CC1CCCCC1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150001
O=C(O)c1csc(N2CCN(Cc3cc4c(Cl)nccc4o3)CC2)n1 REAL300019150002
NC(=O)Cn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150003
Cc1ccccc1-n1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150004
CCSc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150005
O=C(O)c1csc(N2CCN(Cc3cnnn3-c3ccccc3)CC2)n1 REAL300019150006
O=C(O)c1csc(N2CCN(Cc3cc4ccnc(Cl)c4s3)CC2)n1 REAL300019150007
O=C(O)c1csc(N2CCN(Cc3cc(C4CC4)no3)CC2)n1 REAL300019150008
O=C(O)c1csc(N2CCN(CC3C4CC5CC(C4)CC3C5)CC2)n1 REAL300019150009
O=C(O)c1csc(N2CCN(CC3CC3(Cl)Cl)CC2)n1 REAL300019150010
Cn1c(Cl)cnc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150011
CC(C)OC(CN1CCN(c2nc(C(=O)O)cs2)CC1)c1ccccc1 REAL300019150012
CC(C)N(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150013
COCCN(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150014
Cn1nc2c(c1CN1CCN(c3nc(C(=O)O)cs3)CC1)CCCC2 REAL300019150015
O=C(O)c1csc(N2CCN(Cc3scnc3C3CC3)CC2)n1 REAL300019150016
Cc1c[nH]nc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150017
CN(C)Cc1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150018
O=C(O)c1csc(N2CCN(Cc3ccsc3C(F)(F)F)CC2)n1 REAL300019150019
O=C(O)c1csc(N2CCN(C[C@@H]3C[C@H]3c3ccccc3)CC2)n1 REAL300019150020
CC(C)(C)n1nnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150021
O=C(O)c1csc(N2CCN(CC=Cc3ccc(F)cc3)CC2)n1 REAL300019150022
O=C(O)c1csc(N2CCN(Cc3cccc4c3NCCC4)CC2)n1 REAL300019150023
Cn1cc(-c2csc(CN3CCN(c4nc(C(=O)O)cs4)CC3)n2)cn1 REAL300019150024
O=C(O)c1csc(N2CCN(CCC3CCOCC3)CC2)n1 REAL300019150025
O=C(O)c1csc(N2CCN(CC3CCC4(CC3)OCCO4)CC2)n1 REAL300019150026
COc1ccc2nc(CN3CCN(c4nc(C(=O)O)cs4)CC3)sc2c1 REAL300019150027
Cn1c(=O)sc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc21 REAL300019150028
COC(=O)C1C(CN2CCN(c3nc(C(=O)O)cs3)CC2)C1(F)F REAL300019150029
O=C(O)c1csc(N2CCN(Cc3ccsc3Cl)CC2)n1 REAL300019150030
CCN(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150031
O=C(O)c1csc(N2CCN(Cc3ccc(OCC4CC4)cc3)CC2)n1 REAL300019150032
O=C(O)c1csc(N2CCN(Cc3c(O)ccc(Cl)c3F)CC2)n1 REAL300019150033
O=C(O)c1csc(N2CCN(Cc3cc4ccc(F)cc4[nH]3)CC2)n1 REAL300019150034
O=C(O)c1csc(N2CCN(Cc3cnc(C4OCCO4)s3)CC2)n1 REAL300019150035
O=C(O)c1csc(N2CCN(Cc3nc4ccc(F)cc4s3)CC2)n1 REAL300019150036
O=C(O)c1csc(N2CCN(Cc3ccc(F)c(Cl)c3Cl)CC2)n1 REAL300019150037
O=C(O)c1csc(N2CCN(Cc3csc(Cl)c3Cl)CC2)n1 REAL300019150038
CC(CCC#N)CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150039
O=C(O)c1csc(N2CCN(CCc3ccc(F)cc3Cl)CC2)n1 REAL300019150040
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1C#N REAL300019150041
O=C(O)c1csc(N2CCN(Cc3cnc(C(F)(F)F)s3)CC2)n1 REAL300019150042
COc1c([N+](=O)[O-])ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1O REAL300019150043
CC(O)c1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150044
O=C(O)c1csc(N2CCN(Cc3ncc(C4OCCO4)s3)CC2)n1 REAL300019150045
Cn1nc(Br)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150046
CCCCCCCCCC(C)CCN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150047
Cc1nc(F)ccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150048
O=C(O)c1csc(N2CCN(Cc3sccc3Cl)CC2)n1 REAL300019150049
O=C(O)c1csc(N2CCN(Cc3ccc4cnccc4c3)CC2)n1 REAL300019150050
CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150051
O=C(O)c1csc(N2CCN(Cc3cc4ccccc4[nH]3)CC2)n1 REAL300019150052
CC(C)(C)c1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150053
CSc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150054
O=C(O)c1csc(N2CCN(Cc3ccc(OCCCCl)cc3)CC2)n1 REAL300019150055
Cn1cc(-c2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc2)cn1 REAL300019150056
O=C(O)c1csc(N2CCN(Cc3ccc(C(F)F)cc3)CC2)n1 REAL300019150057
CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC REAL300019150058
O=C(O)c1csc(N2CCN(Cc3ccc(-n4cccn4)cc3)CC2)n1 REAL300019150059
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)c1 REAL300019150060
Cc1ccc(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150061
O=C(O)c1csc(N2CCN(Cc3ccc4ncccc4c3)CC2)n1 REAL300019150062
CC(C)(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150063
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1OC(F)F REAL300019150064
CCOc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1OC REAL300019150065
CCCCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150066
CCCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150067
Cc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C REAL300019150068
C=CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC REAL300019150069
CN(CCC#N)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150070
CCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150071
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1OC(C)C REAL300019150072
COC(=O)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150073
COC(=O)c1ccc(Cl)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150074
O=C(O)c1csc(N2CCN(CC3CCC(c4ccccc4)CC3)CC2)n1 REAL300019150075
Cc1nn(C(C)C)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150076
C[C@H](CN1CCN(c2nc(C(=O)O)cs2)CC1)NC(=O)OC(C)(C)C REAL300019150077
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(OC)c1O REAL300019150078
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(C)c1O REAL300019150079
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1C#N REAL300019150080
COC(=O)c1[nH]c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150081
COC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n(C)c1C REAL300019150082
CCc1oc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C(=O)OC REAL300019150083
Cn1cc(-c2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)s2)cn1 REAL300019150084
COCCCn1nccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150085
Cc1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1C REAL300019150086
CC(C)C(CN1CCN(c2nc(C(=O)O)cs2)CC1)C(C)C REAL300019150087
Cn1nnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150088
O=C(O)c1csc(N2CCN(CC=Cc3ccc(F)c(F)c3)CC2)n1 REAL300019150089
O=C(O)c1csc(N2CCN(Cc3cscc3Br)CC2)n1 REAL300019150090
CCOC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)[nH]c1C REAL300019150091
O=C(O)c1csc(N2CCN(C[C@@H]3C[C@H]3c3ccccc3)CC2)n1 REAL300019150092
O=C(O)c1csc(N2CCN(CCc3ccc(Cl)cc3)CC2)n1 REAL300019150093
CC(C)C1CCC(CN2CCN(c3nc(C(=O)O)cs3)CC2)CC1 REAL300019150094
CC(C)n1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150095
CN(C)Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)no1 REAL300019150096
O=C(O)c1csc(N2CCN(Cc3cnccn3)CC2)n1 REAL300019150097
COCCOCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150098
N#Cc1c(F)cccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150099
O=C(O)c1csc(N2CCN(Cc3ccc4ccccc4c3)CC2)n1 REAL300019150100
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(OC)c1 REAL300019150101
COc1ccc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc2c1 REAL300019150102
O=C(O)c1csc(N2CCN(Cc3ccc(N4CCCCC4)cc3)CC2)n1 REAL300019150103
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(Cl)c1OC REAL300019150104
CCOc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1OC REAL300019150105
CCCOc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1OC REAL300019150106
C=CCOc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150107
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC(F)F REAL300019150108
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(C)c1OC(F)F REAL300019150109
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc2c1OCCO2 REAL300019150110
Cc1cc(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150111
O=C(O)c1csc(N2CCN(Cc3cc(-c4ccccn4)n[nH]3)CC2)n1 REAL300019150112
O=C(O)c1csc(N2CCN(Cc3ccc4[nH]ccc4c3)CC2)n1 REAL300019150113
O=C(O)c1csc(N2CCN(Cc3cc(O)cc(C(F)(F)F)c3)CC2)n1 REAL300019150114
O=C(O)c1csc(N2CCN(Cc3cscc3C(F)(F)F)CC2)n1 REAL300019150115
COc1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150116
O=C(O)c1csc(N2CCN(Cc3ccc(C4CCCC4)cc3)CC2)n1 REAL300019150117
Cc1nc(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150118
CCOC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)on1 REAL300019150119
O=C(O)c1csc(N2CCN(CCc3ccc([N+](=O)[O-])cc3)CC2)n1 REAL300019150120
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)CCCC4)CC2)n1 REAL300019150121
Cc1nnsc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150122
O=C(O)c1csc(N2CCN(Cc3cnn(CC(F)F)c3)CC2)n1 REAL300019150123
COCc1ccccc1C=C(C)CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150124
COC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)on1 REAL300019150125
Cn1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150126
COC(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1C REAL300019150127
CSC(C)(C)CCN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150128
O=C(O)c1csc(N2CCN(Cc3ccc4ccc(F)c(F)c4n3)CC2)n1 REAL300019150129
O=C(O)c1csc(N2CCN(Cc3ccc(C4CCC4)cc3)CC2)n1 REAL300019150130
O=C(O)c1csc(N2CCN(Cc3cccc(O)c3Cl)CC2)n1 REAL300019150131
Cc1sccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150132
Cc1cc(Cl)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150133
O=C(O)c1csc(N2CCN(Cc3cc(Cl)c(F)cc3O)CC2)n1 REAL300019150134
CSCc1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150135
O=C(O)c1csc(N2CCN(Cc3ccc(F)cc3O)CC2)n1 REAL300019150136
O=C(O)c1csc(N2CCN(Cc3cc4cccnc4o3)CC2)n1 REAL300019150137
CC(CN1CCN(c2nc(C(=O)O)cs2)CC1)c1cc(F)cc(F)c1 REAL300019150138
COc1cccc2c(CN3CCN(c4nc(C(=O)O)cs4)CC3)cccc12 REAL300019150139
COc1nccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150140
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cs1 REAL300019150141
Cc1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150142
O=C(O)c1csc(N2CCN(Cc3nc(Cl)cs3)CC2)n1 REAL300019150143
CCC(C)C(CN1CCN(c2nc(C(=O)O)cs2)CC1)OC REAL300019150144
COc1cc2ccccc2cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150145
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc2ccccc12 REAL300019150146
Cc1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150147
COC(=O)Cn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150148
Cc1cnccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150149
Cc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1F REAL300019150150
O=C(O)c1csc(N2CCN(Cc3ccnc(Cl)c3F)CC2)n1 REAL300019150151
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc2c1OCO2 REAL300019150152
O=C(O)c1csc(N2CCN(Cc3ccc(-n4ccnc4)cc3)CC2)n1 REAL300019150153
O=C(O)c1csc(N2CCN(Cc3cc(Cl)c4c(c3)OCCO4)CC2)n1 REAL300019150154
O=C(O)c1csc(N2CCN(Cc3ccccc3)CC2)n1 REAL300019150155
O=C(O)c1csc(N2CCN(Cc3ccccc3Cl)CC2)n1 REAL300019150156
O=C(O)c1csc(N2CCN(Cc3cccc4ccccc34)CC2)n1 REAL300019150157
CN(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150158
CCN(CC)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150159
O=C(O)c1csc(N2CCN(Cc3ccc(Br)cc3)CC2)n1 REAL300019150160
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)cc3)CC2)n1 REAL300019150161
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(OC)c1OC REAL300019150162
O=C(O)c1csc(N2CCN(Cc3ccc(F)cc3)CC2)n1 REAL300019150163
COc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1OC REAL300019150164
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150165
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(OC)c1 REAL300019150166
O=C(O)c1csc(N2CCN(Cc3ccc(F)cc3F)CC2)n1 REAL300019150167
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)c(Cl)c3)CC2)n1 REAL300019150168
O=C(O)c1csc(N2CCN(Cc3ccc(OC(F)F)cc3)CC2)n1 REAL300019150169
CCCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150170
CC(C)CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150171
O=C(O)c1csc(N2CCN(Cc3cccc(Oc4ccccc4)c3)CC2)n1 REAL300019150172
O=C(O)c1csc(N2CCN(Cc3cccc(Cl)c3)CC2)n1 REAL300019150173
COc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150174
O=C(O)c1csc(N2CCN(Cc3cccc(C(F)(F)F)c3)CC2)n1 REAL300019150175
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(OC)c1OC REAL300019150176
CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150177
O=C(O)c1csc(N2CCN(Cc3cccc(F)c3)CC2)n1 REAL300019150178
O=C(O)c1csc(N2CCN(Cc3cccc(O)c3)CC2)n1 REAL300019150179
COc1ccccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150180
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccccc4)cc3)CC2)n1 REAL300019150181
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150182
CSc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150183
COc1cc(OC)c(OC)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150184
Cc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150185
O=C(O)c1csc(N2CCN(Cc3ccc(F)c(F)c3)CC2)n1 REAL300019150186
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1O REAL300019150187
Cc1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cs1 REAL300019150188
C#CCCCCCCN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150189
COC(Cc1ccccc1)CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150190
CCCn1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150191
Cn1nc(C2CC2)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150192
O=C(O)c1csc(N2CCN(Cc3cnc4ccccc4n3)CC2)n1 REAL300019150193
O=C(O)c1csc(N2CCN(Cc3ccc4c(n3)CCC4)CC2)n1 REAL300019150194
CCOP(=O)(CCCN1CCN(c2nc(C(=O)O)cs2)CC1)OCC REAL300019150195
CCC(C)(CN1CCN(c2nc(C(=O)O)cs2)CC1)OC REAL300019150196
CCn1nnc(C)c1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150197
O=C(O)c1csc(N2CCN(Cc3cc4cc(Cl)cnc4o3)CC2)n1 REAL300019150198
Cn1cc(CCCN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150199
O=C(O)c1csc(N2CCN(Cc3cccc4ccoc34)CC2)n1 REAL300019150200
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)OCCCCO4)CC2)n1 REAL300019150201
CS(=O)(=O)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150202
O=C(O)c1csc(N2CCN(Cc3ccnn3C3CCCC3)CC2)n1 REAL300019150203
O=C(O)c1csc(N2CCN(Cc3cccn3C3CC3)CC2)n1 REAL300019150204
CC(C)(C)OC(=O)N1CC(CCN2CCN(c3nc(C(=O)O)cs3)CC2)C1 REAL300019150205
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)no1 REAL300019150206
NS(=O)(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150207
COC(CN1CCN(c2nc(C(=O)O)cs2)CC1)C1CCOC1 REAL300019150208
C[C@]1(CN2CCN(c3nc(C(=O)O)cs3)CC2)C[C@@H]1c1ccccc1 REAL300019150209
CCn1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150210
O=C(O)c1csc(N2CCN(Cc3ccc(C4CC4)cc3)CC2)n1 REAL300019150211
O=C(O)c1csc(N2CCN(Cc3ccncc3Br)CC2)n1 REAL300019150212
O=C(O)c1csc(N2CCN(Cc3cccc4c3OC(F)(F)O4)CC2)n1 REAL300019150213
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1C REAL300019150214
CCc1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150215
O=C(O)c1csc(N2CCN(CCCC3CCO3)CC2)n1 REAL300019150216
CS(=O)(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150217
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1C(F)(F)F REAL300019150218
CS(=O)(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150219
O=C(O)c1csc(N2CCN(Cc3ccc(O)nc3)CC2)n1 REAL300019150220
O=C(O)c1csc(N2CCN(Cc3nc4cc([N+](=O)[O-])ccc4o3)CC2)n1 REAL300019150221
O=C(O)c1csc(N2CCN(Cc3cccc(C4CC4)c3)CC2)n1 REAL300019150222
N#Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150223
CC(c1nccc2ccccc12)N1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150224
O=C(O)c1csc(N2CCN(Cc3cnn(-c4ccccc4)n3)CC2)n1 REAL300019150225
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccccc4)s3)CC2)n1 REAL300019150226
O=C(O)c1csc(N2CCN(Cc3ccccn3)CC2)n1 REAL300019150227
O=C(O)c1csc(N2CCN(Cc3cccs3)CC2)n1 REAL300019150228
CC(=O)Nc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150229
O=C(O)c1csc(N2CCN(Cc3ccc([N+](=O)[O-])cc3)CC2)n1 REAL300019150230
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)cc3Cl)CC2)n1 REAL300019150231
O=C(O)c1csc(N2CCN(Cc3cccc(Cl)c3Cl)CC2)n1 REAL300019150232
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150233
O=C(O)c1csc(N2CCN(Cc3ccncc3)CC2)n1 REAL300019150234
Cc1ccsc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150235
O=C(O)c1csc(N2CCN(Cc3ccsc3)CC2)n1 REAL300019150236
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150237
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)o3)CC2)n1 REAL300019150238
Cc1nn(-c2ccccc2)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150239
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccccc4F)o3)CC2)n1 REAL300019150240
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)OC(F)(F)O4)CC2)n1 REAL300019150241
CCOC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)[nH]n1 REAL300019150242
CCC1CCCCC1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150243
CC(C)Cn1nccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150244
O=C(O)c1csc(N2CCN(Cc3ccns3)CC2)n1 REAL300019150245
CN(C)Cc1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cs1 REAL300019150246
CC(C)n1ncnc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150247
Cc1cccc(-n2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)c(C)n2)c1 REAL300019150248
COc1cc(OC)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150249
COc1cc(F)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC REAL300019150250
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(Cl)c1 REAL300019150251
CCc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150252
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(F)c1 REAL300019150253
O=C(O)c1csc(N2CCN(Cc3cccc4c3CCC4)CC2)n1 REAL300019150254
O=C(O)c1csc(N2CCN(Cc3cc4cnccc4o3)CC2)n1 REAL300019150255
O=C(O)c1csc(N2CCN(Cc3cc4nc(Cl)ccc4s3)CC2)n1 REAL300019150256
Nc1c(F)cccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150257
Cc1ccc(-n2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)c(C)n2)cc1 REAL300019150258
CC(C)(C#N)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150259
COC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)o1 REAL300019150260
COc1cc(O)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150261
O=C(O)c1csc(N2CCN(Cc3cc4n(n3)CCCC4)CC2)n1 REAL300019150262
COC(=O)c1[nH]cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C REAL300019150263
COC(=O)C=Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150264
CCc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1O REAL300019150265
O=C(O)c1csc(N2CCN(Cc3cccn(C(F)F)c3=O)CC2)n1 REAL300019150266
O=C(O)c1csc(N2CCN(CC3CCN(c4ccccc4)C3)CC2)n1 REAL300019150267
COC(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150268
COc1ncccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150269
O=C(O)c1csc(N2CCN(Cc3cccc(C4CCCC4)c3)CC2)n1 REAL300019150270
COc1ccc(C)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150271
O=C(O)c1csc(N2CCN(Cc3cc4ccccc4o3)CC2)n1 REAL300019150272
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccccc4)o3)CC2)n1 REAL300019150273
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1[N+](=O)[O-] REAL300019150274
COc1cccc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)oc12 REAL300019150275
CC(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1[N+](=O)[O-] REAL300019150276
O=C(O)c1csc(N2CCN(CC3CC4C=CC3C4)CC2)n1 REAL300019150277
O=C(O)c1csc(N2CCN(Cc3ccc(CSC(F)F)o3)CC2)n1 REAL300019150278
O=C(O)c1csc(N2CCN(Cc3cnn(-c4ccccc4)c3)CC2)n1 REAL300019150279
O=C(O)c1csc(N2CCN(Cc3cnn(Cc4ccccc4)c3)CC2)n1 REAL300019150280
NC(=O)COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150281
O=C(O)c1csc(N2CCN(Cc3cn(C4CCC4)nn3)CC2)n1 REAL300019150282
O=C(O)c1csc(N2CCN(Cc3ccc(CO)cc3)CC2)n1 REAL300019150283
Cc1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)[nH]c1C REAL300019150284
COC(CN1CCN(c2nc(C(=O)O)cs2)CC1)C1CC1 REAL300019150285
O=C(O)c1csc(N2CCN(Cc3cccc(OC4CC4)c3F)CC2)n1 REAL300019150286
CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)c1 REAL300019150287
COc1cncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150288
CCc1cccc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)oc12 REAL300019150289
Cc1c(Br)cncc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150290
COc1cnc(F)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150291
COC(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1Cl REAL300019150292
CCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)c1 REAL300019150293
O=C(O)c1csc(N2CCN(Cc3cnn4c3CCC4)CC2)n1 REAL300019150294
O=C(O)c1csc(N2CCN(Cc3cc4n(n3)CCC4)CC2)n1 REAL300019150295
O=C(O)c1csc(N2CCN(Cc3ccnn3CC3CC3)CC2)n1 REAL300019150296
CN1CCCCC(CN2CCN(c3nc(C(=O)O)cs3)CC2)C1=O REAL300019150297
Cc1cc(O)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1Cl REAL300019150298
O=C(O)c1csc(N2CCN(Cc3ccc(OC4CCOC4)cc3)CC2)n1 REAL300019150299
Cc1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1C REAL300019150300
Cc1cccc2[nH]c(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc12 REAL300019150301
O=C(O)c1csc(N2CCN(Cc3ccc(C(F)(F)F)o3)CC2)n1 REAL300019150302
O=C(O)c1csc(N2CCN(CC3CCSCC3)CC2)n1 REAL300019150303
Cn1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cnc1Br REAL300019150304
O=C(O)c1csc(N2CCN(CC3CC3c3ccc(F)cc3)CC2)n1 REAL300019150305
O=C(O)c1csc(N2CCN(Cc3ccc(Br)cc3O)CC2)n1 REAL300019150306
COCC(C)Oc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150307
Cn1nc(C(F)(F)F)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150308
O=C(O)c1csc(N2CCN(Cc3ccc(F)c(F)c3F)CC2)n1 REAL300019150309
CCCn1nccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150310
Cc1ccc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)[nH]c2c1 REAL300019150311
O=C(O)c1csc(N2CCN(Cc3ccc(-c4cccs4)cc3)CC2)n1 REAL300019150312
O=C(O)c1csc(N2CCN(Cc3cnc4n3CCC4)CC2)n1 REAL300019150313
O=C(O)c1csc(N2CCN(CC3CCC4CC4C3)CC2)n1 REAL300019150314
O=C(O)c1csc(N2CCN(CC3CC4CC4C3)CC2)n1 REAL300019150315
CC(C)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150316
COC(=O)c1oc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150317
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)on1 REAL300019150318
Cc1nccnc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150319
O=C(O)c1csc(N2CCN(CC[C@@H]3C[C@H]3c3ccccc3)CC2)n1 REAL300019150320
CCCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150321
O=C(O)c1csc(N2CCN(Cc3ccnn3CCc3ccccc3)CC2)n1 REAL300019150322
Cn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(Cl)n1 REAL300019150323
O=C(O)c1csc(N2CCN(Cc3ccc(OC(F)(F)F)cc3)CC2)n1 REAL300019150324
CC1CC1c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150325
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(Cl)c1 REAL300019150326
O=C(O)c1csc(N2CCN(Cc3ccc(C(F)(F)F)cc3)CC2)n1 REAL300019150327
O=C(O)c1csc(N2CCN(Cc3ccccc3F)CC2)n1 REAL300019150328
COc1cc2c(cc1CN1CCN(c3nc(C(=O)O)cs3)CC1)OC(C)C2 REAL300019150329
CC(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150330
CCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC REAL300019150331
O=C(O)c1csc(N2CCN(Cc3ccc(Br)s3)CC2)n1 REAL300019150332
O=C(O)c1csc(N2CCN(Cc3ccccc3Br)CC2)n1 REAL300019150333
O=C(O)c1csc(N2CCN(Cc3csc4ccccc34)CC2)n1 REAL300019150334
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150335
N#Cc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150336
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)s3)CC2)n1 REAL300019150337
O=C(O)c1csc(N2CCN(Cc3ccc(-n4cncn4)c(F)c3)CC2)n1 REAL300019150338
O=C(O)c1csc(N2CCN(Cc3cccc4cccnc34)CC2)n1 REAL300019150339
CCN(CC)c1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150340
O=C(NC1CC1)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150341
CNC(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150342
CCN(C(C)=O)c1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cs1 REAL300019150343
O=C(O)c1csc(N2CCN(Cc3cc(F)ccc3F)CC2)n1 REAL300019150344
NC(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150345
CC(C)Oc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150346
N#Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150347
Cn1cccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150348
Cc1nnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150349
O=C(O)c1csc(N2CCN(Cc3ccc(F)cn3)CC2)n1 REAL300019150350
O=C(O)c1csc(N2CCN(C3CCC4(CC3F)OCCO4)CC2)n1 REAL300019150351
CC(C)CCCCN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150352
COC1CCC(CN2CCN(c3nc(C(=O)O)cs3)CC2)CC1 REAL300019150353
O=C(O)c1csc(N2CCN(Cc3cc4c(O)cccc4s3)CC2)n1 REAL300019150354
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC1CC1 REAL300019150355
CN(C)c1cc(F)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150356
O=C(O)c1csc(N2CCN(Cc3ccncc3Cl)CC2)n1 REAL300019150357
O=C(O)c1csc(N2CCN(Cc3cncc(Cl)c3)CC2)n1 REAL300019150358
O=C(O)c1csc(N2CCN(Cc3ccnn3C3CCOCC3)CC2)n1 REAL300019150359
O=C(O)c1csc(N2CCN(Cc3sncc3Br)CC2)n1 REAL300019150360
O=C(O)c1csc(N2CCN(Cc3ccsc3Br)CC2)n1 REAL300019150361
CCOc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(F)cc1OC REAL300019150362
Cn1cc(-c2nc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cs2)cn1 REAL300019150363
O=C(O)c1csc(N2CCN(Cc3ccnc(F)c3)CC2)n1 REAL300019150364
O=C(O)c1csc(N2CCN(Cc3ccc4cc[nH]c4c3)CC2)n1 REAL300019150365
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1Cl REAL300019150366
O=C(O)c1csc(N2CCN(Cc3cn(-c4ccc(F)cc4)nn3)CC2)n1 REAL300019150367
Cn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(Br)n1 REAL300019150368
CCOC(=O)c1[nH]c(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C REAL300019150369
O=C(O)c1csc(N2CCN(Cc3ccnc(O)c3)CC2)n1 REAL300019150370
CCOC(=O)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150371
CC1C(Cl)C1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150372
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ncc1Br REAL300019150373
CCOC(=O)c1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150374
O=C(O)c1csc(N2CCN(Cc3cc4c(=O)[nH]ccc4o3)CC2)n1 REAL300019150375
O=C(O)c1csc(N2CCN(Cc3ccc(F)c4ccccc34)CC2)n1 REAL300019150376
O=C(O)c1csc(N2CCN(Cc3cccnc3Br)CC2)n1 REAL300019150377
O=C(O)c1csc(N2CCN(Cc3ccc(C(F)F)nc3)CC2)n1 REAL300019150378
O=C(O)c1csc(N2CCN(Cc3nc(Br)c[nH]3)CC2)n1 REAL300019150379
CC(C)(C)OC(=O)NC1CC(CN2CCN(c3nc(C(=O)O)cs3)CC2)C1 REAL300019150380
CC(C)(C)OC(=O)N[C@H]1C[C@@H](CN2CCN(c3nc(C(=O)O)cs3)CC2)C1 REAL300019150381
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150382
Cc1ccc(-c2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)o2)cc1 REAL300019150383
O=C(O)c1csc(N2CCN(Cc3ccc(-n4cncn4)cc3)CC2)n1 REAL300019150384
Cn1nccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150385
O=C(O)c1csc(N2CCN(Cc3ccc(N4CCCC4)cc3)CC2)n1 REAL300019150386
O=C(O)c1csc(N2CCN(Cc3csc(-c4ccccn4)n3)CC2)n1 REAL300019150387
Cc1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150388
CC(C)(C)n1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150389
O=C(O)c1csc(N2CCN(Cc3cnc(-c4ccccc4)nc3)CC2)n1 REAL300019150390
COCCOc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150391
O=C(O)c1csc(N2CCN(Cc3cccc4c3OCCCO4)CC2)n1 REAL300019150392
CCCOc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150393
COc1ccc(Cl)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150394
Cc1n[nH]c2ncc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc12 REAL300019150395
Cc1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150396
O=C(O)c1csc(N2CCN(Cc3cnc(N4CCCC4)nc3)CC2)n1 REAL300019150397
CN(C)CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150398
O=C(O)c1csc(N2CCN(Cc3cnc(N4CCOCC4)nc3)CC2)n1 REAL300019150399
Cc1nn(C)c2ncc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc12 REAL300019150400
CN(C)c1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150401
O=C(O)c1csc(N2CCN(Cc3cccc(-c4ccccc4)c3)CC2)n1 REAL300019150402
O=C(O)c1csc(N2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)n1 REAL300019150403
O=C(O)c1csc(N2CCN(Cc3cc(-c4ccccc4)cs3)CC2)n1 REAL300019150404
O=C(O)c1csc(N2CCN(Cc3cnc4ccccn34)CC2)n1 REAL300019150405
O=C(O)c1csc(N2CCN(Cc3cccc4c3OCCO4)CC2)n1 REAL300019150406
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)CCO4)CC2)n1 REAL300019150407
O=C(O)c1csc(N2CCN(Cc3cccc(OC4CCCC4)c3)CC2)n1 REAL300019150408
CS(=O)(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150409
CC(C)c1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cs1 REAL300019150410
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(F)c1 REAL300019150411
CC(=O)Nc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150412
COc1cc(Cl)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC REAL300019150413
O=C(O)c1csc(N2CCN(Cc3ccc(CC(F)(F)F)cc3)CC2)n1 REAL300019150414
Cc1scc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C REAL300019150415
O=C(O)c1csc(N2CCN(Cc3ccnn3CC3CCC3)CC2)n1 REAL300019150416
Cn1ncc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cnc21 REAL300019150417
O=C(O)c1csc(N2CCN(Cc3cnc(Cl)c(F)c3)CC2)n1 REAL300019150418
O=C(O)c1csc(N2CCN(CC#Cc3ccccc3)CC2)n1 REAL300019150419
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(Cl)cc1O REAL300019150420
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C(C)(C)C REAL300019150421
O=C(O)c1csc(N2CCN(Cc3cccc(CC4CCC4)c3)CC2)n1 REAL300019150422
Cc1cc(C)c(C=CCN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)c1 REAL300019150423
COc1c(C)cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C REAL300019150424
COCC1(CN2CCN(c3nc(C(=O)O)cs3)CC2)CCC1 REAL300019150425
NS(=O)(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150426
Nc1c(Cl)cc(Cl)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150427
CCn1ncnc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150428
Cc1ccnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1Br REAL300019150429
CC1(C)OC[C@H](CN2CCN(c3nc(C(=O)O)cs3)CC2)O1 REAL300019150430
CCOc1cc(F)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150431
O=C(O)c1csc(N2CCN(Cc3ccc(OC(F)F)cc3F)CC2)n1 REAL300019150432
CC(C)(C)Oc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150433
Cc1c(Cl)cccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150434
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(F)cc1C REAL300019150435
O=C(O)c1csc(N2CCN(Cc3cn(CC4CCCO4)nn3)CC2)n1 REAL300019150436
CCCn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150437
CC(C)(C)c1csc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150438
COCCc1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150439
O=C(O)c1csc(N2CCN(Cc3cnc4c(F)cccc4c3)CC2)n1 REAL300019150440
Cc1cc(C)c(C=CCN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150441
O=C(O)c1csc(N2CCN(CCCC(F)(F)F)CC2)n1 REAL300019150442
CN1CCC(CN2CCN(c3nc(C(=O)O)cs3)CC2)CC1 REAL300019150443
O=C(O)c1csc(N2CCN(CCc3cc(Cl)cc(Cl)c3)CC2)n1 REAL300019150444
Cc1ccc(CCN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150445
O=C(O)c1csc(N2CCN(Cc3cccc4ncccc34)CC2)n1 REAL300019150446
CCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150447
O=C(O)c1csc(N2CCN(Cc3ccc4nccnc4c3)CC2)n1 REAL300019150448
Cc1n[nH]cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150449
O=C(O)c1csc(N2CCN(Cc3cscn3)CC2)n1 REAL300019150450
Cn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(=O)n(C)c1=O REAL300019150451
O=C(O)c1csc(N2CCN(Cc3ccc(-c4cccnc4)o3)CC2)n1 REAL300019150452
Cc1nn(CCO)c(C)c1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150453
CCc1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cs1 REAL300019150454
O=C(O)c1csc(N2CCN(Cc3csc(-c4ccsc4)n3)CC2)n1 REAL300019150455
CC(C)(C)c1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150456
CC(C)(C)c1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cs1 REAL300019150457
Cc1ccc(-c2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)s2)cc1 REAL300019150458
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1SC REAL300019150459
CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OCC REAL300019150460
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)c(F)c3)CC2)n1 REAL300019150461
Cc1cc(C)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150462
CC(C)Oc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150463
O=C(O)c1csc(N2CCN(Cc3ccccc3O)CC2)n1 REAL300019150464
O=C(O)c1csc(N2CCN(Cc3cc(Br)ccc3O)CC2)n1 REAL300019150465
CCOc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1O REAL300019150466
O=C(O)c1csc(N2CCN(CC=Cc3ccccc3[N+](=O)[O-])CC2)n1 REAL300019150467
O=C(O)c1csc(N2CCN(Cc3cccc(OC(F)F)c3)CC2)n1 REAL300019150468
O=C(O)c1csc(N2CCN(Cc3csc([N+](=O)[O-])c3)CC2)n1 REAL300019150469
CCOCc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1OC REAL300019150470
Cc1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cccc1[N+](=O)[O-] REAL300019150471
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(O)c1 REAL300019150472
COC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)[nH]c1C REAL300019150473
NS(=O)(=O)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150474
COC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cs1 REAL300019150475
COC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)[nH]c1C(C)C REAL300019150476
O=C(O)c1csc(N2CCN(Cc3cccc4c3CCOC4)CC2)n1 REAL300019150477
O=C(O)c1csc(N2CCN(Cc3ccc4oc(=O)oc4c3)CC2)n1 REAL300019150478
Cn1nc2c(c1CN1CCN(c3nc(C(=O)O)cs3)CC1)CSCC2 REAL300019150479
COc1cc(C)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1O REAL300019150480
O=C(O)c1csc(N2CCN(Cc3cc(F)cc(F)c3O)CC2)n1 REAL300019150481
O=C(O)c1csc(N2CCN(CCc3ccc(F)c(F)c3)CC2)n1 REAL300019150482
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)cn3)CC2)n1 REAL300019150483
Cc1[nH]nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C REAL300019150484
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(F)c1OC REAL300019150485
CCc1[nH]c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C(=O)OC REAL300019150486
Cc1coc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150487
O=C(O)c1csc(N2CCN(CC=Cc3cccc(F)c3)CC2)n1 REAL300019150488
COC(=O)c1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150489
COC(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(F)c1 REAL300019150490
O=C(O)c1csc(N2CCN(Cc3cccc(Oc4ccccn4)c3)CC2)n1 REAL300019150491
CC(C)(C)c1coc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150492
CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(O)c1 REAL300019150493
O=C(O)c1csc(N2CCN(Cc3cc(Cl)cc([N+](=O)[O-])c3O)CC2)n1 REAL300019150494
COc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1O REAL300019150495
O=C(O)c1csc(N2CCN(Cc3cc(Cl)ccc3O)CC2)n1 REAL300019150496
O=C(O)c1csc(N2CCN(Cc3cc(Cl)cc(Cl)c3O)CC2)n1 REAL300019150497
O=C(O)c1csc(N2CCN(Cc3cccc([N+](=O)[O-])c3O)CC2)n1 REAL300019150498
O=C(O)c1csc(N2CCN(Cc3cccc(Br)c3O)CC2)n1 REAL300019150499
O=C(O)c1csc(N2CCN(Cc3cc4c(cc3O)OCO4)CC2)n1 REAL300019150500
O=C(O)c1csc(N2CCN(Cc3cc(-c4ccccc4)ccc3O)CC2)n1 REAL300019150501
CC(=Cc1ccccc1)CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150502
O=C(O)c1csc(N2CCN(CC3=Cc4ccccc4OC3)CC2)n1 REAL300019150503
O=C(O)c1csc(N2CCN(Cc3nc(-c4ccccc4)cs3)CC2)n1 REAL300019150504
N#CCCCOc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150505
O=C(O)c1csc(N2CCN(Cc3cnc4ccnn4c3)CC2)n1 REAL300019150506
O=C(O)c1csc(N2CCN(Cc3cccnc3Cl)CC2)n1 REAL300019150507
O=C(O)c1csc(N2CCN(Cc3cnc(N4CCOCC4)s3)CC2)n1 REAL300019150508
O=C(O)c1csc(N2CCN(Cc3cc(F)c(F)c(F)c3)CC2)n1 REAL300019150509
O=C(O)c1csc(N2CCN(Cc3cnn(-c4ccc(F)cc4)c3)CC2)n1 REAL300019150510
COc1cc2c(c(CN3CCN(c4nc(C(=O)O)cs4)CC3)c1)OC(C)C2 REAL300019150511
O=C(O)c1csc(N2CCN(Cc3cccc(OC(F)(F)F)c3)CC2)n1 REAL300019150512
C=CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1Cl REAL300019150513
Cn1ccnc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150514
CC(C#N)Oc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150515
O=C(O)c1csc(N2CCN(Cc3nccn3CC(F)(F)F)CC2)n1 REAL300019150516
O=C(O)c1csc(N2CCN(Cc3cnc(-c4ccccc4)s3)CC2)n1 REAL300019150517
O=C(O)c1csc(N2CCN(Cc3nccc4c3CCCC4)CC2)n1 REAL300019150518
Cc1nn(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1Cl REAL300019150519
COC(=O)c1sccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150520
O=C(O)c1csc(N2CCN(Cc3cnn(CCF)c3)CC2)n1 REAL300019150521
O=C(O)c1csc(N2CCN(Cc3cnc4n3CCOC4)CC2)n1 REAL300019150522
Cn1ccc(-c2nc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cs2)n1 REAL300019150523
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)c1 REAL300019150524
Cc1c(Cl)ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1Cl REAL300019150525
CC1Cc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc2O1 REAL300019150526
O=C(O)c1csc(N2CCN(Cc3cccc4[nH]c(=O)oc34)CC2)n1 REAL300019150527
O=C(O)c1csc(N2CCN(Cc3cccc4c3OCC4)CC2)n1 REAL300019150528
CSCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150529
O=C(O)c1csc(N2CCN(Cc3cnn(CC4CCC4)c3)CC2)n1 REAL300019150530
Cn1nc2c(c1CN1CCN(c3nc(C(=O)O)cs3)CC1)COCC2 REAL300019150531
Cn1nc2c(c1CN1CCN(c3nc(C(=O)O)cs3)CC1)CCC2 REAL300019150532
O=C(O)c1csc(N2CCN(Cc3ccnn3C3CCC3)CC2)n1 REAL300019150533
O=C(O)c1csc(N2CCN(Cc3cnn(C4CCC4)c3)CC2)n1 REAL300019150534
CCc1nnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150535
Cc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1Br REAL300019150536
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)CCCO4)CC2)n1 REAL300019150537
CN(C)C(=O)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150538
O=C(O)c1csc(N2CCN(Cc3ccc(C(F)F)c(F)c3)CC2)n1 REAL300019150539
COC(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150540
C=C(CCC#N)CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150541
O=C(O)c1csc(N2CCN(Cc3cc(C4CC4)[nH]n3)CC2)n1 REAL300019150542
Cn1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C1CC1 REAL300019150543
COCn1ncc(C)c1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150544
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nc1 REAL300019150545
O=C(O)c1csc(N2CCN(Cc3cccnn3)CC2)n1 REAL300019150546
O=C(O)c1csc(N2CCN(Cc3csc(C(F)(F)F)n3)CC2)n1 REAL300019150547
CCn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150548
CC(C)Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150549
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c2c(n1)CCCC2 REAL300019150550
CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150551
O=C(O)c1csc(N2CCN(Cc3cn4ccnc4s3)CC2)n1 REAL300019150552
Cc1oc(C(C)(C)C)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150553
Cc1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)sc1C REAL300019150554
O=C(O)c1csc(N2CCN(Cc3cn(Cc4ccccc4)nn3)CC2)n1 REAL300019150555
O=C(O)c1csc(N2CCN(Cc3cc(O)cc(Cl)c3)CC2)n1 REAL300019150556
COc1nccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1F REAL300019150557
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150558
COCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150559
CCn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)n1 REAL300019150560
O=C(O)c1csc(N2CCN(Cc3cnc(CC(F)(F)F)s3)CC2)n1 REAL300019150561
CC(C)(C)c1nnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150562
CCc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)no1 REAL300019150563
O=C(O)c1csc(N2CCN(Cc3ncc(Br)cc3O)CC2)n1 REAL300019150564
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(O)c1OC REAL300019150565
COC(=O)c1cc2oc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc2[nH]1 REAL300019150566
O=C(O)c1csc(N2CCN(Cc3ccn(CCF)n3)CC2)n1 REAL300019150567
O=C(O)c1csc(N2CCN(Cc3csc(-c4cccs4)n3)CC2)n1 REAL300019150568
O=C(O)c1csc(N2CCN(Cc3cccc4cc[nH]c34)CC2)n1 REAL300019150569
O=C(O)c1csc(N2CCN(Cc3nccs3)CC2)n1 REAL300019150570
O=C(O)c1csc(N2CCN(Cc3cncnc3)CC2)n1 REAL300019150571
O=C(O)c1csc(N2CCN(Cc3cnc4ccccc4c3)CC2)n1 REAL300019150572
Cn1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)nc2ccccc21 REAL300019150573
CS(=O)(=O)Nc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150574
O=C(O)c1csc(N2CCN(Cc3cccc4[nH]ccc34)CC2)n1 REAL300019150575
Cn1cncc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150576
Cc1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c[nH]1 REAL300019150577
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)[nH]n1 REAL300019150578
NC(=O)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150579
CN(C)c1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150580
Cn1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c2ccccc21 REAL300019150581
Cn1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150582
CCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150583
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150584
O=C(O)c1csc(N2CCN(Cc3cccc(F)c3F)CC2)n1 REAL300019150585
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(Cl)c1OC REAL300019150586
CC1(C)Cc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc2O1 REAL300019150587
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1F REAL300019150588
Cc1ccccc1-c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150589
O=C(O)c1csc(N2CCN(Cc3ccnc(-c4ccccc4)n3)CC2)n1 REAL300019150590
Cc1ncccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150591
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1[N+](=O)[O-] REAL300019150592
CC(C)COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150593
Cc1ccc(O)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150594
COCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150595
O=C(O)c1csc(N2CCN(Cc3cc4sccc4nc3Cl)CC2)n1 REAL300019150596
CC1(C)CCc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc2O1 REAL300019150597
O=C(O)c1csc(N2CCN(Cc3cc(C(F)(F)F)ccc3F)CC2)n1 REAL300019150598
CCn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150599
CC(C)n1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150600
O=C(O)c1csc(N2CCN(Cc3cc4ccccc4nc3O)CC2)n1 REAL300019150601
O=C(O)c1csc(N2CCN(Cc3cc(Br)co3)CC2)n1 REAL300019150602
C#CCCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150603
O=C(O)c1csc(N2CCN(Cc3csc(C4CC4)n3)CC2)n1 REAL300019150604
O=C(O)c1csc(N2CCN(Cc3cc(C4CC4)on3)CC2)n1 REAL300019150605
O=C(O)c1csc(N2CCN(Cc3cnc(C4CCOCC4)o3)CC2)n1 REAL300019150606
N#CCc1ccc(O)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150607
O=C(O)c1csc(N2CCN(Cc3cc(C4CCC4)on3)CC2)n1 REAL300019150608
CC1(c2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)no2)CC1 REAL300019150609
CCc1ccccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150610
CN(C)C(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150611
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)c1C REAL300019150612
CCNC(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150613
O=C(O)c1csc(N2CCN(Cc3cnc4n3CCCCC4)CC2)n1 REAL300019150614
O=C(O)c1csc(N2CCN(Cc3ccnc(Cl)c3)CC2)n1 REAL300019150615
Cc1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cnn1C(C)C REAL300019150616
O=C(O)c1csc(N2CCN(Cc3cc(-c4ccccc4)no3)CC2)n1 REAL300019150617
COc1ccc2sc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc2c1 REAL300019150618
CCN1CCc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc21 REAL300019150619
COC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n(C)n1 REAL300019150620
O=C(O)c1csc(N2CCN(Cc3cccc4ccsc34)CC2)n1 REAL300019150621
COc1ccc(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150622
Cc1cc(F)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150623
CCN(C)C(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150624
CSc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1Cl REAL300019150625
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1C1CC1 REAL300019150626
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C1CC1 REAL300019150627
Cc1ccn(-c2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)c(C)c2)n1 REAL300019150628
CCOc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccn1 REAL300019150629
Cn1cnc2cccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)c21 REAL300019150630
COC(=O)CCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150631
O=C(O)c1csc(N2CCN(Cc3ncccc3F)CC2)n1 REAL300019150632
Cc1cc(Br)cnc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150633
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)cc3O)CC2)n1 REAL300019150634
Cc1cc(-n2ccnc2)ccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150635
O=C(O)c1csc(N2CCN(Cc3ccc(OC4CC4)cc3)CC2)n1 REAL300019150636
Cc1cc(-n2ccnc2C)ccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150637
Cc1ncn(-c2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc2)c1C REAL300019150638
CNC(=O)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150639
O=C(O)c1csc(N2CCN(Cc3ccc(C4CC4)c(C4CC4)c3)CC2)n1 REAL300019150640
CN(C)CCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150641
CCNC(=O)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150642
Cc1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)oc2ccc(F)cc12 REAL300019150643
CCCn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)n1 REAL300019150644
CCn1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150645
O=C(O)c1csc(N2CCN(Cc3cc(Cl)ccn3)CC2)n1 REAL300019150646
CC(C)(C)c1c[nH]c(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150647
O=C(O)c1csc(N2CCN(Cc3ccc(CC4CC4)s3)CC2)n1 REAL300019150648
Cn1cc(Cl)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150649
CSc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150650
COC(=O)c1cnc(C(C)N2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150651
C[C@H]1CC(N2CCN(c3nc(C(=O)O)cs3)CC2)c2ccsc2S1 REAL300019150652
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)OCC4)CC2)n1 REAL300019150653
O=C(O)c1csc(N2CCN(Cc3nc4c([nH]3)CCCC4)CC2)n1 REAL300019150654
O=C(O)c1csc(N2CCN(Cc3cn4cc(Cl)ccc4n3)CC2)n1 REAL300019150655
C#CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150656
C=CCc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(OC)c1O REAL300019150657
CCn1ccnc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150658
CN(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150659
Cc1ccc(F)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150660
O=C(O)c1csc(N2CCN(Cc3occc3Br)CC2)n1 REAL300019150661
Cc1csc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150662
O=C(O)c1csc(N2CCN(Cc3ccc(OCC(F)F)cc3)CC2)n1 REAL300019150663
O=C(O)c1csc(N2CCN(CC3CCCCCC3)CC2)n1 REAL300019150664
O=C(O)c1csc(N2CCN(CC3=CCCOC3)CC2)n1 REAL300019150665
Cc1nc(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150666
O=C(O)c1csc(N2CCN(Cc3ccc(Br)cn3)CC2)n1 REAL300019150667
O=C(O)c1csc(N2CCN(Cc3ccc(CO)o3)CC2)n1 REAL300019150668
CCN(CC)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150669
Cn1nnc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc21 REAL300019150670
O=C(O)c1csc(N2CCN(Cc3nccc4ccccc34)CC2)n1 REAL300019150671
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1Cl REAL300019150672
Cn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150673
CC1(C)Cc2cccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)c2O1 REAL300019150674
Cc1cccn2c(CN3CCN(c4nc(C(=O)O)cs4)CC3)cnc12 REAL300019150675
Cc1cc(O)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C REAL300019150676
COCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150677
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)CCC4)CC2)n1 REAL300019150678
O=C(O)c1csc(N2CCN(Cc3cccc(-c4ccncc4)c3)CC2)n1 REAL300019150679
O=C(O)c1csc(N2CCN(Cc3ccc(Oc4cnccn4)cc3)CC2)n1 REAL300019150680
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1C#N REAL300019150681
O=C(O)c1csc(N2CCN(Cc3cc4cc(F)ccc4o3)CC2)n1 REAL300019150682
N#Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150683
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1O REAL300019150684
CC(C)Cn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150685
O=C(O)c1csc(N2CCN(Cc3nc(C4CC4)cs3)CC2)n1 REAL300019150686
Cc1c(C(F)(F)F)n[nH]c1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150687
Cc1ccoc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150688
COCc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150689
CCc1ccc(-c2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)o2)cc1 REAL300019150690
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1-n1cncn1 REAL300019150691
Cc1ncsc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150692
COCCn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150693
Cc1cc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)oc2cc1C REAL300019150694
O=C(O)c1csc(N2CCN(Cc3ccc(-n4ccnc4)nc3)CC2)n1 REAL300019150695
CN(C)C(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)[nH]1 REAL300019150696
CS(=O)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150697
COC(=O)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c[nH]1 REAL300019150698
O=C(O)c1csc(N2CCN(Cc3cnc(-c4ccsc4)s3)CC2)n1 REAL300019150699
O=C(O)c1csc(N2CCN(Cc3ccccc3C3CC3)CC2)n1 REAL300019150700
N#Cc1csc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150701
O=C(O)c1csc(N2CCN(Cc3cnc(-c4cccnc4)s3)CC2)n1 REAL300019150702
O=C(O)c1csc(N2CCN(Cc3cnc(C4CCCCC4)s3)CC2)n1 REAL300019150703
CCc1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150704
COc1cc(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC REAL300019150705
Cn1nncc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150706
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1Br REAL300019150707
O=C(O)c1csc(N2CCN(Cc3cnc(-c4cccs4)s3)CC2)n1 REAL300019150708
N#Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150709
Cc1cccc2ncc(CN3CCN(c4nc(C(=O)O)cs4)CC3)n12 REAL300019150710
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)nc3)CC2)n1 REAL300019150711
CCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150712
O=C(O)c1csc(N2CCN(Cc3cccc(-n4cccn4)c3)CC2)n1 REAL300019150713
O=C(O)c1csc(N2CCN(Cc3cnc(C4CCC4)s3)CC2)n1 REAL300019150714
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cnc1Cl REAL300019150715
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)s1 REAL300019150716
O=C(O)c1csc(N2CCN(Cc3ccc(N4CCCC4)nc3)CC2)n1 REAL300019150717
CC(C)c1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150718
O=C(O)c1csc(N2CCN(Cc3cc4ccccc4s3)CC2)n1 REAL300019150719
O=C(O)c1csc(N2CCN(Cc3ccc(F)cc3Cl)CC2)n1 REAL300019150720
O=C(O)c1csc(N2CCN(Cc3cc(F)c(F)cc3F)CC2)n1 REAL300019150721
NC(=O)c1csc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150722
O=C(O)c1csc(N2CCN(Cc3cncs3)CC2)n1 REAL300019150723
O=C(O)c1csc(N2CCN(Cc3cc(-c4ccccc4)[nH]n3)CC2)n1 REAL300019150724
O=C(O)c1csc(N2CCN(Cc3cnc(C4CC4)s3)CC2)n1 REAL300019150725
O=C(O)c1csc(N2CCN(Cc3cnc(C4CCCC4)s3)CC2)n1 REAL300019150726
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nc1 REAL300019150727
Cc1cc(Br)ccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150728
O=C(O)c1csc(N2CCN(Cc3cccc(Cl)c3F)CC2)n1 REAL300019150729
O=C(O)c1csc(N2CCN(Cc3cccc(-c4cccnc4)c3)CC2)n1 REAL300019150730
Cc1ccc(-c2cccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)c2)cc1 REAL300019150731
O=C(O)c1csc(N2CCN(Cc3cnn(CC(F)(F)F)c3)CC2)n1 REAL300019150732
CCOc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150733
CC(C)Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150734
O=C(O)c1csc(N2CCN(Cc3cc(Cl)cc4cccnc34)CC2)n1 REAL300019150735
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)COC4)CC2)n1 REAL300019150736
COc1ccsc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150737
Cc1ccc(-c2ncc(CN3CCN(c4nc(C(=O)O)cs4)CC3)s2)o1 REAL300019150738
COCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150739
COc1nc2ccccc2cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150740
O=C(O)c1csc(N2CCN(Cc3cc(Cl)ccc3Cl)CC2)n1 REAL300019150741
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1F REAL300019150742
O=C(O)c1csc(N2CCN(Cc3cncc4ccccc34)CC2)n1 REAL300019150743
O=C(O)c1csc(N2CCN(Cc3ncccc3C(F)(F)F)CC2)n1 REAL300019150744
O=C(O)c1csc(N2CCN(CC=Cc3ccc(Cl)cc3)CC2)n1 REAL300019150745
Cc1oc2ccccc2c1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150746
O=C(O)c1csc(N2CCN(CC3CC3c3ccccc3)CC2)n1 REAL300019150747
O=C(O)c1csc(N2CCN(Cc3cscc3Cl)CC2)n1 REAL300019150748
O=C(O)c1csc(N2CCN(Cc3cnc4ccsc4c3)CC2)n1 REAL300019150749
Cc1cc(Cl)cc(C)c1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150750
CCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nc1 REAL300019150751
Cc1nn2c(CN3CCN(c4nc(C(=O)O)cs4)CC3)c(C)nc2s1 REAL300019150752
Cn1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)nc2cc(Cl)ccc21 REAL300019150753
CC1CCc2nc(CN3CCN(c4nc(C(=O)O)cs4)CC3)sc2C1 REAL300019150754
CC(C)Cc1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150755
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccncc4)cc3F)CC2)n1 REAL300019150756
O=C(O)c1csc(N2CCN(Cc3c(Cl)oc4ccccc34)CC2)n1 REAL300019150757
CC1(C)CCc2nc(CN3CCN(c4nc(C(=O)O)cs4)CC3)sc2C1 REAL300019150758
CCc1nn(C)c(CC)c1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150759
O=C(O)c1csc(N2CCN(Cc3cnc(C4CCCO4)s3)CC2)n1 REAL300019150760
CC1(C)CCC(CN2CCN(c3nc(C(=O)O)cs3)CC2)CC1 REAL300019150761
COC(=O)c1occc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150762
COc1ccc(O)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150763
Cc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1O REAL300019150764
O=C(O)c1csc(N2CCN(Cc3cccc(Cl)c3O)CC2)n1 REAL300019150765
O=C(O)c1csc(N2CCN(Cc3cc(Cl)cc(F)c3O)CC2)n1 REAL300019150766
COc1cc(O)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC REAL300019150767
O=C(O)c1csc(N2CCN(Cc3cccc4nccn34)CC2)n1 REAL300019150768
CCCC1CCC(CN2CCN(c3nc(C(=O)O)cs3)CC2)CC1 REAL300019150769
CC(CCc1ccccc1)CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150770
CC(C)COc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150771
Cn1cnc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc21 REAL300019150772
O=C(O)c1csc(N2CCN(Cc3ccn(-c4ccccc4)n3)CC2)n1 REAL300019150773
CCc1nn(C)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150774
O=C(O)c1csc(N2CCN(Cc3nc4c(s3)CCC4)CC2)n1 REAL300019150775
COc1ccc(C(C)CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150776
O=C(O)c1csc(N2CCN(Cc3nc4c(s3)CCCC4)CC2)n1 REAL300019150777
O=C(O)c1csc(N2CCN(Cc3ccn(C(F)F)n3)CC2)n1 REAL300019150778
CC(CCc1cccc(F)c1)N1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150779
CC(Cc1ccsc1)N1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150780
Cc1ccc(F)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150781
COc1c(O)cccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150782
O=C(O)c1csc(N2CCN(Cc3cc(F)ccc3O)CC2)n1 REAL300019150783
O=C(O)c1csc(N2CCN(CCc3ccc(F)cc3)CC2)n1 REAL300019150784
O=C(O)c1csc(N2CCN(Cc3cccc(F)c3O)CC2)n1 REAL300019150785
CC(C)C1CC(CN2CCN(c3nc(C(=O)O)cs3)CC2)CCO1 REAL300019150786
CCC1CC(CN2CCN(c3nc(C(=O)O)cs3)CC2)CCO1 REAL300019150787
O=C(O)c1csc(N2CCN(Cc3c(Cl)ccc4cccnc34)CC2)n1 REAL300019150788
O=C(O)c1csc(N2CCN(Cc3ccc(SC(F)F)cc3)CC2)n1 REAL300019150789
CC(C)Cn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150790
COC(=O)COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150791
CCOCOc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150792
CC(Cc1ccccc1)CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150793
O=C(O)c1csc(N2CCN(Cc3cn(Cc4cccnc4)nn3)CC2)n1 REAL300019150794
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc2cccnc12 REAL300019150795
CC(C)(C)C1CCC(CN2CCN(c3nc(C(=O)O)cs3)CC2)CC1 REAL300019150796
CC(C)c1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150797
COC(=O)c1coc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150798
COc1ccc(CC(C)CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150799
O=C(O)c1csc(N2CCN(CC=Cc3ccc(F)cc3F)CC2)n1 REAL300019150800
CC(CC1CCCCC1)CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150801
CC(C)(C)OC(=O)N1CC(CN2CCN(c3nc(C(=O)O)cs3)CC2)C1 REAL300019150802
O=C(O)c1csc(N2CCN(Cc3ccc([N+](=O)[O-])c(Cl)c3)CC2)n1 REAL300019150803
COc1cc(Cl)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1O REAL300019150804
COc1cc2c(cc1CN1CCN(c3nc(C(=O)O)cs3)CC1)OCO2 REAL300019150805
O=C(O)c1csc(N2CCN(Cc3cnn4ncccc34)CC2)n1 REAL300019150806
O=C(O)c1csc(N2CCN(CC3CC4CCC3C4)CC2)n1 REAL300019150807
O=C(O)c1csc(N2CCN(Cc3cccn4nccc34)CC2)n1 REAL300019150808
O=C(O)c1csc(N2CCN(Cc3sccc3Br)CC2)n1 REAL300019150809
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150810
CC(C)c1ccc(CCN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150811
O=C(O)c1csc(N2CCN(Cc3cncc(Br)c3)CC2)n1 REAL300019150812
CCn1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c2ccccc21 REAL300019150813
O=C(O)c1csc(N2CCN(Cc3ncc(Cl)s3)CC2)n1 REAL300019150814
CCOC(=O)c1nn(C)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150815
O=C(O)c1csc(N2CCN(CCSCc3ccccc3)CC2)n1 REAL300019150816
CN1C(=O)CCc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc21 REAL300019150817
Cc1ccncc1CCCN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150818
COC(=O)C(C)(C)CCN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150819
CC1(c2ccccc2)CCC(N2CCN(c3nc(C(=O)O)cs3)CC2)C1 REAL300019150820
O=C(O)c1csc(N2CCN(Cc3cc4c(F)cccc4[nH]3)CC2)n1 REAL300019150821
O=C(O)c1csc(N2CCN(CC3CCc4ccccc43)CC2)n1 REAL300019150822
CC(C)(C)OC(=O)NCCCN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150823
O=C(O)c1csc(N2CCN(CCC3CCOC3)CC2)n1 REAL300019150824
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)sn1 REAL300019150825
COC(=O)Cc1coc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150826
O=C(O)c1csc(N2CCN(Cc3nc4c([nH]3)COCC4)CC2)n1 REAL300019150827
O=C(O)c1csc(N2CCN(Cc3noc4c3COCC4)CC2)n1 REAL300019150828
Cn1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1Br REAL300019150829
O=C(O)c1csc(N2CCN(CC=Cc3ccccc3)CC2)n1 REAL300019150830
O=C(O)c1csc(N2CCN(Cc3cnnn3C3CC3)CC2)n1 REAL300019150831
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)COCC4)CC2)n1 REAL300019150832
Cc1nc(N2CCCC2)sc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150833
O=C(O)c1csc(N2CCN(Cc3cnn(CCO)c3)CC2)n1 REAL300019150834
Cc1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)sc2cc(F)ccc12 REAL300019150835
O=C(O)c1csc(N2CCN(Cc3cc(-c4ccncc4)n[nH]3)CC2)n1 REAL300019150836
O=C(O)c1csc(N2CCN(CC=Cc3ccncc3)CC2)n1 REAL300019150837
C=Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150838
O=C(O)c1csc(N2CCN(Cc3cccc(OCC4CCC4)c3)CC2)n1 REAL300019150839
CC(F)(F)c1ccccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150840
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1OCCO REAL300019150841
CCc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nc1 REAL300019150842
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OCCO REAL300019150843
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150844
O=C(O)c1csc(N2CCN(Cc3ccc4ccncc4c3)CC2)n1 REAL300019150845
Cc1cc2cccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)c2o1 REAL300019150846
COc1csc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1OC REAL300019150847
CN(C)c1nc(Cl)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150848
Cn1c(=O)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc2ccccc21 REAL300019150849
Cc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150850
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccsc4)cc3)CC2)n1 REAL300019150851
O=C(O)c1csc(N2CCN(Cc3nc4ccccc4s3)CC2)n1 REAL300019150852
O=C(O)c1csc(N2CCN(Cc3[nH]ncc3Br)CC2)n1 REAL300019150853
O=C(O)c1csc(N2CCN(Cc3ccc4nsnc4c3)CC2)n1 REAL300019150854
O=C(O)c1csc(N2CCN(Cc3ccc4nonc4c3)CC2)n1 REAL300019150855
O=C(O)c1csc(N2CCN(Cc3cccc4nsnc34)CC2)n1 REAL300019150856
N#Cc1cnn2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cnc12 REAL300019150857
O=C(O)c1csc(N2CCN(Cc3cn(-c4ccccc4)nn3)CC2)n1 REAL300019150858
Cc1oc(-c2cccs2)nc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150859
Cn1nc(-c2ccccc2)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150860
CC(C)(C)c1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n[nH]1 REAL300019150861
CCN1CCCc2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)ccc21 REAL300019150862
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccsc4)nc3)CC2)n1 REAL300019150863
O=C(O)c1csc(N2CCN(Cc3cc4ccccc4cn3)CC2)n1 REAL300019150864
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(Cl)n1 REAL300019150865
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(C)n1 REAL300019150866
O=C(O)c1csc(N2CCN(Cc3ccc[nH]c3=O)CC2)n1 REAL300019150867
O=C(O)c1csc(N2CCN(Cc3cc4ccc(F)cc4[nH]c3=O)CC2)n1 REAL300019150868
O=C(O)c1csc(N2CCN(Cc3noc4c3CCCC4)CC2)n1 REAL300019150869
Cc1cn(C)nc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150870
Cc1coc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150871
O=C(O)c1csc(N2CCN(Cc3cc4ccncc4s3)CC2)n1 REAL300019150872
COc1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)ccc1C REAL300019150873
O=C(O)c1csc(N2CCN(Cc3cc4ncccc4o3)CC2)n1 REAL300019150874
O=C(O)c1csc(N2CCN(Cc3nc(CO)cs3)CC2)n1 REAL300019150875
O=C(O)c1csc(N2CCN(Cc3cccc4cc(Cl)ccc34)CC2)n1 REAL300019150876
CCCn1cncc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150877
CCc1c[nH]c(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150878
O=C(O)c1csc(N2CCN(Cc3cncc(-c4cccnc4)c3)CC2)n1 REAL300019150879
CC(C)(C)c1cncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150880
O=C(O)c1csc(N2CCN(Cc3ccc4c(c3)CCOC4)CC2)n1 REAL300019150881
O=C(O)c1csc(N2CCN(Cc3cccc(C(F)F)c3F)CC2)n1 REAL300019150882
O=C(O)c1csc(N2CCN(Cc3nc4c(s3)CCCCC4)CC2)n1 REAL300019150883
O=C(O)c1csc(N2CCN(Cc3nc4c(s3)COCC4)CC2)n1 REAL300019150884
CSc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150885
O=C(O)c1csc(N2CCN(Cc3cnn(C4CCCCC4)c3)CC2)n1 REAL300019150886
CC(C)n1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150887
O=C(O)c1csc(N2CCN(Cc3ccn(CC(F)(F)F)n3)CC2)n1 REAL300019150888
CC(F)(F)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150889
Cc1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)oc1C REAL300019150890
CS(=O)(=O)c1coc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150891
O=C(O)c1csc(N2CCN(Cc3cn(CC4CC4)nn3)CC2)n1 REAL300019150892
O=C(O)c1csc(N2CCN(Cc3cccn3C(F)F)CC2)n1 REAL300019150893
O=C(O)c1csc(N2CCN(Cc3cc4c(o3)CCCC4)CC2)n1 REAL300019150894
Cn1cc(Br)nc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150895
COc1nn(C)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150896
CN(CCO)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150897
Cn1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)nc2c1CCCC2 REAL300019150898
O=C(O)c1csc(N2CCN(Cc3cccc4c3COCC4)CC2)n1 REAL300019150899
CC(C)(C#N)c1ncc(CN2CCN(c3nc(C(=O)O)cs3)CC2)s1 REAL300019150900
CCn1nc(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150901
COc1sccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150902
O=C(O)c1csc(N2CCN(Cc3cc(C4CCC4)[nH]n3)CC2)n1 REAL300019150903
C=CCCn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)nn1 REAL300019150904
O=C(O)c1csc(N2CCN(Cc3ccc(CC4CCC4)cc3)CC2)n1 REAL300019150905
COc1nsc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1Cl REAL300019150906
O=C(O)c1csc(N2CCN(Cc3cn(C4CC4)cn3)CC2)n1 REAL300019150907
Cn1nnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C(F)F REAL300019150908
Cc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1OC(F)F REAL300019150909
CC1Oc2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc2C1C REAL300019150910
O=C(O)c1csc(N2CCN(Cc3ccnn3C3CC3(F)F)CC2)n1 REAL300019150911
COCc1nocc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150912
O=C(O)c1csc(N2CCN(Cc3ccc(C(F)F)cn3)CC2)n1 REAL300019150913
O=C(O)c1csc(N2CCN(Cc3ccc(C(F)(F)F)cc3F)CC2)n1 REAL300019150914
CC(C)Oc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1F REAL300019150915
CCn1cc(Cl)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150916
O=C(O)c1csc(N2CCN(Cc3ccc(F)c(Cl)c3F)CC2)n1 REAL300019150917
O=C(O)c1csc(N2CCN(Cc3cccc(C(F)F)c3)CC2)n1 REAL300019150918
O=C(O)c1csc(N2CCN(Cc3ccc4ccccc4c3F)CC2)n1 REAL300019150919
CS(=O)(=O)c1csc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150920
O=C(O)c1csc(N2CCN(Cc3csc(Cl)c3)CC2)n1 REAL300019150921
Cc1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cnn1C1CCC1 REAL300019150922
Cc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n(C2CCCC2)n1 REAL300019150923
O=C(O)c1csc(N2CCN(Cc3ccnn3CC(F)F)CC2)n1 REAL300019150924
COc1ccc(C)nc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150925
O=C(O)c1csc(N2CCN(Cc3cc(Cl)cc(Cl)n3)CC2)n1 REAL300019150926
O=C(O)c1csc(N2CCN(Cc3nccc4cc(Cl)ccc34)CC2)n1 REAL300019150927
O=C(O)c1csc(N2CCN(Cc3cc4cnccc4[nH]3)CC2)n1 REAL300019150928
O=C(O)c1csc(N2CCN(Cc3cccc(C(F)F)n3)CC2)n1 REAL300019150929
O=C(O)c1csc(N2CCN(Cc3cnn(-c4cccc(F)c4)c3)CC2)n1 REAL300019150930
CC(C)N(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(O)c1 REAL300019150931
O=C(O)c1csc(N2CCN(Cc3c(O)ccc4c3OCO4)CC2)n1 REAL300019150932
Cc1nn(-c2ccccc2)nc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150933
O=C(O)c1csc(N2CCN(Cc3ccn(C4CCC4)n3)CC2)n1 REAL300019150934
O=C(O)c1csc(N2CCN(Cc3ccn(CC(F)F)n3)CC2)n1 REAL300019150935
O=C(O)c1csc(N2CCN(Cc3ccn(C4CC4(F)F)n3)CC2)n1 REAL300019150936
Cc1nn(C2CCCCC2)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150937
O=C(O)c1csc(N2CCN(Cc3cnn(C4CCOCC4)c3)CC2)n1 REAL300019150938
Cc1nn(C2CCOCC2)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150939
Cc1cn(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150940
O=C(O)c1csc(N2CCN(Cc3noc4c3CCC4)CC2)n1 REAL300019150941
O=C(O)c1csc(N2CCN(Cc3nc4cccc(F)c4s3)CC2)n1 REAL300019150942
O=C(O)c1csc(N2CCN(Cc3ccn(C4CCCC4)n3)CC2)n1 REAL300019150943
NS(=O)(=O)c1csc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150944
O=C(O)c1csc(N2CCN(Cc3ccc(F)c4ccoc34)CC2)n1 REAL300019150945
O=C(O)c1csc(N2CCN(Cc3cc(Cl)cc4ccoc34)CC2)n1 REAL300019150946
O=C(O)c1csc(N2CCN(Cc3ncc(Cl)cc3Cl)CC2)n1 REAL300019150947
Cc1nn(C2CCCC2)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150948
O=C(O)c1csc(N2CCN(Cc3ccccc3C(F)F)CC2)n1 REAL300019150949
O=C(O)c1csc(N2CCN(Cc3ccc4[nH]ncc4c3)CC2)n1 REAL300019150950
O=C(O)c1csc(N2CCN(Cc3ccc(Cl)c(F)c3F)CC2)n1 REAL300019150951
Cc1c(F)cccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150952
Cn1cc(-c2cccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)c2)cn1 REAL300019150953
Cc1ccc(Br)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150954
COc1c(C#N)cccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150955
COc1nc2ccc(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc2s1 REAL300019150956
O=C(O)c1csc(N2CCN(Cc3ccnc(Br)c3)CC2)n1 REAL300019150957
O=C(O)c1csc(N2CCN(Cc3cc(F)cc(Cl)c3Cl)CC2)n1 REAL300019150958
Cc1nc(Cl)ccc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150959
CC(C)(C)COc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150960
COc1cc(Cl)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150961
COc1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc(F)c1F REAL300019150962
COc1cc(C)ncc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150963
COc1ccc2sc(CN3CCN(c4nc(C(=O)O)cs4)CC3)nc2c1 REAL300019150964
CC(C)n1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150965
Cc1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)nnn1C REAL300019150966
COC(=O)c1c(C)[nH]c(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C REAL300019150967
CC(C)Oc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)o1 REAL300019150968
O=C(O)c1csc(N2CCN(Cc3ccc(C(F)(F)F)cc3O)CC2)n1 REAL300019150969
Cc1oc(-c2ccccc2)nc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150970
Cn1nc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1-c1ccco1 REAL300019150971
N#Cc1cc(F)cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1 REAL300019150972
O=C(O)c1csc(N2CCN(Cc3ccc(C4CCCCC4)cc3)CC2)n1 REAL300019150973
Cc1nc(C)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)nc1C REAL300019150974
NC(=O)c1cnc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150975
Cc1nn(C2CCC2)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150976
Cc1c(CN2CCN(c3nc(C(=O)O)cs3)CC2)cnn1CC(F)F REAL300019150977
COc1ccccc1C=CCN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150978
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccccn4)nc3)CC2)n1 REAL300019150979
CCCn1nc(C)c(Cl)c1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150980
COc1cccc2[nH]c(CN3CCN(c4nc(C(=O)O)cs4)CC3)cc12 REAL300019150981
Cc1ccc(OC(F)F)c(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150982
Cn1nc(-c2ccco2)cc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150983
O=C(O)c1csc(N2CCN(Cc3ccc(Cc4ccccc4)cc3)CC2)n1 REAL300019150984
COc1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)n1 REAL300019150985
CCN(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c(C)c1 REAL300019150986
O=C(O)c1csc(N2CCN(Cc3cc(-c4ccccc4)ccn3)CC2)n1 REAL300019150987
O=C(O)c1csc(N2CCN(Cc3scc(Cl)c3Cl)CC2)n1 REAL300019150988
O=C(O)c1csc(N2CCN(Cc3ccc(CF)cc3)CC2)n1 REAL300019150989
O=C(O)c1csc(N2CCN(Cc3ccc4sccc4c3)CC2)n1 REAL300019150990
O=C(O)c1csc(N2CCN(Cc3ccc(-c4ccncc4)cc3)CC2)n1 REAL300019150991
COc1cc(C)c2cc(CN3CCN(c4nc(C(=O)O)cs4)CC3)[nH]c2c1 REAL300019150992
Cc1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)c1C(F)(F)F REAL300019150993
C=CCn1cc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cn1 REAL300019150994
O=C(O)c1csc(N2CCN(Cc3ccc4cn[nH]c4c3)CC2)n1 REAL300019150995
CCC(C)c1ccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)cc1 REAL300019150996
Cc1oncc1CN1CCN(c2nc(C(=O)O)cs2)CC1 REAL300019150997
CC(F)(F)c1cccc(CN2CCN(c3nc(C(=O)O)cs3)CC2)n1 REAL300019150998
O=C(O)c1csc(N2CCN(Cc3cc4c(nc3Cl)CCOC4)CC2)n1 REAL300019150999
O=C(O)c1csc(N2CCN(Cc3cc4sccc4[nH]3)CC2)n1 REAL300019151000
