Cc1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1-c1ccccc1 REAL300019304001
Cc1nc(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)s1 REAL300019304002
O=C(O)c1csc(CC2CCCN(Cc3ccc(Br)cn3)C2)n1 REAL300019304003
O=C(O)c1csc(CC2CCCN(Cc3ccc(CO)o3)C2)n1 REAL300019304004
O=C(O)c1csc(CC2CCCN(Cc3cccc4cn[nH]c34)C2)n1 REAL300019304005
Cn1nnc2cc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)ccc21 REAL300019304006
O=C(O)c1csc(CC2CCCN(Cc3cc(Cl)ccc3[N+](=O)[O-])C2)n1 REAL300019304007
O=C(O)c1csc(CC2CCCN(Cc3nccc4ccccc34)C2)n1 REAL300019304008
O=C(O)c1csc(CC2CCCN(Cc3cnc4ccc(Cl)cn34)C2)n1 REAL300019304009
COc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1Cl REAL300019304010
CC(C)CCn1cccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304011
Cn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nn1 REAL300019304012
CC1(C)Cc2cccc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)c2O1 REAL300019304013
Cc1cccn2c(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)cnc12 REAL300019304014
CC(C)(CCC#N)CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304015
Cc1cc(O)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1C REAL300019304016
COCc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1 REAL300019304017
O=C(O)c1csc(CC2CCCN(Cc3ccc4c(c3)CCC4)C2)n1 REAL300019304018
O=C(O)c1csc(CC2CCCN(Cc3cccc(-c4ccncc4)c3)C2)n1 REAL300019304019
COc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1C#N REAL300019304020
O=C(O)c1csc(CC2CCCN(Cc3cc4cc(F)ccc4o3)C2)n1 REAL300019304021
N#Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)o1 REAL300019304022
Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1O REAL300019304023
CC(C)Cn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nn1 REAL300019304024
O=C(O)c1csc(CC2CCCN(Cc3nc(C4CC4)cs3)C2)n1 REAL300019304025
Cc1c(C(F)(F)F)n[nH]c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304026
Cc1ccoc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304027
COCc1cccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304028
O=C(O)c1csc(CC2CCCN(CC3CCCCCCC3)C2)n1 REAL300019304029
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)ccc1-n1cncn1 REAL300019304030
CCC(C)(C)CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304031
Cc1ncsc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304032
COCCn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cn1 REAL300019304033
Cc1cc2cc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)oc2cc1C REAL300019304034
O=C(O)c1csc(CC2CCCN(Cc3ccc(-n4ccnc4)nc3)C2)n1 REAL300019304035
CN(C)C(=O)c1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)[nH]1 REAL300019304036
CS(=O)c1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1 REAL300019304037
COC(=O)c1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c[nH]1 REAL300019304038
O=C(O)c1csc(CC2CCCN(Cc3ccccc3C3CC3)C2)n1 REAL300019304039
N#Cc1csc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304040
CCc1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)s1 REAL300019304041
COc1cc(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1OC REAL300019304042
Cn1nncc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304043
N#Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)s1 REAL300019304044
Cc1cccc2ncc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)n12 REAL300019304045
COCCOc1ccccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304046
O=C(O)c1csc(CC2CCCN(Cc3ccc(Cl)nc3)C2)n1 REAL300019304047
CCc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)o1 REAL300019304048
O=C(O)c1csc(CC2CCCN(Cc3cccc(-n4cccn4)c3)C2)n1 REAL300019304049
O=C(O)c1csc(CC2CCCN(Cc3cnc(C4CCC4)s3)C2)n1 REAL300019304050
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cnc1Cl REAL300019304051
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C)s1 REAL300019304052
O=C(O)c1csc(CC2CCCN(Cc3cc(F)cc4cccnc34)C2)n1 REAL300019304053
O=C(O)c1csc(CC2CCCN(Cc3ccc(N4CCCC4)nc3)C2)n1 REAL300019304054
CC(C)c1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)s1 REAL300019304055
O=C(O)c1csc(CC2CCCN(Cc3cc4ccccc4s3)C2)n1 REAL300019304056
O=C(O)c1csc(CC2CCCN(Cc3ccc(F)cc3Cl)C2)n1 REAL300019304057
O=C(O)c1csc(CC2CCCN(Cc3cc(F)c(F)cc3F)C2)n1 REAL300019304058
CCC1(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)COC1 REAL300019304059
NC(=O)c1csc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304060
O=C(O)c1csc(CC2CCCN(Cc3cncs3)C2)n1 REAL300019304061
O=C(O)c1csc(CC2CCCN(Cc3cc(-c4ccccc4)[nH]n3)C2)n1 REAL300019304062
O=C(O)c1csc(CC2CCCN(Cc3cnc(C4CC4)s3)C2)n1 REAL300019304063
O=C(O)c1csc(CC2CCCN(Cc3cnc(C4CCCC4)s3)C2)n1 REAL300019304064
Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nc1 REAL300019304065
O=C(O)c1csc(CC2CCCN(Cc3cccc(Cl)c3F)C2)n1 REAL300019304066
O=C(O)c1csc(CC2CCCN(Cc3ccc(F)c4cccnc34)C2)n1 REAL300019304067
CCCn1nc(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1C REAL300019304068
O=C(O)c1csc(CC2CCCN(Cc3cccc(-c4cccnc4)c3)C2)n1 REAL300019304069
O=C(O)c1csc(CC2CCCN(Cc3cnn(CC(F)(F)F)c3)C2)n1 REAL300019304070
CCOc1cccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304071
CC(C)Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1 REAL300019304072
O=C(O)c1csc(CC2CCCN(Cc3ccc4c(c3)COC4)C2)n1 REAL300019304073
COc1ccsc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304074
COCc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)o1 REAL300019304075
CC(=O)Nc1ccccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304076
COc1nc2ccccc2cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304077
O=C(O)c1csc(CC2CCCN(Cc3cc(Cl)ccc3Cl)C2)n1 REAL300019304078
COc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)ccc1F REAL300019304079
O=C(O)c1csc(CC2CCCN(Cc3cncc4ccccc34)C2)n1 REAL300019304080
O=C(O)c1csc(CC2CCCN(Cc3ncccc3C(F)(F)F)C2)n1 REAL300019304081
O=C(O)c1csc(CC2CCCN(CC=Cc3ccc(Cl)cc3)C2)n1 REAL300019304082
Cc1oc2ccccc2c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304083
O=C(O)c1csc(CC2CCCN(CC3CC3c3ccccc3)C2)n1 REAL300019304084
O=C(O)c1csc(CC2CCCN(Cc3cscc3Cl)C2)n1 REAL300019304085
O=C(O)c1csc(CC2CCCN(Cc3cnc4ccsc4c3)C2)n1 REAL300019304086
Cc1cc(Cl)cc(C)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304087
CCOc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nc1 REAL300019304088
Cc1nn2c(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)c(C)nc2s1 REAL300019304089
CC1CCc2nc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)sc2C1 REAL300019304090
CC(C)Cc1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)s1 REAL300019304091
O=C(O)c1csc(CC2CCCN(Cc3c(Cl)oc4ccccc34)C2)n1 REAL300019304092
CCc1nn(C)c(CC)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304093
O=C(O)c1csc(CC2CCCN(Cc3cnc(C4CCCO4)s3)C2)n1 REAL300019304094
CC1(C)CCC(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)CC1 REAL300019304095
COC(=O)c1occc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304096
COc1ccc(O)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304097
Cc1cccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1O REAL300019304098
O=C(O)c1csc(CC2CCCN(Cc3cccc(Cl)c3O)C2)n1 REAL300019304099
O=C(O)c1csc(CC2CCCN(Cc3cc(Cl)cc(F)c3O)C2)n1 REAL300019304100
COc1cc(O)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1OC REAL300019304101
Cc1cccc(C)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304102
O=C(O)c1csc(CC2CCCN(Cc3cccc4nccn34)C2)n1 REAL300019304103
CCCC1CCC(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)CC1 REAL300019304104
CCCC(C)CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304105
CC(CCc1ccccc1)CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304106
Cn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C(C)(C)C)n1 REAL300019304107
CC(C)COc1cccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304108
Cn1cnc2cc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)ccc21 REAL300019304109
O=C(O)c1csc(CC2CCCN(Cc3ccn(-c4ccccc4)n3)C2)n1 REAL300019304110
CN(C)c1cccc(Cl)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304111
Cn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(-c2ccccc2)n1 REAL300019304112
CCc1nn(C)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304113
CC(C)(CN1CCCC(Cc2nc(C(=O)O)cs2)C1)c1ccccc1 REAL300019304114
O=C(O)c1csc(CC2CCCN(Cc3nc4c(s3)CCC4)C2)n1 REAL300019304115
CCCC(CN1CCCC(Cc2nc(C(=O)O)cs2)C1)c1ccccc1 REAL300019304116
COc1ccc(C(C)CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1 REAL300019304117
O=C(O)c1csc(CC2CCCN(Cc3nc4c(s3)CCCC4)C2)n1 REAL300019304118
O=C(O)c1csc(CC2CCCN(Cc3ccn(C(F)F)n3)C2)n1 REAL300019304119
CC(CCc1cccc(F)c1)N1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304120
CC(Cc1ccsc1)N1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304121
Cc1ccc(F)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304122
COc1c(O)cccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304123
O=C(O)c1csc(CC2CCCN(Cc3cc(F)ccc3O)C2)n1 REAL300019304124
O=C(O)c1csc(CC2CCCN(CCc3ccc(F)cc3)C2)n1 REAL300019304125
O=C(O)c1csc(CC2CCCN(Cc3cccc(F)c3O)C2)n1 REAL300019304126
CC(C)C1CC(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)CCO1 REAL300019304127
CCC1CC(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)CCO1 REAL300019304128
COCCC1(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)CCC1 REAL300019304129
O=C(O)c1csc(CC2CCCN(Cc3ccc(SC(F)F)cc3)C2)n1 REAL300019304130
COc1cc(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C)n1 REAL300019304131
CC(C)Cn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cn1 REAL300019304132
CCOCOc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1 REAL300019304133
CC(Cc1ccccc1)CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304134
O=C(O)c1csc(CC2CCCN(Cc3cn(Cc4cccnc4)nn3)C2)n1 REAL300019304135
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc2cccnc12 REAL300019304136
CC(C)(C)C1CCC(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)CC1 REAL300019304137
CC(C)c1cnc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)s1 REAL300019304138
COC(=O)c1coc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304139
O=C(O)c1csc(CC2CCCN(CC=Cc3ccc(F)cc3F)C2)n1 REAL300019304140
CC(CC1CCCCC1)CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304141
CC(C)(C)OC(=O)N1CC(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)C1 REAL300019304142
O=C(O)c1csc(CC2CCCN(Cc3ccc([N+](=O)[O-])c(Cl)c3)C2)n1 REAL300019304143
CC(C)(CN1CCCC(Cc2nc(C(=O)O)cs2)C1)NC(=O)OC(C)(C)C REAL300019304144
COc1cc(Cl)cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1O REAL300019304145
COc1cc2c(cc1CN1CCCC(Cc3nc(C(=O)O)cs3)C1)OCO2 REAL300019304146
O=C(O)c1csc(CC2CCCN(Cc3cnn4ncccc34)C2)n1 REAL300019304147
O=C(O)c1csc(CC2CCCN(CC3CC4CCC3C4)C2)n1 REAL300019304148
O=C(O)c1csc(CC2CCCN(Cc3cccn4nccc34)C2)n1 REAL300019304149
Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cn1 REAL300019304150
CC(C)c1ccc(CCN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1 REAL300019304151
CCCCOc1ccccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304152
O=C(O)c1csc(CC2CCCN(Cc3cncc(Br)c3)C2)n1 REAL300019304153
CCn1nc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c2ccccc21 REAL300019304154
O=C(O)c1csc(CC2CCCN(Cc3ncc(Cl)s3)C2)n1 REAL300019304155
CCOC(=O)c1nn(C)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304156
CC(C)(C)CCN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304157
O=C(O)c1csc(CC2CCCN(CCSCc3ccccc3)C2)n1 REAL300019304158
CN1C(=O)CCc2cc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)ccc21 REAL300019304159
Cc1ccncc1CCCN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304160
COC(=O)C(C)(C)CCN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304161
CC1(c2ccccc2)CCC(N2CCCC(Cc3nc(C(=O)O)cs3)C2)C1 REAL300019304162
O=C(O)c1csc(CC2CCCN(Cc3cc4c(F)cccc4[nH]3)C2)n1 REAL300019304163
O=C(O)c1csc(CC2CCCN(Cc3c[nH]nc3-c3ccsc3)C2)n1 REAL300019304164
Cn1ncc(Cl)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304165
O=C(O)c1csc(CC2CCCN(CC3CCc4ccccc43)C2)n1 REAL300019304166
CC(C)(C)OC(=O)NCCCN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304167
O=C(O)c1csc(CC2CCCN(CCC3CCOC3)C2)n1 REAL300019304168
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)sn1 REAL300019304169
COC(=O)Cc1coc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304170
O=C(O)c1csc(CC2CCCN(Cc3nc4c([nH]3)COCC4)C2)n1 REAL300019304171
O=C(O)c1csc(CC2CCCN(Cc3noc4c3COCC4)C2)n1 REAL300019304172
Cn1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1Br REAL300019304173
O=C(O)c1csc(CC2CCCN(CC=Cc3ccccc3)C2)n1 REAL300019304174
O=C(O)c1csc(CC2CCCN(Cc3cnnn3C3CC3)C2)n1 REAL300019304175
COCc1ccccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304176
O=C(O)c1csc(CC2CCCN(Cc3ccc4c(c3)COCC4)C2)n1 REAL300019304177
O=C(O)c1csc(CC2CCCN(Cc3cnn(CCO)c3)C2)n1 REAL300019304178
O=C(O)c1csc(CC2CCCN(Cc3cc(-c4ccncc4)n[nH]3)C2)n1 REAL300019304179
COc1ccc(F)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1OC REAL300019304180
O=C(O)c1csc(CC2CCCN(CC=Cc3ccncc3)C2)n1 REAL300019304181
Cn1ccc(-c2n[nH]cc2CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304182
C=Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1 REAL300019304183
CC(F)(F)c1ccccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304184
CCn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C2CC2)n1 REAL300019304185
CCc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nc1 REAL300019304186
COc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nn1 REAL300019304187
CC(C)(C)c1nocc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304188
O=C(O)c1csc(CC2CCCN(Cc3ccc4ccncc4c3)C2)n1 REAL300019304189
Cc1cc2cccc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)c2o1 REAL300019304190
COc1csc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1OC REAL300019304191
O=C(O)c1csc(CC2CCCN(Cc3conc3C3CCC3)C2)n1 REAL300019304192
Cn1c(=O)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc2ccccc21 REAL300019304193
Cc1cccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304194
O=C(O)c1csc(CC2CCCN(Cc3ccc(-c4ccsc4)cc3)C2)n1 REAL300019304195
O=C(O)c1csc(CC2CCCN(Cc3nc4ccccc4s3)C2)n1 REAL300019304196
O=C(O)c1csc(CC2CCCN(Cc3[nH]ncc3Br)C2)n1 REAL300019304197
O=C(O)c1csc(CC2CCCN(Cc3ccc4nsnc4c3)C2)n1 REAL300019304198
O=C(O)c1csc(CC2CCCN(Cc3ccc4nonc4c3)C2)n1 REAL300019304199
O=C(O)c1csc(CC2CCCN(Cc3cccc4nsnc34)C2)n1 REAL300019304200
CCn1cnc(Cl)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304201
N#Cc1cnn2cc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)cnc12 REAL300019304202
O=C(O)c1csc(CC2CCCN(Cc3cn(-c4ccccc4)nn3)C2)n1 REAL300019304203
CCOc1ccc(Cl)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304204
Cn1nc(-c2ccccc2)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304205
CC(C)(C)c1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n[nH]1 REAL300019304206
CCN1CCCc2cc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)ccc21 REAL300019304207
O=C(O)c1csc(CC2CCCN(Cc3ccc(-c4ccsc4)nc3)C2)n1 REAL300019304208
O=C(O)c1csc(CC2CCCN(Cc3cc4ccccc4cn3)C2)n1 REAL300019304209
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc(Cl)n1 REAL300019304210
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc(C)n1 REAL300019304211
COc1cc(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cn1 REAL300019304212
O=C(O)c1csc(CC2CCCN(Cc3ccc[nH]c3=O)C2)n1 REAL300019304213
CCc1c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cnn1CC REAL300019304214
Cn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C(F)(F)F)n1 REAL300019304215
O=C(O)c1csc(CC2CCCN(Cc3noc4c3CCCC4)C2)n1 REAL300019304216
Cc1cn(C)nc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304217
Cc1coc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304218
O=C(O)c1csc(CC2CCCN(Cc3cc4ccncc4s3)C2)n1 REAL300019304219
COc1nc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)ccc1C REAL300019304220
O=C(O)c1csc(CC2CCCN(Cc3cc4ncccc4o3)C2)n1 REAL300019304221
CCC(C)n1nccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304222
O=C(O)c1csc(CC2CCCN(Cc3nc(CO)cs3)C2)n1 REAL300019304223
CCCn1cncc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304224
CCc1c[nH]c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304225
O=C(O)c1csc(CC2CCCN(Cc3cncc(-c4cccnc4)c3)C2)n1 REAL300019304226
CC(C)(C)c1cncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304227
COc1nc(Cl)ccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304228
Cc1c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)ccnc1F REAL300019304229
O=C(O)c1csc(CC2CCCN(Cc3ccc4c(c3)CCOC4)C2)n1 REAL300019304230
O=C(O)c1csc(CC2CCCN(Cc3cccc(C(F)F)c3F)C2)n1 REAL300019304231
Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C)n1 REAL300019304232
O=C(O)c1csc(CC2CCCN(Cc3nc4c(s3)CCCCC4)C2)n1 REAL300019304233
O=C(O)c1csc(CC2CCCN(Cc3nc4c(s3)COCC4)C2)n1 REAL300019304234
CC(C)Cc1ccccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304235
CSc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)o1 REAL300019304236
O=C(O)c1csc(CC2CCCN(Cc3cnn(C4CCCCC4)c3)C2)n1 REAL300019304237
CCCn1nc(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1Cl REAL300019304238
Cn1cc(-c2n[nH]cc2CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cn1 REAL300019304239
CC(C)n1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304240
O=C(O)c1csc(CC2CCCN(Cc3ccn(CC(F)(F)F)n3)C2)n1 REAL300019304241
CC(F)(F)c1cccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304242
Cc1cc(O)ncc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304243
Cc1nc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)oc1C REAL300019304244
CS(=O)(=O)c1coc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304245
O=C(O)c1csc(CC2CCCN(Cc3cn(CC4CC4)nn3)C2)n1 REAL300019304246
O=C(O)c1csc(CC2CCCN(Cc3cccn3C(F)F)C2)n1 REAL300019304247
O=C(O)c1csc(CC2CCCN(Cc3cc4c(o3)CCCC4)C2)n1 REAL300019304248
Cn1cc(Br)nc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304249
C=CCc1ccccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304250
COc1nn(C)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304251
CC(C)(C)n1nccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304252
CN(CCO)c1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cn1 REAL300019304253
Cn1c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nc2c1CCCC2 REAL300019304254
O=C(O)c1csc(CC2CCCN(Cc3cccc4c3COCC4)C2)n1 REAL300019304255
O=C(O)c1csc(CC2CCCN(Cc3ccccc3C3CCC3)C2)n1 REAL300019304256
CC(C)(C#N)c1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)s1 REAL300019304257
CCn1nc(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304258
COc1sccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304259
O=C(O)c1csc(CC2CCCN(Cc3cc(C4CCC4)[nH]n3)C2)n1 REAL300019304260
C=CCCn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nn1 REAL300019304261
O=C(O)c1csc(CC2CCCN(Cc3ccc(CC4CCC4)cc3)C2)n1 REAL300019304262
COc1nsc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1Cl REAL300019304263
O=C(O)c1csc(CC2CCCN(Cc3cn(C4CC4)cn3)C2)n1 REAL300019304264
CC(C)c1cnn(C)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304265
Cn1nnc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1C(F)F REAL300019304266
Cn1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1S(C)(=O)=O REAL300019304267
Cc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1OC(F)F REAL300019304268
CC1Oc2ccc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)cc2C1C REAL300019304269
O=C(O)c1csc(CC2CCCN(Cc3ccccc3-n3cccn3)C2)n1 REAL300019304270
O=C(O)c1csc(CC2CCCN(Cc3ccnn3C3CC3(F)F)C2)n1 REAL300019304271
COCc1nocc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304272
COCc1cnc(OC)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304273
O=C(O)c1csc(CC2CCCN(Cc3ccc(C(F)F)cn3)C2)n1 REAL300019304274
CC(C)Oc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1F REAL300019304275
CCn1cc(Cl)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304276
O=C(O)c1csc(CC2CCCN(Cc3ccc(F)c(Cl)c3F)C2)n1 REAL300019304277
O=C(O)c1csc(CC2CCCN(Cc3cccc(C(F)F)c3)C2)n1 REAL300019304278
O=C(O)c1csc(CC2CCCN(Cc3ccc4ccccc4c3F)C2)n1 REAL300019304279
O=C(O)c1csc(CC2CCCN(Cc3csc(Cl)c3)C2)n1 REAL300019304280
Cc1c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cnn1C1CCC1 REAL300019304281
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n(C2CCCC2)n1 REAL300019304282
O=C(O)c1csc(CC2CCCN(Cc3ccnn3CC(F)F)C2)n1 REAL300019304283
COc1ccc(C)nc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304284
O=C(O)c1csc(CC2CCCN(Cc3cc(Cl)cc(Cl)n3)C2)n1 REAL300019304285
O=C(O)c1csc(CC2CCCN(Cc3cc4cnccc4[nH]3)C2)n1 REAL300019304286
O=C(O)c1csc(CC2CCCN(Cc3c(F)ccnc3Cl)C2)n1 REAL300019304287
O=C(O)c1csc(CC2CCCN(Cc3cccc(C(F)F)n3)C2)n1 REAL300019304288
CN(C)c1cncc(F)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304289
O=C(O)c1csc(CC2CCCN(Cc3c(O)ccc4c3OCO4)C2)n1 REAL300019304290
Cc1nn(-c2ccccc2)nc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304291
O=C(O)c1csc(CC2CCCN(Cc3ccn(C4CCC4)n3)C2)n1 REAL300019304292
O=C(O)c1csc(CC2CCCN(Cc3ccn(CC(F)F)n3)C2)n1 REAL300019304293
O=C(O)c1csc(CC2CCCN(Cc3ccn(C4CC4(F)F)n3)C2)n1 REAL300019304294
O=C(O)c1csc(CC2CCCN(Cc3cnn(C4CCOCC4)c3)C2)n1 REAL300019304295
Cc1cn(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304296
O=C(O)c1csc(CC2CCCN(Cc3noc4c3CCC4)C2)n1 REAL300019304297
O=C(O)c1csc(CC2CCCN(Cc3nc4cccc(F)c4s3)C2)n1 REAL300019304298
O=C(O)c1csc(CC2CCCN(Cc3ccn(C4CCCC4)n3)C2)n1 REAL300019304299
O=C(O)c1csc(CC2CCCN(Cc3ccc(F)c4ccoc34)C2)n1 REAL300019304300
O=C(O)c1csc(CC2CCCN(Cc3cc(Cl)cc4ccoc34)C2)n1 REAL300019304301
O=C(O)c1csc(CC2CCCN(Cc3ncc(Cl)cc3Cl)C2)n1 REAL300019304302
Cc1nn(C2CCCC2)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304303
O=C(O)c1csc(CC2CCCN(Cc3ccccc3C(F)F)C2)n1 REAL300019304304
O=C(O)c1csc(CC2CCCN(Cc3ccc4[nH]ncc4c3)C2)n1 REAL300019304305
O=C(O)c1csc(CC2CCCN(Cc3ccc(Cl)c(F)c3F)C2)n1 REAL300019304306
Cc1c(F)cccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304307
Cn1cc(-c2cccc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)c2)cn1 REAL300019304308
COc1c(C#N)cccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304309
O=C(O)c1csc(CC2CCCN(Cc3ccnc(Br)c3)C2)n1 REAL300019304310
Cc1nc(Cl)ccc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304311
COc1cc(Cl)cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304312
COc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc(F)c1F REAL300019304313
COc1cc(C)ncc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304314
CC(C)n1cnc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304315
Cc1c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nnn1C REAL300019304316
Cn1nccc1-c1n[nH]cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304317
Cc1onc(C2CC2)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304318
COC(=O)c1c(C)[nH]c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1C REAL300019304319
CC(C)Oc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)o1 REAL300019304320
Cc1oc(-c2ccccc2)nc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304321
Cn1nc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1-c1ccco1 REAL300019304322
O=C(O)c1csc(CC2CCCN(Cc3c(Cl)ccc4c3OCO4)C2)n1 REAL300019304323
N#Cc1cc(F)cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1 REAL300019304324
O=C(O)c1csc(CC2CCCN(Cc3ccc(C4CCCCC4)cc3)C2)n1 REAL300019304325
Cc1nc(C)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)nc1C REAL300019304326
NC(=O)c1cnc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cn1 REAL300019304327
Cc1nn(C2CCC2)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304328
Cc1c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cnn1CC(F)F REAL300019304329
COc1ccccc1C=CCN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304330
O=C(O)c1csc(CC2CCCN(Cc3ccc(-c4ccccn4)nc3)C2)n1 REAL300019304331
CCCn1nc(C)c(Cl)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304332
COc1cccc2[nH]c(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)cc12 REAL300019304333
Cc1ccc(OC(F)F)c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304334
Cn1nc(-c2ccco2)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304335
COc1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C)n1 REAL300019304336
CCN(C)c1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C)c1 REAL300019304337
O=C(O)c1csc(CC2CCCN(Cc3cc(-c4ccccc4)ccn3)C2)n1 REAL300019304338
O=C(O)c1csc(CC2CCCN(Cc3scc(Cl)c3Cl)C2)n1 REAL300019304339
COc1cc(C)cc(OC)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304340
O=C(O)c1csc(CC2CCCN(Cc3ccc(CF)cc3)C2)n1 REAL300019304341
O=C(O)c1csc(CC2CCCN(Cc3ccc4sccc4c3)C2)n1 REAL300019304342
O=C(O)c1csc(CC2CCCN(Cc3ccc(-c4ccncc4)cc3)C2)n1 REAL300019304343
O=C(O)c1csc(CC2CCCN(Cc3ccccc3CO)C2)n1 REAL300019304344
CC(C)(C)c1oncc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304345
Cc1cncc(C)c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304346
COc1cc(C)c2cc(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)[nH]c2c1 REAL300019304347
Cc1cccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1C(F)(F)F REAL300019304348
C=CCn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cn1 REAL300019304349
O=C(O)c1csc(CC2CCCN(Cc3ccc4cn[nH]c4c3)C2)n1 REAL300019304350
CCC(C)c1ccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cc1 REAL300019304351
Cc1oncc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304352
CC(F)(F)c1cccc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n1 REAL300019304353
O=C(O)c1csc(CC2CCCN(Cc3cc4sccc4[nH]3)C2)n1 REAL300019304354
O=C(O)c1csc(CC2CCCN(Cc3cccc4c3CCCC4)C2)n1 REAL300019304355
CC(=Cc1cc(F)cc(F)c1)CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304356
O=C(O)c1csc(CC2CCCN(Cc3ccc(-n4ccnn4)cc3)C2)n1 REAL300019304357
Cc1c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)ccc2ccccc12 REAL300019304358
COc1c(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)ccc2[nH]ccc12 REAL300019304359
Cc1nc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C)s1 REAL300019304360
CCCn1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c1C REAL300019304361
Cc1ccc2cccnc2c1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304362
O=C(O)c1csc(CC2CCCN(Cc3c(O)cccc3F)C2)n1 REAL300019304363
Cc1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)cnc1-n1cccn1 REAL300019304364
COC(=O)c1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)n(C)c1 REAL300019304365
O=C(O)c1csc(CC2CCCN(Cc3cc4sc(Cl)cc4[nH]3)C2)n1 REAL300019304366
COc1ccn2c(CN3CCCC(Cc4nc(C(=O)O)cs4)C3)cnc2c1 REAL300019304367
CCCn1nc(C)cc1CN1CCCC(Cc2nc(C(=O)O)cs2)C1 REAL300019304368
Cn1cc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c(C2CCC2)n1 REAL300019304369
CC(C)(C)c1ncc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)o1 REAL300019304370
Cn1nc(CN2CCCC(Cc3nc(C(=O)O)cs3)C2)c2c1CCOC2 REAL300019304371
O=C(O)c1cnc2c(c1)CN(Cc1ccc3c(c1)OCCO3)C2 REAL300019304372
O=C(O)c1cnc2c(c1)CN(Cc1cccc(Br)c1)C2 REAL300019304373
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304374
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1C(F)(F)F)C2 REAL300019304375
COC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304376
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccc(F)cc3)o1)C2 REAL300019304377
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Br)o1)C2 REAL300019304378
O=C(O)c1cnc2c(c1)CN(Cc1cc(Br)cs1)C2 REAL300019304379
CC(C)=CCCC(C)CCN1Cc2cc(C(=O)O)cnc2C1 REAL300019304380
O=C(O)c1cnc2c(c1)CN(Cc1csc(-c3ccc(F)cc3)n1)C2 REAL300019304381
COC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)oc1C REAL300019304382
Cc1nn(C)c(Cl)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304383
O=C(O)c1cnc2c(c1)CN(Cc1cc(C(F)(F)F)ccc1Cl)C2 REAL300019304384
O=C(O)c1cnc2c(c1)CN(Cc1ccc(F)c(Cl)c1)C2 REAL300019304385
O=C(O)c1cnc2c(c1)CN(Cc1ccc(F)c(C(F)(F)F)c1)C2 REAL300019304386
O=C(O)c1cnc2c(c1)CN(Cc1ccc(F)cc1C(F)(F)F)C2 REAL300019304387
O=C(O)c1cnc2c(c1)CN(Cc1cc(F)cc(C(F)(F)F)c1)C2 REAL300019304388
COc1ccc(F)c(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304389
O=C(O)c1cnc2c(c1)CN(Cc1cc(F)cc(Cl)c1)C2 REAL300019304390
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Cl)cc1F)C2 REAL300019304391
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)ccc1F)C2 REAL300019304392
COc1ccc(F)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304393
COC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)cn1C REAL300019304394
Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1Cl REAL300019304395
O=C(O)c1cnc2c(c1)CN(CC1CCN(C(=O)OCc3ccccc3)CC1)C2 REAL300019304396
O=C(O)c1cnc2c(c1)CN(Cc1cccc(-c3ccccn3)c1)C2 REAL300019304397
Cc1nn(C(C)(C)C)c(C)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304398
COC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)o1 REAL300019304399
COc1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1F REAL300019304400
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)cc(C(F)(F)F)c1)C2 REAL300019304401
Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(Br)c1 REAL300019304402
CN(C)c1ncc(CN2Cc3cc(C(=O)O)cnc3C2)n1C REAL300019304403
O=C(O)c1cnc2c(c1)CN(CCCc1c(F)cccc1Cl)C2 REAL300019304404
Cc1cc(Cl)ccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304405
Cn1ncc(Br)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304406
Cc1ccc2cc(CN3Cc4cc(C(=O)O)cnc4C3)ccc2n1 REAL300019304407
COc1cc(F)cc(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304408
CC(C)(C)c1ncc(CN2Cc3cc(C(=O)O)cnc3C2)cn1 REAL300019304409
Cn1c(=O)oc2cc(CN3Cc4cc(C(=O)O)cnc4C3)ccc21 REAL300019304410
O=C(O)c1cnc2c(c1)CN(CCc1cccc(Cl)c1)C2 REAL300019304411
O=C(O)c1cnc2c(c1)CN(Cc1nc3ccccn3c1Br)C2 REAL300019304412
COc1ccc2oc(CN3Cc4cc(C(=O)O)cnc4C3)cc2c1 REAL300019304413
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(C)c1OC REAL300019304414
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Oc3ccccc3)o1)C2 REAL300019304415
Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1Br REAL300019304416
Cc1ccc2nc(CN3Cc4cc(C(=O)O)cnc4C3)cn2c1 REAL300019304417
COCc1csc(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304418
O=C1COc2ccc(CN3Cc4cc(C(=O)O)cnc4C3)cc2N1 REAL300019304419
O=C(O)c1cnc2c(c1)CN(Cc1ccnc(Cl)c1Cl)C2 REAL300019304420
O=C(O)c1cnc2c(c1)CN(CCCc1ccc3c(c1)CCO3)C2 REAL300019304421
O=C(O)c1cnc2c(c1)CN(Cc1cc3c(cn1)OCCO3)C2 REAL300019304422
Cc1ccc2ncc(CN3Cc4cc(C(=O)O)cnc4C3)n2c1 REAL300019304423
O=C(O)c1cnc2c(c1)CN(Cc1cc(C(F)(F)F)[nH]n1)C2 REAL300019304424
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)cc3c1OCC3)C2 REAL300019304425
Cc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1Cl REAL300019304426
O=C(O)c1cnc2c(c1)CN(Cc1nccn1-c1ccccc1)C2 REAL300019304427
CC(CN1Cc2cc(C(=O)O)cnc2C1)c1cccc(Cl)c1 REAL300019304428
CC(C)(C)n1cc(CN2Cc3cc(C(=O)O)cnc3C2)nn1 REAL300019304429
Cn1c(CN2Cc3cc(C(=O)O)cnc3C2)nc2ccc(Cl)cc21 REAL300019304430
CC(C)c1nnc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304431
CC(CN1Cc2cc(C(=O)O)cnc2C1)c1ccc(F)cc1 REAL300019304432
O=C(O)c1cnc2c(c1)CN(CC1CCS(=O)(=O)CC1)C2 REAL300019304433
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C(F)(F)F)s1)C2 REAL300019304434
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OC(F)F)c(F)c1)C2 REAL300019304435
O=C(O)c1cnc2c(c1)CN(Cc1csc(C(F)(F)F)c1)C2 REAL300019304436
CC1(C)OCc2cc(CN3Cc4cc(C(=O)O)cnc4C3)ccc2O1 REAL300019304437
O=C(O)c1cnc2c(c1)CN(Cc1ncc(Br)s1)C2 REAL300019304438
Cc1cc(C(F)(F)F)ccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304439
Cn1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(C(F)F)n1 REAL300019304440
O=C(O)c1cnc2c(c1)CN(Cc1ncc(C(F)(F)F)s1)C2 REAL300019304441
CCOC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)o1 REAL300019304442
COc1ccc(-n2cc(CN3Cc4cc(C(=O)O)cnc4C3)cn2)cc1 REAL300019304443
Cc1noc2ncc(CN3Cc4cc(C(=O)O)cnc4C3)cc12 REAL300019304444
CC(CN1Cc2cc(C(=O)O)cnc2C1)c1cccc(Br)c1 REAL300019304445
CC(CN1Cc2cc(C(=O)O)cnc2C1)c1ccc(C(F)(F)F)cc1 REAL300019304446
O=C(O)c1cnc2c(c1)CN(Cc1cnn(Cc3ccc(F)cc3)c1)C2 REAL300019304447
O=C(O)c1cnc2c(c1)CN(Cc1nnn(-c3ccccc3)c1C1CC1)C2 REAL300019304448
COc1cc(-c2ccccc2)ccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304449
O=C(O)c1cnc2c(c1)CN(Cc1cnc(-c3ccco3)s1)C2 REAL300019304450
Cc1nn(-c2cccc(F)c2)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304451
CC(C)(C)c1ccc(CCN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304452
O=C(O)c1cnc2c(c1)CN(CCCc1c(Cl)cccc1Cl)C2 REAL300019304453
O=C(O)c1cnc2c(c1)CN(CC1CCOc3ccccc31)C2 REAL300019304454
O=C(O)c1cnc2c(c1)CN(CCCCc1cccc(C(F)(F)F)c1)C2 REAL300019304455
CN(c1ccccc1)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cn1 REAL300019304456
COCOc1ccc(OC)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304457
O=C(O)c1cnc2c(c1)CN(Cc1cc3c(Cl)nccc3o1)C2 REAL300019304458
NC(=O)Cn1cc(CN2Cc3cc(C(=O)O)cnc3C2)nn1 REAL300019304459
O=C(O)c1cnc2c(c1)CN(Cc1cn(-c3ccc(F)c(Cl)c3)nn1)C2 REAL300019304460
Cc1ccccc1-n1cc(CN2Cc3cc(C(=O)O)cnc3C2)nn1 REAL300019304461
CCSc1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304462
O=C(O)c1cnc2c(c1)CN(Cc1cnnn1-c1ccccc1)C2 REAL300019304463
O=C(O)c1cnc2c(c1)CN(Cc1cc3ccnc(Cl)c3s1)C2 REAL300019304464
Cn1ncc(I)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304465
O=C(O)c1cnc2c(c1)CN(CC1C3CC4CC(C3)CC1C4)C2 REAL300019304466
COCCC(CN1Cc2cc(C(=O)O)cnc2C1)NC(=O)OC(C)(C)C REAL300019304467
CC(C)OC(CN1Cc2cc(C(=O)O)cnc2C1)c1ccccc1 REAL300019304468
CC(C)N(C)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cn1 REAL300019304469
COCCN(C)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cn1 REAL300019304470
CC(C)(C)OC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304471
Cn1nc2c(c1CN1Cc3cc(C(=O)O)cnc3C1)CCCC2 REAL300019304472
O=C(O)c1cnc2c(c1)CN(Cc1cc(Br)c(Cl)s1)C2 REAL300019304473
O=C(O)c1cnc2c(c1)CN(Cc1cnn(Cc3ccccc3)c1Cl)C2 REAL300019304474
O=C(O)c1cnc2c(c1)CN(Cc1scnc1C1CC1)C2 REAL300019304475
CN(C)Cc1cnc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304476
O=C(O)c1cnc2c(c1)CN(Cc1ccsc1C(F)(F)F)C2 REAL300019304477
CC(C)(C)n1nnc(CN2Cc3cc(C(=O)O)cnc3C2)n1 REAL300019304478
O=C(O)c1cnc2c(c1)CN(Cc1cccc3c1NCCC3)C2 REAL300019304479
Cn1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(I)n1 REAL300019304480
CC(=Cc1cccc([N+](=O)[O-])c1)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304481
Cn1cc(-c2csc(CN3Cc4cc(C(=O)O)cnc4C3)n2)cn1 REAL300019304482
O=C(O)c1cnc2c(c1)CN(Cc1ccncc1[N+](=O)[O-])C2 REAL300019304483
O=C(O)c1cnc2c(c1)CN(CC1CCC3(CC1)OCCO3)C2 REAL300019304484
COc1ccc2nc(CN3Cc4cc(C(=O)O)cnc4C3)sc2c1 REAL300019304485
COC(=O)COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1[N+](=O)[O-] REAL300019304486
CCc1cccc(Cl)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304487
Cn1c(=O)sc2cc(CN3Cc4cc(C(=O)O)cnc4C3)ccc21 REAL300019304488
COC(=O)C1C(CN2Cc3cc(C(=O)O)cnc3C2)C1(F)F REAL300019304489
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3cccc(F)c3F)o1)C2 REAL300019304490
CCN(C)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cn1 REAL300019304491
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OCC3CC3)cc1)C2 REAL300019304492
O=C(O)c1cnc2c(c1)CN(Cc1c(O)ccc(Cl)c1F)C2 REAL300019304493
O=C(O)c1cnc2c(c1)CN(Cc1n[nH]cc1-c1ccccc1)C2 REAL300019304494
O=C(O)c1cnc2c(c1)CN(Cc1cc3ccc(F)cc3[nH]1)C2 REAL300019304495
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Br)c(Cl)c1)C2 REAL300019304496
O=C(O)c1cnc2c(c1)CN(Cc1cnc(C3OCCO3)s1)C2 REAL300019304497
O=C(O)c1cnc2c(c1)CN(Cc1nc3ccc(F)cc3s1)C2 REAL300019304498
O=C(O)c1cnc2c(c1)CN(Cc1ccc(F)c(Cl)c1Cl)C2 REAL300019304499
O=C(O)c1cnc2c(c1)CN(Cc1csc(Cl)c1Cl)C2 REAL300019304500
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Sc3ccccn3)o1)C2 REAL300019304501
O=C(O)c1cnc2c(c1)CN(CCc1ccc(F)cc1Cl)C2 REAL300019304502
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Oc3cccc(F)c3)cc1)C2 REAL300019304503
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(OCc2cccnc2)c1 REAL300019304504
O=C(O)c1cnc2c(c1)CN(Cc1cnc(C(F)(F)F)s1)C2 REAL300019304505
O=C(O)c1cnc2c(c1)CN(Cc1nc3ccc(Br)cc3s1)C2 REAL300019304506
COc1c([N+](=O)[O-])ccc(CN2Cc3cc(C(=O)O)cnc3C2)c1O REAL300019304507
CC(O)c1ncc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304508
O=C(O)c1cnc2c(c1)CN(Cc1ncc(C3OCCO3)s1)C2 REAL300019304509
O=C(O)c1cnc2c(c1)CN(Cc1c[nH]nc1-c1ccc(C(F)(F)F)cc1)C2 REAL300019304510
Cn1nc(Br)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304511
CCOc1c(Cl)cccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304512
CCCCCCCCCC(C)CCN1Cc2cc(C(=O)O)cnc2C1 REAL300019304513
O=C(O)c1cnc2c(c1)CN(Cc1ccc3cnccc3c1)C2 REAL300019304514
CCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1F REAL300019304515
N#CCCn1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(-c2ccncc2)n1 REAL300019304516
O=C(O)c1cnc2c(c1)CN(Cc1ccnn1-c1ccccc1)C2 REAL300019304517
CC(C)(C)c1cnc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304518
Cc1nn(C)c(CN2Cc3cc(C(=O)O)cnc3C2)c1Br REAL300019304519
O=C(O)c1cnc2c(c1)CN(CC1(c3ccccc3)CCOC1)C2 REAL300019304520
CSc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304521
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OCCCCl)cc1)C2 REAL300019304522
CC(C)(C)OC(=O)N(CCN1Cc2cc(C(=O)O)cnc2C1)C(C)(C)C REAL300019304523
CC(C)C(CNC(=O)OC(C)(C)C)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304524
Cn1cc(-c2ccc(CN3Cc4cc(C(=O)O)cnc4C3)cc2)cn1 REAL300019304525
O=C(O)c1cnc2c(c1)CN(Cc1c(F)cccc1Br)C2 REAL300019304526
O=C(O)c1cnc2c(c1)CN(Cc1c(F)ccc(O)c1F)C2 REAL300019304527
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C(F)F)cc1)C2 REAL300019304528
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Cl)cc1-n1cncn1)C2 REAL300019304529
O=C(O)c1cnc2c(c1)CN(CC(c1ccccc1)c1ccccc1)C2 REAL300019304530
CCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304531
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-n3cccn3)cc1)C2 REAL300019304532
CC(C)(C)OC(=O)N1CCCC(CN2Cc3cc(C(=O)O)cnc3C2)C1 REAL300019304533
O=C(O)c1cnc2c(c1)CN(Cc1ccc3ncccc3c1)C2 REAL300019304534
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OCc1ccccc1 REAL300019304535
CC(C)(C)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304536
COc1cc(OC)c(CN2Cc3cc(C(=O)O)cnc3C2)c(OC)c1 REAL300019304537
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OC(F)F)cc1OC(F)F)C2 REAL300019304538
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OC(F)F REAL300019304539
CCCOc1ccc(Br)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304540
CCOc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OC REAL300019304541
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OCc1ccccc1)C2 REAL300019304542
CCCCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304543
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1Br REAL300019304544
CC(C)Oc1ccccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304545
CCCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304546
C=CCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304547
CCCCCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304548
CN(CCC#N)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304549
CCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304550
O=C(O)c1cnc2c(c1)CN(Cc1c(OC(F)F)ccc3ccccc13)C2 REAL300019304551
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OC(C)C REAL300019304552
CCc1cccc(F)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304553
CN(C)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(C(F)(F)F)c1 REAL300019304554
CC(C)C(CN1Cc2cc(C(=O)O)cnc2C1)c1ccccc1 REAL300019304555
O=C(O)c1cnc2c(c1)CN(Cc1ccnn1-c1ccc(F)cc1)C2 REAL300019304556
Cc1ccccc1-n1nccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304557
COC(=O)c1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304558
COC(=O)c1ccc(Cl)c(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304559
COc1ccccc1-n1nccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304560
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)ccc1OCC1CC1)C2 REAL300019304561
O=C(O)c1cnc2c(c1)CN(CC1CCC(c3ccccc3)CC1)C2 REAL300019304562
O=C(O)c1cnc2c(c1)CN(CC(Cc1ccccc1)Cc1ccccc1)C2 REAL300019304563
Cc1nn(C(C)C)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304564
C[C@H](CN1Cc2cc(C(=O)O)cnc2C1)NC(=O)OC(C)(C)C REAL300019304565
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(OC)c1O REAL300019304566
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1C#N REAL300019304567
COC(=O)c1[nH]c(CN2Cc3cc(C(=O)O)cnc3C2)cc1C REAL300019304568
CCc1cc(OC)ccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304569
O=C(O)c1cnc2c(c1)CN(Cc1c(F)ccc(Br)c1F)C2 REAL300019304570
CC(C)(C)OC(=O)Nc1ncc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304571
CC(=Cc1ccccc1C(F)(F)F)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304572
O=C(O)c1cnc2c(c1)CN(CC(c1ccc(F)cc1)c1ccc(F)cc1)C2 REAL300019304573
COC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)n(C)c1C REAL300019304574
CCc1oc(CN2Cc3cc(C(=O)O)cnc3C2)cc1C(=O)OC REAL300019304575
Cn1cc(-c2ccc(CN3Cc4cc(C(=O)O)cnc4C3)s2)cn1 REAL300019304576
CN(C)c1nc(CN2Cc3cc(C(=O)O)cnc3C2)c(Cl)n1-c1ccccc1 REAL300019304577
Cc1nn(-c2ccccn2)c(C)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304578
COCCCn1nccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304579
Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(-c2ccnn2C)c1 REAL300019304580
Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(-c2cnn(C)c2)c1 REAL300019304581
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccc(Cl)cc3)cc1)C2 REAL300019304582
O=C(O)c1cnc2c(c1)CN(Cc1cnc(-c3ccc(Cl)cc3)s1)C2 REAL300019304583
COC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(Br)c1 REAL300019304584
O=C(O)c1cnc2c(c1)CN(Cc1c(F)cccc1OC(F)(F)F)C2 REAL300019304585
O=C(O)c1cnc2c(c1)CN(Cc1cccc(I)c1)C2 REAL300019304586
COc1cccc(OC)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304587
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(Br)c1 REAL300019304588
Cc1nn(-c2ccccn2)c(Cl)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304589
O=C(O)c1cnc2c(c1)CN(CC=Cc1ccc(F)c(F)c1)C2 REAL300019304590
O=C(O)c1cnc2c(c1)CN(Cc1ccc3c(c1)CCN3Cc1ccccc1)C2 REAL300019304591
O=C(O)c1cnc2c(c1)CN(Cc1cscc1Br)C2 REAL300019304592
CCOC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)[nH]c1C REAL300019304593
O=C(O)c1cnc2c(c1)CN(CCc1ccc(Cl)cc1)C2 REAL300019304594
O=C(O)c1cnc2c(c1)CN(Cc1cnn(-c3ccc(C(F)(F)F)cc3)c1)C2 REAL300019304595
CC(C)C1CCC(CN2Cc3cc(C(=O)O)cnc3C2)CC1 REAL300019304596
O=C(O)c1cnc2c(c1)CN(Cc1ncc(I)s1)C2 REAL300019304597
CN(C)Cc1cc(CN2Cc3cc(C(=O)O)cnc3C2)no1 REAL300019304598
CC1CN(C(=O)OC(C)(C)C)CCC1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304599
CC(C)(C)OC(=O)NCC1(CN2Cc3cc(C(=O)O)cnc3C2)CC1 REAL300019304600
CC1CC(CN2Cc3cc(C(=O)O)cnc3C2)CCN1C(=O)OC(C)(C)C REAL300019304601
CCOC(=O)CC(C)(C)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304602
COCCOCc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304603
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(OC)c1OCC(F)F REAL300019304604
CCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OCC REAL300019304605
CCn1c2ccccc2c2cc(CN3Cc4cc(C(=O)O)cnc4C3)ccc21 REAL300019304606
O=C(O)c1cnc2c(c1)CN(Cc1ccc3ccccc3c1)C2 REAL300019304607
O=C(O)c1cnc2c(c1)CN(Cc1cc(Br)c3c(c1)OCO3)C2 REAL300019304608
CCOc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OCC(C)C REAL300019304609
O=C(O)c1cnc2c(c1)CN(Cc1cc(Br)ccc1F)C2 REAL300019304610
COc1cc(Br)c(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304611
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(OC)c1 REAL300019304612
COc1ccc2cc(CN3Cc4cc(C(=O)O)cnc4C3)ccc2c1 REAL300019304613
CCCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OCC REAL300019304614
COc1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1OC(F)F REAL300019304615
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1N1CCCC1)C2 REAL300019304616
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OCC(N)=O REAL300019304617
O=C(O)c1cnc2c(c1)CN(Cc1c(F)cccc1N1CCCC1)C2 REAL300019304618
O=C(O)c1cnc2c(c1)CN(Cc1ccc(F)c(Br)c1)C2 REAL300019304619
Cc1ccc(COc2ccc(CN3Cc4cc(C(=O)O)cnc4C3)cc2)cc1 REAL300019304620
O=C(O)c1cnc2c(c1)CN(Cc1ccc(N3CCCCC3)cc1)C2 REAL300019304621
CN(c1ccccc1)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304622
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(Cl)c1OC REAL300019304623
O=C(O)c1cnc2c(c1)CN(Cc1cc(Br)ccc1OC(F)F)C2 REAL300019304624
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OCC(C)C REAL300019304625
CCOc1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1OC REAL300019304626
CCCOc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OC REAL300019304627
CCOc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(Cl)c1OC REAL300019304628
C=CCOc1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304629
COc1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1OC(C)C REAL300019304630
C#CCOc1ccccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304631
CCOc1c(Cl)cc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304632
CCNC(=O)COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304633
CCCOc1c(CN2Cc3cc(C(=O)O)cnc3C2)cccc1OCC REAL300019304634
CCCCOc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OC REAL300019304635
CCCOc1c(Cl)cc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OCC REAL300019304636
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC(F)F REAL300019304637
CCOc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OC(F)F REAL300019304638
Cc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(C)c1OC(F)F REAL300019304639
CCOc1cc2c(cc1CN1Cc3cc(C(=O)O)cnc3C1)OC(C)C2 REAL300019304640
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc2c1OCCO2 REAL300019304641
CCOc1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1OC(F)F REAL300019304642
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OCC(=O)N1CCCC1)C2 REAL300019304643
O=C(O)c1cnc2c(c1)CN(Cc1cc(-c3ccccn3)n[nH]1)C2 REAL300019304644
CN(C)c1cc(Cl)cc(Cl)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304645
COC(=O)c1ccc([N+](=O)[O-])c(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304646
O=C(O)c1cnc2c(c1)CN(Cc1cc(O)cc(C(F)(F)F)c1)C2 REAL300019304647
CC(=Cc1ccccc1OC(F)F)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304648
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)cc(Cl)c1[N+](=O)[O-])C2 REAL300019304649
O=C(O)c1cnc2c(c1)CN(Cc1cscc1C(F)(F)F)C2 REAL300019304650
O=C(O)c1cnc2c(c1)CN(Cc1c(F)ccc(C3OCCO3)c1Cl)C2 REAL300019304651
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C3CCCC3)cc1)C2 REAL300019304652
CCOC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)on1 REAL300019304653
CC(C)(C)OC(=O)N1CC2CC2(CN2Cc3cc(C(=O)O)cnc3C2)C1 REAL300019304654
O=C(O)c1cnc2c(c1)CN(CCc1ccc([N+](=O)[O-])cc1)C2 REAL300019304655
CC(C)(C)OC(=O)N1CC(F)(F)CC1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304656
O=C(O)c1cnc2c(c1)CN(Cc1ccc3c(c1)CCCC3)C2 REAL300019304657
O=C(O)c1cnc2c(c1)CN(Cc1cnn(CC(F)F)c1)C2 REAL300019304658
COCc1ccccc1C=C(C)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304659
Cn1nccc1-c1ccccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304660
COC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)on1 REAL300019304661
CC(C)(C)OC(=O)NCC1(CN2Cc3cc(C(=O)O)cnc3C2)CCC1 REAL300019304662
O=C(O)c1cnc2c(c1)CN(Cc1conc1Cc1ccccc1)C2 REAL300019304663
CC(C)(C)OC(=O)N1CCC[C@@H]1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304664
COC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)n1C REAL300019304665
O=C(O)c1cnc2c(c1)CN(Cc1ccc3ccc(F)c(F)c3n1)C2 REAL300019304666
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C3CCC3)cc1)C2 REAL300019304667
O=C(O)c1cnc2c(c1)CN(Cc1cccc(O)c1Cl)C2 REAL300019304668
Cc1cc(Cl)cc(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304669
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)c(F)cc1O)C2 REAL300019304670
CSCc1cnc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304671
O=C(O)c1cnc2c(c1)CN(Cc1c(Cl)cccc1N1CCOCC1)C2 REAL300019304672
CC1CN(c2ccccc2CN2Cc3cc(C(=O)O)cnc3C2)CCO1 REAL300019304673
CC(C)(C)OC(=O)NC(CN1Cc2cc(C(=O)O)cnc2C1)CC(F)(F)F REAL300019304674
Cc1c(CN2Cc3cc(C(=O)O)cnc3C2)sc2c(Cl)cccc12 REAL300019304675
O=C(O)c1cnc2c(c1)CN(Cc1ccc(I)s1)C2 REAL300019304676
COC(CN1Cc2cc(C(=O)O)cnc2C1)C1CCOCC1 REAL300019304677
CC(CN1Cc2cc(C(=O)O)cnc2C1)c1cc(F)cc(F)c1 REAL300019304678
COc1cccc2c(CN3Cc4cc(C(=O)O)cnc4C3)cccc12 REAL300019304679
CC(C)(CNC(=O)OC(C)(C)C)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304680
O=C(O)c1cnc2c(c1)CN(Cc1cccc(F)c1Br)C2 REAL300019304681
COc1cc2ccccc2cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304682
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc2ccccc12 REAL300019304683
COC(=O)Cn1cc(CN2Cc3cc(C(=O)O)cnc3C2)nn1 REAL300019304684
CC(C)(C)OC(=O)Nc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304685
O=C(O)c1cnc2c(c1)CN(Cc1ccnc(Cl)c1F)C2 REAL300019304686
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc2c1OCO2 REAL300019304687
CCCOc1c(Cl)cc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304688
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-n3ccnc3)cc1)C2 REAL300019304689
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)c3c(c1)OCCO3)C2 REAL300019304690
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OCc3ccc(Cl)cc3)cc1)C2 REAL300019304691
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OCc1cccs1 REAL300019304692
CCCCCCCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304693
O=C(O)c1cnc2c(c1)CN(Cc1cccc3ccccc13)C2 REAL300019304694
O=C(O)c1cnc2c(c1)CN(Cc1c3ccccc3cc3ccccc13)C2 REAL300019304695
CCN(CC)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304696
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Br)cc1)C2 REAL300019304697
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(OC)c1OC REAL300019304698
O=C(O)c1cnc2c(c1)CN(Cc1c(F)cccc1Cl)C2 REAL300019304699
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OC(F)F)C2 REAL300019304700
COc1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1OC REAL300019304701
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(OC)c1 REAL300019304702
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Cl)c(Cl)c1)C2 REAL300019304703
CCN(Cc1ccccc1)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304704
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OC(F)F)cc1)C2 REAL300019304705
O=C(O)c1cnc2c(c1)CN(Cc1c3ccccc3c(Cl)c3ccccc13)C2 REAL300019304706
CCCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304707
CC(C)CCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304708
CCCCCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304709
O=C(O)c1cnc2c(c1)CN(Cc1cccc(Oc3ccccc3)c1)C2 REAL300019304710
O=C(O)c1cnc2c(c1)CN(Cc1cccc(C(F)(F)F)c1)C2 REAL300019304711
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(OC)c1OC REAL300019304712
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OCc1ccccc1 REAL300019304713
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OCc3ccccc3)cc1)C2 REAL300019304714
COc1ccc(Br)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304715
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccccc3)cc1)C2 REAL300019304716
COc1ccc2ccccc2c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304717
CSc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304718
O=C(O)c1cnc2c(c1)CN(Cc1c(Cl)cccc1Cl)C2 REAL300019304719
COc1cc(OC)c(OC)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304720
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1O REAL300019304721
Cc1ccc(C)c(-n2nc(C)c(CN3Cc4cc(C(=O)O)cnc4C3)c2Cl)c1 REAL300019304722
O=C(O)c1cnc2c(c1)CN(Cc1csc(-c3ccc(Cl)cc3)n1)C2 REAL300019304723
CCCCn1nc(C)c(CN2Cc3cc(C(=O)O)cnc3C2)c1Cl REAL300019304724
CC(C)(CN1Cc2cc(C(=O)O)cnc2C1)Oc1ccccc1 REAL300019304725
COC(Cc1ccccc1)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304726
O=C(O)c1cnc2c(c1)CN(Cc1ccc(I)cc1)C2 REAL300019304727
O=C(O)c1cnc2c(c1)CN(Cc1ccnc3c(Br)cccc13)C2 REAL300019304728
O=C(O)c1cnc2c(c1)CN(Cc1c[nH]c(C(=O)OCc3ccccc3)c1)C2 REAL300019304729
CN(Cc1cccs1)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304730
O=C(O)c1cnc2c(c1)CN(Cc1cnc3ccccc3n1)C2 REAL300019304731
Cc1nc2scc(C3CC3)n2c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304732
O=C(O)c1cnc2c(c1)CN(Cc1sc(N3CCOCC3)nc1Cl)C2 REAL300019304733
CCOP(=O)(CCCN1Cc2cc(C(=O)O)cnc2C1)OCC REAL300019304734
CC(C)(C)CCC(CN1Cc2cc(C(=O)O)cnc2C1)NC(=O)OC(C)(C)C REAL300019304735
Cc1cc(Br)c(CN2Cc3cc(C(=O)O)cnc3C2)cc1Cl REAL300019304736
O=C(O)c1cnc2c(c1)CN(Cc1cnc(-c3c(F)cccc3F)s1)C2 REAL300019304737
CC(CN1Cc2cc(C(=O)O)cnc2C1)c1ccc(S(C)(=O)=O)cc1 REAL300019304738
O=C(O)c1cnc2c(c1)CN(Cc1cc3cc(Cl)cnc3o1)C2 REAL300019304739
O=C(O)c1cnc2c(c1)CN(Cc1cnc(-c3ccccc3F)s1)C2 REAL300019304740
O=C(O)c1cnc2c(c1)CN(Cc1cccc(Br)c1F)C2 REAL300019304741
COc1cccc(Sc2ccccc2CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304742
O=C(O)c1cnc2c(c1)CN(Cc1cnc(CCc3ccccc3)s1)C2 REAL300019304743
O=C(O)c1cnc2c(c1)CN(Cc1ccc3c(c1)OCCCCO3)C2 REAL300019304744
O=C(O)c1cnc2c(c1)CN(Cc1cc(F)cc(Br)c1)C2 REAL300019304745
CC(C)COc1ccccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304746
Cc1ccccc1-c1ccccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304747
CS(=O)(=O)c1cccc(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304748
O=C(O)c1cnc2c(c1)CN(Cc1ccnn1C1CCCC1)C2 REAL300019304749
Cn1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(-c2ccc(F)cc2)n1 REAL300019304750
CC(C)(C)OC(=O)N1CC(CCN2Cc3cc(C(=O)O)cnc3C2)C1 REAL300019304751
Cc1cc(Br)c(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304752
O=C(O)c1cnc2c(c1)CN(Cc1c(-c3ccccc3)nc3sccn13)C2 REAL300019304753
NS(=O)(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)o1 REAL300019304754
CC(C)(C)OC(=O)NC(CC(F)F)CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304755
C[C@]1(CN2Cc3cc(C(=O)O)cnc3C2)C[C@@H]1c1ccccc1 REAL300019304756
O=C(O)c1cnc2c(c1)CN(CC=Cc1ccc(OCc3ccccc3)cc1)C2 REAL300019304757
Cc1cc(F)c(CN2Cc3cc(C(=O)O)cnc3C2)c(Cl)c1 REAL300019304758
COc1ccc(-c2ccccc2C)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304759
O=C(O)c1cnc2c(c1)CN(Cc1ccncc1Br)C2 REAL300019304760
CC(C)(CN1Cc2cc(C(=O)O)cnc2C1)N1CCOCC1 REAL300019304761
Cc1cc(O)c(CN2Cc3cc(C(=O)O)cnc3C2)c(Cl)c1 REAL300019304762
O=C(O)c1cnc2c(c1)CN(Cc1cccc3c1OC(F)(F)O3)C2 REAL300019304763
CCOc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OC(=O)CC REAL300019304764
CS(=O)(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304765
Cc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1C(F)(F)F REAL300019304766
CS(=O)(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)o1 REAL300019304767
CN(C)C(=O)c1ccccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304768
O=C(O)c1cnc2c(c1)CN(Cc1nc3cc([N+](=O)[O-])ccc3o1)C2 REAL300019304769
O=C(O)c1cnc2c(c1)CN(Cc1ccc(F)cc1I)C2 REAL300019304770
O=C(O)c1cnc2c(c1)CN(Cc1cnn(C3CCCC3)c1-c1ccccc1)C2 REAL300019304771
CC(c1nccc2ccccc12)N1Cc2cc(C(=O)O)cnc2C1 REAL300019304772
O=C(O)c1cnc2c(c1)CN(Cc1cnn3cc(Br)cnc13)C2 REAL300019304773
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OCCCCO)C2 REAL300019304774
O=C(O)c1cnc2c(c1)CN(Cc1cnn(-c3ccccc3)n1)C2 REAL300019304775
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccccc3)s1)C2 REAL300019304776
CC(=O)Nc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304777
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Cl)cc1Cl)C2 REAL300019304778
O=C(O)c1cnc2c(c1)CN(Cc1cccc(Cl)c1Cl)C2 REAL300019304779
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1I)C2 REAL300019304780
Cc1nn(-c2ccccc2)c(Cl)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304781
O=C(O)c1cnc2c(c1)CN(Cc1cn(-c3ccccc3)nc1-c1ccccc1)C2 REAL300019304782
O=C(O)c1cnc2c(c1)CN(Cc1c[nH]nc1-c1ccccc1)C2 REAL300019304783
Cc1nn(-c2ccccc2)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304784
N#CCCn1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(-c2ccccc2)n1 REAL300019304785
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3cc(Cl)ccc3Cl)o1)C2 REAL300019304786
O=C(O)c1cnc2c(c1)CN(Cc1cn(-c3ccccc3)nc1-c1cccnc1)C2 REAL300019304787
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccc(Br)cc3)o1)C2 REAL300019304788
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccc(Cl)cc3[N+](=O)[O-])o1)C2 REAL300019304789
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccc(Cl)cc3)o1)C2 REAL300019304790
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccccc3Cl)o1)C2 REAL300019304791
O=C(O)c1cnc2c(c1)CN(Cc1ccc(N3CCCCC3)c([N+](=O)[O-])c1)C2 REAL300019304792
O=C(O)c1cnc2c(c1)CN(Cc1cn(Cc3ccccc3)c3ccccc13)C2 REAL300019304793
Cc1nn(Cc2ccccc2)c(Cl)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304794
O=C(O)c1cnc2c(c1)CN(Cc1c[nH]nc1-c1ccc(Cl)cc1)C2 REAL300019304795
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccccc3F)o1)C2 REAL300019304796
O=C(O)c1cnc2c(c1)CN(Cc1ccc3c(c1)OC(F)(F)O3)C2 REAL300019304797
Cc1cc(F)c(CN2Cc3cc(C(=O)O)cnc3C2)c(F)c1 REAL300019304798
CCOC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)[nH]n1 REAL300019304799
CC(C)Cn1nccc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304800
O=C(O)c1cnc2c(c1)CN(Cc1cc(Br)cnc1Cl)C2 REAL300019304801
O=C(O)c1cnc2c(c1)CN(Cc1cc(OC(F)F)ccc1Br)C2 REAL300019304802
Cc1ccc(-c2nn(C)cc2CN2Cc3cc(C(=O)O)cnc3C2)o1 REAL300019304803
NS(=O)(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1Cl REAL300019304804
O=C(O)c1cnc2c(c1)CN(Cc1cccc(OCc3ccc(F)cc3F)c1)C2 REAL300019304805
CN(C)Cc1nc(CN2Cc3cc(C(=O)O)cnc3C2)cs1 REAL300019304806
O=C(O)c1cnc2c(c1)CN(Cc1cc(Br)c([N+](=O)[O-])s1)C2 REAL300019304807
Cc1cccc(-n2cc(CN3Cc4cc(C(=O)O)cnc4C3)c(C)n2)c1 REAL300019304808
COc1cc(OC)c(CN2Cc3cc(C(=O)O)cnc3C2)cc1F REAL300019304809
COc1cc(F)c(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304810
Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(Cl)c1 REAL300019304811
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(F)c1 REAL300019304812
O=C(O)c1cnc2c(c1)CN(Cc1cc3nc(Cl)ccc3s1)C2 REAL300019304813
Cn1ncc(C(=O)OC(C)(C)C)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304814
Cc1nn(-c2ccccc2F)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304815
Cc1nn(-c2ccccc2Cl)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304816
Cc1ccc(-n2cc(CN3Cc4cc(C(=O)O)cnc4C3)c(C)n2)cc1 REAL300019304817
CC(C)(C#N)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304818
COC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(C)o1 REAL300019304819
COc1cc(O)cc(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304820
COC(=O)c1[nH]cc(CN2Cc3cc(C(=O)O)cnc3C2)c1C REAL300019304821
COC(=O)C=Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)o1 REAL300019304822
Cc1ccc(-c2ncc(CN3Cc4cc(C(=O)O)cnc4C3)s2)cc1C REAL300019304823
O=C(O)c1cnc2c(c1)CN(Cc1cccn(C(F)F)c1=O)C2 REAL300019304824
O=C(O)c1cnc2c(c1)CN(CC1CCN(c3ccccc3)C1)C2 REAL300019304825
COC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1F REAL300019304826
Cn1cc(-c2nn(C)cc2CN2Cc3cc(C(=O)O)cnc3C2)cn1 REAL300019304827
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Oc3ccc(F)cc3)nc1)C2 REAL300019304828
O=C(O)c1cnc2c(c1)CN(Cc1cnc(-c3cccc(Cl)c3)s1)C2 REAL300019304829
O=C(O)c1cnc2c(c1)CN(Cc1cccc(C3CCCC3)c1)C2 REAL300019304830
CCCCc1oc2ccccc2c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304831
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-n3cnc4ccccc43)cc1)C2 REAL300019304832
Cc1nn(-c2ccc(F)cc2)c(C)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304833
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)c3c(c1)OCCCO3)C2 REAL300019304834
O=C(O)c1cnc2c(c1)CN(Cc1cccc(OCc3ccccc3Cl)c1)C2 REAL300019304835
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccccc3)o1)C2 REAL300019304836
Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1[N+](=O)[O-] REAL300019304837
COc1cccc2cc(CN3Cc4cc(C(=O)O)cnc4C3)oc12 REAL300019304838
CC(C)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1[N+](=O)[O-] REAL300019304839
Cc1nn(Cc2ccccc2)c(C)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304840
Cc1nn(Cc2ccccc2Cl)c(C)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304841
Cc1nn(-c2ccccc2)c(C)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304842
Cc1ccc(Cn2nc(C)c(CN3Cc4cc(C(=O)O)cnc4C3)c2C)cc1 REAL300019304843
O=C(O)c1cnc2c(c1)CN(Cc1ccc(CSC(F)F)o1)C2 REAL300019304844
O=C(O)c1cnc2c(c1)CN(Cc1cnn(-c3ccccc3)c1)C2 REAL300019304845
O=C(O)c1cnc2c(c1)CN(Cc1cnn(Cc3ccccc3)c1)C2 REAL300019304846
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3cccc(Br)c3)o1)C2 REAL300019304847
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccc(Cl)cc3)s1)C2 REAL300019304848
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(OC)c1OCC(N)=O REAL300019304849
CCc1oc2ccccc2c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304850
COc1ccc(-c2nc(CN3Cc4cc(C(=O)O)cnc4C3)cs2)cc1 REAL300019304851
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OCc3ccccc3F)cc1)C2 REAL300019304852
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(Cl)c1OCC(N)=O REAL300019304853
NC(=O)COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304854
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OCc3cccc(F)c3)cc1)C2 REAL300019304855
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(O)c(C(C)(C)C)c1 REAL300019304856
O=C(O)c1cnc2c(c1)CN(Cc1cccc(OC3CC3)c1F)C2 REAL300019304857
CCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(C)c1 REAL300019304858
O=C(O)c1cnc2c(c1)CN(Cc1cccc(F)c1OC(F)F)C2 REAL300019304859
O=C(O)c1cnc2c(c1)CN(Cc1cc(F)ccc1OC(F)F)C2 REAL300019304860
CCc1cccc2cc(CN3Cc4cc(C(=O)O)cnc4C3)oc12 REAL300019304861
Cc1c(Br)cncc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304862
O=C(O)c1cnc2c(c1)CN(Cc1c(F)cncc1Br)C2 REAL300019304863
COc1cnc(F)c(CN2Cc3cc(C(=O)O)cnc3C2)c1 REAL300019304864
COc1nsc(CN2Cc3cc(C(=O)O)cnc3C2)c1Br REAL300019304865
O=C(O)c1cnc2c(c1)CN(Cc1cc3cc(Br)ccc3o1)C2 REAL300019304866
COC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1Cl REAL300019304867
COc1cccc(F)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304868
CCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(C)c1 REAL300019304869
Cn1ncc(C(F)(F)F)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304870
Cn1ncc(C2CCC2)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304871
CN1CCCCC(CN2Cc3cc(C(=O)O)cnc3C2)C1=O REAL300019304872
Cc1cc(O)c(CN2Cc3cc(C(=O)O)cnc3C2)cc1Cl REAL300019304873
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OC3CCOC3)cc1)C2 REAL300019304874
Cc1cccc2[nH]c(CN3Cc4cc(C(=O)O)cnc4C3)cc12 REAL300019304875
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C(F)(F)F)o1)C2 REAL300019304876
Cn1c(CN2Cc3cc(C(=O)O)cnc3C2)cnc1Br REAL300019304877
O=C(O)c1cnc2c(c1)CN(Cc1c(C(F)(F)F)nc3n1CCCC3)C2 REAL300019304878
O=C(O)c1cnc2c(c1)CN(CC1CC1c1ccc(F)cc1)C2 REAL300019304879
O=C(O)c1cnc2c(c1)CN(CCc1cccc(OC(F)(F)F)c1)C2 REAL300019304880
CC(C)(C)OC(=O)N1CC2CC1(CN1Cc3cc(C(=O)O)cnc3C1)C2 REAL300019304881
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Br)cc1O)C2 REAL300019304882
COCC(C)Oc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304883
Cn1nc(C(F)(F)F)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304884
O=C(O)c1cnc2c(c1)CN(Cc1ccc(F)c(F)c1F)C2 REAL300019304885
O=C(O)c1cnc2c(c1)CN(Cc1ccnn1-c1ccncc1)C2 REAL300019304886
Cc1ccc2cc(CN3Cc4cc(C(=O)O)cnc4C3)[nH]c2c1 REAL300019304887
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3cccs3)cc1)C2 REAL300019304888
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OCc1ccc(F)cc1F)C2 REAL300019304889
COC(=O)c1oc(CN2Cc3cc(C(=O)O)cnc3C2)cc1C REAL300019304890
CC(C)(C)C1(CN2Cc3cc(C(=O)O)cnc3C2)CCN(Cc2ccccc2)C1 REAL300019304891
O=C(O)c1cnc2c(c1)CN(CC[C@@H]1C[C@H]1c1ccccc1)C2 REAL300019304892
COC(=O)c1cc(CN2Cc3cc(C(=O)O)cnc3C2)n2c1CCCC2 REAL300019304893
CCCc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304894
O=C(O)c1cnc2c(c1)CN(Cc1ccnn1CCc1ccccc1)C2 REAL300019304895
O=C(O)c1cnc2c(c1)CN(Cc1ccc(SC(F)(F)F)cc1)C2 REAL300019304896
O=C(O)c1cnc2c(c1)CN(Cc1cnn(Cc3ccccc3Cl)c1)C2 REAL300019304897
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OC(F)(F)F)C2 REAL300019304898
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OC(F)(F)F)cc1)C2 REAL300019304899
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(Cl)c1 REAL300019304900
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C(F)(F)F)cc1)C2 REAL300019304901
CCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(OCCC)c1 REAL300019304902
O=C(O)c1cnc2c(c1)CN(Cc1cccc(OCc3ccccc3)c1)C2 REAL300019304903
Cc1ccc(Cn2nc(C)c(CN3Cc4cc(C(=O)O)cnc4C3)c2Cl)cc1 REAL300019304904
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3nc4ccccc4s3)o1)C2 REAL300019304905
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Br)cc1F)C2 REAL300019304906
COc1cc2c(cc1CN1Cc3cc(C(=O)O)cnc3C1)OC(C)C2 REAL300019304907
CCCOc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304908
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Br)s1)C2 REAL300019304909
O=C(O)c1cnc2c(c1)CN(Cc1cc3c(cc1Br)OCO3)C2 REAL300019304910
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1Br)C2 REAL300019304911
O=C(O)c1cnc2c(c1)CN(Cc1csc3ccccc13)C2 REAL300019304912
Cc1ccc(-c2n[nH]cc2CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304913
O=C(O)c1cnc2c(c1)CN(Cc1c[nH]nc1-c1ccc(F)cc1)C2 REAL300019304914
O=C(O)c1cnc2c(c1)CN(Cc1c[nH]nc1-c1cccs1)C2 REAL300019304915
COc1ccc(-c2n[nH]cc2CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304916
CCOc1c(CN2Cc3cc(C(=O)O)cnc3C2)c(C)nn1CC(C)C REAL300019304917
Cc1ccc(-c2n[nH]cc2CN2Cc3cc(C(=O)O)cnc3C2)o1 REAL300019304918
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OCC3CCCO3)cc1)C2 REAL300019304919
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-n3cncn3)c(F)c1)C2 REAL300019304920
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OCc1ccccn1)C2 REAL300019304921
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OCc1cscn1)C2 REAL300019304922
O=C(O)c1cnc2c(c1)CN(Cc1c(Cl)ccc(Cl)c1Cl)C2 REAL300019304923
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccc(F)cc3)s1)C2 REAL300019304924
O=C(O)c1cnc2c(c1)CN(Cc1cccc3cccnc13)C2 REAL300019304925
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccccc3Cl)s1)C2 REAL300019304926
O=C(O)c1cnc2c(c1)CN(CC13C4=C5C6=C1[Fe]56431789C3=C1C7C8=C39)C2 REAL300019304927
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccccc3F)s1)C2 REAL300019304928
CCN(CC)c1ncc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304929
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C(=O)NC3CC3)cc1)C2 REAL300019304930
CC(C)c1nn(-c2ccccc2)c(Cl)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304931
CNC(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304932
CCN(C(C)=O)c1nc(CN2Cc3cc(C(=O)O)cnc3C2)cs1 REAL300019304933
O=C(O)c1cnc2c(c1)CN(Cc1ccc(OCCN3CCCC3)cc1)C2 REAL300019304934
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OCc1ccncc1)C2 REAL300019304935
O=C(O)c1cnc2c(c1)CN(Cc1cc(Cl)ccc1OCc1cccnc1)C2 REAL300019304936
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3cccc(Cl)c3)s1)C2 REAL300019304937
CC(C)n1ncc2cc(CN3Cc4cc(C(=O)O)cnc4C3)c(Cl)nc21 REAL300019304938
CC(C)Oc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1 REAL300019304939
O=C(O)c1cnc2c(c1)CN(Cc1cc3ccccc3nc1N1CCOCC1)C2 REAL300019304940
Cc1nc(N2CCCCC2)sc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304941
O=C(O)c1cnc2c(c1)CN(C1CCC3(CC1F)OCCO3)C2 REAL300019304942
O=C(O)c1cnc2c(c1)CN(Cc1cc3c(O)cccc3s1)C2 REAL300019304943
CC(=O)N(c1ccccc1)c1nc(CN2Cc3cc(C(=O)O)cnc3C2)cs1 REAL300019304944
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(C(F)(F)F)c1 REAL300019304945
C=CCOc1c(Cl)cc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC REAL300019304946
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OC1CC1 REAL300019304947
O=C(O)c1cnc2c(c1)CN(Cc1cccc(F)c1OCC(F)(F)F)C2 REAL300019304948
CN(C)c1cc(F)c(CN2Cc3cc(C(=O)O)cnc3C2)cc1F REAL300019304949
O=C(O)c1cnc2c(c1)CN(Cc1c(F)ccc(F)c1Cl)C2 REAL300019304950
CC(C)Oc1cc(Cl)c(CN2Cc3cc(C(=O)O)cnc3C2)cc1Cl REAL300019304951
O=C(O)c1cnc2c(c1)CN(Cc1ccnn1C1CCOCC1)C2 REAL300019304952
CN(C)c1c(CN2Cc3cc(C(=O)O)cnc3C2)ccc(F)c1F REAL300019304953
CC1(CN2Cc3cc(C(=O)O)cnc3C2)CCCN(C(=O)OC(C)(C)C)C1 REAL300019304954
O=C(O)c1cnc2c(c1)CN(Cc1sncc1Br)C2 REAL300019304955
COCCCC1(CN2Cc3cc(C(=O)O)cnc3C2)CCC1 REAL300019304956
CCc1n[nH]c(Cl)c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304957
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-c3ccccc3)c(Cl)c1)C2 REAL300019304958
O=C(O)c1cnc2c(c1)CN(Cc1ccc(Br)c(F)c1F)C2 REAL300019304959
O=C(O)c1cnc2c(c1)CN(Cc1ccsc1Br)C2 REAL300019304960
CCOc1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(F)cc1OC REAL300019304961
Cn1cc(-c2nc(CN3Cc4cc(C(=O)O)cnc4C3)cs2)cn1 REAL300019304962
O=C(O)c1cnc2c(c1)CN(Cc1ncc(Br)cc1F)C2 REAL300019304963
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1Cl REAL300019304964
O=C(O)c1cnc2c(c1)CN(Cc1cn(-c3ccc(F)cc3)nn1)C2 REAL300019304965
Cn1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(Br)n1 REAL300019304966
CCOC(=O)c1[nH]c(C)c(CN2Cc3cc(C(=O)O)cnc3C2)c1C REAL300019304967
COC(=O)c1[nH]c2ccccc2c1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304968
O=C(O)c1cnc2c(c1)CN(CC1CCc3ccccc3C1)C2 REAL300019304969
CCOC(=O)c1cccc(CN2Cc3cc(C(=O)O)cnc3C2)n1 REAL300019304970
Cc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ncc1Br REAL300019304971
Cc1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(Br)cc1F REAL300019304972
CCOC(=O)c1ncc(CN2Cc3cc(C(=O)O)cnc3C2)s1 REAL300019304973
O=C(O)c1cnc2c(c1)CN(Cc1cc3c(=O)[nH]ccc3o1)C2 REAL300019304974
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)c(F)cc1Br REAL300019304975
O=C(O)c1cnc2c(c1)CN(Cc1cccc(Br)c1Cl)C2 REAL300019304976
CC(C)(C)OC(=O)Nc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)nn1 REAL300019304977
CN(C)Cc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c2c1OC(F)(F)O2 REAL300019304978
COc1ncc(Br)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304979
O=C(O)c1cnc2c(c1)CN(Cc1ccc(F)c3ccccc13)C2 REAL300019304980
O=C(O)c1cnc2c(c1)CN(Cc1cccnc1Br)C2 REAL300019304981
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C(F)F)nc1)C2 REAL300019304982
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1CC(F)(F)F)C2 REAL300019304983
CN(C)c1ccc(C#N)cc1CN1Cc2cc(C(=O)O)cnc2C1 REAL300019304984
O=C(O)c1cnc2c(c1)CN(Cc1ccc(C(F)(F)F)cc1[N+](=O)[O-])C2 REAL300019304985
O=C(O)c1cnc2c(c1)CN(Cc1nc(Br)c[nH]1)C2 REAL300019304986
CC(C)(C)OC(=O)N1C2CCC1CC(CN1Cc3cc(C(=O)O)cnc3C1)C2 REAL300019304987
CC(C)(C)OC(=O)NC1CC(CN2Cc3cc(C(=O)O)cnc3C2)C1 REAL300019304988
NS(=O)(=O)c1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c(F)c1 REAL300019304989
CC(C)(C)OC(=O)N[C@H]1C[C@@H](CN2Cc3cc(C(=O)O)cnc3C2)C1 REAL300019304990
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1F REAL300019304991
Cc1ccc(-c2ccc(CN3Cc4cc(C(=O)O)cnc4C3)o2)cc1 REAL300019304992
O=C(O)c1cnc2c(c1)CN(Cc1c[nH]nc1-c1cccnc1)C2 REAL300019304993
O=C(O)c1cnc2c(c1)CN(Cc1ccc(-n3cncn3)cc1)C2 REAL300019304994
Cc1nc(C)c2c(C)c(CN3Cc4cc(C(=O)O)cnc4C3)sc2n1 REAL300019304995
COc1cc(CN2Cc3cc(C(=O)O)cnc3C2)ccc1OCc1ccncc1 REAL300019304996
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)c2ccccc12 REAL300019304997
COc1ccc(CN2Cc3cc(C(=O)O)cnc3C2)cc1OCc1cccnc1 REAL300019304998
O=C(O)c1cnc2c(c1)CN(Cc1ccccc1OCc1cccnc1)C2 REAL300019304999
Cc1cc(CN2Cc3cc(C(=O)O)cnc3C2)cc(C)c1OCc1ccccn1 REAL300019305000
