NC(=O)c1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775001
CN(C)c1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775002
Cn1nc(CN2CCC(CC(F)F)(C(=O)O)CC2)c2ccccc21 REAL300018775003
O=C(O)C1(CC(F)F)CCN(Cc2ccc(OC(F)F)c(Cl)c2)CC1 REAL300018775004
CCc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775005
Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1F REAL300018775006
COc1nc(Cl)c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1C REAL300018775007
O=C(O)C1(CC(F)F)CCN(Cc2cccc(F)c2F)CC1 REAL300018775008
COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(Cl)c1OC REAL300018775009
CC1(C)Cc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)ccc2O1 REAL300018775010
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1F REAL300018775011
Cc1ccccc1-c1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775012
O=C(O)C1(CC(F)F)CCN(Cc2ccnc(-c3ccccc3)n2)CC1 REAL300018775013
Cc1cccc(-c2[nH]ncc2CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775014
COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1[N+](=O)[O-] REAL300018775015
CC(C)COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775016
Cc1ccc(O)c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775017
COCCOc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775018
O=C(O)C1(CC(F)F)CCN(Cc2cc3sccc3nc2Cl)CC1 REAL300018775019
CC1(C)CCc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)ccc2O1 REAL300018775020
O=C(O)C1(CC(F)F)CCN(Cc2cc(C(F)(F)F)ccc2F)CC1 REAL300018775021
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1Oc1cccnc1 REAL300018775022
CCn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775023
CC(C)n1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775024
O=C(O)C1(CC(F)F)CCN(Cc2cc3ccccc3nc2O)CC1 REAL300018775025
O=C(O)C1(CC(F)F)CCN(Cc2cc(Br)co2)CC1 REAL300018775026
O=C(O)C1(CC(F)F)CCN(Cc2c(O)cccc2Cl)CC1 REAL300018775027
CC(C)n1c(CN2CCC(CC(F)F)(C(=O)O)CC2)nc2ccccc21 REAL300018775028
C#CCCOc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775029
Cc1ccc(-c2nc(CN3CCC(CC(F)F)(C(=O)O)CC3)cs2)cc1 REAL300018775030
O=C(O)C1(CC(F)F)CCN(Cc2csc(C3CC3)n2)CC1 REAL300018775031
O=C(O)C1(CC(F)F)CCN(Cc2csc(COc3ccccc3)n2)CC1 REAL300018775032
CS(=O)(=O)c1sccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775033
COC(=O)c1cc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)sc2[nH]1 REAL300018775034
O=C(O)C1(CC(F)F)CCN(Cc2cc(C3CC3)on2)CC1 REAL300018775035
O=C(O)C1(CC(F)F)CCN(Cc2ccc(F)c(Br)c2F)CC1 REAL300018775036
O=C(O)C1(CC(F)F)CCN(Cc2cnc(C3CCOCC3)o2)CC1 REAL300018775037
N#CCc1ccc(O)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775038
O=C(O)C1(CC(F)F)CCN(Cc2cc(C3CCC3)on2)CC1 REAL300018775039
CC1(c2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)no2)CC1 REAL300018775040
CCc1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775041
CN(C)C(=O)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775042
Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)c1C REAL300018775043
CCNC(=O)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775044
CC(C)(C)c1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775045
O=C(O)C1(CC(F)F)CCN(Cc2cnc3n2CCCCC3)CC1 REAL300018775046
O=C(O)C1(CC(F)F)CCN(Cc2ccnc(Cl)c2)CC1 REAL300018775047
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)cnn1C(C)C REAL300018775048
O=C(O)C1(CC(F)F)CCN(Cc2conc2C2CC2)CC1 REAL300018775049
O=C(O)C1(CC(F)F)CCN(Cc2cc(-c3ccccc3)no2)CC1 REAL300018775050
COc1ccc2sc(CN3CCC(CC(F)F)(C(=O)O)CC3)cc2c1 REAL300018775051
CCN1CCc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)ccc21 REAL300018775052
CNS(=O)(=O)c1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1F REAL300018775053
COC(=O)c1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)n(C)n1 REAL300018775054
O=C(O)C1(CC(F)F)CCN(Cc2cccc3ccsc23)CC1 REAL300018775055
Cc1nn(-c2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)cc2)cc1Cl REAL300018775056
COc1ccc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775057
Cc1cc(F)cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775058
CCN(CC)C(=O)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775059
CCN(C)C(=O)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775060
CSc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1Cl REAL300018775061
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1C1CC1 REAL300018775062
Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1C1CC1 REAL300018775063
Cc1ccn(-c2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)c(C)c2)n1 REAL300018775064
Cc1cc(-n2cc(Cl)cn2)ccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775065
CNC(=O)c1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775066
CCNC(=O)c1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775067
O=C(O)C1(CC(F)F)CCN(Cc2ccccc2-c2ccccc2Cl)CC1 REAL300018775068
O=C(O)C1(CC(F)F)CCN(Cc2ccccc2Oc2cccc(F)c2)CC1 REAL300018775069
CCOc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccn1 REAL300018775070
CCc1cc(Br)c(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775071
Cn1cnc2cccc(CN3CCC(CC(F)F)(C(=O)O)CC3)c21 REAL300018775072
COC(=O)CCc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)o1 REAL300018775073
COC(=O)c1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)n2c1COCC2 REAL300018775074
O=C(O)C1(CC(F)F)CCN(Cc2ncccc2F)CC1 REAL300018775075
O=C(O)C1(CC(F)F)CCN(Cc2c(Cl)cccc2Br)CC1 REAL300018775076
Cc1cc(Br)cnc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775077
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Cl)cc2O)CC1 REAL300018775078
O=C(c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1)N1CCCCC1 REAL300018775079
Cc1cc(-n2ccnc2)ccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775080
CC(C)c1nocc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775081
O=C(O)C1(CC(F)F)CCN(Cc2c[nH]nc2-c2ccc(Cl)o2)CC1 REAL300018775082
O=C(O)C1(CC(F)F)CCN(Cc2ccc(OC3CC3)cc2)CC1 REAL300018775083
O=C(O)C1(CC(F)F)CCN(Cc2ccc(OC(F)(F)F)cc2F)CC1 REAL300018775084
Cc1cc(-n2ccnc2C)ccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775085
Cc1ncn(-c2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)cc2)c1C REAL300018775086
CNC(=O)c1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775087
O=C(O)C1(CC(F)F)CCN(Cc2ccc(C3CC3)c(C3CC3)c2)CC1 REAL300018775088
CN(C)CCc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775089
CCNC(=O)c1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775090
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)oc2ccc(F)cc12 REAL300018775091
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(-c2cccc(F)c2)n1 REAL300018775092
CCCn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)n1 REAL300018775093
CCn1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775094
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)ccn2)CC1 REAL300018775095
Cc1sc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1Br REAL300018775096
CC(C)(C)c1c[nH]c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775097
O=C(O)C1(CC(F)F)CCN(Cc2ccc(CC3CC3)s2)CC1 REAL300018775098
Cn1cc(Cl)c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775099
CSc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775100
COC(=O)c1cnc(C(C)N2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775101
C[C@H]1CC(N2CCC(CC(F)F)(C(=O)O)CC2)c2ccsc2S1 REAL300018775102
O=C(O)C1(CC(F)F)CCN(Cc2ccc3c(c2)OCC3)CC1 REAL300018775103
O=C(O)C1(CC(F)F)CCN(Cc2nc3c([nH]2)CCCC3)CC1 REAL300018775104
O=C(O)C1(CC(F)F)CCN(Cc2cn3cc(Cl)ccc3n2)CC1 REAL300018775105
C#CCOc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775106
C=CCc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc(OC)c1O REAL300018775107
CCn1ccnc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775108
CN(C)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1F REAL300018775109
COc1ccc(OC(F)F)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775110
COc1cccc(Cl)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775111
Cc1ccc(F)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775112
O=C(O)C1(CC(F)F)CCN(Cc2occc2Br)CC1 REAL300018775113
O=C(O)C1(CC(F)F)CCN(Cc2ccc(-c3c(F)cccc3F)o2)CC1 REAL300018775114
O=C(O)C1(CC(F)F)CCN(Cc2c(Cl)cccc2OC(F)F)CC1 REAL300018775115
CCc1nn(C)c(Cl)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775116
Cc1csc(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775117
O=C(O)C1(CC(F)F)CCN(Cc2ccc(OCC(F)F)cc2)CC1 REAL300018775118
O=C(O)C1(CC(F)F)CCN(CC2CCCCCC2)CC1 REAL300018775119
CC(=O)N(c1nc(CN2CCC(CC(F)F)(C(=O)O)CC2)cs1)C1CC1 REAL300018775120
Cc1nc2ccccn2c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775121
Cc1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)n1-c1ccccc1 REAL300018775122
Cc1nc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775123
Cc1cc(F)ccc1-c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)o1 REAL300018775124
Cc1ccc(-c2ncc(CN3CCC(CC(F)F)(C(=O)O)CC3)s2)cc1 REAL300018775125
COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(OC(F)F)c1 REAL300018775126
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Br)cn2)CC1 REAL300018775127
O=C(O)C1(CC(F)F)CCN(Cc2ccc(CO)o2)CC1 REAL300018775128
CCN(CC)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1F REAL300018775129
O=C(O)C1(CC(F)F)CCN(Cc2cccc3cn[nH]c23)CC1 REAL300018775130
Cn1nnc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)ccc21 REAL300018775131
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)ccc2[N+](=O)[O-])CC1 REAL300018775132
O=C(O)C1(CC(F)F)CCN(Cc2nccc3ccccc23)CC1 REAL300018775133
O=C(O)C1(CC(F)F)CCN(Cc2cnc3ccc(Cl)cn23)CC1 REAL300018775134
COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1Cl REAL300018775135
CC(C)CCn1cccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775136
CC1(C)Cc2cccc(CN3CCC(CC(F)F)(C(=O)O)CC3)c2O1 REAL300018775137
Cc1cccn2c(CN3CCC(CC(F)F)(C(=O)O)CC3)cnc12 REAL300018775138
CC(C)(CCC#N)CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775139
COc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(SC)cc1OC REAL300018775140
Cc1cc(O)c(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1C REAL300018775141
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)ccc2Br)CC1 REAL300018775142
COCc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775143
O=C(O)C1(CC(F)F)CCN(Cc2ccc3c(c2)CCC3)CC1 REAL300018775144
O=C(O)C1(CC(F)F)CCN(Cc2cccc(-c3ccncc3)c2)CC1 REAL300018775145
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Oc3cnccn3)cc2)CC1 REAL300018775146
COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1C#N REAL300018775147
O=C(O)C1(CC(F)F)CCN(Cc2cc3cc(F)ccc3o2)CC1 REAL300018775148
Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1O REAL300018775149
CC(C)Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)nn1 REAL300018775150
O=C(O)C1(CC(F)F)CCN(Cc2nc(C3CC3)cs2)CC1 REAL300018775151
Cc1c(C(F)(F)F)n[nH]c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775152
O=C(O)C1(CC(F)F)CCN(Cc2cc3c(cc2OC(F)F)OCO3)CC1 REAL300018775153
COCc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775154
CCc1ccc(-c2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)o2)cc1 REAL300018775155
O=C(O)C1(CC(F)F)CCN(CC2CCCCCCC2)CC1 REAL300018775156
COc1ccccc1-c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775157
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(OC(F)F)cc1C REAL300018775158
Cc1cc(C)cc(-c2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)cc2)c1 REAL300018775159
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1-n1cncn1 REAL300018775160
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Br)cc2Cl)CC1 REAL300018775161
Cc1nn(-c2ccc(Cl)cc2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775162
Cc1ncsc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775163
COCCn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775164
Cc1cc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)oc2cc1C REAL300018775165
O=C(O)C1(CC(F)F)CCN(Cc2ccc(-n3ccnc3)nc2)CC1 REAL300018775166
CN(C)C(=O)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)[nH]1 REAL300018775167
CS(=O)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775168
COC(=O)c1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c[nH]1 REAL300018775169
O=C(O)C1(CC(F)F)CCN(Cc2cnc(-c3ccsc3)s2)CC1 REAL300018775170
O=C(O)C1(CC(F)F)CCN(Cc2ccccc2C2CC2)CC1 REAL300018775171
N#Cc1csc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775172
O=C(O)C1(CC(F)F)CCN(Cc2cnc(-c3cccnc3)s2)CC1 REAL300018775173
O=C(O)C1(CC(F)F)CCN(Cc2cnc(C3CCCCC3)s2)CC1 REAL300018775174
CCc1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775175
COc1cc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1OC REAL300018775176
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1Br REAL300018775177
O=C(O)C1(CC(F)F)CCN(Cc2cnc(-c3cccs3)s2)CC1 REAL300018775178
N#Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775179
Cc1cccc2ncc(CN3CCC(CC(F)F)(C(=O)O)CC3)n12 REAL300018775180
COCCOc1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775181
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Cl)nc2)CC1 REAL300018775182
CCc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)o1 REAL300018775183
O=C(O)C1(CC(F)F)CCN(Cc2cccc(-n3cccn3)c2)CC1 REAL300018775184
O=C(O)C1(CC(F)F)CCN(Cc2cnc(C3CCC3)s2)CC1 REAL300018775185
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cnc1Cl REAL300018775186
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)s1 REAL300018775187
O=C(O)C1(CC(F)F)CCN(Cc2cc(F)cc3cccnc23)CC1 REAL300018775188
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Cl)c3cccnc23)CC1 REAL300018775189
COc1ccc(-c2ccccc2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775190
O=C(O)C1(CC(F)F)CCN(Cc2ccc(N3CCCC3)nc2)CC1 REAL300018775191
CC(C)c1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775192
O=C(O)C1(CC(F)F)CCN(Cc2cc3ccccc3s2)CC1 REAL300018775193
O=C(O)C1(CC(F)F)CCN(Cc2ccc(F)cc2Cl)CC1 REAL300018775194
O=C(O)C1(CC(F)F)CCN(Cc2ccc(F)cc2Br)CC1 REAL300018775195
O=C(O)C1(CC(F)F)CCN(Cc2cc(F)c(F)cc2F)CC1 REAL300018775196
O=C(O)C1(CC(F)F)CCN(Cc2cc(Br)ccc2Cl)CC1 REAL300018775197
CC(C)(C)OC(=O)Nc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775198
NC(=O)c1csc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775199
O=C(O)C1(CC(F)F)CCN(Cc2cc(-c3ccccc3)[nH]n2)CC1 REAL300018775200
O=C(O)C1(CC(F)F)CCN(Cc2cnc(C3CC3)s2)CC1 REAL300018775201
O=C(O)C1(CC(F)F)CCN(Cc2cnc(C3CCCC3)s2)CC1 REAL300018775202
Cc1cc(Br)ccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775203
O=C(O)C1(CC(F)F)CCN(Cc2cccc(Cl)c2F)CC1 REAL300018775204
O=C(O)C1(CC(F)F)CCN(Cc2ccc(F)c3cccnc23)CC1 REAL300018775205
CC(C)(C)OC(=O)N1CCC(CN2CCC(CC(F)F)(C(=O)O)CC2)CC1 REAL300018775206
CN1CCN(c2ncc(CN3CCC(CC(F)F)(C(=O)O)CC3)cn2)CC1 REAL300018775207
CCCn1nc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1C REAL300018775208
O=C(O)C1(CC(F)F)CCN(Cc2c[nH]nc2-c2c(F)cccc2F)CC1 REAL300018775209
O=C(O)C1(CC(F)F)CCN(Cc2cccc(-c3cccnc3)c2)CC1 REAL300018775210
Cc1ccc(-c2cccc(CN3CCC(CC(F)F)(C(=O)O)CC3)c2)cc1 REAL300018775211
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Cl)cc2Br)CC1 REAL300018775212
O=C(O)C1(CC(F)F)CCN(Cc2cnn(CC(F)(F)F)c2)CC1 REAL300018775213
CCOc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775214
CC(C)Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775215
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)cc3cccnc23)CC1 REAL300018775216
O=C(O)C1(CC(F)F)CCN(Cc2ccc3c(c2)COC3)CC1 REAL300018775217
O=C(O)C1(CC(F)F)CCN(Cc2c[nH]nc2-c2ccccc2F)CC1 REAL300018775218
O=C(O)C1(CC(F)F)CCN(Cc2c[nH]nc2-c2cccc(Cl)c2)CC1 REAL300018775219
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Br)c(F)c2)CC1 REAL300018775220
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)sc1Br REAL300018775221
COc1ccsc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775222
Cc1ccc(-c2ncc(CN3CCC(CC(F)F)(C(=O)O)CC3)s2)o1 REAL300018775223
COCc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)o1 REAL300018775224
CC(=O)Nc1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775225
COc1nc2ccccc2cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775226
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)ccc2Cl)CC1 REAL300018775227
O=C(O)C1(CC(F)F)CCN(Cc2cc(F)ccc2Br)CC1 REAL300018775228
COc1ccc(Br)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775229
COc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1F REAL300018775230
O=C(O)C1(CC(F)F)CCN(Cc2cncc3ccccc23)CC1 REAL300018775231
O=C(O)C1(CC(F)F)CCN(Cc2ncccc2C(F)(F)F)CC1 REAL300018775232
O=C(O)C1(CC(F)F)CCN(CC=Cc2ccc(Cl)cc2)CC1 REAL300018775233
Cc1oc2ccccc2c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775234
O=C(O)C1(CC(F)F)CCN(CC2CC2c2ccccc2)CC1 REAL300018775235
O=C(O)C1(CC(F)F)CCN(Cc2cscc2Cl)CC1 REAL300018775236
O=C(O)C1(CC(F)F)CCN(Cc2cnc3ccsc3c2)CC1 REAL300018775237
Cc1cc(Cl)cc(C)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775238
CCOc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)nc1 REAL300018775239
Cc1nn2c(CN3CCC(CC(F)F)(C(=O)O)CC3)c(C)nc2s1 REAL300018775240
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Sc3ccccc3)cc2)CC1 REAL300018775241
Cn1c(CN2CCC(CC(F)F)(C(=O)O)CC2)nc2cc(Cl)ccc21 REAL300018775242
CC1CCc2nc(CN3CCC(CC(F)F)(C(=O)O)CC3)sc2C1 REAL300018775243
COc1cc(Cl)c(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1Cl REAL300018775244
CC(C)Cc1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775245
O=C(O)C1(CC(F)F)CCN(Cc2ccc(-c3ccncc3)cc2F)CC1 REAL300018775246
O=C(O)C1(CC(F)F)CCN(Cc2c(Cl)oc3ccccc23)CC1 REAL300018775247
CC1(C)CCc2nc(CN3CCC(CC(F)F)(C(=O)O)CC3)sc2C1 REAL300018775248
CCc1nn(C)c(CC)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775249
O=C(O)C1(CC(F)F)CCN(Cc2cnc(C3CCCO3)s2)CC1 REAL300018775250
CC1(C)CCC(CN2CCC(CC(F)F)(C(=O)O)CC2)CC1 REAL300018775251
COc1sc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1Br REAL300018775252
Cc1nn2c(CN3CCC(CC(F)F)(C(=O)O)CC3)c(C(C)C)nc2s1 REAL300018775253
COc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1OC(=O)C1CC1 REAL300018775254
COC(=O)c1occc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775255
COC(=O)CCn1nc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1C REAL300018775256
CCOC(=O)COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775257
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Cl)c(Br)c2)CC1 REAL300018775258
COc1ccc(O)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775259
Cc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1O REAL300018775260
O=C(O)C1(CC(F)F)CCN(Cc2cccc(Cl)c2O)CC1 REAL300018775261
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)cc(F)c2O)CC1 REAL300018775262
COc1cc(O)c(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1OC REAL300018775263
Cc1cc(Br)cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1O REAL300018775264
O=C(O)C1(CC(F)F)CCN(Cc2c(C3CC3)nc3sccn23)CC1 REAL300018775265
Cc1cccc(C)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775266
O=C(O)C1(CC(F)F)CCN(Cc2cccc3nccn23)CC1 REAL300018775267
CCCC1CCC(CN2CCC(CC(F)F)(C(=O)O)CC2)CC1 REAL300018775268
CC(CCc1ccccc1)CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775269
CC(Cc1ccc(C(C)(C)C)cc1)CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775270
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C(C)(C)C)n1 REAL300018775271
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(-c2cccs2)n1 REAL300018775272
CC(C)COc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775273
Cn1cnc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)ccc21 REAL300018775274
O=C(O)C1(CC(F)F)CCN(Cc2ccn(-c3ccccc3)n2)CC1 REAL300018775275
O=C(O)C1(CC(F)F)CCN(Cc2c(Cl)cccc2N2CCCC2)CC1 REAL300018775276
CN(C)c1cccc(Cl)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775277
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(-c2ccccc2)n1 REAL300018775278
CCc1nn(C)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775279
CC(C)(CN1CCC(CC(F)F)(C(=O)O)CC1)c1ccccc1 REAL300018775280
CN1CCN(c2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)cc2)CC1 REAL300018775281
O=C(O)C1(CC(F)F)CCN(Cc2nc3c(s2)CCC3)CC1 REAL300018775282
CCCC(CN1CCC(CC(F)F)(C(=O)O)CC1)c1ccccc1 REAL300018775283
COc1ccc(C(C)CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775284
O=C(O)C1(CC(F)F)CCN(Cc2nc3c(s2)CCCC3)CC1 REAL300018775285
O=C(O)C1(CC(F)F)CCN(Cc2ccn(C(F)F)n2)CC1 REAL300018775286
CC(CCc1cccc(F)c1)N1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775287
CC(Cc1ccsc1)N1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775288
Cc1ccc(F)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775289
CC(C)(C)OC(=O)c1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775290
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(-c2ccc(C#N)cc2)n1 REAL300018775291
COc1c(O)cccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775292
O=C(O)C1(CC(F)F)CCN(Cc2cc(F)ccc2O)CC1 REAL300018775293
O=C(O)C1(CC(F)F)CCN(CCc2ccc(F)cc2)CC1 REAL300018775294
O=C(O)C1(CC(F)F)CCN(Cc2cccc(F)c2O)CC1 REAL300018775295
CC(C)C1CC(CN2CCC(CC(F)F)(C(=O)O)CC2)CCO1 REAL300018775296
CCC1CC(CN2CCC(CC(F)F)(C(=O)O)CC2)CCO1 REAL300018775297
COCCC1(CN2CCC(CC(F)F)(C(=O)O)CC2)CCC1 REAL300018775298
O=C(O)C1(CC(F)F)CCN(Cc2c(Cl)ccc3cccnc23)CC1 REAL300018775299
Cn1nc(C(F)(F)F)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1Cl REAL300018775300
O=C(O)C1(CC(F)F)CCN(Cc2ccc(SC(F)F)cc2)CC1 REAL300018775301
COc1cc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)n1 REAL300018775302
CC(C)Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775303
COC(=O)COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775304
CCOCOc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775305
CC(Cc1ccccc1)CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775306
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C2CCCCC2)n1 REAL300018775307
O=C(O)C1(CC(F)F)CCN(Cc2cn(Cc3cccnc3)nn2)CC1 REAL300018775308
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc2cccnc12 REAL300018775309
CC(C)(C)C1CCC(CN2CCC(CC(F)F)(C(=O)O)CC2)CC1 REAL300018775310
CC(C)c1cnc(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775311
COC(=O)c1coc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775312
COc1ccc(CC(C)CN2CCC(CC(F)F)(C(=O)O)CC2)cc1F REAL300018775313
O=C(O)C1(CC(F)F)CCN(Cc2ccc(OCC(F)(F)F)c(F)c2)CC1 REAL300018775314
O=C(O)C1(CC(F)F)CCN(CC=Cc2ccc(F)cc2F)CC1 REAL300018775315
CC(CC1CCCCC1)CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775316
CC(C)(C)OC(=O)N1CC(CN2CCC(CC(F)F)(C(=O)O)CC2)C1 REAL300018775317
O=C(O)C1(CC(F)F)CCN(Cc2ccc([N+](=O)[O-])c(Cl)c2)CC1 REAL300018775318
CC(C)(CN1CCC(CC(F)F)(C(=O)O)CC1)NC(=O)OC(C)(C)C REAL300018775319
COc1cc(Cl)cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1O REAL300018775320
COc1cc2c(cc1CN1CCC(CC(F)F)(C(=O)O)CC1)OCO2 REAL300018775321
O=C(O)C1(CC(F)F)CCN(Cc2cnn3ncccc23)CC1 REAL300018775322
O=C(O)C1(CC(F)F)CCN(CC2CC3CCC2C3)CC1 REAL300018775323
O=C(O)C1(CC(F)F)CCN(Cc2cccn3nccc23)CC1 REAL300018775324
O=C(O)C1(CC(F)F)CCN(Cc2sccc2Br)CC1 REAL300018775325
CC(C)c1ccc(CCN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775326
CCCCOc1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775327
O=C(O)C1(CC(F)F)CCN(Cc2cncc(Br)c2)CC1 REAL300018775328
O=C(O)C1(CC(F)F)CCN(CCCCc2ccc(Cl)c(Cl)c2)CC1 REAL300018775329
CCn1nc(CN2CCC(CC(F)F)(C(=O)O)CC2)c2ccccc21 REAL300018775330
O=C(O)C1(CC(F)F)CCN(Cc2ncc(Cl)s2)CC1 REAL300018775331
CCOC(=O)c1nn(C)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775332
O=C(O)C1(CC(F)F)CCN(CCSCc2ccccc2)CC1 REAL300018775333
COc1ccc(-c2ccncc2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775334
CN1C(=O)CCc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)ccc21 REAL300018775335
COc1c(Br)cccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775336
Cc1ccncc1CCCN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775337
COC(=O)C(C)(C)CCN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775338
C#CCOc1cccc(Cl)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775339
CC1(c2ccccc2)CCC(N2CCC(CC(F)F)(C(=O)O)CC2)C1 REAL300018775340
O=C(O)C1(CC(F)F)CCN(Cc2cc3c(F)cccc3[nH]2)CC1 REAL300018775341
O=C(O)C1(CC(F)F)CCN(Cc2c[nH]nc2-c2ccsc2)CC1 REAL300018775342
Cn1ncc(Cl)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775343
O=C(O)C1(CC(F)F)CCN(CC2CCc3ccccc32)CC1 REAL300018775344
CC(C)(C)OC(=O)NCCCN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775345
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)sn1 REAL300018775346
COC(=O)Cc1coc(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775347
O=C(O)C1(CC(F)F)CCN(Cc2nc3c([nH]2)COCC3)CC1 REAL300018775348
O=C(O)C1(CC(F)F)CCN(Cc2noc3c2COCC3)CC1 REAL300018775349
Cn1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1Br REAL300018775350
O=C(O)C1(CC(F)F)CCN(CC=Cc2ccccc2)CC1 REAL300018775351
O=C(O)C1(CC(F)F)CCN(Cc2cnnn2C2CC2)CC1 REAL300018775352
COCc1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775353
O=C(O)C1(CC(F)F)CCN(Cc2cccc(SC(F)(F)F)c2)CC1 REAL300018775354
O=C(O)C1(CC(F)F)CCN(Cc2ccc3c(c2)CCC32OCCO2)CC1 REAL300018775355
O=C(O)C1(CC(F)F)CCN(Cc2ccc3c(c2)COCC3)CC1 REAL300018775356
Cc1nc(N2CCCC2)sc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775357
O=C(O)C1(CC(F)F)CCN(Cc2cnn(CCO)c2)CC1 REAL300018775358
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)sc2cc(F)ccc12 REAL300018775359
O=C(O)C1(CC(F)F)CCN(Cc2cc(-c3ccncc3)n[nH]2)CC1 REAL300018775360
COc1ccc(F)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1OC REAL300018775361
O=C(O)C1(CC(F)F)CCN(CC=Cc2ccncc2)CC1 REAL300018775362
Cn1ccc(-c2n[nH]cc2CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775363
Cc1ccc(F)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1Br REAL300018775364
C=Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775365
O=C(O)C1(CC(F)F)CCN(Cc2cccc(OCC3CCC3)c2)CC1 REAL300018775366
CC(F)(F)c1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775367
COc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1OCCO REAL300018775368
CCn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C2CC2)n1 REAL300018775369
CCc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)nc1 REAL300018775370
COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1OCCO REAL300018775371
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(-c2ccnn2C)n1 REAL300018775372
COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)nn1 REAL300018775373
CC(C)(C)c1nocc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775374
O=C(O)C1(CC(F)F)CCN(Cc2ccc3ccncc3c2)CC1 REAL300018775375
Cc1cc2cccc(CN3CCC(CC(F)F)(C(=O)O)CC3)c2o1 REAL300018775376
O=C(O)C1(CC(F)F)CCN(Cc2cccc(F)c2C(F)(F)F)CC1 REAL300018775377
O=C(O)C1(CC(F)F)CCN(Cc2c(F)cccc2OCC(F)(F)F)CC1 REAL300018775378
COc1csc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1OC REAL300018775379
O=C(O)C1(CC(F)F)CCN(Cc2conc2C2CCC2)CC1 REAL300018775380
CS(=O)(=O)c1ccsc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775381
CN(C)c1nc(Cl)c(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775382
Cn1c(=O)c(CN2CCC(CC(F)F)(C(=O)O)CC2)cc2ccccc21 REAL300018775383
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)c(=O)n(-c2ccccc2)n1C REAL300018775384
O=C(O)C1(CC(F)F)CCN(Cc2ccc(-c3ccsc3)cc2)CC1 REAL300018775385
O=C(O)C1(CC(F)F)CCN(Cc2nc3ccccc3s2)CC1 REAL300018775386
O=C(O)C1(CC(F)F)CCN(Cc2[nH]ncc2Br)CC1 REAL300018775387
O=C(O)C1(CC(F)F)CCN(Cc2ccc3nsnc3c2)CC1 REAL300018775388
O=C(O)C1(CC(F)F)CCN(Cc2ccc3nonc3c2)CC1 REAL300018775389
O=C(O)C1(CC(F)F)CCN(Cc2cccc3nsnc23)CC1 REAL300018775390
CCn1cnc(Cl)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775391
N#Cc1cnn2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)cnc12 REAL300018775392
O=C(O)C1(CC(F)F)CCN(Cc2cn(-c3ccccc3)nn2)CC1 REAL300018775393
CCOc1ccc(Cl)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775394
O=C(O)C1(CC(F)F)CCN(Cc2sc(N3CCCC3)nc2Cl)CC1 REAL300018775395
O=C(O)C1(CC(F)F)CCN(Cc2c[nH]nc2-c2cccc(F)c2)CC1 REAL300018775396
Cc1oc(-c2cccs2)nc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775397
Cn1nc(-c2ccccc2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775398
CC(C)(C)c1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)n[nH]1 REAL300018775399
CCN1CCCc2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)ccc21 REAL300018775400
O=C(O)C1(CC(F)F)CCN(Cc2ccc(-c3ccsc3)nc2)CC1 REAL300018775401
O=C(O)C1(CC(F)F)CCN(Cc2cc3ccccc3cn2)CC1 REAL300018775402
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc(Cl)n1 REAL300018775403
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc(C)n1 REAL300018775404
COc1cc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775405
O=C(O)C1(CC(F)F)CCN(Cc2ccc[nH]c2=O)CC1 REAL300018775406
CCc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)cnn1CC REAL300018775407
O=C(O)C1(CC(F)F)CCN(Cc2cc3ccc(F)cc3[nH]c2=O)CC1 REAL300018775408
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C(F)(F)F)n1 REAL300018775409
O=C(O)C1(CC(F)F)CCN(Cc2noc3c2CCCC3)CC1 REAL300018775410
Cc1cn(C)nc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775411
O=C(O)C1(CC(F)F)CCN(Cc2cc3ccncc3s2)CC1 REAL300018775412
COc1nc(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc1C REAL300018775413
O=C(O)C1(CC(F)F)CCN(Cc2cc3ncccc3o2)CC1 REAL300018775414
CCC(C)n1nccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775415
O=C(O)C1(CC(F)F)CCN(Cc2nc(CO)cs2)CC1 REAL300018775416
O=C(O)C1(CC(F)F)CCN(Cc2cccc3cc(Cl)ccc23)CC1 REAL300018775417
CCCn1cncc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775418
CCc1c[nH]c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775419
O=C(O)C1(CC(F)F)CCN(Cc2cncc(-c3cccnc3)c2)CC1 REAL300018775420
CC(C)(C)c1cncc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775421
COc1nc(Cl)ccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775422
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)ccnc1F REAL300018775423
O=C(O)C1(CC(F)F)CCN(Cc2ccc3c(c2)CCOC3)CC1 REAL300018775424
O=C(O)C1(CC(F)F)CCN(Cc2cccc(C(F)F)c2F)CC1 REAL300018775425
Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)n1 REAL300018775426
O=C(O)C1(CC(F)F)CCN(Cc2nc3c(s2)CCCCC3)CC1 REAL300018775427
O=C(O)C1(CC(F)F)CCN(Cc2nc3c(s2)COCC3)CC1 REAL300018775428
CC(C)Cc1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775429
CSc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)o1 REAL300018775430
O=C(O)C1(CC(F)F)CCN(Cc2cnn(C3CCCCC3)c2)CC1 REAL300018775431
CCCn1nc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1Cl REAL300018775432
Cn1cc(-c2n[nH]cc2CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775433
CC(C)n1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775434
O=C(O)C1(CC(F)F)CCN(Cc2ccn(CC(F)(F)F)n2)CC1 REAL300018775435
CC(F)(F)c1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775436
O=C(O)C1(CC(F)F)CCN(Cc2cnn(-c3ccccc3)c2Cl)CC1 REAL300018775437
Cc1cc(O)ncc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775438
Cc1nc(CN2CCC(CC(F)F)(C(=O)O)CC2)oc1C REAL300018775439
CS(=O)(=O)c1coc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775440
O=C(O)C1(CC(F)F)CCN(Cc2cn(CC3CC3)nn2)CC1 REAL300018775441
O=C(O)C1(CC(F)F)CCN(Cc2cccn2C(F)F)CC1 REAL300018775442
O=C(O)C1(CC(F)F)CCN(Cc2cc3c(o2)CCCC3)CC1 REAL300018775443
O=C(O)C1(CC(F)F)CCN(Cc2c(Cl)nc3cc(Cl)ccn23)CC1 REAL300018775444
Cn1cc(Br)nc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775445
C=CCc1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775446
COc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)cccc1C(C)(C)C REAL300018775447
COc1nn(C)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775448
CC(C)(C)n1nccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775449
CN(CCO)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775450
Cn1c(CN2CCC(CC(F)F)(C(=O)O)CC2)nc2c1CCCC2 REAL300018775451
O=C(O)C1(CC(F)F)CCN(Cc2cccc3c2COCC3)CC1 REAL300018775452
O=C(O)C1(CC(F)F)CCN(Cc2ccccc2C2CCC2)CC1 REAL300018775453
CC(C)(C#N)c1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)s1 REAL300018775454
CCn1nc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775455
COc1sccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775456
O=C(O)C1(CC(F)F)CCN(Cc2cc(C3CCC3)[nH]n2)CC1 REAL300018775457
C=CCCn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)nn1 REAL300018775458
O=C(O)C1(CC(F)F)CCN(Cc2ccc(CC3CCC3)cc2)CC1 REAL300018775459
COc1nsc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1Cl REAL300018775460
O=C(O)C1(CC(F)F)CCN(Cc2cn(C3CC3)cn2)CC1 REAL300018775461
O=C(O)C1(CC(F)F)CCN(Cc2nc(C(F)(F)F)n3c2CCCC3)CC1 REAL300018775462
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C2CCOCC2)n1 REAL300018775463
CC(C)c1cnn(C)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775464
Cn1nnc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1C(F)F REAL300018775465
Cn1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1S(C)(=O)=O REAL300018775466
Cc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1OC(F)F REAL300018775467
CC1Oc2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)cc2C1C REAL300018775468
O=C(O)C1(CC(F)F)CCN(Cc2ccccc2-n2cccn2)CC1 REAL300018775469
O=C(O)C1(CC(F)F)CCN(Cc2ccnn2C2CC2(F)F)CC1 REAL300018775470
COCc1nocc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775471
COCc1cnc(OC)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775472
O=C(O)C1(CC(F)F)CCN(Cc2ccc(C(F)F)cn2)CC1 REAL300018775473
O=C(O)C1(CC(F)F)CCN(Cc2ccc(C(F)(F)F)cc2F)CC1 REAL300018775474
CC(C)Oc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1F REAL300018775475
CCn1cc(Cl)c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775476
O=C(O)C1(CC(F)F)CCN(Cc2ccc(F)c(Cl)c2F)CC1 REAL300018775477
O=C(O)C1(CC(F)F)CCN(Cc2cccc(C(F)F)c2)CC1 REAL300018775478
O=C(O)C1(CC(F)F)CCN(Cc2ccc3ccccc3c2F)CC1 REAL300018775479
CS(=O)(=O)c1csc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775480
O=C(O)C1(CC(F)F)CCN(Cc2csc(Cl)c2)CC1 REAL300018775481
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)cnn1C1CCC1 REAL300018775482
O=C(O)C1(CC(F)F)CCN(Cc2cnn(-c3cccc(Cl)c3)c2)CC1 REAL300018775483
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)n(C2CCCC2)n1 REAL300018775484
O=C(O)C1(CC(F)F)CCN(Cc2ccnn2CC(F)F)CC1 REAL300018775485
COc1ccc(C)nc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775486
N#Cc1ccc(Br)c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775487
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)cc(Cl)n2)CC1 REAL300018775488
O=C(O)C1(CC(F)F)CCN(Cc2nccc3cc(Cl)ccc23)CC1 REAL300018775489
O=C(O)C1(CC(F)F)CCN(Cc2cc3cnccc3[nH]2)CC1 REAL300018775490
CN(C)c1ccc([N+](=O)[O-])cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775491
O=C(O)C1(CC(F)F)CCN(Cc2cccc(Cl)c2C(F)(F)F)CC1 REAL300018775492
O=C(O)C1(CC(F)F)CCN(Cc2c(F)ccnc2Cl)CC1 REAL300018775493
O=C(O)C1(CC(F)F)CCN(Cc2cccc(C(F)F)n2)CC1 REAL300018775494
O=C(O)C1(CC(F)F)CCN(Cc2cnn(-c3cccc(F)c3)c2)CC1 REAL300018775495
CN(C)c1cncc(F)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775496
COc1nc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)c1Cl REAL300018775497
CC(C)N(C)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(O)c1 REAL300018775498
O=C(O)C1(CC(F)F)CCN(Cc2c(O)ccc3c2OCO3)CC1 REAL300018775499
Cc1nn(-c2ccccc2)nc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775500
O=C(O)C1(CC(F)F)CCN(Cc2ccn(C3CCC3)n2)CC1 REAL300018775501
O=C(O)C1(CC(F)F)CCN(Cc2ccn(CC(F)F)n2)CC1 REAL300018775502
O=C(O)C1(CC(F)F)CCN(Cc2ccn(C3CC3(F)F)n2)CC1 REAL300018775503
Cc1nn(C2CCCCC2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775504
O=C(O)C1(CC(F)F)CCN(Cc2cnn(C3CCOCC3)c2)CC1 REAL300018775505
Cc1nn(C2CCOCC2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775506
Cc1cn(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775507
O=C(O)C1(CC(F)F)CCN(Cc2noc3c2CCC3)CC1 REAL300018775508
O=C(O)C1(CC(F)F)CCN(Cc2nc3cccc(F)c3s2)CC1 REAL300018775509
O=C(O)C1(CC(F)F)CCN(Cc2ccn(C3CCCC3)n2)CC1 REAL300018775510
NS(=O)(=O)c1csc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775511
O=C(O)C1(CC(F)F)CCN(Cc2ccc(F)c3ccoc23)CC1 REAL300018775512
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)cc3ccoc23)CC1 REAL300018775513
O=C(O)C1(CC(F)F)CCN(Cc2ncc(Cl)cc2Cl)CC1 REAL300018775514
O=C(c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1)N1CCOCC1 REAL300018775515
Cc1nn(C2CCCC2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775516
O=C(O)C1(CC(F)F)CCN(Cc2ccccc2C(F)F)CC1 REAL300018775517
Cc1cc(Br)c(F)c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775518
COc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1Br REAL300018775519
O=C(O)C1(CC(F)F)CCN(Cc2ccc3[nH]ncc3c2)CC1 REAL300018775520
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Cl)c(F)c2F)CC1 REAL300018775521
Cc1c(F)cccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775522
Cn1cc(-c2cccc(CN3CCC(CC(F)F)(C(=O)O)CC3)c2)cn1 REAL300018775523
O=C(O)C1(CC(F)F)CCN(Cc2ccc([N+](=O)[O-])c(OC3CC3)c2)CC1 REAL300018775524
Cc1ccc(Br)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775525
COc1c(C#N)cccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775526
COc1nc2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)cc2s1 REAL300018775527
O=C(O)C1(CC(F)F)CCN(Cc2ccnc(Br)c2)CC1 REAL300018775528
O=C(O)C1(CC(F)F)CCN(Cc2cc(F)cc(Cl)c2Cl)CC1 REAL300018775529
Cc1nc(Cl)ccc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775530
CC(C)(C)COc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775531
COc1cc(Cl)cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775532
COc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc(F)c1F REAL300018775533
COc1cc(C)ncc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775534
COc1ccc2sc(CN3CCC(CC(F)F)(C(=O)O)CC3)nc2c1 REAL300018775535
CC(C)n1cnc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775536
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)nnn1C REAL300018775537
Cn1nccc1-c1n[nH]cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775538
Cc1onc(C2CC2)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775539
COC(=O)c1c(C)[nH]c(CN2CCC(CC(F)F)(C(=O)O)CC2)c1C REAL300018775540
CC(C)Oc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)o1 REAL300018775541
Cc1cc(Br)cc(C)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775542
O=C(O)C1(CC(F)F)CCN(Cc2ccc(C(F)(F)F)cc2O)CC1 REAL300018775543
Cc1oc(-c2ccccc2)nc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775544
Cn1nc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1-c1ccco1 REAL300018775545
O=C(O)C1(CC(F)F)CCN(Cc2c(Cl)ccc3c2OCO3)CC1 REAL300018775546
N#Cc1cc(F)cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1 REAL300018775547
O=C(O)C1(CC(F)F)CCN(Cc2ccc(C3CCCCC3)cc2)CC1 REAL300018775548
Cc1nc(C)c(CN2CCC(CC(F)F)(C(=O)O)CC2)nc1C REAL300018775549
NC(=O)c1cnc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775550
Cc1cc(Br)sc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775551
Cc1nn(C2CCC2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775552
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)cnn1CC(F)F REAL300018775553
COc1ccccc1C=CCN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775554
O=C(O)C1(CC(F)F)CCN(Cc2ccc(-c3ccccn3)nc2)CC1 REAL300018775555
CCCn1nc(C)c(Cl)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775556
COc1cccc2[nH]c(CN3CCC(CC(F)F)(C(=O)O)CC3)cc12 REAL300018775557
CC(C)n1c(CN2CCC(CC(F)F)(C(=O)O)CC2)nc2cc(Cl)ccc21 REAL300018775558
Cc1ccc(OC(F)F)c(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775559
Cn1nc(-c2ccco2)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775560
O=C(O)C1(CC(F)F)CCN(Cc2ccc(Cc3ccccc3)cc2)CC1 REAL300018775561
CCCCC(=O)Nc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775562
COc1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)n1 REAL300018775563
COC(=O)[C@H]1C[C@H](n2ccc(CN3CCC(CC(F)F)(C(=O)O)CC3)n2)C1 REAL300018775564
COC(=O)[C@H]1C[C@H](n2nccc2CN2CCC(CC(F)F)(C(=O)O)CC2)C1 REAL300018775565
CCN(C)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)c1 REAL300018775566
O=C(O)C1(CC(F)F)CCN(Cc2cc(Cl)cnc2Br)CC1 REAL300018775567
O=C(O)C1(CC(F)F)CCN(Cc2cc(-c3ccccc3)ccn2)CC1 REAL300018775568
O=C(O)C1(CC(F)F)CCN(Cc2scc(Cl)c2Cl)CC1 REAL300018775569
CC(C)(C)c1nn(C(C)(C)C)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775570
COc1cc(C)cc(OC)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775571
O=C(O)C1(CC(F)F)CCN(Cc2ccc(CF)cc2)CC1 REAL300018775572
O=C(O)C1(CC(F)F)CCN(Cc2ccc3sccc3c2)CC1 REAL300018775573
O=C(O)C1(CC(F)F)CCN(Cc2ccc(-c3ccncc3)cc2)CC1 REAL300018775574
O=C(O)C1(CC(F)F)CCN(Cc2ccccc2CO)CC1 REAL300018775575
CC(C)(C)c1oncc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775576
Cc1cncc(C)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775577
COc1cc(C)c2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)[nH]c2c1 REAL300018775578
Cc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1C(F)(F)F REAL300018775579
C=CCn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cn1 REAL300018775580
O=C(O)C1(CC(F)F)CCN(Cc2ccc3cn[nH]c3c2)CC1 REAL300018775581
CCC(C)c1ccc(CN2CCC(CC(F)F)(C(=O)O)CC2)cc1 REAL300018775582
O=C(O)C1(CC(F)F)CCN(Cc2cccc3nc(C(F)F)sc23)CC1 REAL300018775583
CC(F)(F)c1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)n1 REAL300018775584
O=C(O)C1(CC(F)F)CCN(Cc2cc3c(nc2Cl)CCOC3)CC1 REAL300018775585
COc1cc(OC)c2cc(CN3CCC(CC(F)F)(C(=O)O)CC3)[nH]c2c1 REAL300018775586
O=C(O)C1(CC(F)F)CCN(Cc2cc3sccc3[nH]2)CC1 REAL300018775587
Cn1c(Cc2ccccc2)cnc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775588
O=C(O)C1(CC(F)F)CCN(Cc2cc(Br)cc(F)c2F)CC1 REAL300018775589
O=C(O)C1(CC(F)F)CCN(Cc2cccc3c2CCCC3)CC1 REAL300018775590
CC(=Cc1cc(F)cc(F)c1)CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775591
O=C(O)C1(CC(F)F)CCN(Cc2cccc(C(F)(F)F)c2F)CC1 REAL300018775592
O=C(O)C1(CC(F)F)CCN(Cc2ccc(-n3ccnn3)cc2)CC1 REAL300018775593
Cc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc2ccccc12 REAL300018775594
CC(C)c1nn(C(C)(C)C)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775595
COc1c(CN2CCC(CC(F)F)(C(=O)O)CC2)ccc2[nH]ccc12 REAL300018775596
Cc1nc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C)s1 REAL300018775597
O=C(O)C1(CC(F)F)CCN(Cc2ccc(N3CCC(O)C3)cc2)CC1 REAL300018775598
COc1ccc(OC)c(OC)c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775599
CCCn1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1C REAL300018775600
O=C(O)C1(CC(F)F)CCN(Cc2nccc(Br)c2F)CC1 REAL300018775601
O=C(c1ccccc1CN1CCC(CC(F)F)(C(=O)O)CC1)N1CCCCC1 REAL300018775602
Cc1ccc2cccnc2c1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775603
O=C(O)C1(CC(F)F)CCN(Cc2[nH]nc(C3CC3)c2Br)CC1 REAL300018775604
O=C(O)C1(CC(F)F)CCN(Cc2c(O)cccc2F)CC1 REAL300018775605
Cc1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)cnc1-n1cccn1 REAL300018775606
COC(=O)c1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)n(C)c1 REAL300018775607
O=C(O)C1(CC(F)F)CCN(Cc2cc3sc(Cl)cc3[nH]2)CC1 REAL300018775608
COc1ccc2ccnc(C(C)N3CCC(CC(F)F)(C(=O)O)CC3)c2c1 REAL300018775609
COc1ccn2c(CN3CCC(CC(F)F)(C(=O)O)CC3)cnc2c1 REAL300018775610
CCCn1nc(C)cc1CN1CCC(CC(F)F)(C(=O)O)CC1 REAL300018775611
Cn1cc(CN2CCC(CC(F)F)(C(=O)O)CC2)c(C2CCC2)n1 REAL300018775612
CC(C)(C)c1ncc(CN2CCC(CC(F)F)(C(=O)O)CC2)o1 REAL300018775613
Cn1nc(CN2CCC(CC(F)F)(C(=O)O)CC2)c2c1CCOC2 REAL300018775614
O=C(O)c1csc(C2CCCN(Cc3cccnc3)C2)n1 REAL300018775615
CC(CN1CCCC(c2nc(C(=O)O)cs2)C1)c1ccccc1 REAL300018775616
O=C(O)c1csc(C2CCCN(Cc3ccc4c(c3)OCCO4)C2)n1 REAL300018775617
O=C(O)c1csc(C2CCCN(Cc3cccc(Br)c3)C2)n1 REAL300018775618
COc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1OC REAL300018775619
O=C(O)c1csc(C2CCCN(CC3CC=CCC3)C2)n1 REAL300018775620
O=C(O)c1csc(C2CCCN(Cc3ccccc3C(F)(F)F)C2)n1 REAL300018775621
Cc1ccccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775622
CCc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775623
COC(=O)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775624
O=C(O)c1csc(C2CCCN(Cc3ccc(-c4ccc(F)cc4)o3)C2)n1 REAL300018775625
O=C(O)c1csc(C2CCCN(CC3CCCCC3)C2)n1 REAL300018775626
O=C(O)c1csc(C2CCCN(Cc3ccc(Br)o3)C2)n1 REAL300018775627
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1C REAL300018775628
O=C(O)c1csc(C2CCCN(Cc3cc(Br)cs3)C2)n1 REAL300018775629
CC(C)=CCCC(C)CCN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775630
Cn1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cn1 REAL300018775631
COC(=O)c1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)oc1C REAL300018775632
Cc1nn(C)c(Cl)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775633
O=C(O)c1csc(C2CCCN(CC3CCC=CO3)C2)n1 REAL300018775634
CC(CCN1CCCC(c2nc(C(=O)O)cs2)C1)c1ccccc1 REAL300018775635
O=C(O)c1csc(C2CCCN(Cc3ccc(F)c(Cl)c3)C2)n1 REAL300018775636
O=C(O)c1csc(C2CCCN(Cc3ccc(F)c(C(F)(F)F)c3)C2)n1 REAL300018775637
CCOc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775638
O=C(O)c1csc(C2CCCN(Cc3ccc(F)cc3C(F)(F)F)C2)n1 REAL300018775639
O=C(O)c1csc(C2CCCN(Cc3cc(F)cc(C(F)(F)F)c3)C2)n1 REAL300018775640
COc1ccc(F)c(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775641
O=C(O)c1csc(C2CCCN(Cc3cc(F)cc(Cl)c3)C2)n1 REAL300018775642
O=C(O)c1csc(C2CCCN(Cc3ccc(Cl)cc3F)C2)n1 REAL300018775643
O=C(O)c1csc(C2CCCN(Cc3cccc4c3OCO4)C2)n1 REAL300018775644
O=C(O)c1csc(C2CCCN(Cc3cc(Cl)ccc3F)C2)n1 REAL300018775645
COc1ccc(F)cc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775646
O=C(O)c1csc(C2CCCN(Cc3cc(F)cc(F)c3)C2)n1 REAL300018775647
COc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cn1 REAL300018775648
O=C(O)c1csc(C2CCCN(Cc3ccc4occc4c3)C2)n1 REAL300018775649
Cc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n(C)n1 REAL300018775650
COC(=O)c1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cn1C REAL300018775651
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1Cl REAL300018775652
O=C(O)c1csc(C2CCCN(Cc3csnn3)C2)n1 REAL300018775653
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)ccc1C REAL300018775654
O=C(O)c1csc(C2CCCN(Cc3cccc(-c4ccccn4)c3)C2)n1 REAL300018775655
Cc1nn(C(C)(C)C)c(C)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775656
N#Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(F)c1 REAL300018775657
COC(=O)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)o1 REAL300018775658
Cc1nn(C)cc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775659
CCC(CN1CCCC(c2nc(C(=O)O)cs2)C1)c1ccccc1 REAL300018775660
COc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1F REAL300018775661
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(Br)c1 REAL300018775662
CN(C)c1ncc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1C REAL300018775663
CC1(C)CCCC(CN2CCCC(c3nc(C(=O)O)cs3)C2)C1 REAL300018775664
O=C(O)c1csc(C2CCCN(CCCc3c(F)cccc3Cl)C2)n1 REAL300018775665
CC1=CCCC(C)C1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775666
Cc1cc(Cl)ccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775667
O=C(O)c1csc(C2CCCN(CCC3CCCCC3)C2)n1 REAL300018775668
Cn1ncc(Br)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775669
CCn1nccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775670
C#Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775671
COc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1 REAL300018775672
CCn1cncc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775673
O=C(O)c1csc(C2CCCN(Cc3ccncc3F)C2)n1 REAL300018775674
Cc1ccc2cc(CN3CCCC(c4nc(C(=O)O)cs4)C3)ccc2n1 REAL300018775675
COc1cc(F)cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775676
CC(C)(C)c1ncc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cn1 REAL300018775677
Cc1occc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775678
Cn1c(=O)oc2cc(CN3CCCC(c4nc(C(=O)O)cs4)C3)ccc21 REAL300018775679
O=C(O)c1csc(C2CCCN(CCc3cccc(Cl)c3)C2)n1 REAL300018775680
COc1ccc2oc(CN3CCCC(c4nc(C(=O)O)cs4)C3)cc2c1 REAL300018775681
Cc1ccc(C(C)CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775682
N#Cc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1 REAL300018775683
Cn1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775684
CC(C)n1nccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775685
O=C(O)c1csc(C2CCCN(Cc3coc4ccccc34)C2)n1 REAL300018775686
COc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(C)c1OC REAL300018775687
O=C(O)c1csc(C2CCCN(Cc3ccc(Oc4ccccc4)o3)C2)n1 REAL300018775688
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1Br REAL300018775689
Cc1ccc2nc(CN3CCCC(c4nc(C(=O)O)cs4)C3)cn2c1 REAL300018775690
Cc1c[nH]c(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1 REAL300018775691
COc1cc(C)ccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775692
COCc1csc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775693
COCc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)no1 REAL300018775694
O=C1COc2ccc(CN3CCCC(c4nc(C(=O)O)cs4)C3)cc2N1 REAL300018775695
CC(C)n1ccnc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775696
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)nn1 REAL300018775697
O=C(O)c1csc(C2CCCN(Cc3ccnc(Cl)c3Cl)C2)n1 REAL300018775698
O=C(O)c1csc(C2CCCN(Cc3cnc4cnccn34)C2)n1 REAL300018775699
O=C(O)c1csc(C2CCCN(CCCc3ccc4c(c3)CCO4)C2)n1 REAL300018775700
O=C(O)c1csc(C2CCCN(Cc3cc4c(cn3)OCCO4)C2)n1 REAL300018775701
Cc1ccc2ncc(CN3CCCC(c4nc(C(=O)O)cs4)C3)n2c1 REAL300018775702
Cn1c(CN2CCCC(c3nc(C(=O)O)cs3)C2)cnc1Cl REAL300018775703
O=C(O)c1csc(C2CCCN(Cc3cc(C(F)(F)F)[nH]n3)C2)n1 REAL300018775704
O=C(O)c1csc(C2CCCN(Cc3cc(Cl)cc4c3OCC4)C2)n1 REAL300018775705
Cc1nocc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775706
Cc1ncoc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775707
O=C(O)c1csc(C2CCCN(Cc3cc(Cl)cs3)C2)n1 REAL300018775708
Cc1cnn(C)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775709
Cc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)ccc1Cl REAL300018775710
O=C(O)c1csc(C2CCCN(Cc3nccn3-c3ccccc3)C2)n1 REAL300018775711
C=Cn1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cn1 REAL300018775712
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)sn1 REAL300018775713
CCCc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775714
CC(CN1CCCC(c2nc(C(=O)O)cs2)C1)c1cccc(Cl)c1 REAL300018775715
Cn1ncc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1Cl REAL300018775716
Cc1c(CN2CCCC(c3nc(C(=O)O)cs3)C2)cnn1C REAL300018775717
O=C(O)c1csc(C2CCCN(Cc3cnc(C4CC4)nc3)C2)n1 REAL300018775718
O=C(O)c1csc(C2CCCN(Cc3cnc(C4CC4)o3)C2)n1 REAL300018775719
CCOc1cncc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775720
CC(C)(C)n1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)nn1 REAL300018775721
Cn1c(CN2CCCC(c3nc(C(=O)O)cs3)C2)nc2ccc(Cl)cc21 REAL300018775722
Cn1ncnc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775723
CC(C)c1nnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775724
COc1cncc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1C REAL300018775725
CC(CN1CCCC(c2nc(C(=O)O)cs2)C1)c1ccc(F)cc1 REAL300018775726
O=C(O)c1csc(C2CCCN(CC3CCS(=O)(=O)CC3)C2)n1 REAL300018775727
O=C(O)c1csc(C2CCCN(Cc3ccc(C(F)(F)F)s3)C2)n1 REAL300018775728
O=C(O)c1csc(C2CCCN(Cc3ccc(OC(F)F)c(F)c3)C2)n1 REAL300018775729
O=C(O)c1csc(C2CCCN(Cc3csc(C(F)(F)F)c3)C2)n1 REAL300018775730
CC1(C)OCc2cc(CN3CCCC(c4nc(C(=O)O)cs4)C3)ccc2O1 REAL300018775731
O=C(O)c1csc(C2CCCN(CC3Cc4ccccc4C3)C2)n1 REAL300018775732
O=C(O)c1csc(C2CCCN(Cc3ncc(Br)s3)C2)n1 REAL300018775733
O=C(O)c1csc(C2CCCN(Cc3cc(F)ncc3F)C2)n1 REAL300018775734
Cc1cc(C(F)(F)F)ccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775735
Cn1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(C(F)F)n1 REAL300018775736
O=C(O)c1csc(C2CCCN(Cc3ncc(C(F)(F)F)s3)C2)n1 REAL300018775737
CCOC(=O)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)o1 REAL300018775738
O=C(O)c1csc(C2CCCN(CCCC3CCCCC3)C2)n1 REAL300018775739
Cc1ccc(CCN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775740
COc1ccc(-n2cc(CN3CCCC(c4nc(C(=O)O)cs4)C3)cn2)cc1 REAL300018775741
Cc1noc2ncc(CN3CCCC(c4nc(C(=O)O)cs4)C3)cc12 REAL300018775742
CC(CN1CCCC(c2nc(C(=O)O)cs2)C1)c1ccc(C(F)(F)F)cc1 REAL300018775743
CCc1cnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775744
O=C(O)c1csc(C2CCCN(CC3CCSC3)C2)n1 REAL300018775745
Cc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(C)o1 REAL300018775746
O=C(O)c1csc(C2CCCN(Cc3cnc(-c4ccco4)s3)C2)n1 REAL300018775747
CC(C)(C)c1ccc(CCN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775748
O=C(O)c1csc(C2CCCN(CCCc3c(Cl)cccc3Cl)C2)n1 REAL300018775749
O=C(O)c1csc(C2CCCN(CC3CCOc4ccccc43)C2)n1 REAL300018775750
CC1CCC(CN2CCCC(c3nc(C(=O)O)cs3)C2)CC1 REAL300018775751
CC(C)CC(C)CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775752
CCC1CCCC(CN2CCCC(c3nc(C(=O)O)cs3)C2)C1 REAL300018775753
Cc1ccc(CCCN2CCCC(c3nc(C(=O)O)cs3)C2)cn1 REAL300018775754
O=C(O)c1csc(C2CCCN(CCC3CCCCCC3)C2)n1 REAL300018775755
COCOc1ccc(OC)cc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775756
CC1CCCCC1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775757
O=C(O)c1csc(C2CCCN(Cc3cc4c(Cl)nccc4o3)C2)n1 REAL300018775758
NC(=O)Cn1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)nn1 REAL300018775759
Cc1ccccc1-n1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)nn1 REAL300018775760
CCSc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775761
O=C(O)c1csc(C2CCCN(Cc3cnnn3-c3ccccc3)C2)n1 REAL300018775762
O=C(O)c1csc(C2CCCN(Cc3cc4ccnc(Cl)c4s3)C2)n1 REAL300018775763
O=C(O)c1csc(C2CCCN(Cc3cc(C4CC4)no3)C2)n1 REAL300018775764
O=C(O)c1csc(C2CCCN(CC3C4CC5CC(C4)CC3C5)C2)n1 REAL300018775765
O=C(O)c1csc(C2CCCN(CC3CC3(Cl)Cl)C2)n1 REAL300018775766
Cn1c(Cl)cnc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775767
CC(C)OC(CN1CCCC(c2nc(C(=O)O)cs2)C1)c1ccccc1 REAL300018775768
CC(C)N(C)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cn1 REAL300018775769
COCCN(C)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cn1 REAL300018775770
Cn1nc2c(c1CN1CCCC(c3nc(C(=O)O)cs3)C1)CCCC2 REAL300018775771
O=C(O)c1csc(C2CCCN(Cc3scnc3C3CC3)C2)n1 REAL300018775772
Cc1c[nH]nc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775773
CN(C)Cc1cnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775774
O=C(O)c1csc(C2CCCN(Cc3ccsc3C(F)(F)F)C2)n1 REAL300018775775
O=C(O)c1csc(C2CCCN(C[C@@H]3C[C@H]3c3ccccc3)C2)n1 REAL300018775776
CC(C)(C)n1nnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1 REAL300018775777
O=C(O)c1csc(C2CCCN(CC=Cc3ccc(F)cc3)C2)n1 REAL300018775778
O=C(O)c1csc(C2CCCN(Cc3cccc4c3NCCC4)C2)n1 REAL300018775779
CC(=Cc1cccc([N+](=O)[O-])c1)CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775780
Cn1cc(-c2csc(CN3CCCC(c4nc(C(=O)O)cs4)C3)n2)cn1 REAL300018775781
O=C(O)c1csc(C2CCCN(Cc3ccncc3[N+](=O)[O-])C2)n1 REAL300018775782
O=C(O)c1csc(C2CCCN(CCC3CCOCC3)C2)n1 REAL300018775783
O=C(O)c1csc(C2CCCN(CC3CCC4(CC3)OCCO4)C2)n1 REAL300018775784
COc1ccc2nc(CN3CCCC(c4nc(C(=O)O)cs4)C3)sc2c1 REAL300018775785
CCc1cccc(Cl)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775786
Cn1c(=O)sc2cc(CN3CCCC(c4nc(C(=O)O)cs4)C3)ccc21 REAL300018775787
COC(=O)C1C(CN2CCCC(c3nc(C(=O)O)cs3)C2)C1(F)F REAL300018775788
O=C(O)c1csc(C2CCCN(Cc3ccsc3Cl)C2)n1 REAL300018775789
CCN(C)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cn1 REAL300018775790
COC1(CN2CCCC(c3nc(C(=O)O)cs3)C2)CCCC1 REAL300018775791
COC1(CN2CCCC(c3nc(C(=O)O)cs3)C2)CCCCC1 REAL300018775792
O=C(O)c1csc(C2CCCN(Cc3ccc(OCC4CC4)cc3)C2)n1 REAL300018775793
O=C(O)c1csc(C2CCCN(Cc3c(O)ccc(Cl)c3F)C2)n1 REAL300018775794
O=C(O)c1csc(C2CCCN(Cc3n[nH]cc3-c3ccccc3)C2)n1 REAL300018775795
O=C(O)c1csc(C2CCCN(Cc3cc4ccc(F)cc4[nH]3)C2)n1 REAL300018775796
COCC(C)(C)CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775797
O=C(O)c1csc(C2CCCN(Cc3cnc(C4OCCO4)s3)C2)n1 REAL300018775798
O=C(O)c1csc(C2CCCN(Cc3nc4ccc(F)cc4s3)C2)n1 REAL300018775799
O=C(O)c1csc(C2CCCN(Cc3ccc(F)c(Cl)c3Cl)C2)n1 REAL300018775800
O=C(O)c1csc(C2CCCN(Cc3csc(Cl)c3Cl)C2)n1 REAL300018775801
CC(CCC#N)CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775802
O=C(O)c1csc(C2CCCN(CCc3ccc(F)cc3Cl)C2)n1 REAL300018775803
Cc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)ccc1C#N REAL300018775804
O=C(O)c1csc(C2CCCN(Cc3cnc(C(F)(F)F)s3)C2)n1 REAL300018775805
COc1c([N+](=O)[O-])ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1O REAL300018775806
CC(O)c1ncc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775807
O=C(O)c1csc(C2CCCN(Cc3ncc(C4OCCO4)s3)C2)n1 REAL300018775808
Cn1nc(Br)cc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775809
CCOc1c(Cl)cccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775810
CCCCCCCCCC(C)CCN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775811
Cc1nc(F)ccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775812
O=C(O)c1csc(C2CCCN(Cc3sccc3Cl)C2)n1 REAL300018775813
O=C(O)c1csc(C2CCCN(Cc3ccc4cnccc4c3)C2)n1 REAL300018775814
CCOc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1F REAL300018775815
O=C(O)c1csc(C2CCCN(Cc3cc4ccccc4[nH]3)C2)n1 REAL300018775816
O=C(O)c1csc(C2CCCN(CC3(C(F)F)CC3)C2)n1 REAL300018775817
O=C(O)c1csc(C2CCCN(Cc3ccnn3-c3ccccc3)C2)n1 REAL300018775818
CC(C)(C)c1cnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775819
Cc1nn(C)c(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1Br REAL300018775820
O=C(O)c1csc(C2CCCN(CC3(c4ccccc4)CCOC3)C2)n1 REAL300018775821
CSc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775822
O=C(O)c1csc(C2CCCN(Cc3ccc(OCCCCl)cc3)C2)n1 REAL300018775823
Cn1cc(-c2ccc(CN3CCCC(c4nc(C(=O)O)cs4)C3)cc2)cn1 REAL300018775824
O=C(O)c1csc(C2CCCN(Cc3c(F)cccc3Br)C2)n1 REAL300018775825
O=C(O)c1csc(C2CCCN(Cc3c(F)ccc(O)c3F)C2)n1 REAL300018775826
O=C(O)c1csc(C2CCCN(Cc3ccc(C(F)F)cc3)C2)n1 REAL300018775827
O=C(O)c1csc(C2CCCN(CC(c3ccccc3)c3ccccc3)C2)n1 REAL300018775828
CCOc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1OC REAL300018775829
O=C(O)c1csc(C2CCCN(Cc3ccc(-n4cccn4)cc3)C2)n1 REAL300018775830
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(C)c1 REAL300018775831
Cc1ccc(C)c(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775832
O=C(O)c1csc(C2CCCN(Cc3ccc4ncccc4c3)C2)n1 REAL300018775833
CC(C)(C)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775834
COc1cc(OC)c(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(OC)c1 REAL300018775835
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)ccc1OC(F)F REAL300018775836
CCOc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)ccc1OC REAL300018775837
CCCCCOc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775838
CCCc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775839
Cc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1C REAL300018775840
CC(C)Oc1ccccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775841
C=CCOc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1OC REAL300018775842
CN(CCC#N)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775843
CCCOc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775844
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)ccc1OC(C)C REAL300018775845
CCc1cccc(F)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775846
CC(C)C(CN1CCCC(c2nc(C(=O)O)cs2)C1)c1ccccc1 REAL300018775847
O=C(O)c1csc(C2CCCN(Cc3ccnn3-c3ccc(F)cc3)C2)n1 REAL300018775848
Cc1ccccc1-n1nccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775849
COC(=O)c1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775850
COC(=O)c1ccc(Cl)c(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775851
COc1ccccc1-n1nccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775852
O=C(O)c1csc(C2CCCN(CC3CCC(c4ccccc4)CC3)C2)n1 REAL300018775853
Cc1nn(C(C)C)cc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775854
C[C@H](CN1CCCC(c2nc(C(=O)O)cs2)C1)NC(=O)OC(C)(C)C REAL300018775855
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc(OC)c1O REAL300018775856
Cc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc(C)c1O REAL300018775857
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)ccc1C#N REAL300018775858
COC(=O)c1[nH]c(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1C REAL300018775859
CCc1cc(OC)ccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775860
CSC1(CN2CCCC(c3nc(C(=O)O)cs3)C2)CC1 REAL300018775861
CSC1(CN2CCCC(c3nc(C(=O)O)cs3)C2)CCC1 REAL300018775862
COC(=O)c1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n(C)c1C REAL300018775863
CCc1oc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1C(=O)OC REAL300018775864
Cn1cc(-c2ccc(CN3CCCC(c4nc(C(=O)O)cs4)C3)s2)cn1 REAL300018775865
Cc1nn(-c2ccccn2)c(C)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775866
COCCCn1nccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775867
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(-c2ccnn2C)c1 REAL300018775868
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(-c2cnn(C)c2)c1 REAL300018775869
Cc1cnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1C REAL300018775870
CC(C)C(CN1CCCC(c2nc(C(=O)O)cs2)C1)C(C)C REAL300018775871
COc1cccc(OC)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775872
Cn1nnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1 REAL300018775873
O=C(O)c1csc(C2CCCN(CC=Cc3ccc(F)c(F)c3)C2)n1 REAL300018775874
O=C(O)c1csc(C2CCCN(Cc3cscc3Br)C2)n1 REAL300018775875
CCOC(=O)c1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)[nH]c1C REAL300018775876
O=C(O)c1csc(C2CCCN(C[C@@H]3C[C@H]3c3ccccc3)C2)n1 REAL300018775877
O=C(O)c1csc(C2CCCN(CCc3ccc(Cl)cc3)C2)n1 REAL300018775878
CC(C)C1CCC(CN2CCCC(c3nc(C(=O)O)cs3)C2)CC1 REAL300018775879
CC(C)n1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)nn1 REAL300018775880
CN(C)Cc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)no1 REAL300018775881
CN(C)c1ncccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775882
O=C(O)c1csc(C2CCCN(Cc3cnccn3)C2)n1 REAL300018775883
CC(C)(C)OC(=O)NCC1(CN2CCCC(c3nc(C(=O)O)cs3)C2)CC1 REAL300018775884
CCOC(=O)CC(C)(C)CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775885
COCCOCc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775886
N#Cc1c(F)cccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775887
O=C(O)c1csc(C2CCCN(Cc3ccc4ccccc4c3)C2)n1 REAL300018775888
O=C(O)c1csc(C2CCCN(Cc3cc(Br)ccc3F)C2)n1 REAL300018775889
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc(OC)c1 REAL300018775890
COc1ccc2cc(CN3CCCC(c4nc(C(=O)O)cs4)C3)ccc2c1 REAL300018775891
COc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1OC(F)F REAL300018775892
O=C(O)c1csc(C2CCCN(Cc3ccccc3N3CCCC3)C2)n1 REAL300018775893
O=C(O)c1csc(C2CCCN(Cc3c(F)cccc3N3CCCC3)C2)n1 REAL300018775894
O=C(O)c1csc(C2CCCN(Cc3ccc(F)c(Br)c3)C2)n1 REAL300018775895
O=C(O)c1csc(C2CCCN(Cc3ccc(N4CCCCC4)cc3)C2)n1 REAL300018775896
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc(Cl)c1OC REAL300018775897
CCOc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1OC REAL300018775898
CCCOc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)ccc1OC REAL300018775899
C=CCOc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775900
COc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1OC(C)C REAL300018775901
C#CCOc1ccccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775902
COc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1OC(F)F REAL300018775903
Cc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc(C)c1OC(F)F REAL300018775904
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc2c1OCCO2 REAL300018775905
Cc1cc(C)c(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1C REAL300018775906
O=C(O)c1csc(C2CCCN(Cc3cc(-c4ccccn4)n[nH]3)C2)n1 REAL300018775907
O=C(O)c1csc(C2CCCN(Cc3ccc4[nH]ccc4c3)C2)n1 REAL300018775908
O=C(O)c1csc(C2CCCN(Cc3cc(O)cc(C(F)(F)F)c3)C2)n1 REAL300018775909
O=C(O)c1csc(C2CCCN(Cc3cscc3C(F)(F)F)C2)n1 REAL300018775910
COc1ncc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775911
O=C(O)c1csc(C2CCCN(Cc3ccc(C4CCCC4)cc3)C2)n1 REAL300018775912
Cc1nc(C)c(CN2CCCC(c3nc(C(=O)O)cs3)C2)o1 REAL300018775913
CCOC(=O)c1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)on1 REAL300018775914
O=C(O)c1csc(C2CCCN(CCc3ccc([N+](=O)[O-])cc3)C2)n1 REAL300018775915
CC1(CN2CCCC(c3nc(C(=O)O)cs3)C2)CCCS1 REAL300018775916
O=C(O)c1csc(C2CCCN(Cc3ccc4c(c3)CCCC4)C2)n1 REAL300018775917
Cc1nnsc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775918
O=C(O)c1csc(C2CCCN(Cc3cnn(CC(F)F)c3)C2)n1 REAL300018775919
COCc1ccccc1C=C(C)CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775920
Cn1nccc1-c1ccccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775921
COC(=O)c1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)on1 REAL300018775922
O=C(O)c1csc(C2CCCN(Cc3conc3Cc3ccccc3)C2)n1 REAL300018775923
CCc1nocc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775924
Cn1ncc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1 REAL300018775925
CC(C)(C)OC(=O)N1CCC[C@@H]1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775926
CC(CN1CCCC(c2nc(C(=O)O)cs2)C1)C1CCCCC1 REAL300018775927
COC(=O)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1C REAL300018775928
CSC(C)(C)CCN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775929
COC(C)(CN1CCCC(c2nc(C(=O)O)cs2)C1)C1CC1 REAL300018775930
O=C(O)c1csc(C2CCCN(Cc3ccc4ccc(F)c(F)c4n3)C2)n1 REAL300018775931
O=C(O)c1csc(C2CCCN(Cc3ccc(C4CCC4)cc3)C2)n1 REAL300018775932
O=C(O)c1csc(C2CCCN(Cc3cccc(O)c3Cl)C2)n1 REAL300018775933
Cc1sccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775934
Cc1cc(Cl)cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775935
O=C(O)c1csc(C2CCCN(Cc3cc(Cl)c(F)cc3O)C2)n1 REAL300018775936
CSCc1cnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775937
O=C(O)c1csc(C2CCCN(Cc3ccc(F)cc3O)C2)n1 REAL300018775938
COC(CN1CCCC(c2nc(C(=O)O)cs2)C1)C1CCOCC1 REAL300018775939
O=C(O)c1csc(C2CCCN(Cc3cc4cccnc4o3)C2)n1 REAL300018775940
CC(CN1CCCC(c2nc(C(=O)O)cs2)C1)c1cc(F)cc(F)c1 REAL300018775941
COc1cccc2c(CN3CCCC(c4nc(C(=O)O)cs4)C3)cccc12 REAL300018775942
COc1nccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)n1 REAL300018775943
Cc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cs1 REAL300018775944
Cc1cnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)o1 REAL300018775945
COc1cccc(C)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775946
O=C(O)c1csc(C2CCCN(Cc3nc(Cl)cs3)C2)n1 REAL300018775947
CC(C)(CNC(=O)OC(C)(C)C)CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775948
CCC(C)C(CN1CCCC(c2nc(C(=O)O)cs2)C1)OC REAL300018775949
O=C(O)c1csc(C2CCCN(Cc3cccc(F)c3Br)C2)n1 REAL300018775950
COc1cc2ccccc2cc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775951
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc2ccccc12 REAL300018775952
Cc1cnc(CN2CCCC(c3nc(C(=O)O)cs3)C2)s1 REAL300018775953
COC(=O)Cn1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)nn1 REAL300018775954
Cc1cccc(O)c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775955
Cc1cnccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775956
Cc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1F REAL300018775957
O=C(O)c1csc(C2CCCN(Cc3ccnc(Cl)c3F)C2)n1 REAL300018775958
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc2c1OCO2 REAL300018775959
O=C(O)c1csc(C2CCCN(Cc3ccc(-n4ccnc4)cc3)C2)n1 REAL300018775960
O=C(O)c1csc(C2CCCN(Cc3cc(Cl)c4c(c3)OCCO4)C2)n1 REAL300018775961
O=C(O)c1csc(C2CCCN(Cc3ccccc3)C2)n1 REAL300018775962
O=C(O)c1csc(C2CCCN(Cc3ccccc3Cl)C2)n1 REAL300018775963
O=C(O)c1csc(C2CCCN(Cc3cccc4ccccc34)C2)n1 REAL300018775964
CN(C)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775965
CCN(CC)c1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775966
O=C(O)c1csc(C2CCCN(Cc3ccc(Br)cc3)C2)n1 REAL300018775967
O=C(O)c1csc(C2CCCN(Cc3ccc(Cl)cc3)C2)n1 REAL300018775968
COc1cc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc(OC)c1OC REAL300018775969
O=C(O)c1csc(C2CCCN(Cc3c(F)cccc3Cl)C2)n1 REAL300018775970
O=C(O)c1csc(C2CCCN(Cc3ccc(F)cc3)C2)n1 REAL300018775971
O=C(O)c1csc(C2CCCN(Cc3ccccc3OC(F)F)C2)n1 REAL300018775972
COc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1OC REAL300018775973
COc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775974
COc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(OC)c1 REAL300018775975
O=C(O)c1csc(C2CCCN(Cc3ccc(F)cc3F)C2)n1 REAL300018775976
O=C(O)c1csc(C2CCCN(Cc3ccc(Cl)c(Cl)c3)C2)n1 REAL300018775977
O=C(O)c1csc(C2CCCN(Cc3ccc(OC(F)F)cc3)C2)n1 REAL300018775978
CCCCOc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775979
CC(C)CCOc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775980
O=C(O)c1csc(C2CCCN(Cc3cccc(Oc4ccccc4)c3)C2)n1 REAL300018775981
O=C(O)c1csc(C2CCCN(Cc3cccc(Cl)c3)C2)n1 REAL300018775982
COc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775983
O=C(O)c1csc(C2CCCN(Cc3cccc(C(F)(F)F)c3)C2)n1 REAL300018775984
COc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(OC)c1OC REAL300018775985
CCOc1ccccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775986
CCOc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775987
O=C(O)c1csc(C2CCCN(Cc3cccc(F)c3)C2)n1 REAL300018775988
O=C(O)c1csc(C2CCCN(Cc3cccc(O)c3)C2)n1 REAL300018775989
COc1ccccc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775990
O=C(O)c1csc(C2CCCN(Cc3ccc(-c4ccccc4)cc3)C2)n1 REAL300018775991
COc1ccc2ccccc2c1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775992
Cc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775993
CSc1ccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)cc1 REAL300018775994
O=C(O)c1csc(C2CCCN(Cc3c(Cl)cccc3Cl)C2)n1 REAL300018775995
COc1cc(OC)c(OC)cc1CN1CCCC(c2nc(C(=O)O)cs2)C1 REAL300018775996
Cc1cccc(CN2CCCC(c3nc(C(=O)O)cs3)C2)c1 REAL300018775997
Cc1cc(C)c(CN2CCCC(c3nc(C(=O)O)cs3)C2)c(C)c1 REAL300018775998
O=C(O)c1csc(C2CCCN(Cc3c(F)cccc3F)C2)n1 REAL300018775999
O=C(O)c1csc(C2CCCN(Cc3ccc(F)c(F)c3)C2)n1 REAL300018776000
