O=C(O)Cc1csc(C2CCN(Cc3cnnn3C3CC3)CC2)n1 REAL300018778001
COCc1ccccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778002
O=C(O)Cc1csc(C2CCN(Cc3ccc4c(c3)COCC4)CC2)n1 REAL300018778003
O=C(O)Cc1csc(C2CCN(Cc3cnn(CCO)c3)CC2)n1 REAL300018778004
O=C(O)Cc1csc(C2CCN(Cc3cc(-c4ccncc4)n[nH]3)CC2)n1 REAL300018778005
COc1ccc(F)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1OC REAL300018778006
O=C(O)Cc1csc(C2CCN(CC=Cc3ccncc3)CC2)n1 REAL300018778007
Cn1ccc(-c2n[nH]cc2CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778008
C=Cc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc1 REAL300018778009
CC(F)(F)c1ccccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778010
CCn1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c(C2CC2)n1 REAL300018778011
CCc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)nc1 REAL300018778012
COc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)nn1 REAL300018778013
CC(C)(C)c1nocc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778014
O=C(O)Cc1csc(C2CCN(Cc3ccc4ccncc4c3)CC2)n1 REAL300018778015
Cc1cc2cccc(CN3CCC(c4nc(CC(=O)O)cs4)CC3)c2o1 REAL300018778016
COc1csc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1OC REAL300018778017
O=C(O)Cc1csc(C2CCN(Cc3conc3C3CCC3)CC2)n1 REAL300018778018
Cn1c(=O)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc2ccccc21 REAL300018778019
Cc1cccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778020
O=C(O)Cc1csc(C2CCN(Cc3ccc(-c4ccsc4)cc3)CC2)n1 REAL300018778021
O=C(O)Cc1csc(C2CCN(Cc3nc4ccccc4s3)CC2)n1 REAL300018778022
O=C(O)Cc1csc(C2CCN(Cc3[nH]ncc3Br)CC2)n1 REAL300018778023
O=C(O)Cc1csc(C2CCN(Cc3ccc4nsnc4c3)CC2)n1 REAL300018778024
O=C(O)Cc1csc(C2CCN(Cc3ccc4nonc4c3)CC2)n1 REAL300018778025
O=C(O)Cc1csc(C2CCN(Cc3cccc4nsnc34)CC2)n1 REAL300018778026
CCn1cnc(Cl)c1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778027
N#Cc1cnn2cc(CN3CCC(c4nc(CC(=O)O)cs4)CC3)cnc12 REAL300018778028
O=C(O)Cc1csc(C2CCN(Cc3cn(-c4ccccc4)nn3)CC2)n1 REAL300018778029
CCOc1ccc(Cl)cc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778030
Cn1nc(-c2ccccc2)cc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778031
CC(C)(C)c1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n[nH]1 REAL300018778032
CCN1CCCc2cc(CN3CCC(c4nc(CC(=O)O)cs4)CC3)ccc21 REAL300018778033
O=C(O)Cc1csc(C2CCN(Cc3ccc(-c4ccsc4)nc3)CC2)n1 REAL300018778034
O=C(O)Cc1csc(C2CCN(Cc3cc4ccccc4cn3)CC2)n1 REAL300018778035
Cc1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc(Cl)n1 REAL300018778036
Cc1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc(C)n1 REAL300018778037
COc1cc(C)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cn1 REAL300018778038
O=C(O)Cc1csc(C2CCN(Cc3ccc[nH]c3=O)CC2)n1 REAL300018778039
CCc1c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cnn1CC REAL300018778040
Cn1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c(C(F)(F)F)n1 REAL300018778041
O=C(O)Cc1csc(C2CCN(Cc3noc4c3CCCC4)CC2)n1 REAL300018778042
Cc1cn(C)nc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778043
Cc1coc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778044
O=C(O)Cc1csc(C2CCN(Cc3cc4ccncc4s3)CC2)n1 REAL300018778045
COc1nc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)ccc1C REAL300018778046
O=C(O)Cc1csc(C2CCN(Cc3cc4ncccc4o3)CC2)n1 REAL300018778047
CCC(C)n1nccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778048
O=C(O)Cc1csc(C2CCN(Cc3nc(CO)cs3)CC2)n1 REAL300018778049
CCCn1cncc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778050
CCc1c[nH]c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778051
O=C(O)Cc1csc(C2CCN(Cc3cncc(-c4cccnc4)c3)CC2)n1 REAL300018778052
CC(C)(C)c1cncc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1 REAL300018778053
COc1nc(Cl)ccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778054
Cc1c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)ccnc1F REAL300018778055
O=C(O)Cc1csc(C2CCN(Cc3ccc4c(c3)CCOC4)CC2)n1 REAL300018778056
O=C(O)Cc1csc(C2CCN(Cc3cccc(C(F)F)c3F)CC2)n1 REAL300018778057
Cc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c(C)n1 REAL300018778058
O=C(O)Cc1csc(C2CCN(Cc3nc4c(s3)CCCCC4)CC2)n1 REAL300018778059
O=C(O)Cc1csc(C2CCN(Cc3nc4c(s3)COCC4)CC2)n1 REAL300018778060
CC(C)Cc1ccccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778061
CSc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)o1 REAL300018778062
O=C(O)Cc1csc(C2CCN(Cc3cnn(C4CCCCC4)c3)CC2)n1 REAL300018778063
CCCn1nc(C)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1Cl REAL300018778064
Cn1cc(-c2n[nH]cc2CN2CCC(c3nc(CC(=O)O)cs3)CC2)cn1 REAL300018778065
CC(C)n1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778066
O=C(O)Cc1csc(C2CCN(Cc3ccn(CC(F)(F)F)n3)CC2)n1 REAL300018778067
CC(F)(F)c1cccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1 REAL300018778068
Cc1cc(O)ncc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778069
Cc1nc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)oc1C REAL300018778070
CS(=O)(=O)c1coc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1 REAL300018778071
O=C(O)Cc1csc(C2CCN(Cc3cn(CC4CC4)nn3)CC2)n1 REAL300018778072
O=C(O)Cc1csc(C2CCN(Cc3cccn3C(F)F)CC2)n1 REAL300018778073
O=C(O)Cc1csc(C2CCN(Cc3cc4c(o3)CCCC4)CC2)n1 REAL300018778074
Cn1cc(Br)nc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778075
C=CCc1ccccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778076
COc1nn(C)cc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778077
CC(C)(C)n1nccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778078
CN(CCO)c1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cn1 REAL300018778079
Cn1c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)nc2c1CCCC2 REAL300018778080
O=C(O)Cc1csc(C2CCN(Cc3cccc4c3COCC4)CC2)n1 REAL300018778081
O=C(O)Cc1csc(C2CCN(Cc3ccccc3C3CCC3)CC2)n1 REAL300018778082
CC(C)(C#N)c1ncc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)s1 REAL300018778083
CCn1nc(C)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778084
COc1sccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778085
O=C(O)Cc1csc(C2CCN(Cc3cc(C4CCC4)[nH]n3)CC2)n1 REAL300018778086
C=CCCn1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)nn1 REAL300018778087
O=C(O)Cc1csc(C2CCN(Cc3ccc(CC4CCC4)cc3)CC2)n1 REAL300018778088
COc1nsc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1Cl REAL300018778089
O=C(O)Cc1csc(C2CCN(Cc3cn(C4CC4)cn3)CC2)n1 REAL300018778090
CC(C)c1cnn(C)c1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778091
Cn1nnc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1C(F)F REAL300018778092
Cn1ncc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1S(C)(=O)=O REAL300018778093
Cc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc1OC(F)F REAL300018778094
CC1Oc2ccc(CN3CCC(c4nc(CC(=O)O)cs4)CC3)cc2C1C REAL300018778095
O=C(O)Cc1csc(C2CCN(Cc3ccccc3-n3cccn3)CC2)n1 REAL300018778096
O=C(O)Cc1csc(C2CCN(Cc3ccnn3C3CC3(F)F)CC2)n1 REAL300018778097
COCc1nocc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778098
COCc1cnc(OC)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1 REAL300018778099
O=C(O)Cc1csc(C2CCN(Cc3ccc(C(F)F)cn3)CC2)n1 REAL300018778100
CC(C)Oc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc1F REAL300018778101
CCn1cc(Cl)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778102
O=C(O)Cc1csc(C2CCN(Cc3ccc(F)c(Cl)c3F)CC2)n1 REAL300018778103
O=C(O)Cc1csc(C2CCN(Cc3cccc(C(F)F)c3)CC2)n1 REAL300018778104
O=C(O)Cc1csc(C2CCN(Cc3ccc4ccccc4c3F)CC2)n1 REAL300018778105
O=C(O)Cc1csc(C2CCN(Cc3csc(Cl)c3)CC2)n1 REAL300018778106
Cc1c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cnn1C1CCC1 REAL300018778107
Cc1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n(C2CCCC2)n1 REAL300018778108
O=C(O)Cc1csc(C2CCN(Cc3ccnn3CC(F)F)CC2)n1 REAL300018778109
COc1ccc(C)nc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778110
O=C(O)Cc1csc(C2CCN(Cc3cc(Cl)cc(Cl)n3)CC2)n1 REAL300018778111
O=C(O)Cc1csc(C2CCN(Cc3cc4cnccc4[nH]3)CC2)n1 REAL300018778112
O=C(O)Cc1csc(C2CCN(Cc3c(F)ccnc3Cl)CC2)n1 REAL300018778113
O=C(O)Cc1csc(C2CCN(Cc3cccc(C(F)F)n3)CC2)n1 REAL300018778114
CN(C)c1cncc(F)c1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778115
O=C(O)Cc1csc(C2CCN(Cc3c(O)ccc4c3OCO4)CC2)n1 REAL300018778116
Cc1nn(-c2ccccc2)nc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778117
O=C(O)Cc1csc(C2CCN(Cc3ccn(C4CCC4)n3)CC2)n1 REAL300018778118
O=C(O)Cc1csc(C2CCN(Cc3ccn(CC(F)F)n3)CC2)n1 REAL300018778119
O=C(O)Cc1csc(C2CCN(Cc3ccn(C4CC4(F)F)n3)CC2)n1 REAL300018778120
O=C(O)Cc1csc(C2CCN(Cc3cnn(C4CCOCC4)c3)CC2)n1 REAL300018778121
Cc1cn(C)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778122
O=C(O)Cc1csc(C2CCN(Cc3noc4c3CCC4)CC2)n1 REAL300018778123
O=C(O)Cc1csc(C2CCN(Cc3nc4cccc(F)c4s3)CC2)n1 REAL300018778124
O=C(O)Cc1csc(C2CCN(Cc3ccn(C4CCCC4)n3)CC2)n1 REAL300018778125
O=C(O)Cc1csc(C2CCN(Cc3ccc(F)c4ccoc34)CC2)n1 REAL300018778126
O=C(O)Cc1csc(C2CCN(Cc3cc(Cl)cc4ccoc34)CC2)n1 REAL300018778127
O=C(O)Cc1csc(C2CCN(Cc3ncc(Cl)cc3Cl)CC2)n1 REAL300018778128
Cc1nn(C2CCCC2)cc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778129
O=C(O)Cc1csc(C2CCN(Cc3ccccc3C(F)F)CC2)n1 REAL300018778130
O=C(O)Cc1csc(C2CCN(Cc3ccc4[nH]ncc4c3)CC2)n1 REAL300018778131
O=C(O)Cc1csc(C2CCN(Cc3ccc(Cl)c(F)c3F)CC2)n1 REAL300018778132
Cc1c(F)cccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778133
Cn1cc(-c2cccc(CN3CCC(c4nc(CC(=O)O)cs4)CC3)c2)cn1 REAL300018778134
COc1c(C#N)cccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778135
O=C(O)Cc1csc(C2CCN(Cc3ccnc(Br)c3)CC2)n1 REAL300018778136
Cc1nc(Cl)ccc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778137
COc1cc(Cl)cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1 REAL300018778138
COc1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc(F)c1F REAL300018778139
COc1cc(C)ncc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778140
CC(C)n1cnc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1 REAL300018778141
Cc1c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)nnn1C REAL300018778142
Cn1nccc1-c1n[nH]cc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778143
Cc1onc(C2CC2)c1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778144
COC(=O)c1c(C)[nH]c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1C REAL300018778145
CC(C)Oc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)o1 REAL300018778146
Cc1oc(-c2ccccc2)nc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778147
Cn1nc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc1-c1ccco1 REAL300018778148
O=C(O)Cc1csc(C2CCN(Cc3c(Cl)ccc4c3OCO4)CC2)n1 REAL300018778149
N#Cc1cc(F)cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1 REAL300018778150
O=C(O)Cc1csc(C2CCN(Cc3ccc(C4CCCCC4)cc3)CC2)n1 REAL300018778151
Cc1nc(C)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)nc1C REAL300018778152
NC(=O)c1cnc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cn1 REAL300018778153
Cc1nn(C2CCC2)cc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778154
Cc1c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cnn1CC(F)F REAL300018778155
COc1ccccc1C=CCN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778156
O=C(O)Cc1csc(C2CCN(Cc3ccc(-c4ccccn4)nc3)CC2)n1 REAL300018778157
CCCn1nc(C)c(Cl)c1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778158
COc1cccc2[nH]c(CN3CCC(c4nc(CC(=O)O)cs4)CC3)cc12 REAL300018778159
Cc1ccc(OC(F)F)c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778160
Cn1nc(-c2ccco2)cc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778161
COc1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c(C)n1 REAL300018778162
CCN(C)c1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c(C)c1 REAL300018778163
O=C(O)Cc1csc(C2CCN(Cc3cc(-c4ccccc4)ccn3)CC2)n1 REAL300018778164
O=C(O)Cc1csc(C2CCN(Cc3scc(Cl)c3Cl)CC2)n1 REAL300018778165
COc1cc(C)cc(OC)c1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778166
O=C(O)Cc1csc(C2CCN(Cc3ccc(CF)cc3)CC2)n1 REAL300018778167
O=C(O)Cc1csc(C2CCN(Cc3ccc4sccc4c3)CC2)n1 REAL300018778168
O=C(O)Cc1csc(C2CCN(Cc3ccc(-c4ccncc4)cc3)CC2)n1 REAL300018778169
O=C(O)Cc1csc(C2CCN(Cc3ccccc3CO)CC2)n1 REAL300018778170
CC(C)(C)c1oncc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778171
Cc1cncc(C)c1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778172
COc1cc(C)c2cc(CN3CCC(c4nc(CC(=O)O)cs4)CC3)[nH]c2c1 REAL300018778173
Cc1cccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1C(F)(F)F REAL300018778174
C=CCn1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cn1 REAL300018778175
O=C(O)Cc1csc(C2CCN(Cc3ccc4cn[nH]c4c3)CC2)n1 REAL300018778176
CCC(C)c1ccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cc1 REAL300018778177
Cc1oncc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778178
CC(F)(F)c1cccc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n1 REAL300018778179
O=C(O)Cc1csc(C2CCN(Cc3cc4sccc4[nH]3)CC2)n1 REAL300018778180
O=C(O)Cc1csc(C2CCN(Cc3cccc4c3CCCC4)CC2)n1 REAL300018778181
CC(=Cc1cc(F)cc(F)c1)CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778182
O=C(O)Cc1csc(C2CCN(Cc3ccc(-n4ccnn4)cc3)CC2)n1 REAL300018778183
Cc1c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)ccc2ccccc12 REAL300018778184
COc1c(CN2CCC(c3nc(CC(=O)O)cs3)CC2)ccc2[nH]ccc12 REAL300018778185
Cc1nc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c(C)s1 REAL300018778186
CCCn1ncc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c1C REAL300018778187
Cc1ccc2cccnc2c1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778188
O=C(O)Cc1csc(C2CCN(Cc3c(O)cccc3F)CC2)n1 REAL300018778189
Cc1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)cnc1-n1cccn1 REAL300018778190
COC(=O)c1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)n(C)c1 REAL300018778191
O=C(O)Cc1csc(C2CCN(Cc3cc4sc(Cl)cc4[nH]3)CC2)n1 REAL300018778192
COc1ccn2c(CN3CCC(c4nc(CC(=O)O)cs4)CC3)cnc2c1 REAL300018778193
CCCn1nc(C)cc1CN1CCC(c2nc(CC(=O)O)cs2)CC1 REAL300018778194
Cn1cc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c(C2CCC2)n1 REAL300018778195
CC(C)(C)c1ncc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)o1 REAL300018778196
Cn1nc(CN2CCC(c3nc(CC(=O)O)cs3)CC2)c2c1CCOC2 REAL300018778197
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccnc1)CC2 REAL300018778198
CC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1ccccc1 REAL300018778199
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3c(c1)OCCO3)CC2 REAL300018778200
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1OC REAL300018778201
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CC=CCC1)CC2 REAL300018778202
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1C(F)(F)F)CC2 REAL300018778203
Cc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778204
CCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778205
COC(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778206
CCC(CC)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778207
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCCCC1)CC2 REAL300018778208
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Br)o1)CC2 REAL300018778209
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778210
CC(C)=CCCC(C)CCN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778211
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778212
COC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)oc1C REAL300018778213
Cc1nn(C)c(Cl)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778214
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCC=CO1)CC2 REAL300018778215
CC(CCN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1ccccc1 REAL300018778216
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)c(Cl)c1)CC2 REAL300018778217
CCOc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778218
COc1ccc(F)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778219
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(F)cc(Cl)c1)CC2 REAL300018778220
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)cc1F)CC2 REAL300018778221
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3c1OCO3)CC2 REAL300018778222
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Cl)ccc1F)CC2 REAL300018778223
COc1ccc(F)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778224
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(F)cc(F)c1)CC2 REAL300018778225
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778226
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3occc3c1)CC2 REAL300018778227
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n(C)n1 REAL300018778228
COC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1C REAL300018778229
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1Cl REAL300018778230
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1csnn1)CC2 REAL300018778231
COc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1C REAL300018778232
Cc1nn(C(C)(C)C)c(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778233
N#Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(F)c1 REAL300018778234
COC(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778235
Cc1nn(C)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778236
CCC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1ccccc1 REAL300018778237
COc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1F REAL300018778238
CN(C)c1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1C REAL300018778239
CC1(C)CCCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)C1 REAL300018778240
CC1=CCCC(C)C1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778241
Cc1cc(Cl)ccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778242
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCC1CCCCC1)CC2 REAL300018778243
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cocn1)CC2 REAL300018778244
CCn1nccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778245
C#Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778246
COc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778247
CCn1cncc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778248
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccncc1F)CC2 REAL300018778249
Cc1ccc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)ccc2n1 REAL300018778250
COc1cc(F)cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778251
CC(C)(C)c1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778252
Cc1occc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778253
Cn1c(=O)oc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)ccc21 REAL300018778254
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCc1cccc(Cl)c1)CC2 REAL300018778255
COc1ccc2oc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cc2c1 REAL300018778256
Cc1ccc(C(C)CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778257
N#Cc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778258
Cn1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778259
CC(C)n1nccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778260
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1coc3ccccc13)CC2 REAL300018778261
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)c1OC REAL300018778262
Cc1ccc2nc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cn2c1 REAL300018778263
Cc1c[nH]c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778264
COc1cc(C)ccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778265
COCc1csc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778266
COCc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)no1 REAL300018778267
O=C1COc2ccc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cc2N1 REAL300018778268
CC(C)n1ccnc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778269
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778270
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnc(Cl)c1Cl)CC2 REAL300018778271
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3cnccn13)CC2 REAL300018778272
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCCc1ccc3c(c1)CCO3)CC2 REAL300018778273
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3c(cn1)OCCO3)CC2 REAL300018778274
Cc1ccc2ncc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)n2c1 REAL300018778275
Cn1c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cnc1Cl REAL300018778276
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(C(F)(F)F)[nH]n1)CC2 REAL300018778277
Cc1nocc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778278
Cc1ncoc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778279
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Cl)cs1)CC2 REAL300018778280
Cc1cnn(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778281
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1Cl REAL300018778282
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nccn1-c1ccccc1)CC2 REAL300018778283
C=Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778284
COc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)sn1 REAL300018778285
CCCc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778286
CC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1cccc(Cl)c1 REAL300018778287
Cn1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1Cl REAL300018778288
Cc1c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cnn1C REAL300018778289
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc(C3CC3)nc1)CC2 REAL300018778290
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc(C3CC3)o1)CC2 REAL300018778291
CCOc1cncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778292
CC(C)(C)n1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778293
Cn1ncnc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778294
CC(C)c1nnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778295
COc1cncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C REAL300018778296
CC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1ccc(F)cc1 REAL300018778297
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCS(=O)(=O)CC1)CC2 REAL300018778298
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C(F)(F)F)s1)CC2 REAL300018778299
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1csc(C(F)(F)F)c1)CC2 REAL300018778300
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1Cc3ccccc3C1)CC2 REAL300018778301
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(F)ncc1F)CC2 REAL300018778302
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C(F)F)n1 REAL300018778303
CCOC(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778304
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCCC1CCCCC1)CC2 REAL300018778305
Cc1ccc(CCN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778306
Cc1noc2ncc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cc12 REAL300018778307
CCc1cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778308
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCSC1)CC2 REAL300018778309
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)o1 REAL300018778310
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc(-c3ccco3)s1)CC2 REAL300018778311
CC(C)(C)c1ccc(CCN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778312
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCOc3ccccc31)CC2 REAL300018778313
CC1CC1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778314
CC1CCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CC1 REAL300018778315
CC(C)CC(C)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778316
CCC1CCCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)C1 REAL300018778317
Cc1ccc(CCCN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778318
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCC1CCCCCC1)CC2 REAL300018778319
CC1CCCCC1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778320
NC(=O)Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778321
CCSc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778322
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnnn1-c1ccccc1)CC2 REAL300018778323
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(C3CC3)no1)CC2 REAL300018778324
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1C3CC4CC(C3)CC1C4)CC2 REAL300018778325
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CC1(Cl)Cl)CC2 REAL300018778326
Cn1c(Cl)cnc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778327
CC(C)OC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1ccccc1 REAL300018778328
CC(C)N(C)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778329
Cn1nc2c(c1CN1CCn3c(C(F)(F)F)nc(C(=O)O)c3C1)CCCC2 REAL300018778330
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1scnc1C1CC1)CC2 REAL300018778331
Cc1c[nH]nc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778332
CN(C)Cc1cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778333
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccsc1C(F)(F)F)CC2 REAL300018778334
O=C(O)c1nc(C(F)(F)F)n2c1CN(C[C@@H]1C[C@H]1c1ccccc1)CC2 REAL300018778335
CC(C)(C)n1nnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778336
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC=Cc1ccc(F)cc1)CC2 REAL300018778337
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3c1NCCC3)CC2 REAL300018778338
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccncc1[N+](=O)[O-])CC2 REAL300018778339
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCC1CCOCC1)CC2 REAL300018778340
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCC3(CC1)OCCO3)CC2 REAL300018778341
CCc1cccc(Cl)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778342
COC(=O)C1C(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)C1(F)F REAL300018778343
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccsc1Cl)CC2 REAL300018778344
CCN(C)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778345
COC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CCCC1 REAL300018778346
COC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CCCCC1 REAL300018778347
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(OCC3CC3)cc1)CC2 REAL300018778348
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(O)ccc(Cl)c1F)CC2 REAL300018778349
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1n[nH]cc1-c1ccccc1)CC2 REAL300018778350
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3ccc(F)cc3[nH]1)CC2 REAL300018778351
COCC(C)(C)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778352
CC(CCC#N)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778353
CC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CCC1 REAL300018778354
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCc1ccc(F)cc1Cl)CC2 REAL300018778355
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1C#N REAL300018778356
CC(O)c1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778357
CC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CC1 REAL300018778358
Cc1nc(F)ccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778359
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1sccc1Cl)CC2 REAL300018778360
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3cnccc3c1)CC2 REAL300018778361
CCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1F REAL300018778362
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3ccccc3[nH]1)CC2 REAL300018778363
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1(C(F)F)CC1)CC2 REAL300018778364
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnn1-c1ccccc1)CC2 REAL300018778365
CC(C)(C)c1cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778366
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1(c3ccccc3)CCOC1)CC2 REAL300018778367
CSc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778368
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1(F)CC1)CC2 REAL300018778369
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(F)ccc(O)c1F)CC2 REAL300018778370
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C(F)F)cc1)CC2 REAL300018778371
CCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1OC REAL300018778372
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(-n3cccn3)cc1)CC2 REAL300018778373
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)c1 REAL300018778374
Cc1ccc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778375
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3ncccc3c1)CC2 REAL300018778376
CC(C)(C)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778377
CCOc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1OC REAL300018778378
CCCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778379
Cc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C REAL300018778380
CC(C)Oc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778381
CCCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778382
CCc1cccc(F)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778383
CC(C)C(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1ccccc1 REAL300018778384
COC(=O)c1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778385
Cc1nn(C(C)C)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778386
C[C@H](CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)NC(=O)OC(C)(C)C REAL300018778387
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc(C)c1O REAL300018778388
COc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1C#N REAL300018778389
COC(=O)c1[nH]c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778390
CCc1cc(OC)ccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778391
CSC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CC1 REAL300018778392
CSC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CCC1 REAL300018778393
COCCCn1nccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778394
Cc1cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1C REAL300018778395
CC(C)C(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)C(C)C REAL300018778396
COc1cccc(OC)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778397
Cn1nnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778398
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC=Cc1ccc(F)c(F)c1)CC2 REAL300018778399
O=C(O)c1nc(C(F)(F)F)n2c1CN(C[C@@H]1C[C@H]1c1ccccc1)CC2 REAL300018778400
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCc1ccc(Cl)cc1)CC2 REAL300018778401
CC(C)C1CCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CC1 REAL300018778402
CC(C)n1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778403
CN(C)Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)no1 REAL300018778404
CN(C)c1ncccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778405
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnccn1)CC2 REAL300018778406
CCOC(=O)CC(C)(C)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778407
N#Cc1c(F)cccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778408
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3ccccc3c1)CC2 REAL300018778409
COc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc(OC)c1 REAL300018778410
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1N1CCCC1)CC2 REAL300018778411
CCOc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1OC REAL300018778412
C=CCOc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778413
C#CCOc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778414
Cc1cc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778415
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(-c3ccccn3)n[nH]1)CC2 REAL300018778416
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3[nH]ccc3c1)CC2 REAL300018778417
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccon1)CC2 REAL300018778418
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cscc1C(F)(F)F)CC2 REAL300018778419
COc1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778420
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C3CCCC3)cc1)CC2 REAL300018778421
Cc1nc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778422
CCOC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)on1 REAL300018778423
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCc1ccc([N+](=O)[O-])cc1)CC2 REAL300018778424
CC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CCCS1 REAL300018778425
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3c(c1)CCCC3)CC2 REAL300018778426
Cc1nnsc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778427
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnn(CC(F)F)c1)CC2 REAL300018778428
COC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)on1 REAL300018778429
CCc1nocc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778430
Cn1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778431
CC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)C1CCCCC1 REAL300018778432
COC(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1C REAL300018778433
CSC(C)(C)CCN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778434
COC(C)(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)C1CC1 REAL300018778435
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C3CCC3)cc1)CC2 REAL300018778436
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(O)c1Cl)CC2 REAL300018778437
Cc1sccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778438
Cc1cc(Cl)cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778439
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Cl)c(F)cc1O)CC2 REAL300018778440
CSCc1cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778441
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)cc1O)CC2 REAL300018778442
COC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)C1CCOCC1 REAL300018778443
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3cccnc3o1)CC2 REAL300018778444
CC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1cc(F)cc(F)c1 REAL300018778445
COc1nccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778446
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cs1 REAL300018778447
Cc1cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778448
COc1cccc(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778449
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nc(Cl)cs1)CC2 REAL300018778450
CCC(C)C(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)OC REAL300018778451
Cc1cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778452
COC(=O)Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778453
Cc1cccc(O)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778454
Cc1cnccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778455
Cc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1F REAL300018778456
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnc(Cl)c1F)CC2 REAL300018778457
COc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc2c1OCO2 REAL300018778458
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(-n3ccnc3)cc1)CC2 REAL300018778459
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1)CC2 REAL300018778460
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1Cl)CC2 REAL300018778461
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3ccccc13)CC2 REAL300018778462
CN(C)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778463
CCN(CC)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778464
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)cc1)CC2 REAL300018778465
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(F)cccc1Cl)CC2 REAL300018778466
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)cc1)CC2 REAL300018778467
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1OC(F)F)CC2 REAL300018778468
COc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1OC REAL300018778469
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778470
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(OC)c1 REAL300018778471
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)cc1F)CC2 REAL300018778472
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)c(Cl)c1)CC2 REAL300018778473
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(OC(F)F)cc1)CC2 REAL300018778474
CCCCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778475
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(Cl)c1)CC2 REAL300018778476
COc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778477
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(C(F)(F)F)c1)CC2 REAL300018778478
CCOc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778479
CCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778480
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(F)c1)CC2 REAL300018778481
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(O)c1)CC2 REAL300018778482
COc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778483
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778484
CSc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778485
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(Cl)cccc1Cl)CC2 REAL300018778486
Cc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778487
Cc1cc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)c1 REAL300018778488
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(F)cccc1F)CC2 REAL300018778489
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)c(F)c1)CC2 REAL300018778490
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1O REAL300018778491
Cc1noc(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778492
Cc1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cs1 REAL300018778493
C#CCCCCCCN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778494
CC(C)(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)Oc1ccccc1 REAL300018778495
COC(Cc1ccccc1)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778496
CCCn1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778497
Cn1nc(C2CC2)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778498
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3ccccc3n1)CC2 REAL300018778499
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3c(n1)CCC3)CC2 REAL300018778500
CCC(C)(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)OC REAL300018778501
CCn1nnc(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778502
Cn1cc(CCCN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778503
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3ccoc13)CC2 REAL300018778504
CC(C)COc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778505
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnn1C1CCCC1)CC2 REAL300018778506
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccn1C1CC1)CC2 REAL300018778507
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)no1 REAL300018778508
NS(=O)(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778509
COC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)C1CCOC1 REAL300018778510
C[C@]1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)C[C@@H]1c1ccccc1 REAL300018778511
CCn1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778512
Cc1cc(F)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(Cl)c1 REAL300018778513
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C3CC3)cc1)CC2 REAL300018778514
CC(C)(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)N1CCOCC1 REAL300018778515
COC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CCOC1 REAL300018778516
Cc1cc(O)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(Cl)c1 REAL300018778517
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1C REAL300018778518
CCc1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778519
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCCC1CCO1)CC2 REAL300018778520
CS(=O)(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778521
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(O)nc1)CC2 REAL300018778522
CN(C)C(=O)c1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778523
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(C3CC3)c1)CC2 REAL300018778524
N#Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1F REAL300018778525
CC(c1nccc2ccccc12)N1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778526
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnn(-c3ccccc3)n1)CC2 REAL300018778527
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccn1)CC2 REAL300018778528
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccs1)CC2 REAL300018778529
CC(=O)Nc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778530
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc([N+](=O)[O-])cc1)CC2 REAL300018778531
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccco1)CC2 REAL300018778532
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1[N+](=O)[O-])CC2 REAL300018778533
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)cc1Cl)CC2 REAL300018778534
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(Cl)c1Cl)CC2 REAL300018778535
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778536
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccncc1)CC2 REAL300018778537
Cc1ccsc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778538
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccsc1)CC2 REAL300018778539
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778540
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c[nH]nc1-c1ccccc1)CC2 REAL300018778541
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)o1)CC2 REAL300018778542
Cc1cc(F)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(F)c1 REAL300018778543
CCOC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)[nH]n1 REAL300018778544
CCC1CCCCC1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778545
CC(C)Cn1nccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778546
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccns1)CC2 REAL300018778547
CN(C)Cc1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cs1 REAL300018778548
CC(C)n1ncnc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778549
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(Cl)c1 REAL300018778550
CCc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778551
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(F)c1 REAL300018778552
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3c1CCC3)CC2 REAL300018778553
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3cnccc3o1)CC2 REAL300018778554
Nc1c(F)cccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778555
CC(C)(C#N)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778556
COC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)o1 REAL300018778557
CC(C)c1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778558
COc1cc(O)cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778559
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3n(n1)CCCC3)CC2 REAL300018778560
COC(=O)c1[nH]cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C REAL300018778561
COC(=O)C=Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778562
CCc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1O REAL300018778563
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccn(C(F)F)c1=O)CC2 REAL300018778564
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCN(c3ccccc3)C1)CC2 REAL300018778565
COc1ncccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778566
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(C3CCCC3)c1)CC2 REAL300018778567
COc1ccc(C)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778568
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3ccccc3o1)CC2 REAL300018778569
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(-c3ccccc3)o1)CC2 REAL300018778570
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1[N+](=O)[O-] REAL300018778571
COc1cccc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)oc12 REAL300018778572
Cc1nn(C)c(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778573
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CC3C=CC1C3)CC2 REAL300018778574
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnn(-c3ccccc3)c1)CC2 REAL300018778575
CCc1oc2ccccc2c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778576
NC(=O)COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778577
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cn(C3CCC3)nn1)CC2 REAL300018778578
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(CO)cc1)CC2 REAL300018778579
Cc1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)[nH]c1C REAL300018778580
COC(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)C1CC1 REAL300018778581
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(OC3CC3)c1F)CC2 REAL300018778582
CCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)c1 REAL300018778583
COc1cncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778584
CCc1cccc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)oc12 REAL300018778585
COc1cnc(F)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778586
COc1cccc(F)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778587
CCCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)c1 REAL300018778588
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnn3c1CCC3)CC2 REAL300018778589
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3n(n1)CCC3)CC2 REAL300018778590
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnn1CC1CC1)CC2 REAL300018778591
Cn1ncc(C(F)(F)F)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778592
Cn1ncc(C2CC2)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778593
Cn1ncc(C2CCC2)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778594
CN1CCCCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)C1=O REAL300018778595
Cc1cc(O)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1Cl REAL300018778596
Cc1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1C REAL300018778597
Cc1cccc2[nH]c(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cc12 REAL300018778598
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C(F)(F)F)o1)CC2 REAL300018778599
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCSCC1)CC2 REAL300018778600
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CC1c1ccc(F)cc1)CC2 REAL300018778601
Cn1nc(C(F)(F)F)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778602
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)c(F)c1F)CC2 REAL300018778603
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnn1-c1ccncc1)CC2 REAL300018778604
CCCn1nccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778605
Cc1ccc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)[nH]c2c1 REAL300018778606
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3n1CCC3)CC2 REAL300018778607
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCC3CC3C1)CC2 REAL300018778608
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CC3CC3C1)CC2 REAL300018778609
CC(C)c1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778610
COC(=O)c1oc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778611
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)on1 REAL300018778612
Cc1nccnc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778613
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC[C@@H]1C[C@H]1c1ccccc1)CC2 REAL300018778614
CCCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778615
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(Cl)n1 REAL300018778616
CC1CC1c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778617
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(Cl)c1 REAL300018778618
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C(F)(F)F)cc1)CC2 REAL300018778619
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1F)CC2 REAL300018778620
CC(C)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778621
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1csc3ccccc13)CC2 REAL300018778622
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778623
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c[nH]nc1-c1cccs1)CC2 REAL300018778624
Cc1ccc(-c2n[nH]cc2CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778625
N#Cc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778626
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)s1)CC2 REAL300018778627
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3cccnc13)CC2 REAL300018778628
CNC(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778629
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(F)ccc1F)CC2 REAL300018778630
NC(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778631
CC(C)Oc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778632
N#Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778633
Cn1cccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778634
Cc1nnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778635
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)cn1)CC2 REAL300018778636
O=C(O)c1nc(C(F)(F)F)n2c1CN(C1CCC3(CC1F)OCCO3)CC2 REAL300018778637
CC(C)CCCCN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778638
COC1CCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CC1 REAL300018778639
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3c(O)cccc3s1)CC2 REAL300018778640
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccncc1Cl)CC2 REAL300018778641
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(F)ccc(F)c1Cl)CC2 REAL300018778642
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cncc(Cl)c1)CC2 REAL300018778643
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnn1C1CCOCC1)CC2 REAL300018778644
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3[nH]ncc13)CC2 REAL300018778645
COCCCC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CCC1 REAL300018778646
CCc1n[nH]c(Cl)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778647
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnc(F)c1)CC2 REAL300018778648
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3cc[nH]c3c1)CC2 REAL300018778649
COc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1Cl REAL300018778650
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnc(O)c1)CC2 REAL300018778651
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCc3ccccc3C1)CC2 REAL300018778652
CCOC(=O)c1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778653
CC1C(Cl)C1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778654
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3c(=O)[nH]ccc3o1)CC2 REAL300018778655
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)c3ccccc13)CC2 REAL300018778656
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C(F)F)nc1)CC2 REAL300018778657
CN(C)c1ccc(C#N)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778658
Cc1ccnc(N)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778659
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nc(Br)c[nH]1)CC2 REAL300018778660
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1F REAL300018778661
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c[nH]nc1-c1cccnc1)CC2 REAL300018778662
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(-n3cncn3)cc1)CC2 REAL300018778663
Cn1nccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778664
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(N3CCCC3)cc1)CC2 REAL300018778665
Cc1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778666
CC(C)(C)n1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778667
CC(C)c1nn(C)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778668
COCCOc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778669
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3c1OCCCO3)CC2 REAL300018778670
CCCOc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778671
COc1ccc(Cl)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778672
Cc1n[nH]c2ncc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cc12 REAL300018778673
Cc1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778674
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc(N3CCCC3)nc1)CC2 REAL300018778675
Cc1nn(C)c2ncc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cc12 REAL300018778676
CN(C)c1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778677
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Cl)cc(Cl)c1)CC2 REAL300018778678
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3ccccn13)CC2 REAL300018778679
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3c1OCCO3)CC2 REAL300018778680
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3c(c1)CCO3)CC2 REAL300018778681
CC(C)c1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cs1 REAL300018778682
CC(C)(C)c1n[nH]cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778683
Cc1n[nH]c(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778684
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(F)c1 REAL300018778685
CC(=O)Nc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778686
Cc1scc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C REAL300018778687
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnn1CC1CCC1)CC2 REAL300018778688
Cn1ncc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cnc21 REAL300018778689
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc(Cl)c(F)c1)CC2 REAL300018778690
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC#Cc1ccccc1)CC2 REAL300018778691
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(CC3CCC3)c1)CC2 REAL300018778692
Cc1cc(C)c(C=CCN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)c1 REAL300018778693
COc1c(C)cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C REAL300018778694
COCC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CCC1 REAL300018778695
CCn1ncnc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778696
CC1(C)OC[C@H](CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)O1 REAL300018778697
CCOc1cc(F)cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778698
CC(C)(C)Oc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778699
Cc1c(Cl)cccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778700
COc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(F)cc1C REAL300018778701
CCCn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778702
CN(C)c1ccc(F)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778703
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(Cl)cncc1Cl)CC2 REAL300018778704
CC(C)(C)c1csc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778705
COCCc1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778706
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3c(F)cccc3c1)CC2 REAL300018778707
Cc1cc(C)c(C=CCN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778708
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCCC(F)(F)F)CC2 REAL300018778709
CN1CCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CC1 REAL300018778710
Cc1ccc(CCN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778711
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3ncccc13)CC2 REAL300018778712
CCCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778713
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3nccnc3c1)CC2 REAL300018778714
CCOc1cccc(F)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778715
Cc1n[nH]cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778716
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cscn1)CC2 REAL300018778717
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(=O)n(C)c1=O REAL300018778718
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(-c3cccnc3)o1)CC2 REAL300018778719
Cc1nn(CCO)c(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778720
CCc1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cs1 REAL300018778721
CC(C)(C)c1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778722
CC(C)(C)c1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cs1 REAL300018778723
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)c(F)c1)CC2 REAL300018778724
Cc1cc(C)cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778725
CC(C)Oc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778726
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1O)CC2 REAL300018778727
CCOc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1O REAL300018778728
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC=Cc1ccccc1[N+](=O)[O-])CC2 REAL300018778729
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(OC(F)F)c1)CC2 REAL300018778730
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1csc([N+](=O)[O-])c1)CC2 REAL300018778731
Cc1c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cccc1[N+](=O)[O-] REAL300018778732
Cc1ccc([N+](=O)[O-])c(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778733
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(O)c1 REAL300018778734
COC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)[nH]c1C REAL300018778735
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c([N+](=O)[O-])n1 REAL300018778736
COC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cs1 REAL300018778737
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3c1CCOC3)CC2 REAL300018778738
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3oc(=O)oc3c1)CC2 REAL300018778739
COc1cc(C)cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1O REAL300018778740
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(F)cc(F)c1O)CC2 REAL300018778741
O=C(O)c1nc(C(F)(F)F)n2c1CN(CCc1ccc(F)c(F)c1)CC2 REAL300018778742
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)cn1)CC2 REAL300018778743
Cc1[nH]nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C REAL300018778744
Cc1coc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778745
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC=Cc1cccc(F)c1)CC2 REAL300018778746
COC(=O)c1cnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778747
Cc1cc(C#N)cc(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778748
CC(C)(C)c1coc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778749
Cc1cc(F)ccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778750
CCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(O)c1 REAL300018778751
COc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1O REAL300018778752
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Cl)ccc1O)CC2 REAL300018778753
COc1cccc(O)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778754
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc([N+](=O)[O-])c1O)CC2 REAL300018778755
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3c(cc1O)OCO3)CC2 REAL300018778756
CC(=Cc1ccccc1)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778757
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1=Cc3ccccc3OC1)CC2 REAL300018778758
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1-n1cncn1)CC2 REAL300018778759
CCn1nc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C REAL300018778760
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3ccnn3c1)CC2 REAL300018778761
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccnc1Cl)CC2 REAL300018778762
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cn[nH]c1)CC2 REAL300018778763
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(F)c(F)c(F)c1)CC2 REAL300018778764
Cn1c(Cl)nc(Cl)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778765
Cn1ccnc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778766
CC(C#N)Oc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778767
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nccn1CC(F)(F)F)CC2 REAL300018778768
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C2CCCC2)n1 REAL300018778769
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nccc3c1CCCC3)CC2 REAL300018778770
Cc1nn(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1Cl REAL300018778771
COC(=O)c1sccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778772
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnn(CCF)c1)CC2 REAL300018778773
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3n1CCOC3)CC2 REAL300018778774
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)c1 REAL300018778775
CC1Cc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)ccc2O1 REAL300018778776
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3[nH]c(=O)oc13)CC2 REAL300018778777
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3c1OCC3)CC2 REAL300018778778
CSCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778779
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnn(CC3CCC3)c1)CC2 REAL300018778780
Cn1nc2c(c1CN1CCn3c(C(F)(F)F)nc(C(=O)O)c3C1)COCC2 REAL300018778781
Cn1nc2c(c1CN1CCn3c(C(F)(F)F)nc(C(=O)O)c3C1)CCC2 REAL300018778782
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnn1C1CCC1)CC2 REAL300018778783
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnn(C3CCC3)c1)CC2 REAL300018778784
CCc1nnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778785
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3c(c1)CCCO3)CC2 REAL300018778786
CN(C)C(=O)c1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778787
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(C3CC3)n[nH]c1Cl)CC2 REAL300018778788
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(C(F)F)c(F)c1)CC2 REAL300018778789
COC(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778790
C=C(CCC#N)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778791
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(C3CC3)[nH]n1)CC2 REAL300018778792
Cn1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C1CC1 REAL300018778793
COCn1ncc(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778794
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nc1 REAL300018778795
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccnn1)CC2 REAL300018778796
CCc1onc(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778797
CCn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778798
CC(C)Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778799
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c2c(n1)CCCC2 REAL300018778800
CCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778801
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cn3ccnc3s1)CC2 REAL300018778802
Cc1oc(C(C)(C)C)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778803
Cc1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)sc1C REAL300018778804
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(O)cc(Cl)c1)CC2 REAL300018778805
COc1nccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1F REAL300018778806
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778807
COCCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778808
CCn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)n1 REAL300018778809
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C2CC2)n1 REAL300018778810
CC(C)(C)c1nnc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778811
CCc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)no1 REAL300018778812
Cc1nn(C(C)C)c(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778813
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccn(CCF)n1)CC2 REAL300018778814
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3cc[nH]c13)CC2 REAL300018778815
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nccs1)CC2 REAL300018778816
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cncnc1)CC2 REAL300018778817
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3ccccc3c1)CC2 REAL300018778818
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc[nH]n1)CC2 REAL300018778819
Cn1c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nc2ccccc21 REAL300018778820
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3[nH]ccc13)CC2 REAL300018778821
Cn1cncc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778822
Cc1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c[nH]1 REAL300018778823
CN(C)c1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778824
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)[nH]n1 REAL300018778825
NC(=O)c1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778826
CN(C)c1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778827
Cn1nc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c2ccccc21 REAL300018778828
Cn1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778829
CCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778830
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1F REAL300018778831
COc1nc(Cl)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1C REAL300018778832
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(F)c1F)CC2 REAL300018778833
CC1(C)Cc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)ccc2O1 REAL300018778834
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1F REAL300018778835
Cc1ncccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778836
CC(C)COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778837
Cc1ccc(O)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778838
COCCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778839
CCn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778840
CC(C)n1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778841
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3ccccc3nc1O)CC2 REAL300018778842
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Br)co1)CC2 REAL300018778843
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(O)cccc1Cl)CC2 REAL300018778844
C#CCCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778845
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1csc(C3CC3)n1)CC2 REAL300018778846
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(C3CC3)on1)CC2 REAL300018778847
N#CCc1ccc(O)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778848
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(C3CCC3)on1)CC2 REAL300018778849
CC1(c2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)no2)CC1 REAL300018778850
CCc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778851
CN(C)C(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778852
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)c1C REAL300018778853
CCNC(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778854
CC(C)(C)c1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778855
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3n1CCCCC3)CC2 REAL300018778856
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccnc(Cl)c1)CC2 REAL300018778857
Cc1c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cnn1C(C)C REAL300018778858
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1conc1C1CC1)CC2 REAL300018778859
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(-c3ccccc3)no1)CC2 REAL300018778860
CCN1CCc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)ccc21 REAL300018778861
COC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n(C)n1 REAL300018778862
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3ccsc13)CC2 REAL300018778863
COc1ccc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778864
Cc1cc(F)cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778865
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1C1CC1 REAL300018778866
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C1CC1 REAL300018778867
CNC(=O)c1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778868
CCNC(=O)c1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778869
CCOc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccn1 REAL300018778870
Cn1cnc2cccc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)c21 REAL300018778871
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ncccc1F)CC2 REAL300018778872
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)cc1O)CC2 REAL300018778873
CC(C)c1nocc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778874
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(OC3CC3)cc1)CC2 REAL300018778875
CNC(=O)c1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778876
CN(C)CCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778877
CCNC(=O)c1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778878
Cc1c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)oc2ccc(F)cc12 REAL300018778879
CCCn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)n1 REAL300018778880
CCn1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778881
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Cl)ccn1)CC2 REAL300018778882
CC(C)(C)c1c[nH]c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778883
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(CC3CC3)s1)CC2 REAL300018778884
Cn1cc(Cl)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778885
CSc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778886
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3c(c1)OCC3)CC2 REAL300018778887
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nc3c([nH]1)CCCC3)CC2 REAL300018778888
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cn3cc(Cl)ccc3n1)CC2 REAL300018778889
C#CCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778890
CCn1ccnc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778891
CN(C)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1F REAL300018778892
COc1cccc(Cl)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778893
Cc1ccc(F)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778894
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1occc1Br)CC2 REAL300018778895
CCc1nn(C)c(Cl)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778896
Cc1csc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778897
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCCCCC1)CC2 REAL300018778898
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1=CCCOC1)CC2 REAL300018778899
Cc1nc2ccccn2c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778900
Cc1nc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778901
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(CO)o1)CC2 REAL300018778902
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3cn[nH]c13)CC2 REAL300018778903
Cn1nnc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)ccc21 REAL300018778904
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nccc3ccccc13)CC2 REAL300018778905
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3ccc(Cl)cn13)CC2 REAL300018778906
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1Cl REAL300018778907
CC(C)CCn1cccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778908
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778909
CC1(C)Cc2cccc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)c2O1 REAL300018778910
Cc1cccn2c(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)cnc12 REAL300018778911
CC(C)(CCC#N)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778912
Cc1cc(O)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C REAL300018778913
COCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778914
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3c(c1)CCC3)CC2 REAL300018778915
COc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1C#N REAL300018778916
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3cc(F)ccc3o1)CC2 REAL300018778917
N#Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778918
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1O REAL300018778919
CC(C)Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nn1 REAL300018778920
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1nc(C3CC3)cs1)CC2 REAL300018778921
Cc1c(C(F)(F)F)n[nH]c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778922
Cc1ccoc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778923
COCc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778924
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CCCCCCC1)CC2 REAL300018778925
CCC(C)(C)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778926
Cc1ncsc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778927
COCCn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cn1 REAL300018778928
Cc1cc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)oc2cc1C REAL300018778929
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(-n3ccnc3)nc1)CC2 REAL300018778930
CN(C)C(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)[nH]1 REAL300018778931
CS(=O)c1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778932
COC(=O)c1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c[nH]1 REAL300018778933
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccccc1C1CC1)CC2 REAL300018778934
N#Cc1csc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778935
CCc1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778936
COc1cc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1OC REAL300018778937
Cn1nncc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778938
N#Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778939
Cc1cccc2ncc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)n12 REAL300018778940
COCCOc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778941
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(Cl)nc1)CC2 REAL300018778942
CCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778943
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(-n3cccn3)c1)CC2 REAL300018778944
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc(C3CCC3)s1)CC2 REAL300018778945
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cnc1Cl REAL300018778946
Cc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C)s1 REAL300018778947
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(F)cc3cccnc13)CC2 REAL300018778948
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(N3CCCC3)nc1)CC2 REAL300018778949
CC(C)c1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778950
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc3ccccc3s1)CC2 REAL300018778951
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)cc1Cl)CC2 REAL300018778952
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(F)c(F)cc1F)CC2 REAL300018778953
CCC1(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)COC1 REAL300018778954
NC(=O)c1csc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778955
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cncs1)CC2 REAL300018778956
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(-c3ccccc3)[nH]n1)CC2 REAL300018778957
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc(C3CC3)s1)CC2 REAL300018778958
Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nc1 REAL300018778959
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(Cl)c1F)CC2 REAL300018778960
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc(F)c3cccnc13)CC2 REAL300018778961
CCCn1nc(C)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1C REAL300018778962
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnn(CC(F)(F)F)c1)CC2 REAL300018778963
CCOc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)n1 REAL300018778964
CC(C)Cc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)cc1 REAL300018778965
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccc3c(c1)COC3)CC2 REAL300018778966
COc1ccsc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778967
COCc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)o1 REAL300018778968
CC(=O)Nc1ccccc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778969
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Cl)ccc1Cl)CC2 REAL300018778970
COc1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)ccc1F REAL300018778971
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cncc3ccccc13)CC2 REAL300018778972
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ncccc1C(F)(F)F)CC2 REAL300018778973
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC=Cc1ccc(Cl)cc1)CC2 REAL300018778974
Cc1oc2ccccc2c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778975
O=C(O)c1nc(C(F)(F)F)n2c1CN(CC1CC1c1ccccc1)CC2 REAL300018778976
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cscc1Cl)CC2 REAL300018778977
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cnc3ccsc3c1)CC2 REAL300018778978
Cc1cc(Cl)cc(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778979
CCOc1ccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)nc1 REAL300018778980
CC(C)Cc1ncc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)s1 REAL300018778981
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1c(Cl)oc3ccccc13)CC2 REAL300018778982
CCc1nn(C)c(CC)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778983
CC1(C)CCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CC1 REAL300018778984
COC(=O)c1occc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778985
COc1ccc(O)c(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778986
Cc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1O REAL300018778987
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc(Cl)c1O)CC2 REAL300018778988
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cc(Cl)cc(F)c1O)CC2 REAL300018778989
Cc1cccc(C)c1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778990
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1cccc3nccn13)CC2 REAL300018778991
CCCC1CCC(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)CC1 REAL300018778992
CCCC(C)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778993
CC(CCc1ccccc1)CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778994
Cn1cc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c(C(C)(C)C)n1 REAL300018778995
CC(C)COc1cccc(CN2CCn3c(C(F)(F)F)nc(C(=O)O)c3C2)c1 REAL300018778996
Cn1cnc2cc(CN3CCn4c(C(F)(F)F)nc(C(=O)O)c4C3)ccc21 REAL300018778997
O=C(O)c1nc(C(F)(F)F)n2c1CN(Cc1ccn(-c3ccccc3)n1)CC2 REAL300018778998
CCc1nn(C)cc1CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1 REAL300018778999
CC(C)(CN1CCn2c(C(F)(F)F)nc(C(=O)O)c2C1)c1ccccc1 REAL300018779000
