C(F)(F)F)c1 REAL300018133972
CCCCC(CC)CNCc1cnc2c(C(=O)O)cc(Br)cn12 REAL300018133973
CCCCC(CC)CNC1CC(C(=O)O)(c2cccc(Br)c2)C1 REAL300018133974
CCCCC(CC)CNCc1cc(Br)cc(C(=O)O)c1 REAL300018133975
O=C(O)c1ccc(COc2ccccc2CN2CCCCCC2)cc1 REAL300018133976
COc1ccc(CN2CCCCCC2)c2cc(C(=O)O)oc12 REAL300018133977
O=C(O)c1ccc(CN2CCCCCC2)c(C(F)(F)F)c1 REAL300018133978
Cc1cc(Br)c(OCC(=O)O)c(CN2CCCCCC2)c1 REAL300018133979
O=C(O)c1ccc(CN2CCCCCC2)cc1Br REAL300018133980
O=C(O)Cn1cc(CN2CCCCCC2)c(-c2ccccc2)n1 REAL300018133981
CC(Oc1ccc(Cl)cc1CN1CCCCCC1)C(=O)O REAL300018133982
O=C(O)c1cc(Br)c2ncc(CN3CCCCCC3)n2c1 REAL300018133983
O=C(O)c1cccc(CN2CCCCCC2)c1Br REAL300018133984
O=C(O)c1cc(CN2CCCCCC2)cc(C(F)(F)F)c1 REAL300018133985
O=C(O)c1cc(Br)cn2c(CN3CCCCCC3)cnc12 REAL300018133986
O=C(O)c1cc(Br)cc(CN2CCCCCC2)c1 REAL300018133987
COCCNCc1ccccc1OCc1ccc(C(=O)O)cc1 REAL300018133988
COCCNCc1cc(C)cc(Br)c1OCC(=O)O REAL300018133989
COCCNCc1cnc2c(Br)cc(C(=O)O)cn12 REAL300018133990
COCCNCc1cnc2c(C(=O)O)cc(Br)cn12 REAL300018133991
COCCNC1CC(C(=O)O)(c2cccc(Br)c2)C1 REAL300018133992
CCC(C)NCc1ccccc1OCc1ccc(C(=O)O)cc1 REAL300018133993
CCC(C)NCc1cc(C)cc(Br)c1OCC(=O)O REAL300018133994
CCC(C)NCc1cnc2c(Br)cc(C(=O)O)cn12 REAL300018133995
CCC(C)NCc1cnc2c(C(=O)O)cc(Br)cn12 REAL300018133996
CCC(C)NC1CC(C(=O)O)(c2cccc(Br)c2)C1 REAL300018133997
CCCCCNCc1ccccc1OCc1ccc(C(=O)O)cc1 REAL300018133998
CCCCCNCc1cc(C)cc(Br)c1OCC(=O)O REAL300018133999
CCCCCNCc1ccc(C(=O)O)c(Br)c1 REAL300018134000
