COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C(C)(C)C REAL300018772001
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(CC4CCC4)c3)C[C@H]12 REAL300018772002
Cc1cc(C)c(C=CCN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)c1 REAL300018772003
COc1c(C)cnc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C REAL300018772004
COCC1(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)CCC1 REAL300018772005
NS(=O)(=O)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772006
Nc1c(Cl)cc(Cl)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772007
CCn1ncnc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772008
CC1(C)OC[C@H](CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)O1 REAL300018772009
CC(C)Oc1ccc(F)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772010
CCOc1cc(F)cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772011
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(OC(F)F)cc3F)C[C@H]12 REAL300018772012
CC(C)(C)Oc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772013
Cc1c(Cl)cccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772014
COc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(F)cc1C REAL300018772015
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cn(CC4CCCO4)nn3)C[C@H]12 REAL300018772016
CCCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nn1 REAL300018772017
CN(C)c1ccc(F)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772018
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(Cl)cncc3Cl)C[C@H]12 REAL300018772019
CC(C)(C)c1csc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772020
COCCc1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772021
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc4c(F)cccc4c3)C[C@H]12 REAL300018772022
Cc1cc(C)c(C=CCN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C REAL300018772023
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CCCC(F)(F)F)C[C@H]12 REAL300018772024
CN1CCC(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)CC1 REAL300018772025
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CCc3cc(Cl)cc(Cl)c3)C[C@H]12 REAL300018772026
Cc1ccc(CCN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C REAL300018772027
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4ncccc34)C[C@H]12 REAL300018772028
CCCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C REAL300018772029
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4nccnc4c3)C[C@H]12 REAL300018772030
CCOc1cccc(F)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772031
Cc1n[nH]cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772032
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cscn3)C[C@H]12 REAL300018772033
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(-c2cccnc2)n1 REAL300018772034
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(-c2ccncc2)n1 REAL300018772035
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(=O)n(C)c1=O REAL300018772036
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(-c4cccnc4)o3)C[C@H]12 REAL300018772037
Cc1nn(CCO)c(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772038
CCc1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cs1 REAL300018772039
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3csc(-c4ccsc4)n3)C[C@H]12 REAL300018772040
CC(C)(C)c1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772041
CC(C)(C)c1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cs1 REAL300018772042
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3OC3CCCC3)C[C@H]12 REAL300018772043
COCCCOc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772044
COc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc1SC REAL300018772045
CCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1OCC REAL300018772046
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Cl)c(F)c3)C[C@H]12 REAL300018772047
Cc1cc(C)cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772048
CC(C)Oc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772049
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3O)C[C@H]12 REAL300018772050
CCOc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1O REAL300018772051
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC=Cc3ccccc3[N+](=O)[O-])C[C@H]12 REAL300018772052
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(OC(F)F)c3)C[C@H]12 REAL300018772053
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3csc([N+](=O)[O-])c3)C[C@H]12 REAL300018772054
CCOc1ccc([N+](=O)[O-])cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772055
CCOCc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc1OC REAL300018772056
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cccc1[N+](=O)[O-] REAL300018772057
Cc1ccc([N+](=O)[O-])c(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772058
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(O)c1 REAL300018772059
COC(=O)c1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)[nH]c1C REAL300018772060
NS(=O)(=O)c1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772061
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c([N+](=O)[O-])n1 REAL300018772062
COC(=O)c1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cs1 REAL300018772063
COC(=O)c1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)[nH]c1C(C)C REAL300018772064
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4c3CCOC4)C[C@H]12 REAL300018772065
COCc1c(C)cc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C REAL300018772066
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4oc(=O)oc4c3)C[C@H]12 REAL300018772067
Cn1nc2c(c1CN1C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C1)CSCC2 REAL300018772068
COc1cc(C)cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1O REAL300018772069
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(F)cc(F)c3O)C[C@H]12 REAL300018772070
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CCc3ccc(F)c(F)c3)C[C@H]12 REAL300018772071
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Cl)cn3)C[C@H]12 REAL300018772072
Cc1[nH]nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C REAL300018772073
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(F)c1OC REAL300018772074
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3OCC(F)F)C[C@H]12 REAL300018772075
CCc1[nH]c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C(=O)OC REAL300018772076
Cc1coc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772077
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC=Cc3cccc(F)c3)C[C@H]12 REAL300018772078
COC(=O)c1cnc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772079
COC(=O)c1c[nH]c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C1CC1 REAL300018772080
COC(=O)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(F)c1 REAL300018772081
Cc1cc(C#N)cc(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772082
CC(C)(C)c1coc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772083
Cc1cc(F)ccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772084
CCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(O)c1 REAL300018772085
COc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1O REAL300018772086
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)ccc3O)C[C@H]12 REAL300018772087
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)cc(Cl)c3O)C[C@H]12 REAL300018772088
COc1cccc(O)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772089
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc([N+](=O)[O-])c3O)C[C@H]12 REAL300018772090
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4c(cc3O)OCO4)C[C@H]12 REAL300018772091
CC(=Cc1ccccc1)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772092
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC3=Cc4ccccc4OC3)C[C@H]12 REAL300018772093
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3-n3cncn3)C[C@H]12 REAL300018772094
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc(-c4ccccc4)cs3)C[C@H]12 REAL300018772095
CCn1nc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C REAL300018772096
N#CCCCOc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772097
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc4ccnn4c3)C[C@H]12 REAL300018772098
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccnc3Cl)C[C@H]12 REAL300018772099
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(F)c(F)c(F)c3)C[C@H]12 REAL300018772100
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(-c4ccc(F)cc4)c3)C[C@H]12 REAL300018772101
COc1cc2c(c(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)c1)OC(C)C2 REAL300018772102
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(OC(F)(F)F)c3)C[C@H]12 REAL300018772103
C=CCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1Cl REAL300018772104
Cn1c(Cl)nc(Cl)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772105
Cn1ccnc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772106
CC(C#N)Oc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772107
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nccn3CC(F)(F)F)C[C@H]12 REAL300018772108
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(-c4ccccc4)s3)C[C@H]12 REAL300018772109
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C2CCCC2)n1 REAL300018772110
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nccc4c3CCCC4)C[C@H]12 REAL300018772111
Cc1nn(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1Cl REAL300018772112
COC(=O)c1sccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772113
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(CCF)c3)C[C@H]12 REAL300018772114
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc4n3CCOC4)C[C@H]12 REAL300018772115
Cn1ccc(-c2nc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cs2)n1 REAL300018772116
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)c1 REAL300018772117
Cc1c(Cl)ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1Cl REAL300018772118
CC1Cc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)ccc2O1 REAL300018772119
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4[nH]c(=O)oc34)C[C@H]12 REAL300018772120
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4c3OCC4)C[C@H]12 REAL300018772121
CSCc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772122
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(CC4CCC4)c3)C[C@H]12 REAL300018772123
Cn1nc2c(c1CN1C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C1)COCC2 REAL300018772124
Cn1nc2c(c1CN1C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C1)CCC2 REAL300018772125
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccnn3C3CCC3)C[C@H]12 REAL300018772126
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(C4CCC4)c3)C[C@H]12 REAL300018772127
COC(=O)COc1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772128
CCc1nnc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772129
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4c(c3)CCCO4)C[C@H]12 REAL300018772130
CN(C)C(=O)c1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772131
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(C4CC4)n[nH]c3Cl)C[C@H]12 REAL300018772132
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(C(F)F)c(F)c3)C[C@H]12 REAL300018772133
COC(=O)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C REAL300018772134
C=C(CCC#N)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772135
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(C4CC4)[nH]n3)C[C@H]12 REAL300018772136
Cn1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C1CC1 REAL300018772137
COCn1ncc(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772138
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc1 REAL300018772139
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccnn3)C[C@H]12 REAL300018772140
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3N3CCCCC3)C[C@H]12 REAL300018772141
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3csc(C(F)(F)F)n3)C[C@H]12 REAL300018772142
CCc1onc(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772143
CCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nn1 REAL300018772144
CC(C)Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772145
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c2c(n1)CCCC2 REAL300018772146
CCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772147
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cn4ccnc4s3)C[C@H]12 REAL300018772148
Cc1oc(C(C)(C)C)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772149
Cc1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)sc1C REAL300018772150
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cn(Cc4ccccc4)nn3)C[C@H]12 REAL300018772151
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(O)cc(Cl)c3)C[C@H]12 REAL300018772152
COc1nccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1F REAL300018772153
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772154
COCCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772155
CCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)n1 REAL300018772156
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C2CC2)n1 REAL300018772157
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(CC(F)(F)F)s3)C[C@H]12 REAL300018772158
CC(C)(C)c1nnc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772159
CCc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)no1 REAL300018772160
Cc1nn(C(C)C)c(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772161
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Cl)cc3[N+](=O)[O-])C[C@H]12 REAL300018772162
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(O)c1OC REAL300018772163
COC(=O)c1cc2oc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cc2[nH]1 REAL300018772164
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccn(CCF)n3)C[C@H]12 REAL300018772165
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3csc(-c4cccs4)n3)C[C@H]12 REAL300018772166
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4cc[nH]c34)C[C@H]12 REAL300018772167
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3N3CCOCC3)C[C@H]12 REAL300018772168
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nccs3)C[C@H]12 REAL300018772169
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cncnc3)C[C@H]12 REAL300018772170
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc4ccccc4c3)C[C@H]12 REAL300018772171
Cn1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc2ccccc21 REAL300018772172
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4[nH]ccc34)C[C@H]12 REAL300018772173
Cn1cncc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772174
Cc1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c[nH]1 REAL300018772175
CN(C)c1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772176
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)[nH]n1 REAL300018772177
NC(=O)c1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772178
CN(C)c1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772179
Cn1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c2ccccc21 REAL300018772180
Cn1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772181
CCc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772182
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1F REAL300018772183
COc1nc(Cl)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1C REAL300018772184
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(F)c3F)C[C@H]12 REAL300018772185
CC1(C)Cc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)ccc2O1 REAL300018772186
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc1F REAL300018772187
Cc1ccccc1-c1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772188
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccnc(-c4ccccc4)n3)C[C@H]12 REAL300018772189
Cc1ncccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772190
Cc1cccc(-c2[nH]ncc2CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772191
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1[N+](=O)[O-] REAL300018772192
CC(C)COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772193
Cc1ccc(O)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772194
COCCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772195
CC1(C)CCc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)ccc2O1 REAL300018772196
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(C(F)(F)F)ccc3F)C[C@H]12 REAL300018772197
CCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772198
CC(C)n1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772199
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4ccccc4nc3O)C[C@H]12 REAL300018772200
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Br)co3)C[C@H]12 REAL300018772201
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(O)cccc3Cl)C[C@H]12 REAL300018772202
CC(C)n1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc2ccccc21 REAL300018772203
C#CCCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772204
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3csc(C4CC4)n3)C[C@H]12 REAL300018772205
CS(=O)(=O)c1sccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772206
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(C4CC4)on3)C[C@H]12 REAL300018772207
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(C4CCOCC4)o3)C[C@H]12 REAL300018772208
N#CCc1ccc(O)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772209
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(C4CCC4)on3)C[C@H]12 REAL300018772210
CC1(c2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)no2)CC1 REAL300018772211
CCc1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772212
CN(C)C(=O)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772213
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)c1C REAL300018772214
CCNC(=O)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772215
CC(C)(C)c1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772216
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc4n3CCCCC4)C[C@H]12 REAL300018772217
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccnc(Cl)c3)C[C@H]12 REAL300018772218
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cnn1C(C)C REAL300018772219
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3conc3C3CC3)C[C@H]12 REAL300018772220
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(-c4ccccc4)no3)C[C@H]12 REAL300018772221
COc1ccc2sc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cc2c1 REAL300018772222
CCN1CCc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)ccc21 REAL300018772223
COC(=O)c1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n(C)n1 REAL300018772224
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4ccsc34)C[C@H]12 REAL300018772225
COc1ccc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772226
Cc1cc(F)cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772227
CCN(C)C(=O)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772228
CSc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1Cl REAL300018772229
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc1C1CC1 REAL300018772230
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C1CC1 REAL300018772231
CNC(=O)c1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772232
CCNC(=O)c1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772233
CCOc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccn1 REAL300018772234
Cn1cnc2cccc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)c21 REAL300018772235
COC(=O)CCc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772236
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ncccc3F)C[C@H]12 REAL300018772237
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Cl)cc3O)C[C@H]12 REAL300018772238
Cc1cc(-n2ccnc2)ccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772239
CC(C)c1nocc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772240
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c[nH]nc3-c3ccc(Cl)o3)C[C@H]12 REAL300018772241
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(OC4CC4)cc3)C[C@H]12 REAL300018772242
CNC(=O)c1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772243
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(C4CC4)c(C4CC4)c3)C[C@H]12 REAL300018772244
CN(C)CCc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772245
CCNC(=O)c1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772246
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)oc2ccc(F)cc12 REAL300018772247
CCCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)n1 REAL300018772248
CCn1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772249
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)ccn3)C[C@H]12 REAL300018772250
CC(C)(C)c1c[nH]c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772251
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(CC4CC4)s3)C[C@H]12 REAL300018772252
Cn1cc(Cl)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772253
CSc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772254
COC(=O)c1cnc(C(C)N2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772255
C[C@H]1CC(N2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c2ccsc2S1 REAL300018772256
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4c(c3)OCC4)C[C@H]12 REAL300018772257
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc4c([nH]3)CCCC4)C[C@H]12 REAL300018772258
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cn4cc(Cl)ccc4n3)C[C@H]12 REAL300018772259
C#CCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772260
C=CCc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc(OC)c1O REAL300018772261
CCn1ccnc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772262
CN(C)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1F REAL300018772263
COc1cccc(Cl)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772264
Cc1ccc(F)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772265
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3occc3Br)C[C@H]12 REAL300018772266
CCc1nn(C)c(Cl)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772267
Cc1csc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772268
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(OCC(F)F)cc3)C[C@H]12 REAL300018772269
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC3CCCCCC3)C[C@H]12 REAL300018772270
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC3=CCCOC3)C[C@H]12 REAL300018772271
Cc1nc2ccccn2c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772272
Cc1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1-c1ccccc1 REAL300018772273
Cc1nc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772274
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Br)cn3)C[C@H]12 REAL300018772275
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(CO)o3)C[C@H]12 REAL300018772276
CCN(CC)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1F REAL300018772277
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4cn[nH]c34)C[C@H]12 REAL300018772278
Cn1nnc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)ccc21 REAL300018772279
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)ccc3[N+](=O)[O-])C[C@H]12 REAL300018772280
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nccc4ccccc34)C[C@H]12 REAL300018772281
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc4ccc(Cl)cn34)C[C@H]12 REAL300018772282
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1Cl REAL300018772283
CC(C)CCn1cccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772284
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nn1 REAL300018772285
CC1(C)Cc2cccc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)c2O1 REAL300018772286
Cc1cccn2c(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cnc12 REAL300018772287
CC(C)(CCC#N)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772288
Cc1cc(O)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C REAL300018772289
COCc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772290
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4c(c3)CCC4)C[C@H]12 REAL300018772291
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(-c4ccncc4)c3)C[C@H]12 REAL300018772292
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1C#N REAL300018772293
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4cc(F)ccc4o3)C[C@H]12 REAL300018772294
N#Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772295
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1O REAL300018772296
CC(C)Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nn1 REAL300018772297
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc(C4CC4)cs3)C[C@H]12 REAL300018772298
Cc1c(C(F)(F)F)n[nH]c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772299
Cc1ccoc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772300
COCc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772301
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC3CCCCCCC3)C[C@H]12 REAL300018772302
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc1-n1cncn1 REAL300018772303
CCC(C)(C)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772304
Cc1ncsc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772305
COCCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772306
Cc1cc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)oc2cc1C REAL300018772307
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(-n4ccnc4)nc3)C[C@H]12 REAL300018772308
CN(C)C(=O)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)[nH]1 REAL300018772309
CS(=O)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772310
COC(=O)c1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c[nH]1 REAL300018772311
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(-c4ccsc4)s3)C[C@H]12 REAL300018772312
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3C3CC3)C[C@H]12 REAL300018772313
N#Cc1csc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772314
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(-c4cccnc4)s3)C[C@H]12 REAL300018772315
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(C4CCCCC4)s3)C[C@H]12 REAL300018772316
CCc1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772317
COc1cc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1OC REAL300018772318
Cn1nncc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772319
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(-c4cccs4)s3)C[C@H]12 REAL300018772320
N#Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772321
Cc1cccc2ncc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)n12 REAL300018772322
COCCOc1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772323
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Cl)nc3)C[C@H]12 REAL300018772324
CCc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772325
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(-n4cccn4)c3)C[C@H]12 REAL300018772326
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(C4CCC4)s3)C[C@H]12 REAL300018772327
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cnc1Cl REAL300018772328
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)s1 REAL300018772329
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(F)cc4cccnc34)C[C@H]12 REAL300018772330
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Cl)c4cccnc34)C[C@H]12 REAL300018772331
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(N4CCCC4)nc3)C[C@H]12 REAL300018772332
CC(C)c1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772333
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4ccccc4s3)C[C@H]12 REAL300018772334
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(F)cc3Cl)C[C@H]12 REAL300018772335
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(F)c(F)cc3F)C[C@H]12 REAL300018772336
CCC1(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)COC1 REAL300018772337
NC(=O)c1csc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772338
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cncs3)C[C@H]12 REAL300018772339
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(-c4ccccc4)[nH]n3)C[C@H]12 REAL300018772340
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(C4CC4)s3)C[C@H]12 REAL300018772341
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(C4CCCC4)s3)C[C@H]12 REAL300018772342
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc1 REAL300018772343
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(Cl)c3F)C[C@H]12 REAL300018772344
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(F)c4cccnc34)C[C@H]12 REAL300018772345
CCCn1nc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C REAL300018772346
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(-c4cccnc4)c3)C[C@H]12 REAL300018772347
Cc1ccc(-c2cccc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)c2)cc1 REAL300018772348
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(CC(F)(F)F)c3)C[C@H]12 REAL300018772349
CCOc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772350
CC(C)Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772351
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)cc4cccnc34)C[C@H]12 REAL300018772352
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4c(c3)COC4)C[C@H]12 REAL300018772353
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c[nH]nc3-c3ccccc3F)C[C@H]12 REAL300018772354
COc1ccsc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772355
Cc1ccc(-c2ncc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)s2)o1 REAL300018772356
COCc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772357
CC(=O)Nc1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772358
COc1nc2ccccc2cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772359
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)ccc3Cl)C[C@H]12 REAL300018772360
COc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc1F REAL300018772361
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cncc4ccccc34)C[C@H]12 REAL300018772362
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ncccc3C(F)(F)F)C[C@H]12 REAL300018772363
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC=Cc3ccc(Cl)cc3)C[C@H]12 REAL300018772364
Cc1oc2ccccc2c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772365
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC3CC3c3ccccc3)C[C@H]12 REAL300018772366
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cscc3Cl)C[C@H]12 REAL300018772367
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc4ccsc4c3)C[C@H]12 REAL300018772368
Cc1cc(Cl)cc(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772369
CCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc1 REAL300018772370
Cc1nn2c(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)c(C)nc2s1 REAL300018772371
Cn1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc2cc(Cl)ccc21 REAL300018772372
CC1CCc2nc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)sc2C1 REAL300018772373
CC(C)Cc1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772374
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(Cl)oc4ccccc34)C[C@H]12 REAL300018772375
CC1(C)CCc2nc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)sc2C1 REAL300018772376
CCc1nn(C)c(CC)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772377
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnc(C4CCCO4)s3)C[C@H]12 REAL300018772378
CC1(C)CCC(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)CC1 REAL300018772379
COC(=O)c1occc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772380
COc1ccc(O)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772381
Cc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1O REAL300018772382
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(Cl)c3O)C[C@H]12 REAL300018772383
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)cc(F)c3O)C[C@H]12 REAL300018772384
COc1cc(O)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1OC REAL300018772385
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(C4CC4)nc4sccn34)C[C@H]12 REAL300018772386
Cc1cccc(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772387
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4nccn34)C[C@H]12 REAL300018772388
CCCC1CCC(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)CC1 REAL300018772389
CCCC(C)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772390
CC(CCc1ccccc1)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772391
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C(C)(C)C)n1 REAL300018772392
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(-c2cccs2)n1 REAL300018772393
CC(C)COc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772394
Cn1cnc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)ccc21 REAL300018772395
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccn(-c4ccccc4)n3)C[C@H]12 REAL300018772396
CN(C)c1cccc(Cl)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772397
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(-c2ccccc2)n1 REAL300018772398
CCc1nn(C)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772399
CC(C)(CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1)c1ccccc1 REAL300018772400
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc4c(s3)CCC4)C[C@H]12 REAL300018772401
CCCC(CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1)c1ccccc1 REAL300018772402
COc1ccc(C(C)CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772403
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc4c(s3)CCCC4)C[C@H]12 REAL300018772404
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccn(C(F)F)n3)C[C@H]12 REAL300018772405
CC(CCc1cccc(F)c1)N1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772406
CC(Cc1ccsc1)N1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772407
Cc1ccc(F)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772408
COc1c(O)cccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772409
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(F)ccc3O)C[C@H]12 REAL300018772410
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CCc3ccc(F)cc3)C[C@H]12 REAL300018772411
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(F)c3O)C[C@H]12 REAL300018772412
CC(C)C1CC(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)CCO1 REAL300018772413
CCC1CC(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)CCO1 REAL300018772414
COCCC1(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)CCC1 REAL300018772415
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(Cl)ccc4cccnc34)C[C@H]12 REAL300018772416
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(SC(F)F)cc3)C[C@H]12 REAL300018772417
COc1cc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)n1 REAL300018772418
CC(C)Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772419
COC(=O)COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772420
CCOCOc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772421
CC(Cc1ccccc1)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772422
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C2CCCCC2)n1 REAL300018772423
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cn(Cc4cccnc4)nn3)C[C@H]12 REAL300018772424
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc2cccnc12 REAL300018772425
CC(C)(C)C1CCC(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)CC1 REAL300018772426
CC(C)c1cnc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772427
COC(=O)c1coc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772428
COc1ccc(CC(C)CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1F REAL300018772429
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC=Cc3ccc(F)cc3F)C[C@H]12 REAL300018772430
CC(CC1CCCCC1)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772431
CC(C)(C)OC(=O)N1CC(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)C1 REAL300018772432
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc([N+](=O)[O-])c(Cl)c3)C[C@H]12 REAL300018772433
CC(C)(CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1)NC(=O)OC(C)(C)C REAL300018772434
COc1cc(Cl)cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1O REAL300018772435
COc1cc2c(cc1CN1C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C1)OCO2 REAL300018772436
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn4ncccc34)C[C@H]12 REAL300018772437
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC3CC4CCC3C4)C[C@H]12 REAL300018772438
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccn4nccc34)C[C@H]12 REAL300018772439
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3sccc3Br)C[C@H]12 REAL300018772440
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772441
CC(C)c1ccc(CCN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772442
CCCCOc1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772443
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cncc(Br)c3)C[C@H]12 REAL300018772444
CCn1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c2ccccc21 REAL300018772445
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ncc(Cl)s3)C[C@H]12 REAL300018772446
CCOC(=O)c1nn(C)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772447
CC(C)(C)CCN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772448
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CCSCc3ccccc3)C[C@H]12 REAL300018772449
CN1C(=O)CCc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)ccc21 REAL300018772450
Cc1ccncc1CCCN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772451
COC(=O)C(C)(C)CCN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772452
C#CCOc1cccc(Cl)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772453
CC1(c2ccccc2)CCC(N2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)C1 REAL300018772454
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4c(F)cccc4[nH]3)C[C@H]12 REAL300018772455
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c[nH]nc3-c3ccsc3)C[C@H]12 REAL300018772456
Cn1ncc(Cl)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772457
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC3CCc4ccccc43)C[C@H]12 REAL300018772458
CC(C)(C)OC(=O)NCCCN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772459
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CCC3CCOC3)C[C@H]12 REAL300018772460
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)sn1 REAL300018772461
COC(=O)Cc1coc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772462
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc4c([nH]3)COCC4)C[C@H]12 REAL300018772463
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3noc4c3COCC4)C[C@H]12 REAL300018772464
Cn1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1Br REAL300018772465
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC=Cc3ccccc3)C[C@H]12 REAL300018772466
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnnn3C3CC3)C[C@H]12 REAL300018772467
COCc1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772468
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4c(c3)COCC4)C[C@H]12 REAL300018772469
Cc1nc(N2CCCC2)sc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772470
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(CCO)c3)C[C@H]12 REAL300018772471
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)sc2cc(F)ccc12 REAL300018772472
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(-c4ccncc4)n[nH]3)C[C@H]12 REAL300018772473
COc1ccc(F)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1OC REAL300018772474
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(CC=Cc3ccncc3)C[C@H]12 REAL300018772475
Cn1ccc(-c2n[nH]cc2CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772476
C=Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772477
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(OCC4CCC4)c3)C[C@H]12 REAL300018772478
CC(F)(F)c1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772479
COc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc1OCCO REAL300018772480
CCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C2CC2)n1 REAL300018772481
CCc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc1 REAL300018772482
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1OCCO REAL300018772483
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(-c2ccnn2C)n1 REAL300018772484
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nn1 REAL300018772485
CC(C)(C)c1nocc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772486
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4ccncc4c3)C[C@H]12 REAL300018772487
Cc1cc2cccc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)c2o1 REAL300018772488
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(F)c3C(F)(F)F)C[C@H]12 REAL300018772489
COc1csc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1OC REAL300018772490
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3conc3C3CCC3)C[C@H]12 REAL300018772491
CS(=O)(=O)c1ccsc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772492
CN(C)c1nc(Cl)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772493
Cn1c(=O)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc2ccccc21 REAL300018772494
Cc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772495
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(-c4ccsc4)cc3)C[C@H]12 REAL300018772496
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc4ccccc4s3)C[C@H]12 REAL300018772497
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3[nH]ncc3Br)C[C@H]12 REAL300018772498
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4nsnc4c3)C[C@H]12 REAL300018772499
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4nonc4c3)C[C@H]12 REAL300018772500
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4nsnc34)C[C@H]12 REAL300018772501
CCn1cnc(Cl)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772502
N#Cc1cnn2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cnc12 REAL300018772503
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cn(-c4ccccc4)nn3)C[C@H]12 REAL300018772504
CCOc1ccc(Cl)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772505
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c[nH]nc3-c3cccc(F)c3)C[C@H]12 REAL300018772506
Cc1oc(-c2cccs2)nc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772507
Cn1nc(-c2ccccc2)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772508
CC(C)(C)c1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n[nH]1 REAL300018772509
CCN1CCCc2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)ccc21 REAL300018772510
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(-c4ccsc4)nc3)C[C@H]12 REAL300018772511
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4ccccc4cn3)C[C@H]12 REAL300018772512
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc(Cl)n1 REAL300018772513
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc(C)n1 REAL300018772514
COc1cc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772515
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc[nH]c3=O)C[C@H]12 REAL300018772516
CCc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cnn1CC REAL300018772517
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4ccc(F)cc4[nH]c3=O)C[C@H]12 REAL300018772518
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C(F)(F)F)n1 REAL300018772519
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3noc4c3CCCC4)C[C@H]12 REAL300018772520
Cc1cn(C)nc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772521
Cc1coc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772522
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4ccncc4s3)C[C@H]12 REAL300018772523
COc1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc1C REAL300018772524
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4ncccc4o3)C[C@H]12 REAL300018772525
CCC(C)n1nccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772526
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc(CO)cs3)C[C@H]12 REAL300018772527
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4cc(Cl)ccc34)C[C@H]12 REAL300018772528
CCCn1cncc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772529
CCc1c[nH]c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772530
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cncc(-c4cccnc4)c3)C[C@H]12 REAL300018772531
CC(C)(C)c1cncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772532
COc1nc(Cl)ccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772533
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccnc1F REAL300018772534
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4c(c3)CCOC4)C[C@H]12 REAL300018772535
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(C(F)F)c3F)C[C@H]12 REAL300018772536
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)n1 REAL300018772537
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc4c(s3)CCCCC4)C[C@H]12 REAL300018772538
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc4c(s3)COCC4)C[C@H]12 REAL300018772539
CC(C)Cc1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772540
CSc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772541
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(C4CCCCC4)c3)C[C@H]12 REAL300018772542
CCCn1nc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1Cl REAL300018772543
Cn1cc(-c2n[nH]cc2CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772544
CC(C)n1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772545
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccn(CC(F)(F)F)n3)C[C@H]12 REAL300018772546
CC(F)(F)c1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772547
Cc1cc(O)ncc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772548
Cc1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)oc1C REAL300018772549
CS(=O)(=O)c1coc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772550
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cn(CC4CC4)nn3)C[C@H]12 REAL300018772551
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccn3C(F)F)C[C@H]12 REAL300018772552
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4c(o3)CCCC4)C[C@H]12 REAL300018772553
Cn1cc(Br)nc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772554
C=CCc1ccccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772555
COc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cccc1C(C)(C)C REAL300018772556
COc1nn(C)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772557
CC(C)(C)n1nccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772558
CN(CCO)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772559
Cn1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc2c1CCCC2 REAL300018772560
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4c3COCC4)C[C@H]12 REAL300018772561
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3C3CCC3)C[C@H]12 REAL300018772562
CC(C)(C#N)c1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)s1 REAL300018772563
CCn1nc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772564
COc1sccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772565
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(C4CCC4)[nH]n3)C[C@H]12 REAL300018772566
C=CCCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nn1 REAL300018772567
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(CC4CCC4)cc3)C[C@H]12 REAL300018772568
COc1nsc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1Cl REAL300018772569
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cn(C4CC4)cn3)C[C@H]12 REAL300018772570
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C2CCOCC2)n1 REAL300018772571
CC(C)c1cnn(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772572
Cn1nnc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C(F)F REAL300018772573
Cn1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1S(C)(=O)=O REAL300018772574
Cc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1OC(F)F REAL300018772575
CC1Oc2ccc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cc2C1C REAL300018772576
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3-n3cccn3)C[C@H]12 REAL300018772577
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccnn3C3CC3(F)F)C[C@H]12 REAL300018772578
COCc1nocc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772579
COCc1cnc(OC)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772580
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(C(F)F)cn3)C[C@H]12 REAL300018772581
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(C(F)(F)F)cc3F)C[C@H]12 REAL300018772582
CC(C)Oc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1F REAL300018772583
CCn1cc(Cl)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772584
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(F)c(Cl)c3F)C[C@H]12 REAL300018772585
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(C(F)F)c3)C[C@H]12 REAL300018772586
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4ccccc4c3F)C[C@H]12 REAL300018772587
CS(=O)(=O)c1csc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772588
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3csc(Cl)c3)C[C@H]12 REAL300018772589
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cnn1C1CCC1 REAL300018772590
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n(C2CCCC2)n1 REAL300018772591
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccnn3CC(F)F)C[C@H]12 REAL300018772592
COc1ccc(C)nc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772593
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)cc(Cl)n3)C[C@H]12 REAL300018772594
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nccc4cc(Cl)ccc34)C[C@H]12 REAL300018772595
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4cnccc4[nH]3)C[C@H]12 REAL300018772596
CN(C)c1ccc([N+](=O)[O-])cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772597
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(F)ccnc3Cl)C[C@H]12 REAL300018772598
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(C(F)F)n3)C[C@H]12 REAL300018772599
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(-c4cccc(F)c4)c3)C[C@H]12 REAL300018772600
CN(C)c1cncc(F)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772601
CC(C)N(C)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(O)c1 REAL300018772602
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(O)ccc4c3OCO4)C[C@H]12 REAL300018772603
Cc1nn(-c2ccccc2)nc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772604
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccn(C4CCC4)n3)C[C@H]12 REAL300018772605
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccn(CC(F)F)n3)C[C@H]12 REAL300018772606
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccn(C4CC4(F)F)n3)C[C@H]12 REAL300018772607
Cc1nn(C2CCCCC2)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772608
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cnn(C4CCOCC4)c3)C[C@H]12 REAL300018772609
Cc1nn(C2CCOCC2)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772610
Cc1cn(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772611
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3noc4c3CCC4)C[C@H]12 REAL300018772612
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3nc4cccc(F)c4s3)C[C@H]12 REAL300018772613
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccn(C4CCCC4)n3)C[C@H]12 REAL300018772614
NS(=O)(=O)c1csc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772615
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(F)c4ccoc34)C[C@H]12 REAL300018772616
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(Cl)cc4ccoc34)C[C@H]12 REAL300018772617
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ncc(Cl)cc3Cl)C[C@H]12 REAL300018772618
Cc1nn(C2CCCC2)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772619
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3C(F)F)C[C@H]12 REAL300018772620
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4[nH]ncc4c3)C[C@H]12 REAL300018772621
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Cl)c(F)c3F)C[C@H]12 REAL300018772622
Cc1c(F)cccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772623
Cn1cc(-c2cccc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)c2)cn1 REAL300018772624
COc1c(C#N)cccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772625
COc1nc2ccc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cc2s1 REAL300018772626
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccnc(Br)c3)C[C@H]12 REAL300018772627
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(F)cc(Cl)c3Cl)C[C@H]12 REAL300018772628
Cc1nc(Cl)ccc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772629
CC(C)(C)COc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772630
COc1cc(Cl)cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772631
COc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc(F)c1F REAL300018772632
COc1cc(C)ncc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772633
COc1ccc2sc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)nc2c1 REAL300018772634
CC(C)n1cnc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772635
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nnn1C REAL300018772636
Cn1nccc1-c1n[nH]cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772637
Cc1onc(C2CC2)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772638
COC(=O)c1c(C)[nH]c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C REAL300018772639
CC(C)Oc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772640
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(C(F)(F)F)cc3O)C[C@H]12 REAL300018772641
Cc1oc(-c2ccccc2)nc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772642
Cn1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1-c1ccco1 REAL300018772643
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(Cl)ccc4c3OCO4)C[C@H]12 REAL300018772644
N#Cc1cc(F)cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1 REAL300018772645
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(C4CCCCC4)cc3)C[C@H]12 REAL300018772646
Cc1nc(C)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)nc1C REAL300018772647
NC(=O)c1cnc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772648
Cc1nn(C2CCC2)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772649
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cnn1CC(F)F REAL300018772650
COc1ccccc1C=CCN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772651
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(-c4ccccn4)nc3)C[C@H]12 REAL300018772652
CCCn1nc(C)c(Cl)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772653
COc1cccc2[nH]c(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cc12 REAL300018772654
Cc1ccc(OC(F)F)c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772655
Cn1nc(-c2ccco2)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772656
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(Cc4ccccc4)cc3)C[C@H]12 REAL300018772657
COc1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)n1 REAL300018772658
CCN(C)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)c1 REAL300018772659
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc(-c4ccccc4)ccn3)C[C@H]12 REAL300018772660
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3scc(Cl)c3Cl)C[C@H]12 REAL300018772661
COc1cc(C)cc(OC)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772662
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(CF)cc3)C[C@H]12 REAL300018772663
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4sccc4c3)C[C@H]12 REAL300018772664
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(-c4ccncc4)cc3)C[C@H]12 REAL300018772665
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccccc3CO)C[C@H]12 REAL300018772666
CC(C)(C)c1oncc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772667
Cc1cncc(C)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772668
COc1cc(C)c2cc(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)[nH]c2c1 REAL300018772669
Cc1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C(F)(F)F REAL300018772670
C=CCn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cn1 REAL300018772671
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc4cn[nH]c4c3)C[C@H]12 REAL300018772672
CCC(C)c1ccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cc1 REAL300018772673
Cc1oncc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772674
CC(F)(F)c1cccc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n1 REAL300018772675
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4sccc4[nH]3)C[C@H]12 REAL300018772676
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc4c3CCCC4)C[C@H]12 REAL300018772677
CC(=Cc1cc(F)cc(F)c1)CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772678
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cccc(C(F)(F)F)c3F)C[C@H]12 REAL300018772679
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(-n4ccnn4)cc3)C[C@H]12 REAL300018772680
Cc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc2ccccc12 REAL300018772681
CC(C)c1nn(C(C)(C)C)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772682
COc1c(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)ccc2[nH]ccc12 REAL300018772683
Cc1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C)s1 REAL300018772684
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3ccc(N4CCC(O)C4)cc3)C[C@H]12 REAL300018772685
COc1ccc(OC)c(OC)c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772686
CCCn1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c1C REAL300018772687
Cc1ccc2cccnc2c1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772688
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3c(O)cccc3F)C[C@H]12 REAL300018772689
Cc1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)cnc1-n1cccn1 REAL300018772690
COC(=O)c1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)n(C)c1 REAL300018772691
O=C(O)C[C@@H]1CS(=O)(=O)[C@@H]2CN(Cc3cc4sc(Cl)cc4[nH]3)C[C@H]12 REAL300018772692
COc1ccn2c(CN3C[C@@H]4[C@H](CC(=O)O)CS(=O)(=O)[C@@H]4C3)cnc2c1 REAL300018772693
CCCn1nc(C)cc1CN1C[C@@H]2[C@H](CC(=O)O)CS(=O)(=O)[C@@H]2C1 REAL300018772694
Cn1cc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c(C2CCC2)n1 REAL300018772695
CC(C)(C)c1ncc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)o1 REAL300018772696
Cn1nc(CN2C[C@@H]3[C@H](CC(=O)O)CS(=O)(=O)[C@@H]3C2)c2c1CCOC2 REAL300018772697
O=C(O)C1(C2CCN(Cc3cccnc3)CC2)CC(F)(F)C1 REAL300018772698
CC(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)c1ccccc1 REAL300018772699
O=C(O)C1(C2CCN(Cc3ccc4c(c3)OCCO4)CC2)CC(F)(F)C1 REAL300018772700
O=C(O)C1(C2CCN(Cc3cccc(Br)c3)CC2)CC(F)(F)C1 REAL300018772701
COc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1OC REAL300018772702
O=C(O)C1(C2CCN(CC3CC=CCC3)CC2)CC(F)(F)C1 REAL300018772703
O=C(O)C1(C2CCN(Cc3ccccc3C(F)(F)F)CC2)CC(F)(F)C1 REAL300018772704
Cc1ccccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772705
CCc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772706
COC(=O)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772707
CCC(CC)CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772708
O=C(O)C1(C2CCN(Cc3ccc(-c4ccc(F)cc4)o3)CC2)CC(F)(F)C1 REAL300018772709
O=C(O)C1(C2CCN(CC3CCCCC3)CC2)CC(F)(F)C1 REAL300018772710
O=C(O)C1(C2CCN(Cc3ccc(Br)o3)CC2)CC(F)(F)C1 REAL300018772711
Cc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1C REAL300018772712
O=C(O)C1(C2CCN(Cc3cc(Br)cs3)CC2)CC(F)(F)C1 REAL300018772713
CC(C)=CCCC(C)CCN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772714
Cn1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1 REAL300018772715
COC(=O)c1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)oc1C REAL300018772716
Cc1nn(C)c(Cl)c1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772717
O=C(O)C1(C2CCN(CC3CCC=CO3)CC2)CC(F)(F)C1 REAL300018772718
CC(CCN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)c1ccccc1 REAL300018772719
O=C(O)C1(C2CCN(Cc3ccc(F)c(Cl)c3)CC2)CC(F)(F)C1 REAL300018772720
O=C(O)C1(C2CCN(Cc3ccc(F)c(C(F)(F)F)c3)CC2)CC(F)(F)C1 REAL300018772721
CCOc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772722
O=C(O)C1(C2CCN(Cc3ccc(F)cc3C(F)(F)F)CC2)CC(F)(F)C1 REAL300018772723
O=C(O)C1(C2CCN(Cc3cc(F)cc(C(F)(F)F)c3)CC2)CC(F)(F)C1 REAL300018772724
COc1ccc(F)c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772725
O=C(O)C1(C2CCN(Cc3cc(F)cc(Cl)c3)CC2)CC(F)(F)C1 REAL300018772726
O=C(O)C1(C2CCN(Cc3ccc(Cl)cc3F)CC2)CC(F)(F)C1 REAL300018772727
O=C(O)C1(C2CCN(Cc3cccc4c3OCO4)CC2)CC(F)(F)C1 REAL300018772728
O=C(O)C1(C2CCN(Cc3cc(Cl)ccc3F)CC2)CC(F)(F)C1 REAL300018772729
COc1ccc(F)cc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772730
O=C(O)C1(C2CCN(Cc3cc(F)cc(F)c3)CC2)CC(F)(F)C1 REAL300018772731
COc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1 REAL300018772732
O=C(O)C1(C2CCN(Cc3ccc4occc4c3)CC2)CC(F)(F)C1 REAL300018772733
Cc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n(C)n1 REAL300018772734
COC(=O)c1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1C REAL300018772735
Cc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1Cl REAL300018772736
O=C(O)C1(C2CCN(Cc3csnn3)CC2)CC(F)(F)C1 REAL300018772737
COc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)ccc1C REAL300018772738
O=C(O)C1(C2CCN(Cc3cccc(-c4ccccn4)c3)CC2)CC(F)(F)C1 REAL300018772739
Cc1nn(C(C)(C)C)c(C)c1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772740
N#Cc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c(F)c1 REAL300018772741
COC(=O)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)o1 REAL300018772742
Cc1nn(C)cc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772743
CCC(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)c1ccccc1 REAL300018772744
COc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1F REAL300018772745
CN(C)c1ncc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1C REAL300018772746
CC1(C)CCCC(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)C1 REAL300018772747
O=C(O)C1(C2CCN(CCCc3c(F)cccc3Cl)CC2)CC(F)(F)C1 REAL300018772748
CC1=CCCC(C)C1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772749
Cc1cc(Cl)ccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772750
O=C(O)C1(C2CCN(CCC3CCCCC3)CC2)CC(F)(F)C1 REAL300018772751
O=C(O)C1(C2CCN(Cc3cocn3)CC2)CC(F)(F)C1 REAL300018772752
Cn1ncc(Br)c1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772753
CCn1nccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772754
C#Cc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772755
COc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1 REAL300018772756
CCn1cncc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772757
O=C(O)C1(C2CCN(Cc3ccncc3F)CC2)CC(F)(F)C1 REAL300018772758
Cc1ccc2cc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)ccc2n1 REAL300018772759
COc1cc(F)cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772760
CC(C)(C)c1ncc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1 REAL300018772761
Cc1occc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772762
Cn1c(=O)oc2cc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)ccc21 REAL300018772763
O=C(O)C1(C2CCN(CCc3cccc(Cl)c3)CC2)CC(F)(F)C1 REAL300018772764
COc1ccc2oc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)cc2c1 REAL300018772765
Cc1ccc(C(C)CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772766
N#Cc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1 REAL300018772767
Cn1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772768
CC(C)n1nccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772769
O=C(O)C1(C2CCN(Cc3coc4ccccc34)CC2)CC(F)(F)C1 REAL300018772770
COc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c(C)c1OC REAL300018772771
O=C(O)C1(C2CCN(Cc3ccc(Oc4ccccc4)o3)CC2)CC(F)(F)C1 REAL300018772772
Cc1ccc2nc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)cn2c1 REAL300018772773
Cc1c[nH]c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1 REAL300018772774
COc1cc(C)ccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772775
COCc1csc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772776
COCc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)no1 REAL300018772777
O=C1COc2ccc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)cc2N1 REAL300018772778
CC(C)n1ccnc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772779
Cc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)nn1 REAL300018772780
O=C(O)C1(C2CCN(Cc3ccnc(Cl)c3Cl)CC2)CC(F)(F)C1 REAL300018772781
O=C(O)C1(C2CCN(Cc3cnc4cnccn34)CC2)CC(F)(F)C1 REAL300018772782
O=C(O)C1(C2CCN(CCCc3ccc4c(c3)CCO4)CC2)CC(F)(F)C1 REAL300018772783
O=C(O)C1(C2CCN(Cc3cc4c(cn3)OCCO4)CC2)CC(F)(F)C1 REAL300018772784
Cc1ccc2ncc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)n2c1 REAL300018772785
Cn1c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cnc1Cl REAL300018772786
O=C(O)C1(C2CCN(Cc3cc(C(F)(F)F)[nH]n3)CC2)CC(F)(F)C1 REAL300018772787
O=C(O)C1(C2CCN(Cc3cc(Cl)cc4c3OCC4)CC2)CC(F)(F)C1 REAL300018772788
Cc1nocc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772789
Cc1ncoc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772790
O=C(O)C1(C2CCN(Cc3cc(Cl)cs3)CC2)CC(F)(F)C1 REAL300018772791
Cc1cnn(C)c1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772792
Cc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)ccc1Cl REAL300018772793
O=C(O)C1(C2CCN(Cc3nccn3-c3ccccc3)CC2)CC(F)(F)C1 REAL300018772794
C=Cn1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1 REAL300018772795
COc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)sn1 REAL300018772796
CCCc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772797
CC(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)c1cccc(Cl)c1 REAL300018772798
Cn1ncc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1Cl REAL300018772799
Cc1c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cnn1C REAL300018772800
O=C(O)C1(C2CCN(Cc3cnc(C4CC4)nc3)CC2)CC(F)(F)C1 REAL300018772801
O=C(O)C1(C2CCN(Cc3cnc(C4CC4)o3)CC2)CC(F)(F)C1 REAL300018772802
CCOc1cncc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772803
CC(C)(C)n1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)nn1 REAL300018772804
Cn1c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)nc2ccc(Cl)cc21 REAL300018772805
Cn1ncnc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772806
CC(C)c1nnc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)s1 REAL300018772807
COc1cncc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1C REAL300018772808
CC(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)c1ccc(F)cc1 REAL300018772809
O=C(O)C1(C2CCN(CC3CCS(=O)(=O)CC3)CC2)CC(F)(F)C1 REAL300018772810
O=C(O)C1(C2CCN(Cc3ccc(C(F)(F)F)s3)CC2)CC(F)(F)C1 REAL300018772811
O=C(O)C1(C2CCN(Cc3ccc(OC(F)F)c(F)c3)CC2)CC(F)(F)C1 REAL300018772812
O=C(O)C1(C2CCN(Cc3csc(C(F)(F)F)c3)CC2)CC(F)(F)C1 REAL300018772813
CC1(C)OCc2cc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)ccc2O1 REAL300018772814
O=C(O)C1(C2CCN(CC3Cc4ccccc4C3)CC2)CC(F)(F)C1 REAL300018772815
O=C(O)C1(C2CCN(Cc3ncc(Br)s3)CC2)CC(F)(F)C1 REAL300018772816
O=C(O)C1(C2CCN(Cc3cc(F)ncc3F)CC2)CC(F)(F)C1 REAL300018772817
Cc1cc(C(F)(F)F)ccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772818
Cn1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c(C(F)F)n1 REAL300018772819
O=C(O)C1(C2CCN(Cc3ncc(C(F)(F)F)s3)CC2)CC(F)(F)C1 REAL300018772820
CCOC(=O)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)o1 REAL300018772821
O=C(O)C1(C2CCN(CCCC3CCCCC3)CC2)CC(F)(F)C1 REAL300018772822
Cc1ccc(CCN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772823
Cc1noc2ncc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)cc12 REAL300018772824
CCc1cnc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)s1 REAL300018772825
O=C(O)C1(C2CCN(CC3CCSC3)CC2)CC(F)(F)C1 REAL300018772826
Cc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c(C)o1 REAL300018772827
O=C(O)C1(C2CCN(Cc3cnc(-c4ccco4)s3)CC2)CC(F)(F)C1 REAL300018772828
CC(C)(C)c1ccc(CCN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772829
O=C(O)C1(C2CCN(CC3CCOc4ccccc43)CC2)CC(F)(F)C1 REAL300018772830
CC1CCC(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)CC1 REAL300018772831
CC(C)CC(C)CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772832
CCC1CCCC(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)C1 REAL300018772833
Cc1ccc(CCCN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1 REAL300018772834
O=C(O)C1(C2CCN(CCC3CCCCCC3)CC2)CC(F)(F)C1 REAL300018772835
COCOc1ccc(OC)cc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772836
CC1CCCCC1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772837
O=C(O)C1(C2CCN(Cc3cc4c(Cl)nccc4o3)CC2)CC(F)(F)C1 REAL300018772838
NC(=O)Cn1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)nn1 REAL300018772839
Cc1ccccc1-n1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)nn1 REAL300018772840
CCSc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772841
O=C(O)C1(C2CCN(Cc3cnnn3-c3ccccc3)CC2)CC(F)(F)C1 REAL300018772842
O=C(O)C1(C2CCN(Cc3cc(C4CC4)no3)CC2)CC(F)(F)C1 REAL300018772843
O=C(O)C1(C2CCN(CC3C4CC5CC(C4)CC3C5)CC2)CC(F)(F)C1 REAL300018772844
O=C(O)C1(C2CCN(CC3CC3(Cl)Cl)CC2)CC(F)(F)C1 REAL300018772845
Cn1c(Cl)cnc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772846
CC(C)OC(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)c1ccccc1 REAL300018772847
CC(C)N(C)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1 REAL300018772848
COCCN(C)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1 REAL300018772849
Cn1nc2c(c1CN1CCC(C3(C(=O)O)CC(F)(F)C3)CC1)CCCC2 REAL300018772850
O=C(O)C1(C2CCN(Cc3scnc3C3CC3)CC2)CC(F)(F)C1 REAL300018772851
Cc1c[nH]nc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772852
CN(C)Cc1cnc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)s1 REAL300018772853
O=C(O)C1(C2CCN(Cc3ccsc3C(F)(F)F)CC2)CC(F)(F)C1 REAL300018772854
O=C(O)C1(C2CCN(C[C@@H]3C[C@H]3c3ccccc3)CC2)CC(F)(F)C1 REAL300018772855
CC(C)(C)n1nnc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1 REAL300018772856
O=C(O)C1(C2CCN(CC=Cc3ccc(F)cc3)CC2)CC(F)(F)C1 REAL300018772857
O=C(O)C1(C2CCN(Cc3cccc4c3NCCC4)CC2)CC(F)(F)C1 REAL300018772858
CC(=Cc1cccc([N+](=O)[O-])c1)CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772859
Cn1cc(-c2csc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)n2)cn1 REAL300018772860
O=C(O)C1(C2CCN(Cc3ccncc3[N+](=O)[O-])CC2)CC(F)(F)C1 REAL300018772861
O=C(O)C1(C2CCN(CCC3CCOCC3)CC2)CC(F)(F)C1 REAL300018772862
O=C(O)C1(C2CCN(CC3CCC4(CC3)OCCO4)CC2)CC(F)(F)C1 REAL300018772863
COc1ccc2nc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)sc2c1 REAL300018772864
CCc1cccc(Cl)c1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772865
Cn1c(=O)sc2cc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)ccc21 REAL300018772866
COC(=O)C1C(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)C1(F)F REAL300018772867
O=C(O)C1(C2CCN(Cc3ccsc3Cl)CC2)CC(F)(F)C1 REAL300018772868
CCN(C)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cn1 REAL300018772869
COC1(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)CCCC1 REAL300018772870
COC1(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)CCCCC1 REAL300018772871
O=C(O)C1(C2CCN(Cc3ccc(OCC4CC4)cc3)CC2)CC(F)(F)C1 REAL300018772872
O=C(O)C1(C2CCN(Cc3c(O)ccc(Cl)c3F)CC2)CC(F)(F)C1 REAL300018772873
O=C(O)C1(C2CCN(Cc3n[nH]cc3-c3ccccc3)CC2)CC(F)(F)C1 REAL300018772874
O=C(O)C1(C2CCN(Cc3cc4ccc(F)cc4[nH]3)CC2)CC(F)(F)C1 REAL300018772875
COCC(C)(C)CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772876
O=C(O)C1(C2CCN(Cc3cnc(C4OCCO4)s3)CC2)CC(F)(F)C1 REAL300018772877
O=C(O)C1(C2CCN(Cc3nc4ccc(F)cc4s3)CC2)CC(F)(F)C1 REAL300018772878
O=C(O)C1(C2CCN(Cc3ccc(F)c(Cl)c3Cl)CC2)CC(F)(F)C1 REAL300018772879
O=C(O)C1(C2CCN(Cc3csc(Cl)c3Cl)CC2)CC(F)(F)C1 REAL300018772880
CC(CCC#N)CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772881
CC1(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)CCC1 REAL300018772882
O=C(O)C1(C2CCN(CCc3ccc(F)cc3Cl)CC2)CC(F)(F)C1 REAL300018772883
Cc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)ccc1C#N REAL300018772884
O=C(O)C1(C2CCN(Cc3cnc(C(F)(F)F)s3)CC2)CC(F)(F)C1 REAL300018772885
CC(O)c1ncc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)s1 REAL300018772886
O=C(O)C1(C2CCN(Cc3ncc(C4OCCO4)s3)CC2)CC(F)(F)C1 REAL300018772887
Cn1nc(Br)cc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772888
CCOc1c(Cl)cccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772889
Cc1nc(F)ccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772890
O=C(O)C1(C2CCN(Cc3sccc3Cl)CC2)CC(F)(F)C1 REAL300018772891
O=C(O)C1(C2CCN(Cc3ccc4cnccc4c3)CC2)CC(F)(F)C1 REAL300018772892
CCOc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1F REAL300018772893
O=C(O)C1(C2CCN(Cc3cc4ccccc4[nH]3)CC2)CC(F)(F)C1 REAL300018772894
O=C(O)C1(C2CCN(CC3(C(F)F)CC3)CC2)CC(F)(F)C1 REAL300018772895
O=C(O)C1(C2CCN(Cc3ccnn3-c3ccccc3)CC2)CC(F)(F)C1 REAL300018772896
CC(C)(C)c1cnc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)s1 REAL300018772897
O=C(O)C1(C2CCN(CC3(c4ccccc4)CCOC3)CC2)CC(F)(F)C1 REAL300018772898
CSc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)s1 REAL300018772899
Cn1cc(-c2ccc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)cc2)cn1 REAL300018772900
O=C(O)C1(C2CCN(Cc3c(F)ccc(O)c3F)CC2)CC(F)(F)C1 REAL300018772901
O=C(O)C1(C2CCN(Cc3ccc(C(F)F)cc3)CC2)CC(F)(F)C1 REAL300018772902
O=C(O)C1(C2CCN(CC(c3ccccc3)c3ccccc3)CC2)CC(F)(F)C1 REAL300018772903
CCOc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1OC REAL300018772904
O=C(O)C1(C2CCN(Cc3ccc(-n4cccn4)cc3)CC2)CC(F)(F)C1 REAL300018772905
Cc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c(C)c1 REAL300018772906
Cc1ccc(C)c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772907
O=C(O)C1(C2CCN(Cc3ccc4ncccc4c3)CC2)CC(F)(F)C1 REAL300018772908
CC(C)(C)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772909
COc1cc(OC)c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c(OC)c1 REAL300018772910
CCOc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)ccc1OC REAL300018772911
CCCCCOc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772912
CCCc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772913
Cc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1C REAL300018772914
CC(C)Oc1ccccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772915
C=CCOc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1OC REAL300018772916
CN(CCC#N)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772917
CCCOc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772918
COc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)ccc1OC(C)C REAL300018772919
CCc1cccc(F)c1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772920
CC(C)C(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)c1ccccc1 REAL300018772921
O=C(O)C1(C2CCN(Cc3ccnn3-c3ccc(F)cc3)CC2)CC(F)(F)C1 REAL300018772922
Cc1ccccc1-n1nccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772923
COC(=O)c1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772924
O=C(O)C1(C2CCN(CC3CCC(c4ccccc4)CC3)CC2)CC(F)(F)C1 REAL300018772925
Cc1nn(C(C)C)cc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772926
C[C@H](CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)NC(=O)OC(C)(C)C REAL300018772927
COc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc(OC)c1O REAL300018772928
Cc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc(C)c1O REAL300018772929
COc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)ccc1C#N REAL300018772930
COC(=O)c1[nH]c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1C REAL300018772931
CCc1cc(OC)ccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772932
CSC1(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)CC1 REAL300018772933
CSC1(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)CCC1 REAL300018772934
COC(=O)c1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n(C)c1C REAL300018772935
CCc1oc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1C(=O)OC REAL300018772936
Cn1cc(-c2ccc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)s2)cn1 REAL300018772937
COCCCn1nccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772938
Cc1cnc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1C REAL300018772939
CC(C)C(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)C(C)C REAL300018772940
COc1cccc(OC)c1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772941
Cn1nnc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1 REAL300018772942
O=C(O)C1(C2CCN(CC=Cc3ccc(F)c(F)c3)CC2)CC(F)(F)C1 REAL300018772943
O=C(O)C1(C2CCN(Cc3cscc3Br)CC2)CC(F)(F)C1 REAL300018772944
CCOC(=O)c1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)[nH]c1C REAL300018772945
O=C(O)C1(C2CCN(C[C@@H]3C[C@H]3c3ccccc3)CC2)CC(F)(F)C1 REAL300018772946
O=C(O)C1(C2CCN(CCc3ccc(Cl)cc3)CC2)CC(F)(F)C1 REAL300018772947
CC(C)C1CCC(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)CC1 REAL300018772948
CC(C)n1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)nn1 REAL300018772949
CN(C)Cc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)no1 REAL300018772950
CN(C)c1ncccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772951
O=C(O)C1(C2CCN(Cc3cnccn3)CC2)CC(F)(F)C1 REAL300018772952
CCOC(=O)CC(C)(C)CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772953
COCCOCc1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1 REAL300018772954
N#Cc1c(F)cccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772955
O=C(O)C1(C2CCN(Cc3ccc4ccccc4c3)CC2)CC(F)(F)C1 REAL300018772956
COc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc(OC)c1 REAL300018772957
COc1ccc2cc(CN3CCC(C4(C(=O)O)CC(F)(F)C4)CC3)ccc2c1 REAL300018772958
O=C(O)C1(C2CCN(Cc3ccccc3N3CCCC3)CC2)CC(F)(F)C1 REAL300018772959
O=C(O)C1(C2CCN(Cc3c(F)cccc3N3CCCC3)CC2)CC(F)(F)C1 REAL300018772960
O=C(O)C1(C2CCN(Cc3ccc(N4CCCCC4)cc3)CC2)CC(F)(F)C1 REAL300018772961
CCOc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1OC REAL300018772962
CCCOc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)ccc1OC REAL300018772963
C=CCOc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772964
COc1cccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1OC(C)C REAL300018772965
C#CCOc1ccccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772966
COc1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc2c1OCCO2 REAL300018772967
Cc1cc(C)c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)cc1C REAL300018772968
O=C(O)C1(C2CCN(Cc3cc(-c4ccccn4)n[nH]3)CC2)CC(F)(F)C1 REAL300018772969
O=C(O)C1(C2CCN(Cc3ccc4[nH]ccc4c3)CC2)CC(F)(F)C1 REAL300018772970
O=C(O)C1(C2CCN(Cc3ccon3)CC2)CC(F)(F)C1 REAL300018772971
O=C(O)C1(C2CCN(Cc3cc(O)cc(C(F)(F)F)c3)CC2)CC(F)(F)C1 REAL300018772972
O=C(O)C1(C2CCN(Cc3cscc3C(F)(F)F)CC2)CC(F)(F)C1 REAL300018772973
COc1ncc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)s1 REAL300018772974
O=C(O)C1(C2CCN(Cc3ccc(C4CCCC4)cc3)CC2)CC(F)(F)C1 REAL300018772975
Cc1nc(C)c(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)o1 REAL300018772976
CCOC(=O)c1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)on1 REAL300018772977
O=C(O)C1(C2CCN(CCc3ccc([N+](=O)[O-])cc3)CC2)CC(F)(F)C1 REAL300018772978
CC1(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)CCCS1 REAL300018772979
O=C(O)C1(C2CCN(Cc3ccc4c(c3)CCCC4)CC2)CC(F)(F)C1 REAL300018772980
Cc1nnsc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772981
O=C(O)C1(C2CCN(Cc3cnn(CC(F)F)c3)CC2)CC(F)(F)C1 REAL300018772982
COCc1ccccc1C=C(C)CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772983
Cn1nccc1-c1ccccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772984
COC(=O)c1cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)on1 REAL300018772985
O=C(O)C1(C2CCN(Cc3conc3Cc3ccccc3)CC2)CC(F)(F)C1 REAL300018772986
CCc1nocc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772987
Cn1ncc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1 REAL300018772988
CC(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)C1CCCCC1 REAL300018772989
COC(=O)c1ccc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)n1C REAL300018772990
CSC(C)(C)CCN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772991
COC(C)(CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1)C1CC1 REAL300018772992
O=C(O)C1(C2CCN(Cc3ccc4ccc(F)c(F)c4n3)CC2)CC(F)(F)C1 REAL300018772993
O=C(O)C1(C2CCN(Cc3ccc(C4CCC4)cc3)CC2)CC(F)(F)C1 REAL300018772994
O=C(O)C1(C2CCN(Cc3cccc(O)c3Cl)CC2)CC(F)(F)C1 REAL300018772995
Cc1sccc1CN1CCC(C2(C(=O)O)CC(F)(F)C2)CC1 REAL300018772996
Cc1cc(Cl)cc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)c1 REAL300018772997
O=C(O)C1(C2CCN(Cc3cc(Cl)c(F)cc3O)CC2)CC(F)(F)C1 REAL300018772998
CSCc1cnc(CN2CCC(C3(C(=O)O)CC(F)(F)C3)CC2)s1 REAL300018772999
O=C(O)C1(C2CCN(Cc3ccc(F)cc3O)CC2)CC(F)(F)C1 REAL300018773000
