COc1ccc(C=CC(=O)NCc2ncc(C(=O)O)s2)cc1OC REAL300004040001
O=C(C=Cc1ccc(SC(F)F)cc1)NCc1ncc(C(=O)O)s1 REAL300004040002
COc1ccc(OC)c(C=CC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040003
CC1(C)CCc2onc(C(=O)NCc3ncc(C(=O)O)s3)c2C1 REAL300004040004
Cc1ccc(-c2nc(C)c(C(=O)NCc3ncc(C(=O)O)s3)s2)cc1 REAL300004040005
O=C(Cc1csc(C2CCCC2)n1)NCc1ncc(C(=O)O)s1 REAL300004040006
O=C(Cc1csc(C2CC2)n1)NCc1ncc(C(=O)O)s1 REAL300004040007
CC1CCC(OCC(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040008
Cc1occ(C(F)(F)F)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040009
O=C(CCC1CCc2ccccc21)NCc1ncc(C(=O)O)s1 REAL300004040010
O=C(NCc1ncc(C(=O)O)s1)c1cc(C(F)(F)F)ccn1 REAL300004040011
CC1(C)COC(CCC(=O)NCc2ncc(C(=O)O)s2)C1 REAL300004040012
CC(C)(CC(=O)NCc1ncc(C(=O)O)s1)CC(F)(F)F REAL300004040013
COc1ccc(CCCCC(=O)NCc2ncc(C(=O)O)s2)cc1OC REAL300004040014
COc1ccc2c(c1)CCC(C(=O)NCc1ncc(C(=O)O)s1)C2 REAL300004040015
O=C(NCc1ncc(C(=O)O)s1)c1ccc(Cn2ccnc2)cc1 REAL300004040016
Cc1nc(CN2CCC(C(=O)NCc3ncc(C(=O)O)s3)CC2)cs1 REAL300004040017
CC(C(=O)NCc1ncc(C(=O)O)s1)N1CCN(C)CC1 REAL300004040018
O=C(CC1CCC2(CCC2)CO1)NCc1ncc(C(=O)O)s1 REAL300004040019
O=C(CC1CCC2(CCOCC2)CO1)NCc1ncc(C(=O)O)s1 REAL300004040020
Cc1cc(C)c(CC(=O)NCc2ncc(C(=O)O)s2)c(C)c1Br REAL300004040021
O=C(O)c1cnc(CNC(=O)C2CC3CCC(C2)S3)s1 REAL300004040022
O=C(O)c1cnc(CNC(=O)c2cscc2C(F)F)s1 REAL300004040023
COc1ccc(CCCC(=O)NCc2ncc(C(=O)O)s2)cc1OC REAL300004040024
O=C(O)c1cnc(CNC(=O)[C@@H]2[C@@H](c3ccccc3)C2(F)F)s1 REAL300004040025
CCOc1ccc(CCCC(=O)NCc2ncc(C(=O)O)s2)cc1OCC REAL300004040026
O=C(CCCc1ccc(Br)cc1)NCc1ncc(C(=O)O)s1 REAL300004040027
O=C(NCc1ncc(C(=O)O)s1)c1ccn(-c2cc(F)cc(F)c2)n1 REAL300004040028
O=C(CCCCc1ccccc1)NCc1ncc(C(=O)O)s1 REAL300004040029
Cc1c(Cl)ccc2c(CC(=O)NCc3ncc(C(=O)O)s3)coc12 REAL300004040030
Cc1cnc2c(C(=O)NCc3ncc(C(=O)O)s3)cnn2c1 REAL300004040031
Nc1c(C(=O)NCc2ncc(C(=O)O)s2)cc2ccccc2c1[N+](=O)[O-] REAL300004040032
O=C(CC1CCC2(CCC2)O1)NCc1ncc(C(=O)O)s1 REAL300004040033
O=C(O)c1cnc(CNC(=O)C2CCOC3(CCC3)C2)s1 REAL300004040034
O=C(C=Cc1cc(Br)ccc1F)NCc1ncc(C(=O)O)s1 REAL300004040035
COc1ccc2cc(C=CC(=O)NCc3ncc(C(=O)O)s3)ccc2c1 REAL300004040036
CCn1nc(C2CC2)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040037
Cn1nc2c(c1C(=O)NCc1ncc(C(=O)O)s1)CCC2 REAL300004040038
Cc1ccc([N+](=O)[O-])c(C(=O)NCc2ncc(C(=O)O)s2)c1C REAL300004040039
O=C(CCc1cccc(OCc2ccccc2)c1)NCc1ncc(C(=O)O)s1 REAL300004040040
O=C(NCc1ncc(C(=O)O)s1)c1cnc2ccccc2c1 REAL300004040041
O=C(O)c1cnc(CNC(=O)C2CC3(C2)CC(F)(F)C3)s1 REAL300004040042
CCSc1ccccc1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040043
C=CCOc1ccc(C=CC(=O)NCc2ncc(C(=O)O)s2)cc1OC REAL300004040044
CCCCc1oc2ccccc2c1C=CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040045
Cc1cc(C=CC(=O)NCc2ncc(C(=O)O)s2)c(C)n1C1CCCCC1 REAL300004040046
Cc1ccc(C=CC(=O)NCc2ncc(C(=O)O)s2)c(Br)c1 REAL300004040047
Cc1cccc(-c2cccc(C(=O)NCc3ncc(C(=O)O)s3)c2)c1 REAL300004040048
O=C(CC1CCc2sccc2C1=O)NCc1ncc(C(=O)O)s1 REAL300004040049
O=C(O)c1cnc(CNC(=O)c2ccc3c(c2[N+](=O)[O-])OCCCO3)s1 REAL300004040050
COC1(C(=O)NCc2ncc(C(=O)O)s2)CCSC1 REAL300004040051
CC12CC3CC(C1)CC(C(=O)NCc1ncc(C(=O)O)s1)(C3)C2 REAL300004040052
O=C(O)c1cnc(CNC(=O)C2(C3CCCCC3)CC2)s1 REAL300004040053
O=C(O)c1cnc(CNC(=O)C2(c3ccc4c(c3)OCCO4)CC2)s1 REAL300004040054
COc1cccc(C(F)F)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040055
Cc1ccc(F)c(Br)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040056
COc1cccc2c(C(=O)NCc3ncc(C(=O)O)s3)cnn12 REAL300004040057
CCn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(-c2ccccc2)n1 REAL300004040058
CC1CCc2n[nH]c(C(=O)NCc3ncc(C(=O)O)s3)c2C1 REAL300004040059
O=C(O)c1cnc(CNC(=O)c2ccc(Cn3cc(Cl)cn3)s2)s1 REAL300004040060
Cn1nc2c(c1C(=O)NCc1ncc(C(=O)O)s1)CCCC2 REAL300004040061
Cn1nc(-c2ccccc2)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040062
Cn1nc(C(F)(F)F)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040063
O=C(COCCc1ccc(Br)cc1)NCc1ncc(C(=O)O)s1 REAL300004040064
O=C(CCCc1ccc(C2CC2)cc1)NCc1ncc(C(=O)O)s1 REAL300004040065
O=C(O)c1cnc(CNC(=O)c2cc3c([nH]c2=O)CCOC3)s1 REAL300004040066
CCn1cc(Cl)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040067
COc1cc(OC)nc(C(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040068
CC1(C(=O)NCc2ncc(C(=O)O)s2)CCCS1(=O)=O REAL300004040069
O=C(NCc1ncc(C(=O)O)s1)c1cc(Cc2ccccc2)on1 REAL300004040070
COc1ccc2cc(C(=O)NCc3ncc(C(=O)O)s3)cnc2c1 REAL300004040071
CC(=O)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1C REAL300004040072
CCn1nc(C(=O)NCc2ncc(C(=O)O)s2)cc1C1CC1 REAL300004040073
CCc1cc(C(=O)NCc2ncc(C(=O)O)s2)ccc1Br REAL300004040074
Cc1onc(-c2cccc(F)c2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040075
N#CC1(C(=O)NCc2ncc(C(=O)O)s2)CC2CCC1C2 REAL300004040076
COc1ncc(C=CC(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040077
COC(C(=O)NCc1ncc(C(=O)O)s1)c1ccc(Br)s1 REAL300004040078
Cc1n[nH]c2c(C(=O)NCc3ncc(C(=O)O)s3)cccc12 REAL300004040079
O=C(O)c1cnc(CNC(=O)C2CCOC3(CCCC3)C2)s1 REAL300004040080
COc1cccc2[nH]c(C(=O)NCc3ncc(C(=O)O)s3)cc12 REAL300004040081
Cc1cc(C)c(CC(=O)NCc2ncc(C(=O)O)s2)c(=O)[nH]1 REAL300004040082
O=C(NCc1ncc(C(=O)O)s1)c1ccc2[nH]ccc2n1 REAL300004040083
Cn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C2CCCC2)n1 REAL300004040084
O=C(O)c1cnc(CNC(=O)C2(CCCOCc3ccccc3)CC2)s1 REAL300004040085
O=C(NCc1ncc(C(=O)O)s1)c1ccc(N2CCCCCC2)cc1 REAL300004040086
CC(Sc1ccc(F)cc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040087
O=C(O)c1cnc(CNC(=O)c2ccsc2C(F)F)s1 REAL300004040088
O=C(C[C@@H]1C[C@H]1Cc1ccccc1)NCc1ncc(C(=O)O)s1 REAL300004040089
O=C(NCc1ncc(C(=O)O)s1)c1ccc(Cn2ccnn2)o1 REAL300004040090
O=C(NCc1ncc(C(=O)O)s1)c1cnn(-c2ccccn2)c1 REAL300004040091
Cc1ccc(CC(=O)NCc2ncc(C(=O)O)s2)cc1Cl REAL300004040092
Cc1cc(C)n(CCCC(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040093
O=C(O)c1cnc(CNC(=O)c2nccc3cccnc23)s1 REAL300004040094
CC1(CC(=O)NCc2ncc(C(=O)O)s2)CCS(=O)(=O)N1 REAL300004040095
O=C(O)c1cnc(CNC(=O)c2ccnc3cc(Cl)ccc23)s1 REAL300004040096
COc1cccc(CC(C)CC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040097
CC(C)C1CC(C(=O)NCc2ncc(C(=O)O)s2)CCO1 REAL300004040098
O=C(O)c1cnc(CNC(=O)c2cccc3c2CCOC3)s1 REAL300004040099
O=C(CC1CCCC(C(F)(F)F)O1)NCc1ncc(C(=O)O)s1 REAL300004040100
O=C(CC1CCC(C2CC2)O1)NCc1ncc(C(=O)O)s1 REAL300004040101
O=C(O)c1cnc(CNC(=O)[C@H]2CC[C@H](Nc3cnccn3)CC2)s1 REAL300004040102
O=C(O)c1cnc(CNC(=O)[C@H]2CC[C@H](Nc3ncccn3)CC2)s1 REAL300004040103
CN(C)CCOc1ccc(CCC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040104
Cn1nc(C(F)(F)F)c2cc(C(=O)NCc3ncc(C(=O)O)s3)cnc21 REAL300004040105
O=C(O)c1cnc(CNC(=O)C2(CCc3ccccc3)CC2)s1 REAL300004040106
COc1ccc(CCC(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040107
CC1(C(=O)NCc2ncc(C(=O)O)s2)CCOc2ccccc21 REAL300004040108
O=C(O)c1cnc(CNC(=O)C2(c3ccccc3)CCCO2)s1 REAL300004040109
Cc1c(C)c2c(c(C)c1O)CCC(C)(C(=O)NCc1ncc(C(=O)O)s1)O2 REAL300004040110
COc1ccc2[nH]ccc2c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040111
Nc1nc(C2CCCC2)ncc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040112
Cn1cnc(-c2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)n1 REAL300004040113
O=C(O)c1cnc(CNC(=O)c2scnc2C2CCCC2)s1 REAL300004040114
CC1=C(C(=O)NCc2ncc(C(=O)O)s2)C(C)n2ncnc2N1C REAL300004040115
CN(Cc1ccccc1)Cc1cccc(C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040116
Cc1ccncc1C=CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040117
CC1(C(=O)NCc2ncc(C(=O)O)s2)CCN(Cc2ccccc2)CC1 REAL300004040118
Cc1cc(=O)cc(C)n1CCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040119
Cn1ccc(Nc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)n1 REAL300004040120
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)nnn1-c1cnn(C)c1 REAL300004040121
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)nnn1-c1ccn(C)n1 REAL300004040122
CCOc1nc(C(F)(F)F)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040123
CCOc1nc2cc(C(=O)NCc3ncc(C(=O)O)s3)ccc2[nH]1 REAL300004040124
CCC(CC)Oc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040125
Cc1cc(F)c(CC(=O)NCc2ncc(C(=O)O)s2)cc1F REAL300004040126
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2ccoc2)s1 REAL300004040127
Cn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(-c2ccoc2)n1 REAL300004040128
O=C(Cc1ccccc1OC1CCCC1)NCc1ncc(C(=O)O)s1 REAL300004040129
O=C(Cc1ccccc1OC1CCOC1)NCc1ncc(C(=O)O)s1 REAL300004040130
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)c2nccn2c1 REAL300004040131
O=C(O)c1cnc(CNC(=O)C2CCS(=O)(=O)c3ccccc32)s1 REAL300004040132
CC(C)(C)CCC1(O)CC(C(=O)NCc2ncc(C(=O)O)s2)C1 REAL300004040133
CCOc1nccc(C)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040134
CSc1ccc([N+](=O)[O-])cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040135
CNc1snc(C)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040136
O=C(NCc1ncc(C(=O)O)s1)c1ccc(Oc2ccc(F)cc2)cc1 REAL300004040137
O=C(Cc1cc(F)cc2c1OCOC2)NCc1ncc(C(=O)O)s1 REAL300004040138
CS(=O)(=O)NCCc1ccc(C(=O)NCc2ncc(C(=O)O)s2)s1 REAL300004040139
CS(=O)(=O)NCCc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040140
Cn1cc(S(N)(=O)=O)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040141
NS(=O)(=O)c1ccc(C=CC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040142
Cc1nc(COc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)no1 REAL300004040143
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2ccccc2)s1 REAL300004040144
O=C(O)c1cnc(CNC(=O)c2cnn(-c3ccccc3)c2C(F)(F)F)s1 REAL300004040145
O=C(NCc1ncc(C(=O)O)s1)c1cc(-c2cccs2)on1 REAL300004040146
COCCCOc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040147
O=C(CCCOc1cccc(Cl)c1Cl)NCc1ncc(C(=O)O)s1 REAL300004040148
NS(=O)(=O)c1cnn(CCC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040149
NS(=O)(=O)Cc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040150
NS(=O)(=O)c1cnn(CC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040151
NS(=O)(=O)c1ccc(OCC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040152
CC(C)Cc1nc(C(=O)NCc2ncc(C(=O)O)s2)cs1 REAL300004040153
NS(=O)(=O)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)s1 REAL300004040154
O=C(NCc1ncc(C(=O)O)s1)c1ccnc(-n2cncn2)c1 REAL300004040155
Cc1nc(S(=O)(=O)NCC(=O)NCc2ncc(C(=O)O)s2)cn1C REAL300004040156
Cc1nc(S(=O)(=O)NCCC(=O)NCc2ncc(C(=O)O)s2)cn1C REAL300004040157
Cc1noc(C(F)F)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040158
O=C(NCc1ncc(C(=O)O)s1)c1ccc2nc[nH]c2n1 REAL300004040159
Cc1nc(C(=O)NCc2ncc(C(=O)O)s2)c(=O)[nH]c1C REAL300004040160
O=C(O)c1cnc(CNC(=O)C2CCN(c3ccccc3)C2)s1 REAL300004040161
Cc1ccc(CC(=O)NCc2ncc(C(=O)O)s2)c(Cl)c1 REAL300004040162
O=C(Cc1ccc2cnccc2c1)NCc1ncc(C(=O)O)s1 REAL300004040163
O=C(Cc1ccc2[nH]ncc2c1)NCc1ncc(C(=O)O)s1 REAL300004040164
O=C(Cc1cccc(C(F)F)c1)NCc1ncc(C(=O)O)s1 REAL300004040165
Cc1cccc(CC(=O)NCc2ncc(C(=O)O)s2)c1Cl REAL300004040166
O=C(NCc1ncc(C(=O)O)s1)c1ccn2ccnc2c1 REAL300004040167
O=C(O)c1cnc(CNC(=O)c2cccc3nccn23)s1 REAL300004040168
O=C(NCc1ncc(C(=O)O)s1)c1ccc2nnnn2c1 REAL300004040169
Cc1ccc2ncc(C(=O)NCc3ncc(C(=O)O)s3)n2c1 REAL300004040170
Cc1nc(C(=O)NCc2ncc(C(=O)O)s2)c2ccccn12 REAL300004040171
O=C(O)c1cnc(CNC(=O)c2ncc3ccccn23)s1 REAL300004040172
O=C(O)c1cnc(CNC(=O)c2onc3c2CCCC3)s1 REAL300004040173
Cc1ccc2c(c1)CCC(C(=O)NCc1ncc(C(=O)O)s1)O2 REAL300004040174
COc1ccn2c(C(=O)NCc3ncc(C(=O)O)s3)cnc2c1 REAL300004040175
COc1coc(C(=O)NCc2ncc(C(=O)O)s2)cc1=O REAL300004040176
O=C(NCc1ncc(C(=O)O)s1)c1ccc2cncn2c1 REAL300004040177
Cc1csc(CCC(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040178
O=C(NCc1ncc(C(=O)O)s1)c1cnc2cnccc2c1 REAL300004040179
O=C(NCc1ncc(C(=O)O)s1)c1cnc2c(F)cccc2c1 REAL300004040180
O=C(NCc1ncc(C(=O)O)s1)c1ccc(C2CCCC2)cc1 REAL300004040181
Cc1[nH]nc(C(F)(F)F)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040182
O=C(O)c1cnc(CNC(=O)C2CCC(=O)c3cccn32)s1 REAL300004040183
O=C(O)c1cnc(CNC(=O)c2cccc3ccc(O)nc23)s1 REAL300004040184
Cc1cc(S(N)(=O)=O)cc(C(=O)NCc2ncc(C(=O)O)s2)c1C REAL300004040185
COCCOc1cncc(C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040186
CNS(=O)(=O)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040187
NS(=O)(=O)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040188
CN(C)S(=O)(=O)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040189
Cn1cnc(S(=O)(=O)NCC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040190
O=C(CC(O)c1cc(Cl)cc(Cl)c1)NCc1ncc(C(=O)O)s1 REAL300004040191
CCC(C)(C)C1CCC2(CC1)CC2C(=O)NCc1ncc(C(=O)O)s1 REAL300004040192
COc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1C1CC1 REAL300004040193
Cc1ccc(OCCCC(=O)NCc2ncc(C(=O)O)s2)c(Cl)c1 REAL300004040194
CSCc1noc(CCC(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040195
CCOc1nc(C)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040196
CCCOc1nc(C)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040197
O=C(O)c1cnc(CNC(=O)C2(Cc3cccs3)CCCCC2)s1 REAL300004040198
O=C(O)c1cnc(CNC(=O)c2cccnc2OCc2ccccc2F)s1 REAL300004040199
COc1cc(OC2CC2)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040200
O=C(NCc1ncc(C(=O)O)s1)c1ccc(Oc2ccccc2)cn1 REAL300004040201
CC(C)(C)Oc1ccc(C(=O)NCc2ncc(C(=O)O)s2)nc1 REAL300004040202
Cc1nccc(CCC(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040203
O=C(O)c1cnc(CNC(=O)C2CCn3c(cnc3-c3ccccc3)C2)s1 REAL300004040204
O=C(CCCCc1c[nH]nn1)NCc1ncc(C(=O)O)s1 REAL300004040205
O=C(Cc1cc(Cl)cc2c1OCC2)NCc1ncc(C(=O)O)s1 REAL300004040206
CN(C)CC1(C(=O)NCc2ncc(C(=O)O)s2)CCCCC1 REAL300004040207
CCc1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C)nn1 REAL300004040208
CC1(Cn2cc(C(=O)NCc3ncc(C(=O)O)s3)nn2)COC1 REAL300004040209
O=C(O)c1cnc(CNC(=O)c2ocnc2C(F)(F)F)s1 REAL300004040210
CN(CCC(=O)NCc1ncc(C(=O)O)s1)C1CCCCC1 REAL300004040211
O=C(O)c1cnc(CNC(=O)C2COCCN2CC(F)F)s1 REAL300004040212
O=C(O)c1cnc(CNC(=O)c2ccc(C(F)(F)F)cc2N2CCCC2)s1 REAL300004040213
COc1cccc(Oc2ccc(C(=O)NCc3ncc(C(=O)O)s3)nc2)c1 REAL300004040214
O=C(NCc1ncc(C(=O)O)s1)c1cncc(-n2ccnn2)c1 REAL300004040215
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2ccc(Cl)cc2)s1 REAL300004040216
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2ccc3c(c2)OCCO3)s1 REAL300004040217
CC(C)(C)C(Br)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040218
CC1CN(c2ccnc(C(=O)NCc3ncc(C(=O)O)s3)c2)CC(C)O1 REAL300004040219
Cc1cc(C)n(CCC(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040220
O=C(O)c1cnc(CNC(=O)c2ccc(C(F)(F)F)[nH]c2=O)s1 REAL300004040221
O=C(CNS(=O)(=O)c1cccnc1)NCc1ncc(C(=O)O)s1 REAL300004040222
Cc1ccc(C(O)(CC(=O)NCc2ncc(C(=O)O)s2)C(F)(F)F)o1 REAL300004040223
O=C(NCc1ncc(C(=O)O)s1)c1cc2ccsc2[nH]1 REAL300004040224
Cc1nc(C(=O)NCc2ncc(C(=O)O)s2)nn1-c1nnc[nH]1 REAL300004040225
O=C(NCc1ncc(C(=O)O)s1)c1ccc(-n2ccnc2)nc1 REAL300004040226
O=C(O)c1cnc(CNC(=O)c2cnc3ccccc3c2C(F)(F)F)s1 REAL300004040227
Cc1noc2ncc(C(=O)NCc3ncc(C(=O)O)s3)cc12 REAL300004040228
CCCN(CC)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040229
CCN(Cc1ccccc1)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040230
CCN(c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1)C(C)C REAL300004040231
CCOc1cc(C=CC(=O)NCc2ncc(C(=O)O)s2)ccc1O REAL300004040232
CCCN(C)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040233
O=C(O)c1cnc(CNC(=O)C2CCCCN2Cc2ccc(F)cc2)s1 REAL300004040234
O=C(O)c1cnc(CNC(=O)C2CCCN2Cc2ccc(F)cc2)s1 REAL300004040235
CCCS(=O)(=O)Nc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040236
CC(C)c1ccc(C2(C(=O)NCc3ncc(C(=O)O)s3)CCCC2)cc1 REAL300004040237
O=C(NCc1ncc(C(=O)O)s1)c1cccc(Cn2cncn2)c1 REAL300004040238
Cc1noc(C2CC2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040239
Cn1nnc2cc(C(=O)NCc3ncc(C(=O)O)s3)cnc21 REAL300004040240
O=C(NCc1ncc(C(=O)O)s1)c1cccc(-c2ncn[nH]2)c1 REAL300004040241
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C)cc1Cl REAL300004040242
Cn1cnc2cc(C(=O)NCc3ncc(C(=O)O)s3)cnc21 REAL300004040243
O=C(NCc1ncc(C(=O)O)s1)c1csc(NC2CC2)n1 REAL300004040244
Cc1nc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2n1C REAL300004040245
Cc1ccn(C(C)CC(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040246
CCNc1nc(C(=O)NCc2ncc(C(=O)O)s2)cs1 REAL300004040247
Cc1ccc2snc(C(=O)NCc3ncc(C(=O)O)s3)c2c1 REAL300004040248
Cc1oc(S(N)(=O)=O)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040249
CC(C)(CC(=O)NCc1ncc(C(=O)O)s1)Cc1ccc(Cl)cc1 REAL300004040250
CC(Cc1ccccc1)n1cccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040251
CC(C)(C(=O)NCc1ncc(C(=O)O)s1)c1csc(-c2cccs2)n1 REAL300004040252
O=C(COCc1cccc(Cl)c1)NCc1ncc(C(=O)O)s1 REAL300004040253
Cc1nc(O)c(C(=O)NCc2ncc(C(=O)O)s2)cc1Br REAL300004040254
Cn1nc(C(F)F)c2cc(C(=O)NCc3ncc(C(=O)O)s3)sc21 REAL300004040255
O=C(NCc1ncc(C(=O)O)s1)c1coc(C2CCOCC2)n1 REAL300004040256
CCc1nc(-c2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)n[nH]1 REAL300004040257
COCCOc1ccc(C(=O)NCc2ncc(C(=O)O)s2)c(Cl)c1 REAL300004040258
O=C(O)c1cnc(CNC(=O)C2(Cc3ccccc3)CCOCC2)s1 REAL300004040259
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)nc(-c2ccc(Cl)cc2)n1 REAL300004040260
O=C(CC1CCCS(=O)(=O)C1)NCc1ncc(C(=O)O)s1 REAL300004040261
O=C(NCc1ncc(C(=O)O)s1)c1cn(C2CCOCC2)nn1 REAL300004040262
CC(C)C1CC(CC(=O)NCc2ncc(C(=O)O)s2)CCO1 REAL300004040263
CCC1CC(CC(=O)NCc2ncc(C(=O)O)s2)CCO1 REAL300004040264
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)nnn1Cc1ccc(F)cc1F REAL300004040265
CCc1onc(-c2ccccc2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040266
Nc1nc(C2CC2)ncc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040267
O=C(O)c1cnc(CNC(=O)c2occ3c2CCOC3)s1 REAL300004040268
O=C(NCc1ncc(C(=O)O)s1)c1ccc(C(=O)c2cccc(O)c2)cc1 REAL300004040269
COC(C(=O)NCc1ncc(C(=O)O)s1)c1cnn(C)c1 REAL300004040270
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)cc(NCC(F)(F)F)n1 REAL300004040271
CC(C)(C(=O)NCc1ncc(C(=O)O)s1)S(=O)(=O)C1CC1 REAL300004040272
Cn1cc(Oc2ccccc2C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040273
Cn1ncc2c(=O)[nH]c(CCC(=O)NCc3ncc(C(=O)O)s3)nc21 REAL300004040274
COc1cc(CC(=O)NCc2ncc(C(=O)O)s2)ccc1O REAL300004040275
O=C(Cc1ccc(O)c(F)c1)NCc1ncc(C(=O)O)s1 REAL300004040276
O=C(NCc1ncc(C(=O)O)s1)c1cc(-c2ccncc2)on1 REAL300004040277
O=C(Cc1c[nH]c2ccc(Br)cc12)NCc1ncc(C(=O)O)s1 REAL300004040278
COc1ccccc1-c1cc(C(=O)NCc2ncc(C(=O)O)s2)no1 REAL300004040279
O=C(O)c1cnc(CNC(=O)C(O)CCc2ccccc2)s1 REAL300004040280
O=C(NCc1ncc(C(=O)O)s1)c1ccc2c(c1)OC(F)(F)O2 REAL300004040281
O=C(O)c1cnc(CNC(=O)C2(c3ccc(Cl)cc3)CCCCC2)s1 REAL300004040282
CCCOc1cccnc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040283
CS(=O)(=O)Nc1cc(C(=O)NCc2ncc(C(=O)O)s2)ccc1Cl REAL300004040284
CC(C)(C)c1ccc(C2(C(=O)NCc3ncc(C(=O)O)s3)CCC2)cc1 REAL300004040285
O=C(O)c1cnc(CNC(=O)c2cnc(-c3ccccn3)s2)s1 REAL300004040286
O=C(NCc1ncc(C(=O)O)s1)c1ccc(-n2ccnc2)nn1 REAL300004040287
CCC(Nc1nnnn1-c1ccccc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040288
O=C(NCc1ncc(C(=O)O)s1)c1cccc(-n2nccc2C(F)(F)F)c1 REAL300004040289
O=C(NCc1ncc(C(=O)O)s1)c1ccc(Oc2cccc(Cl)c2)cc1 REAL300004040290
O=C(NCc1ncc(C(=O)O)s1)c1ccc(Nc2ccncc2)cc1 REAL300004040291
O=C(O)c1cnc(CNC(=O)C2(Cc3cccc(F)c3)CCCCC2)s1 REAL300004040292
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1-c1ccccc1OC REAL300004040293
CCn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C(F)(F)F)n1 REAL300004040294
Cn1ccnc1CNc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040295
CN(C)CCn1ncc(C(=O)NCc2ncc(C(=O)O)s2)c1-c1ccccc1 REAL300004040296
O=C(NCc1ncc(C(=O)O)s1)c1cc(F)c(N2CCOCC2)c(F)c1 REAL300004040297
Cc1ccc(-n2cc(C(=O)NCc3ncc(C(=O)O)s3)c(C(C)(C)C)n2)cc1 REAL300004040298
CCOCCS(=O)(=O)NCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040299
Cc1cn2ccnc(C(=O)NCc3ncc(C(=O)O)s3)c2n1 REAL300004040300
O=C(NCc1ncc(C(=O)O)s1)c1cncc(N2CCOCC2)c1 REAL300004040301
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1-c1ccccc1Cl REAL300004040302
COc1ccccc1-n1ncc(C(=O)NCc2ncc(C(=O)O)s2)c1C REAL300004040303
Cc1nc(C(=O)NCc2ncc(C(=O)O)s2)c(-c2ccccc2)s1 REAL300004040304
O=C(O)c1cnc(CNC(=O)c2ncsc2-c2ccccc2)s1 REAL300004040305
CN(C)c1cc(C(=O)NCc2ncc(C(=O)O)s2)nc2ccccc12 REAL300004040306
O=C(NCc1ncc(C(=O)O)s1)c1ccc(OC2CCOC2)cc1 REAL300004040307
O=C(Cc1ccc(Br)c(Cl)c1)NCc1ncc(C(=O)O)s1 REAL300004040308
Cc1c(Br)cccc1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040309
O=C(O)c1cnc(CNC(=O)c2cccc(O)c2OC(F)(F)F)s1 REAL300004040310
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)c(O)nc2ccccc12 REAL300004040311
O=C(O)c1cnc(CNC(=O)c2cc3sc(N4CCCC4)nc3s2)s1 REAL300004040312
O=C(O)c1cnc(CNC(=O)c2nc(C(F)(F)F)n3ccccc23)s1 REAL300004040313
Cc1noc(C)c1C(C)(C)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040314
O=C(O)c1cnc(CNC(=O)c2nc3ccccc3nc2C2CC2)s1 REAL300004040315
O=C(O)c1cnc(CNC(=O)C2(c3cccnc3)CC2)s1 REAL300004040316
CN(C)c1cccc(CCC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040317
Cc1nc(O)c(Br)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040318
CC(C(=O)NCc1ncc(C(=O)O)s1)N(C)CC(F)(F)F REAL300004040319
O=C(O)c1cnc(CNC(=O)C2CCCCN2C2CCCC2)s1 REAL300004040320
O=C(O)c1cnc(CNC(=O)C2CCC(N3CCOCC3)CC2)s1 REAL300004040321
O=C(O)c1cnc(CNC(=O)c2cc(F)cc3[nH]nnc23)s1 REAL300004040322
Cc1nn(C)c(-n2ccnc2C)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040323
O=C(Cc1cncn1Cc1ccccc1)NCc1ncc(C(=O)O)s1 REAL300004040324
O=C(O)c1cnc(CNC(=O)C(CO)c2ccccc2)s1 REAL300004040325
Nc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1OC(F)(F)F REAL300004040326
O=C(O)c1cnc(CNC(=O)C(O)c2ccc(Cl)cc2)s1 REAL300004040327
O=C(O)c1cnc(CNC(=O)c2ccc(F)c3ccccc23)s1 REAL300004040328
Cc1ccc(C(=O)NCc2ncc(C(=O)O)s2)c(Cl)c1 REAL300004040329
CC(C)Cc1ccc(C(C)C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040330
O=C(O)c1cnc(CNC(=O)c2cccc3cc(O)ccc23)s1 REAL300004040331
O=C(CCCn1cnc2ccccc21)NCc1ncc(C(=O)O)s1 REAL300004040332
COc1cc(C(=O)NCc2ncc(C(=O)O)s2)cc(OC)c1O REAL300004040333
Cc1nn(-c2ccccc2)c2ncc(C(=O)NCc3ncc(C(=O)O)s3)cc12 REAL300004040334
CC(C(=O)NCc1ncc(C(=O)O)s1)c1cccc(C(=O)c2ccccc2)c1 REAL300004040335
O=C(O)c1cnc(CNC(=O)c2ccccc2NCc2ccccc2)s1 REAL300004040336
O=C(O)c1cnc(CNC(=O)C2Cc3ccccc3C2)s1 REAL300004040337
O=C(O)c1cnc(CNC(=O)c2cccnc2N2CCCCC2)s1 REAL300004040338
O=C(O)c1cnc(CNC(=O)c2ccc(C(F)(F)F)cc2O)s1 REAL300004040339
O=C(O)c1cnc(CNC(=O)C2CCC(C(F)(F)F)CC2)s1 REAL300004040340
O=C(Cc1cc(Cl)ccc1Br)NCc1ncc(C(=O)O)s1 REAL300004040341
CC(NS(C)(=O)=O)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040342
O=C(O)c1cnc(CNC(=O)[C@H](O)c2ccccc2Cl)s1 REAL300004040343
CC(C)(C)c1ccc(CC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040344
C[C@@H](OCc1ccccc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040345
Nc1c(Cl)cc(C(=O)NCc2ncc(C(=O)O)s2)cc1Cl REAL300004040346
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C(F)(F)F)o1 REAL300004040347
O=C(CNc1cccc(C(F)(F)F)c1)NCc1ncc(C(=O)O)s1 REAL300004040348
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)c2c(C)n[nH]c2n1 REAL300004040349
O=C(NCc1ncc(C(=O)O)s1)c1cc(C(F)(F)F)n[nH]1 REAL300004040350
Cc1cccn2cc(CC(=O)NCc3ncc(C(=O)O)s3)nc12 REAL300004040351
O=C(Cc1cn2cc(Cl)cc(Cl)c2n1)NCc1ncc(C(=O)O)s1 REAL300004040352
Cc1nccn1CCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040353
O=C(CCCCN1CCOCC1)NCc1ncc(C(=O)O)s1 REAL300004040354
CC(C)(C(=O)NCc1ncc(C(=O)O)s1)N1CCOCC1 REAL300004040355
CCN(Cc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1)C(C)C REAL300004040356
O=C(O)c1cnc(CNC(=O)C2CC3COCC(C2)C3=O)s1 REAL300004040357
Cc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1Oc1ccncc1 REAL300004040358
CC(=CC(=O)NCc1ncc(C(=O)O)s1)c1ccccc1C REAL300004040359
CC(O)(Cc1ccccc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040360
CC(Oc1cccnc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040361
CCc1nc(C(=O)NCc2ncc(C(=O)O)s2)nn1-c1ccccc1 REAL300004040362
O=C(CN(Cc1cccnc1)c1ccccc1)NCc1ncc(C(=O)O)s1 REAL300004040363
Cn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(-c2ccccc2)n1 REAL300004040364
CNS(=O)(=O)N1CCC(C(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040365
COCCOc1cc(C(=O)NCc2ncc(C(=O)O)s2)nc2ccccc12 REAL300004040366
COc1cccc(-c2nc(C(=O)NCc3ncc(C(=O)O)s3)c(C)[nH]2)c1 REAL300004040367
O=C(NCc1ncc(C(=O)O)s1)c1cncc(-c2ccc(Cl)cc2)c1 REAL300004040368
Cc1ccc(-c2cncc(C(=O)NCc3ncc(C(=O)O)s3)c2)cc1 REAL300004040369
Cc1onc(-c2ccccn2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040370
Cc1onc(-c2cccnc2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040371
Cc1onc(-c2ccncc2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040372
O=C(NCc1ncc(C(=O)O)s1)c1coc(C2CCC2)n1 REAL300004040373
O=C(CC1(Cn2cnnn2)CCCCC1)NCc1ncc(C(=O)O)s1 REAL300004040374
O=C(O)c1cnc(CNC(=O)c2ncccc2Oc2ccccc2)s1 REAL300004040375
O=C(O)c1cnc(CNC(=O)C(O)c2ccc(Cl)cc2F)s1 REAL300004040376
O=C(O)c1cnc(CNC(=O)C(O)c2cc(Cl)cc(Cl)c2)s1 REAL300004040377
Cc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1N1CCOCC1 REAL300004040378
Cn1cc(-c2ccc(C(=O)NCc3ncc(C(=O)O)s3)o2)cn1 REAL300004040379
O=C(O)c1cnc(CNC(=O)C2CCN(Cc3ccccc3)C2)s1 REAL300004040380
O=C(O)c1cnc(CNC(=O)C2CCN(C3CCSC3)CC2)s1 REAL300004040381
O=C(NCc1ncc(C(=O)O)s1)c1cc(Cn2cccn2)on1 REAL300004040382
O=C(CN(Cc1ccccc1)c1ccccc1)NCc1ncc(C(=O)O)s1 REAL300004040383
Cc1nn(CC(F)(F)F)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040384
COc1cccc(C(C)CCCC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040385
CC1Cc2cn[nH]c2C(C(=O)NCc2ncc(C(=O)O)s2)C1 REAL300004040386
Cc1cc(C2(C(=O)NCc3ncc(C(=O)O)s3)CC2)on1 REAL300004040387
O=C(CCc1ccc(=O)[nH]c1)NCc1ncc(C(=O)O)s1 REAL300004040388
COc1ccc(CC(=O)NCc2ncc(C(=O)O)s2)nc1 REAL300004040389
Cn1ncc2c1CC(C(=O)NCc1ncc(C(=O)O)s1)CC2 REAL300004040390
O=C(CCc1ccc(O)cc1)NCc1ncc(C(=O)O)s1 REAL300004040391
O=C(NCc1ncc(C(=O)O)s1)c1ccc2cccnc2n1 REAL300004040392
CCS(=O)(=O)NC(C)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040393
Cc1nc2c(c(C)nn2C)c(C)c1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040394
Cc1nn(-c2ccccn2)c(C)c1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040395
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C)n1-c1ccccn1 REAL300004040396
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C)n1-c1cccnc1 REAL300004040397
CCS(=O)(=O)NCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040398
CS(=O)(=O)NCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040399
CC(C)(C)c1ccc(C(O)CCC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040400
O=C(NCc1ncc(C(=O)O)s1)c1csc(Cc2ccc(F)cc2)n1 REAL300004040401
O=C(NCc1ncc(C(=O)O)s1)c1ccc(C(F)F)cc1 REAL300004040402
CC1CCN(c2ccc(C(=O)NCc3ncc(C(=O)O)s3)cn2)CC1 REAL300004040403
COc1ccc(Cn2cc(C(=O)NCc3ncc(C(=O)O)s3)cn2)cc1 REAL300004040404
O=C(NCc1ncc(C(=O)O)s1)c1ccc(N2CCCC2)nc1 REAL300004040405
O=C(NCc1ncc(C(=O)O)s1)c1ccc(-n2cnc3ccccc32)cc1 REAL300004040406
O=C1NC(=O)C2(CCC(C(=O)NCc3ncc(C(=O)O)s3)CC2)N1 REAL300004040407
O=C(NCc1ncc(C(=O)O)s1)c1ccc(N2CCCC2)nn1 REAL300004040408
CN1CCN(C(C(=O)NCc2ncc(C(=O)O)s2)c2ccccc2)CC1 REAL300004040409
O=C(CC1(N2CCOCC2)CCCC1)NCc1ncc(C(=O)O)s1 REAL300004040410
O=C(NCc1ncc(C(=O)O)s1)c1cc2cccnc2[nH]1 REAL300004040411
O=C(NCc1ncc(C(=O)O)s1)c1cc(C(F)F)[nH]n1 REAL300004040412
Cn1cnc2c(C(=O)NCc3ncc(C(=O)O)s3)ccnc21 REAL300004040413
O=C(NCc1ncc(C(=O)O)s1)c1ccnc(-n2cccn2)c1 REAL300004040414
CC(C(=O)NCc1ncc(C(=O)O)s1)N(C)Cc1ccccc1 REAL300004040415
CC(C)Cc1ccc([C@H](C)C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040416
O=C(O)c1cnc(CNC(=O)C2CCN(CC(F)(F)F)CC2)s1 REAL300004040417
CCNc1ccc(Cl)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040418
CNc1cc(Cl)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040419
CC(C)CCn1cc(C(=O)NCc2ncc(C(=O)O)s2)nn1 REAL300004040420
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)nnn1CC REAL300004040421
O=C(O)c1cnc(CNC(=O)c2cc3occc3s2)s1 REAL300004040422
O=C(CN1CCN(c2ccccn2)CC1)NCc1ncc(C(=O)O)s1 REAL300004040423
O=C(NCc1ncc(C(=O)O)s1)c1c[nH]c(-c2ccccc2)n1 REAL300004040424
COc1cc(C(=O)NCc2ncc(C(=O)O)s2)cc(OC)c1OC(F)F REAL300004040425
O=C(O)c1cnc(CNC(=O)C2CCCN(CCc3ccccc3)C2)s1 REAL300004040426
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2ccccc2Cl)s1 REAL300004040427
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2cccc(Cl)c2)s1 REAL300004040428
O=C(O)c1cnc(CNC(=O)C2(c3ccccc3Br)CC2)s1 REAL300004040429
O=C(O)c1cnc(CNC(=O)c2cnc(-c3cccnc3)s2)s1 REAL300004040430
Cc1onc(-c2cccc(Cl)c2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040431
O=C(NCc1ncc(C(=O)O)s1)c1cc(-c2ccccc2C(F)(F)F)on1 REAL300004040432
O=C(CCCOc1ccc2c(c1)CCCC2)NCc1ncc(C(=O)O)s1 REAL300004040433
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)[nH]c2c(Cl)cccc12 REAL300004040434
O=C(O)c1cnc(CNC(=O)c2cnn(CCO)c2-c2ccccc2)s1 REAL300004040435
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1-c1ccc(OC)cc1 REAL300004040436
CCC(O)(C(=O)NCc1ncc(C(=O)O)s1)c1cccc(Cl)c1 REAL300004040437
COc1cccc(C(=O)c2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)c1 REAL300004040438
Cc1[nH]c2ccc(Cl)cc2c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040439
CCCc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1C1CCCC1 REAL300004040440
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1C1CCCC1 REAL300004040441
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1C1CCCCC1 REAL300004040442
CCCCn1ncc(C(=O)NCc2ncc(C(=O)O)s2)c1C REAL300004040443
CCCCn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C)n1 REAL300004040444
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1C(CC)CC REAL300004040445
CS(=O)(=O)Nc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040446
COc1cccnc1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040447
O=C(O)c1cnc(CNC(=O)c2ccoc2C2(O)CCOCC2)s1 REAL300004040448
CN(C)C(C(=O)NCc1ncc(C(=O)O)s1)c1cncn1C REAL300004040449
Cn1nnc2c1CC(C(=O)NCc1ncc(C(=O)O)s1)CC2 REAL300004040450
Cn1cc2c(n1)CCCC2C(=O)NCc1ncc(C(=O)O)s1 REAL300004040451
O=C(NCc1ncc(C(=O)O)s1)c1cn(-c2ccc(Cl)c(Cl)c2)cn1 REAL300004040452
C[C@H](Oc1ccc(Br)cc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040453
CN(C)Cc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040454
O=C(Cn1nc(C(F)(F)F)c2c1CCOC2)NCc1ncc(C(=O)O)s1 REAL300004040455
CC1(c2ccccc2C(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040456
CCC(C)(C)c1ccccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040457
O=C(NCc1ncc(C(=O)O)s1)c1ccc(OCc2cccnc2)cc1 REAL300004040458
O=C(O)c1cnc(CNC(=O)c2ccccc2OCc2ccncc2)s1 REAL300004040459
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C)n1Cc1ccccn1 REAL300004040460
CCCc1noc2nc(C3CC3)cc(C(=O)NCc3ncc(C(=O)O)s3)c12 REAL300004040461
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1-c1ccccn1 REAL300004040462
O=C(O)c1cnc(CNC(=O)c2cnn(-c3ccccn3)c2C(F)(F)F)s1 REAL300004040463
O=C(NCc1ncc(C(=O)O)s1)c1cccc(CN2CCOCC2)c1 REAL300004040464
CCCN(CCC)CCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040465
O=C(O)c1cnc(CNC(=O)C(c2ccccc2)N2CCC(O)CC2)s1 REAL300004040466
CCN(C)C(C(=O)NCc1ncc(C(=O)O)s1)c1ccccc1 REAL300004040467
O=C(Cc1csc(-c2nnc[nH]2)n1)NCc1ncc(C(=O)O)s1 REAL300004040468
CCCOc1cn(-c2ccccc2)nc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040469
CCn1nc(C)c(CC(=O)NCc2ncc(C(=O)O)s2)c1C REAL300004040470
CC(C(=O)NCc1ncc(C(=O)O)s1)c1ccc(S(C)(=O)=O)cc1 REAL300004040471
CCN(CC)C(C(=O)NCc1ncc(C(=O)O)s1)c1ccccc1 REAL300004040472
CC(C)COc1ncccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040473
O=C(NCc1ncc(C(=O)O)s1)c1nc2n(n1)CCCN2 REAL300004040474
CSC(C(=O)NCc1ncc(C(=O)O)s1)c1ccccc1 REAL300004040475
O=C(Cn1cc(Cl)cn1)NCc1ncc(C(=O)O)s1 REAL300004040476
COc1cccc(C2(C(=O)NCc3ncc(C(=O)O)s3)CC2)c1 REAL300004040477
CN(C)S(=O)(=O)NCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040478
CC(C)c1nccn1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040479
O=C(O)c1cnc(CNC(=O)c2cnc(C3CC3)[nH]c2=O)s1 REAL300004040480
CN(C)C(C(=O)NCc1ncc(C(=O)O)s1)c1ccc(Cl)cc1 REAL300004040481
CCn1ncc(C(=O)NCc2ncc(C(=O)O)s2)c1-c1ccccc1 REAL300004040482
CC(C)(C)OCc1cc(C(=O)NCc2ncc(C(=O)O)s2)no1 REAL300004040483
CC=CCOc1cccc(CC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040484
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1CCC(C)C REAL300004040485
O=C(NCc1ncc(C(=O)O)s1)c1ccc2c(Br)cccc2c1 REAL300004040486
CC(C)Cc1cccc(C(C)C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040487
Cc1nn(-c2cccc(F)c2)cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040488
COc1ccc(C(=O)NCc2ncc(C(=O)O)s2)c(OC(F)F)c1 REAL300004040489
COCCOc1cccc(CC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040490
O=C(NCc1ncc(C(=O)O)s1)c1ccc(OC(F)F)c(F)c1 REAL300004040491
Cc1cc(C(=O)NCc2ncc(C(=O)O)s2)nn1-c1ccc(F)cc1 REAL300004040492
CC(C)c1cc(C(=O)NCc2ncc(C(=O)O)s2)nn1-c1ccccc1 REAL300004040493
O=C(NCc1ncc(C(=O)O)s1)c1cn(CCc2ccccc2)nn1 REAL300004040494
O=C(NCc1ncc(C(=O)O)s1)c1ccc(CN2CCCC2)cc1 REAL300004040495
O=C(CCCOc1ccc2c(c1)CCC2)NCc1ncc(C(=O)O)s1 REAL300004040496
Cc1nn(CC(F)F)c(C)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040497
Cn1cc(CNc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)cn1 REAL300004040498
Cc1nn(C(C)C)c(C)c1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040499
CCSCc1cc(C(=O)NCc2ncc(C(=O)O)s2)no1 REAL300004040500
O=C(O)c1cnc(CNC(=O)c2cc(F)ccc2-n2cccn2)s1 REAL300004040501
O=C(NCc1ncc(C(=O)O)s1)c1cccc(CN2CCCCC2)c1 REAL300004040502
O=C(Cn1c(C2CCCCC2)nc2ccccc21)NCc1ncc(C(=O)O)s1 REAL300004040503
CC(C)(C)c1n[nH]cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040504
Nc1ncnc2c1ncn2CCCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040505
CCC1CN(C(CC)C(=O)NCc2ncc(C(=O)O)s2)CCO1 REAL300004040506
CCN(CC(=O)NCc1ncc(C(=O)O)s1)Cc1ccccc1Cl REAL300004040507
O=C(CC1CCN(CC(F)(F)F)CC1)NCc1ncc(C(=O)O)s1 REAL300004040508
CCN1CCC(N2CCC(C(=O)NCc3ncc(C(=O)O)s3)CC2)CC1 REAL300004040509
O=C(O)c1cnc(CNC(=O)C2CCCN(CC(F)F)C2)s1 REAL300004040510
O=C(O)c1cnc(CNC(=O)C2CCCc3[nH]nnc32)s1 REAL300004040511
O=C(CC(c1ccccc1)c1ncc[nH]1)NCc1ncc(C(=O)O)s1 REAL300004040512
O=C(O)c1cnc(CNC(=O)c2coc3cc(O)ccc23)s1 REAL300004040513
COc1ccc(C=CC(=O)NCc2ncc(C(=O)O)s2)cc1S(N)(=O)=O REAL300004040514
CC1CN(c2ccc(C(=O)NCc3ncc(C(=O)O)s3)cn2)CC(C)O1 REAL300004040515
CC1CN(Cc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)CC(C)O1 REAL300004040516
O=C(NCc1ncc(C(=O)O)s1)c1cncc(-c2ccccc2)c1 REAL300004040517
CN(CC(=O)NCc1ncc(C(=O)O)s1)c1nc2ccccc2s1 REAL300004040518
O=C(NCc1ncc(C(=O)O)s1)c1cccc(Nc2ncccn2)c1 REAL300004040519
CC(Oc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1)c1ccccc1 REAL300004040520
O=C(O)c1cnc(CNC(=O)[C@@H](O)Cc2ccccc2)s1 REAL300004040521
O=C(O)c1cnc(CNC(=O)C(O)c2cccc(C(F)(F)F)c2)s1 REAL300004040522
COc1cc(C)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040523
Cc1ccc(F)c(CC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040524
O=C(O)c1cnc(CNC(=O)c2cc(O)ccc2Cl)s1 REAL300004040525
Cc1ccc(-n2nc(C(=O)NCc3ncc(C(=O)O)s3)c3c2CCC3)c(C)c1 REAL300004040526
O=C(CC1CN(Cc2ccccc2)CCO1)NCc1ncc(C(=O)O)s1 REAL300004040527
O=C(O)c1cnc(CNC(=O)c2ccccc2CN2CCOCC2)s1 REAL300004040528
COc1ccc(Nc2nc(C(=O)NCc3ncc(C(=O)O)s3)cs2)cc1 REAL300004040529
O=C(O)c1cnc(CNC(=O)c2ccc3cccnn23)s1 REAL300004040530
O=C(O)c1cnc(CNC(=O)c2cnn3c(=O)cc[nH]c23)s1 REAL300004040531
O=C(O)c1cnc(CNC(=O)c2cnc3cccnn23)s1 REAL300004040532
Cc1cc(C(F)(F)F)nn1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040533
O=C(NCc1ncc(C(=O)O)s1)c1cccc(OCC(F)(F)F)c1 REAL300004040534
CC(CC(=O)NCc1ncc(C(=O)O)s1)c1c[nH]c2ccccc12 REAL300004040535
O=C(NCc1ncc(C(=O)O)s1)c1cc(-c2cccc(O)c2)on1 REAL300004040536
Cc1c(NCC(C)(C)C)cccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040537
COCCNS(=O)(=O)c1c[nH]c(C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040538
CC(C)c1cccc(-n2cc(O)c(C(=O)NCc3ncc(C(=O)O)s3)n2)c1 REAL300004040539
CC(C)c1ccc(-n2cc(O)c(C(=O)NCc3ncc(C(=O)O)s3)n2)cc1 REAL300004040540
Cc1c(NC(C)C(C)C)cccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040541
O=C(O)c1cnc(CNC(=O)C2CC(OCc3ccccc3)C2)s1 REAL300004040542
O=C(O)c1cnc(CNC(=O)C2CCCCN2Cc2ccccc2)s1 REAL300004040543
CC(Oc1cccc(CO)c1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040544
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1-c1ccncc1 REAL300004040545
O=C(O)c1cnc(CNC(=O)c2c[nH]cc2-c2ccccc2F)s1 REAL300004040546
Cn1cc(-c2n[nH]cc2C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040547
CCn1cc(-c2n[nH]cc2C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040548
Cn1cc(-c2nn(C)cc2C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040549
CCn1cc(-c2nn(C)cc2C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040550
O=C(Cc1c[nH]c2cccc(Br)c12)NCc1ncc(C(=O)O)s1 REAL300004040551
CC(C(=O)NCc1ncc(C(=O)O)s1)c1cn(C)c2ccccc12 REAL300004040552
O=C(NCc1ncc(C(=O)O)s1)c1ccc(CN2CCCCC2)cc1 REAL300004040553
Cc1cccc(-c2nc(C(=O)NCc3ncc(C(=O)O)s3)c(C)[nH]2)c1 REAL300004040554
Cc1nc2ccccc2n1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040555
O=C(Cc1ccc2c(c1)OC(F)(F)O2)NCc1ncc(C(=O)O)s1 REAL300004040556
NS(=O)(=O)N1CCCC(C(=O)NCc2ncc(C(=O)O)s2)C1 REAL300004040557
O=C(Cc1c[nH]c2cc(Br)ccc12)NCc1ncc(C(=O)O)s1 REAL300004040558
CC(C)[C@@H](NS(=O)(=O)C1CC1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040559
CC(C(=O)NCc1ncc(C(=O)O)s1)C1OCCc2sccc21 REAL300004040560
Nc1nc(C(=O)NCc2ncc(C(=O)O)s2)nc(N2CCOCC2)n1 REAL300004040561
Cc1cn2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2n1 REAL300004040562
CNc1ccc(Cl)c(C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040563
Cn1cc(-c2ncccc2C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040564
O=C(NCc1ncc(C(=O)O)s1)c1cc(CN2CCCC2)on1 REAL300004040565
CN(C)CCc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040566
N#CC1(C(=O)NCc2ncc(C(=O)O)s2)CCSCC1 REAL300004040567
CC(C)(C)Cc1ccccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040568
O=C(O)c1cnc(CNC(=O)C2(c3ccc4c(c3)OCO4)CC2)s1 REAL300004040569
O=C(O)c1cnc(CNC(=O)[C@]23C[C@H]2COC32CCC2)s1 REAL300004040570
CC1(C(=O)NCc2ncc(C(=O)O)s2)CCC2(CC1)OCCO2 REAL300004040571
O=C(O)c1cnc(CNC(=O)c2coc3c2C(=O)CCC3)s1 REAL300004040572
CC(C)Cc1ccc(C=CC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040573
CS(=O)(=O)Nc1cccc(CC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040574
Cc1nc(CC(=O)NCc2ncc(C(=O)O)s2)c(C)s1 REAL300004040575
COc1ccc(-c2ocnc2C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040576
CNc1nc(C)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040577
O=C(O)c1cnc(CNC(=O)C2CN(Cc3ccccc3)CCO2)s1 REAL300004040578
O=C(O)c1cnc(CNC(=O)c2ccnn2-c2ccccc2)s1 REAL300004040579
COc1cc(CC(=O)NCc2ncc(C(=O)O)s2)cc(OC)c1O REAL300004040580
O=C(O)c1cnc(CNC(=O)C2(C(F)(F)F)CCC2)s1 REAL300004040581
COCCS(=O)(=O)CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040582
COc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1OCCO REAL300004040583
CN(CC(=O)NCc1ncc(C(=O)O)s1)c1ncnc2nc[nH]c12 REAL300004040584
O=C(CCCc1ccccn1)NCc1ncc(C(=O)O)s1 REAL300004040585
CCc1ccccc1OC(C(=O)NCc1ncc(C(=O)O)s1)c1ccccc1 REAL300004040586
Cc1cccc(COc2cccc(CC(=O)NCc3ncc(C(=O)O)s3)c2)c1 REAL300004040587
CC(C)Nc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040588
O=C(NCc1ncc(C(=O)O)s1)c1ccc(N2CCCC2)c(F)c1 REAL300004040589
O=C(NCc1ncc(C(=O)O)s1)c1ccc(N2CCOCC2)c(F)c1 REAL300004040590
O=C(O)c1cnc(CNC(=O)c2cc(F)ccc2N2CCOCC2)s1 REAL300004040591
CC(C(=O)NCc1ncc(C(=O)O)s1)N1CCC(Cc2ccccc2)CC1 REAL300004040592
COc1cccc(C(O)C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040593
O=C(O)c1cnc(CNC(=O)C2(Cc3ccc(F)cc3)CC2)s1 REAL300004040594
O=C(O)c1cnc(CNC(=O)C2(CO)CCOCC2)s1 REAL300004040595
CC(C)c1ncsc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040596
COCc1ncsc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040597
CC(C)(C(=O)NCc1ncc(C(=O)O)s1)C1CCCCC1 REAL300004040598
COCC1(C(=O)NCc2ncc(C(=O)O)s2)CCOCC1 REAL300004040599
O=C(NCc1ncc(C(=O)O)s1)c1ccc2[nH]nnc2n1 REAL300004040600
O=C(CCCc1ccccc1Cl)NCc1ncc(C(=O)O)s1 REAL300004040601
CC(C)(C)n1cc(C(=O)NCc2ncc(C(=O)O)s2)nn1 REAL300004040602
Cc1cc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cn2c1 REAL300004040603
O=C(O)c1cnc(CNC(=O)c2ccccc2-c2cn[nH]c2)s1 REAL300004040604
O=C(O)c1cnc(CNC(=O)c2ccccc2OC2CC2)s1 REAL300004040605
O=C(NCc1ncc(C(=O)O)s1)c1ccnc(OC(F)F)c1 REAL300004040606
O=C(O)c1cnc(CNC(=O)c2nc3cccnc3s2)s1 REAL300004040607
O=C(NCc1ncc(C(=O)O)s1)c1cnn(CC(F)(F)F)c1 REAL300004040608
O=C(O)c1cnc(CNC(=O)c2cnn3ccncc23)s1 REAL300004040609
O=C(NCc1ncc(C(=O)O)s1)c1cnc2[nH]nnc2c1 REAL300004040610
O=C(O)c1cnc(CNC(=O)c2cnn3ncccc23)s1 REAL300004040611
Cn1cc(C(=O)NCc2ncc(C(=O)O)s2)c2cc(F)ccc21 REAL300004040612
COc1ccc2c(c1)C(C(=O)NCc1ncc(C(=O)O)s1)CC2 REAL300004040613
Cn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C(F)F)n1 REAL300004040614
O=C(NCc1ncc(C(=O)O)s1)c1csc(C2CCCCC2)n1 REAL300004040615
Cc1nc(C2CCCCC2)sc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040616
COc1ccc2onc(CC(=O)NCc3ncc(C(=O)O)s3)c2c1 REAL300004040617
CN(C)S(=O)(=O)c1ccc(CC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040618
O=C(CCc1ccccc1N1CCOCC1)NCc1ncc(C(=O)O)s1 REAL300004040619
O=C(CC(O)c1ccc(Cl)cc1)NCc1ncc(C(=O)O)s1 REAL300004040620
CC1(C)CC(C(=O)NCc2ncc(C(=O)O)s2)c2ccccc2O1 REAL300004040621
COc1cccc(CC2(C(=O)NCc3ncc(C(=O)O)s3)CCCCC2)c1 REAL300004040622
O=C(O)c1cnc(CNC(=O)C2(Cc3cccc(Cl)c3)CCCCC2)s1 REAL300004040623
COCCn1cc(C(=O)NCc2ncc(C(=O)O)s2)nn1 REAL300004040624
COc1cccc(-n2cc(C(=O)NCc3ncc(C(=O)O)s3)nn2)c1 REAL300004040625
CC(C(=O)NCc1ncc(C(=O)O)s1)c1ccc2ccccc2c1 REAL300004040626
CC(C)(C(=O)NCc1ncc(C(=O)O)s1)c1ccc2c(c1)OCO2 REAL300004040627
CC(O)(C(=O)NCc1ncc(C(=O)O)s1)c1ccc(Cl)cc1 REAL300004040628
CNc1ncnc2cc(C(=O)NCc3ncc(C(=O)O)s3)ccc12 REAL300004040629
O=C(O)c1cnc(CNC(=O)C2Cc3cc(Br)ccc3O2)s1 REAL300004040630
Cc1cc(F)ccc1-n1cc(O)c(C(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040631
O=C(NCc1ncc(C(=O)O)s1)c1ccc(NCc2ccsc2)cc1 REAL300004040632
CC(C(=O)NCc1ncc(C(=O)O)s1)N1CCSCC1 REAL300004040633
CC(C)Cc1ccc(CCCC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040634
O=C(NCc1ncc(C(=O)O)s1)c1ccc(NCC2CC2)nc1 REAL300004040635
O=C(O)c1cnc(CNC(=O)c2nn(-c3cccc(F)c3)cc2O)s1 REAL300004040636
CC(C)(C)Sc1cc(C(=O)NCc2ncc(C(=O)O)s2)ccn1 REAL300004040637
COc1ccc(COCCCC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040638
O=C(NCc1ncc(C(=O)O)s1)c1ccnc(-c2ncc[nH]2)c1 REAL300004040639
CN(CCc1ccccc1)CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040640
COCCOCCN(C)CCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040641
Cc1cn(C2CCOCC2)nc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040642
O=C(Cn1nnc2c1CCCC2)NCc1ncc(C(=O)O)s1 REAL300004040643
NS(=O)(=O)C1(C(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040644
CN1CCCC(O)(CC(=O)NCc2ncc(C(=O)O)s2)C1 REAL300004040645
O=C(O)c1cnc(CNC(=O)c2nccn3ccnc23)s1 REAL300004040646
COCCOCCc1nc(C(=O)NCc2ncc(C(=O)O)s2)c[nH]1 REAL300004040647
Cc1nc(C2CC2)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040648
O=C(O)c1cnc(CNC(=O)c2cccnc2N2CCOCC2)s1 REAL300004040649
NS(=O)(=O)N1CCC(C(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040650
O=C(CCNS(=O)(=O)c1cccnc1)NCc1ncc(C(=O)O)s1 REAL300004040651
CN(C)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040652
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1-c1ccccn1 REAL300004040653
CC(C)c1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1-c1ccccn1 REAL300004040654
O=C(CCCN1CCN(c2ccccc2)CC1)NCc1ncc(C(=O)O)s1 REAL300004040655
O=C(O)c1cnc(CNC(=O)C2CCCCN2Cc2ccncc2)s1 REAL300004040656
O=C(O)c1cnc(CNC(=O)C2CCCCN2Cc2cccnc2)s1 REAL300004040657
Cc1n[nH]c(C)c1C(C)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040658
CCCCCCN(C)CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040659
COc1cc(C)cnc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040660
CC(C)(C)c1cnc(CCC(=O)NCc2ncc(C(=O)O)s2)o1 REAL300004040661
CSc1ccccc1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040662
CCc1nn(C)c(CC)c1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040663
CCSc1ccc(CC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040664
O=C(O)c1cnc(CNC(=O)c2scnc2C(F)(F)F)s1 REAL300004040665
O=C(O)c1cnc(CNC(=O)c2cccc3cccc(O)c23)s1 REAL300004040666
O=C(O)c1cnc(CNC(=O)c2ncc3ccccc3c2O)s1 REAL300004040667
O=C(O)c1cnc(CNC(=O)c2cccnc2C2CC2)s1 REAL300004040668
Cc1cccc(Cl)c1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040669
O=C(O)c1cnc(CNC(=O)c2cnn3c2OCCC3)s1 REAL300004040670
O=C(NCc1ncc(C(=O)O)s1)c1ccn2cncc2c1 REAL300004040671
Cn1nc(C(=O)NCc2ncc(C(=O)O)s2)cc1OC(F)F REAL300004040672
CC(C)c1cccc(C(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040673
O=C(NCc1ncc(C(=O)O)s1)c1ccc(OC(F)F)cn1 REAL300004040674
CC(C)(C(=O)NCc1ncc(C(=O)O)s1)C1CCOCC1 REAL300004040675
CCc1ccccc1-n1cc(C(=O)NCc2ncc(C(=O)O)s2)nn1 REAL300004040676
Cc1cc(F)ccc1-n1cc(C(=O)NCc2ncc(C(=O)O)s2)nn1 REAL300004040677
O=C(Cc1coc2cc(F)ccc12)NCc1ncc(C(=O)O)s1 REAL300004040678
CN(C)S(=O)(=O)N(C)CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040679
O=C(NCc1ncc(C(=O)O)s1)c1cccc(NCc2ccccn2)c1 REAL300004040680
CC(C)S(=O)(=O)c1cccc(C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040681
Cc1nn(C)c(-n2cccn2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040682
Cc1ccccc1-c1nc(C)c(C(=O)NCc2ncc(C(=O)O)s2)s1 REAL300004040683
Cc1nc(-c2c(C)noc2C)sc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040684
O=C(NCc1ncc(C(=O)O)s1)c1ccnc(-c2ccc(Cl)cc2)n1 REAL300004040685
O=C(Cc1ccc(OCc2ccccn2)cc1)NCc1ncc(C(=O)O)s1 REAL300004040686
CC(Oc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1)c1ccccc1 REAL300004040687
Cc1cc(C(C)(C)C)ccc1OCCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040688
CN(CC(=O)NCc1ncc(C(=O)O)s1)C1CCSC1 REAL300004040689
CC(C)Cn1ccc2c(C(=O)NCc3ncc(C(=O)O)s3)cccc21 REAL300004040690
Cc1ccc(-c2c[nH]cc2C(=O)NCc2ncc(C(=O)O)s2)s1 REAL300004040691
O=C(NCc1ncc(C(=O)O)s1)c1ccn(-c2ccc(Cl)cc2Cl)n1 REAL300004040692
Cc1ccccc1-n1cc(C(=O)NCc2ncc(C(=O)O)s2)nn1 REAL300004040693
O=C(NCc1ncc(C(=O)O)s1)c1cccc(-c2c(F)cccc2F)c1 REAL300004040694
Cc1oc(C(C)C)nc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040695
CC(OCc1ccncc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040696
Cn1cncc1[C@@H]1C[C@H]1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040697
O=C(NCc1ncc(C(=O)O)s1)c1cnn(CC(O)CO)c1 REAL300004040698
CCc1ccc(CC(=O)NCc2ncc(C(=O)O)s2)nc1 REAL300004040699
Cn1nc(C(=O)NCc2ncc(C(=O)O)s2)c2c1CCCC2 REAL300004040700
CCON1CCC(CC(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040701
O=C(O)c1cnc(CNC(=O)[C@@H]2C[C@H]2c2cccnc2)s1 REAL300004040702
CN(C)c1cccnc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040703
CC(C)N1CCN(CCC(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040704
CC(C)N1CCN(CCCC(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040705
O=C(O)c1cnc(CNC(=O)C2CCCC3CCCN32)s1 REAL300004040706
Cc1cc(N(C)C)cc(C)c1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040707
CN(C)CCn1cc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040708
N#CC1(C(=O)NCc2ncc(C(=O)O)s2)CC12CCCC2 REAL300004040709
N#CC1(C(=O)NCc2ncc(C(=O)O)s2)CC2CCC1CC2 REAL300004040710
Cc1nc2c(cc1C(=O)NCc1ncc(C(=O)O)s1)c(C)nn2C REAL300004040711
Cc1ccnc2sc(C(=O)NCc3ncc(C(=O)O)s3)c(C)c12 REAL300004040712
CCCc1c(C(=O)NCc2ncc(C(=O)O)s2)cnn1C REAL300004040713
Cn1ncc(C(=O)NCc2ncc(C(=O)O)s2)c1C(F)(F)F REAL300004040714
Cc1cccc(N2CCN(CCC(=O)NCc3ncc(C(=O)O)s3)CC2)c1 REAL300004040715
O=C(CNc1cccc(Cl)c1)NCc1ncc(C(=O)O)s1 REAL300004040716
O=C(CCN1CCN(c2ccccc2)CC1)NCc1ncc(C(=O)O)s1 REAL300004040717
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2ccncc2)s1 REAL300004040718
O=C(NCc1ncc(C(=O)O)s1)c1cc(-c2cccc(F)c2)no1 REAL300004040719
O=C(O)c1cnc(CNC(=O)C2CCCN(Cc3cccnc3)C2)s1 REAL300004040720
CC(=O)c1ccc(CC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040721
Cn1cc(S(=O)(=O)NCC(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040722
Cn1cc(-c2cncc(C(=O)NCc3ncc(C(=O)O)s3)c2)cn1 REAL300004040723
O=C(CCc1nc2cccnc2[nH]1)NCc1ncc(C(=O)O)s1 REAL300004040724
CC(C(=O)NCc1ncc(C(=O)O)s1)N1CCc2ccccc2C1 REAL300004040725
O=C(O)c1cnc(CNC(=O)c2nccn3ccnc23)s1 REAL300004040726
CC(C(=O)NCc1ncc(C(=O)O)s1)N1CCN(c2ccc(F)cc2)CC1 REAL300004040727
Cc1nc(C)c(C(=O)NCc2ncc(C(=O)O)s2)nc1C REAL300004040728
Cc1ccc2nc(C(=O)NCc3ncc(C(=O)O)s3)ccc2c1 REAL300004040729
Cc1cncc(CCC(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040730
O=C(O)c1cnc(CNC(=O)c2nc3cnccc3s2)s1 REAL300004040731
O=C(O)c1cnc(CNC(=O)C2CCCC2c2ccccc2)s1 REAL300004040732
COc1ccc2occ(C(=O)NCc3ncc(C(=O)O)s3)c2c1 REAL300004040733
Cc1cnc(COCC(=O)NCc2ncc(C(=O)O)s2)o1 REAL300004040734
O=C(O)c1cnc(CNC(=O)c2ccnc3nn[nH]c23)s1 REAL300004040735
O=C(NCc1ncc(C(=O)O)s1)c1cc2n(n1)CCCO2 REAL300004040736
CC1(C)COc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc21 REAL300004040737
O=C(O)c1cnc(CNC(=O)c2c[nH]cc2-c2ccc(F)cc2)s1 REAL300004040738
O=C(O)c1cnc(CNC(=O)C2CC23CCOc2ccccc23)s1 REAL300004040739
Cc1cc(Br)cc(C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040740
COC(Cc1ccccc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040741
O=C(O)c1cnc(CNC(=O)C(c2ccccc2F)N2CCOCC2)s1 REAL300004040742
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2cccc(OC(F)F)c2)s1 REAL300004040743
CCC(CC)C(C(=O)NCc1ncc(C(=O)O)s1)N1CCOCC1 REAL300004040744
O=C(NCc1ncc(C(=O)O)s1)c1ccc(-c2nc(C3CC3)n[nH]2)cc1 REAL300004040745
O=C(NCc1ncc(C(=O)O)s1)c1ccc(N2CCCc3ccccc32)cc1 REAL300004040746
O=C(NCc1ncc(C(=O)O)s1)c1ccc(-c2cccc3cccnc23)cc1 REAL300004040747
CN(C)c1ccc(-c2cncc(C(=O)NCc3ncc(C(=O)O)s3)c2)cc1 REAL300004040748
O=C(NCc1ncc(C(=O)O)s1)c1ccn2cc(C(F)(F)F)nc2c1 REAL300004040749
O=C(NCc1ncc(C(=O)O)s1)c1ccc2nc(C(F)(F)F)cn2c1 REAL300004040750
O=C(O)c1cnc(CNC(=O)c2cnn3cc(Br)cnc23)s1 REAL300004040751
O=C(NCc1ncc(C(=O)O)s1)c1cc(-c2ccc3c(c2)CCO3)no1 REAL300004040752
O=C(CC1CCN(Cc2ccccc2)C1)NCc1ncc(C(=O)O)s1 REAL300004040753
O=C(O)c1cnc(CNC(=O)c2cccc3scnc23)s1 REAL300004040754
COCCn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C)n1 REAL300004040755
O=C(NCc1ncc(C(=O)O)s1)c1cnc(OCc2ccccc2)cn1 REAL300004040756
O=C(O)c1cnc(CNC(=O)C2CC3CSCC(C2)C3=O)s1 REAL300004040757
O=C(O)c1cnc(CNC(=O)C2(c3ccccn3)CC2)s1 REAL300004040758
O=C(CS(=O)(=O)C1CC1)NCc1ncc(C(=O)O)s1 REAL300004040759
Cc1ccc(C(C)C(O)C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040760
CC(c1ccccc1)C(C)(O)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040761
O=C(NCc1ncc(C(=O)O)s1)c1ccn(Cc2ccccc2)n1 REAL300004040762
O=C(NCc1ncc(C(=O)O)s1)c1ccn(C2CCCCC2)n1 REAL300004040763
NS(=O)(=O)c1ccc(NCC(=O)NCc2ncc(C(=O)O)s2)c(F)c1 REAL300004040764
CN(C)c1cnc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040765
O=C(NCc1ncc(C(=O)O)s1)c1cnc(Oc2ccccc2)cn1 REAL300004040766
CC(C)Oc1cnc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040767
CN(C)CCn1ccc(C(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040768
CN(C)CCn1nccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040769
O=C(O)c1cnc(CNC(=O)c2c(C(F)(F)F)nc3n2CCCC3)s1 REAL300004040770
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)nnn1Cc1ccccc1 REAL300004040771
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2C2CCOCC2)s1 REAL300004040772
CCn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C2CCOCC2)n1 REAL300004040773
CC(C)(C)c1nc[nH]c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040774
CCc1nccn1C(C)CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040775
O=C(NCc1ncc(C(=O)O)s1)c1ccnc(NC2CCC2)c1 REAL300004040776
O=C(O)c1cnc(CNC(=O)c2cncc3nc[nH]c23)s1 REAL300004040777
O=C(O)c1cnc(CNC(=O)C2CCCn3cc(C(F)(F)F)nc32)s1 REAL300004040778
CN1CCCC1c1cc(C(=O)NCc2ncc(C(=O)O)s2)[nH]n1 REAL300004040779
O=C(Cc1ccc(-n2ccnc2)cc1)NCc1ncc(C(=O)O)s1 REAL300004040780
O=C(O)c1cnc(CNC(=O)c2cncc3nc(C(F)(F)F)[nH]c23)s1 REAL300004040781
CN1CCC(C(=O)NCc2ncc(C(=O)O)s2)c2ccccc21 REAL300004040782
CC(C)[C@H](NCC(F)(F)F)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040783
O=C(O)c1cnc(CNC(=O)c2nc(C(F)(F)F)n3c2CCCC3)s1 REAL300004040784
Cn1cc(C(=O)NCc2ncc(C(=O)O)s2)c(=O)[nH]c1=O REAL300004040785
Cc1oc(C)c(S(N)(=O)=O)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040786
O=C(O)c1cnc(CNC(=O)c2cc(C(F)(F)F)c[nH]c2=O)s1 REAL300004040787
CN(C)c1ncccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040788
CN(CCO)S(=O)(=O)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040789
O=C(Cc1nc2ncccn2n1)NCc1ncc(C(=O)O)s1 REAL300004040790
O=C(O)c1cnc(CNC(=O)C2CCCN(Cc3cccc(F)c3)C2)s1 REAL300004040791
O=C(O)c1cnc(CNC(=O)C2CCCN2Cc2ccccn2)s1 REAL300004040792
Cc1[nH]nc2ncc(C(=O)NCc3ncc(C(=O)O)s3)cc12 REAL300004040793
Cc1nn(C)c(C)c1-c1cc(C(=O)NCc2ncc(C(=O)O)s2)[nH]n1 REAL300004040794
O=C(O)c1cnc(CNC(=O)c2n[nH]c3c2CCCCC3)s1 REAL300004040795
CC(CN1CCOCC1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040796
O=C(CCN1CCN(c2ccccn2)CC1)NCc1ncc(C(=O)O)s1 REAL300004040797
CCN1CCc2nc3ccccc3c(C(=O)NCc3ncc(C(=O)O)s3)c2C1 REAL300004040798
O=C(NCc1ncc(C(=O)O)s1)c1ccc2cccnc2c1 REAL300004040799
O=C(NCc1ncc(C(=O)O)s1)c1cc2ncccn2n1 REAL300004040800
Cc1ccc2cc(C(=O)NCc3ncc(C(=O)O)s3)ccc2n1 REAL300004040801
COc1cc(Cl)cc(C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040802
O=C(O)c1cnc(CNC(=O)c2cccc3[nH]cnc23)s1 REAL300004040803
Cc1nc(-c2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)cs1 REAL300004040804
COc1cccc(-c2cc(C(=O)NCc3ncc(C(=O)O)s3)[nH]n2)c1 REAL300004040805
O=C(NCc1ncc(C(=O)O)s1)c1cccc(N2CCCC2)c1 REAL300004040806
O=C(Cc1ccc(F)cc1Br)NCc1ncc(C(=O)O)s1 REAL300004040807
O=C(Cc1coc2ccccc12)NCc1ncc(C(=O)O)s1 REAL300004040808
Cc1ncsc1CCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040809
CC(C)C(Oc1ccc(Cl)cc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040810
Cc1ccc2sc(C(=O)NCc3ncc(C(=O)O)s3)cc2c1 REAL300004040811
O=C(CCc1ccc(F)cc1F)NCc1ncc(C(=O)O)s1 REAL300004040812
O=C(NCc1ncc(C(=O)O)s1)c1cc(Cl)cc(Br)c1 REAL300004040813
Cc1cccc(C)c1NCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040814
O=C(NCc1ncc(C(=O)O)s1)c1ccc(OC2CCC2)cc1 REAL300004040815
O=C(O)c1cnc(CNC(=O)C2CCc3cn[nH]c3C2)s1 REAL300004040816
O=C(O)c1cnc(CNC(=O)c2cnc(NC3CC3)s2)s1 REAL300004040817
O=C(O)c1cnc(CNC(=O)C(c2cccc(F)c2)N2CCOCC2)s1 REAL300004040818
O=C(CCCOc1cccnc1)NCc1ncc(C(=O)O)s1 REAL300004040819
O=C(O)c1cnc(CNC(=O)c2cc(-c3ccccc3)ns2)s1 REAL300004040820
O=C(O)c1cnc(CNC(=O)C2CCSc3ccccc32)s1 REAL300004040821
Cc1ccc(F)c(-n2cc(O)c(C(=O)NCc3ncc(C(=O)O)s3)n2)c1 REAL300004040822
CCc1ccccc1-n1cc(O)c(C(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040823
C[C@H](Cc1ccccc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040824
C=CCC(C(=O)NCc1ncc(C(=O)O)s1)c1ccccc1 REAL300004040825
CC(O)(CC(=O)NCc1ncc(C(=O)O)s1)c1ccccc1 REAL300004040826
CC(C)(C)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)s1 REAL300004040827
O=C(Cc1nsc2ccccc12)NCc1ncc(C(=O)O)s1 REAL300004040828
CCC(O)(CC(=O)NCc1ncc(C(=O)O)s1)c1ccccc1 REAL300004040829
O=C(O)c1cnc(CNC(=O)C23CC4CC(CC(F)(C4)C2)C3)s1 REAL300004040830
CC(C)(C)C1CCC(=CC(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040831
O=C(O)c1cnc(CNC(=O)c2nn[nH]c2-c2ccccc2)s1 REAL300004040832
CC(C(=O)NCc1ncc(C(=O)O)s1)c1ccc2c(c1)OCO2 REAL300004040833
Cc1ccc(C(=O)NCc2ncc(C(=O)O)s2)c2c1CCC2 REAL300004040834
O=C(COc1cc(F)cc(F)c1)NCc1ncc(C(=O)O)s1 REAL300004040835
CN(C)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)nc1 REAL300004040836
COc1cc(CO)ccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040837
CC(=O)c1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1O REAL300004040838
CCSCc1ccccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040839
O=C(CCc1cccc2c1OCO2)NCc1ncc(C(=O)O)s1 REAL300004040840
CC1(C)CCCC(O)(C(=O)NCc2ncc(C(=O)O)s2)C1 REAL300004040841
O=C(NCc1ncc(C(=O)O)s1)c1ccn(CCn2cccn2)n1 REAL300004040842
O=C(O)c1cnc(CNC(=O)c2ccnn2CC(F)F)s1 REAL300004040843
Cc1cccc(=O)n1CC(C)(O)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040844
Cc1ccn(CC(C)(O)C(=O)NCc2ncc(C(=O)O)s2)c(=O)c1 REAL300004040845
O=C(O)c1cnc(CNC(=O)c2ncsc2Nc2ccccc2)s1 REAL300004040846
O=C(NCc1ncc(C(=O)O)s1)c1ccc(Cn2ccnn2)cc1 REAL300004040847
NS(=O)(=O)c1cc(C(=O)NCc2ncc(C(=O)O)s2)ccn1 REAL300004040848
O=C(Cc1n[nH]c2c1CCCC2)NCc1ncc(C(=O)O)s1 REAL300004040849
O=C(O)c1cnc(CNC(=O)C2CCCc3[nH]ncc32)s1 REAL300004040850
Cn1ccnc1CN1CCC(C(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040851
O=C(O)c1cnc(CNC(=O)C2CCN(C3CCCCC3)C2)s1 REAL300004040852
O=C(NCc1ncc(C(=O)O)s1)c1ccc(NCCn2ccnc2)cc1 REAL300004040853
O=C(CC(O)COCc1ccccc1)NCc1ncc(C(=O)O)s1 REAL300004040854
CS(=O)(=O)CCC(C(=O)NCc1ncc(C(=O)O)s1)c1ccccc1 REAL300004040855
O=C(O)c1cnc(CNC(=O)c2cccn2-c2c(Cl)cccc2Cl)s1 REAL300004040856
O=C(O)c1cnc(CNC(=O)C(O)C(O)(c2ccccc2)C(F)(F)F)s1 REAL300004040857
O=C(Cc1cncc2ccccc12)NCc1ncc(C(=O)O)s1 REAL300004040858
Cn1cnc2cncc(C(=O)NCc3ncc(C(=O)O)s3)c21 REAL300004040859
CSc1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C)o1 REAL300004040860
Cn1c(C(F)(F)F)nc2cncc(C(=O)NCc3ncc(C(=O)O)s3)c21 REAL300004040861
O=C(O)c1cnc(CNC(=O)C2CCCN2c2ncccn2)s1 REAL300004040862
O=C(NCc1ncc(C(=O)O)s1)c1ccc(Nn2ccnc2)cc1 REAL300004040863
Nc1nnnn1-c1cccc(C(=O)NCc2ncc(C(=O)O)s2)c1 REAL300004040864
O=C(O)c1cnc(CNC(=O)c2nccc3ccsc23)s1 REAL300004040865
O=C(O)c1cnc(CNC(=O)c2cnc3n2CCOC3)s1 REAL300004040866
O=C(Cc1cnn2c1CCCC2)NCc1ncc(C(=O)O)s1 REAL300004040867
O=C(C=Cc1ccc2ccccc2n1)NCc1ncc(C(=O)O)s1 REAL300004040868
COc1ccc([C@]2(C(=O)NCc3ncc(C(=O)O)s3)C[C@H](O)C2)cc1 REAL300004040869
Cc1cn(C(C)(C)C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040870
O=C(O)c1cnc(CNC(=O)C23CCCN(CCC2)C3)s1 REAL300004040871
O=C(O)c1cnc(CNC(=O)c2cnc3n2CCCCC3)s1 REAL300004040872
CC(C)n1cc(C(=O)NCc2ncc(C(=O)O)s2)c(C2CCOCC2)n1 REAL300004040873
O=C(O)c1cnc(CNC(=O)c2cn(CCO)nc2C2CCOCC2)s1 REAL300004040874
O=C(O)c1cnc(CNC(=O)C2CCC3CCCCN32)s1 REAL300004040875
O=C(O)c1cnc(CNC(=O)c2cnn3c(-c4cccnc4)ccnc23)s1 REAL300004040876
O=C(NCc1ncc(C(=O)O)s1)c1cn([C@@H]2CC[C@H]2O)nn1 REAL300004040877
COc1cc(COCC(=O)NCc2ncc(C(=O)O)s2)ccn1 REAL300004040878
COc1ccc(COCC(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040879
O=C(COCc1cc[nH]c(=O)c1)NCc1ncc(C(=O)O)s1 REAL300004040880
CC1CCc2nc(C(=O)NCc3ncc(C(=O)O)s3)cn2C1 REAL300004040881
O=C(O)c1cnc(CNC(=O)c2ccccc2-c2ccncc2)s1 REAL300004040882
CC(C)(CN1CCOCC1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040883
O=C(O)c1cnc(CNC(=O)[C@]2(c3ccccc3)C[C@H](O)C2)s1 REAL300004040884
COc1cncc(C(=O)NCc2ncc(C(=O)O)s2)c1C REAL300004040885
O=C(Cc1cccc2cnccc12)NCc1ncc(C(=O)O)s1 REAL300004040886
O=C(NCc1ncc(C(=O)O)s1)c1cn2c(n1)COCC2 REAL300004040887
CC(C)N1CCC(C(=O)NCc2ncc(C(=O)O)s2)C(c2cnn(C)c2)C1 REAL300004040888
CN1CCC(C(=O)NCc2ncc(C(=O)O)s2)C(c2cnn(C)c2)C1 REAL300004040889
Cc1ccc(F)c2oc(C(=O)NCc3ncc(C(=O)O)s3)cc12 REAL300004040890
O=C(O)c1cnc(CNC(=O)[C@@H]2CC[C@H](C(F)(F)F)O2)s1 REAL300004040891
Cc1ccc2c(C(=O)NCc3ncc(C(=O)O)s3)cnn2c1C REAL300004040892
Cc1nc(-c2ccncc2)[nH]c(=O)c1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040893
CN1CCN(Cc2cccc(C(=O)NCc3ncc(C(=O)O)s3)c2)CC1 REAL300004040894
CN1CCN(Cc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc2)CC1 REAL300004040895
CCN(CC)CCOc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040896
Cc1nc2ccnn2c(C)c1CCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040897
O=C(CCSCc1ccccn1)NCc1ncc(C(=O)O)s1 REAL300004040898
O=C(NCc1ncc(C(=O)O)s1)c1ccnc(-n2ccnc2)c1 REAL300004040899
CC(C)(C)NS(=O)(=O)CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040900
O=C(O)c1cnc(CNC(=O)c2c[nH]c3ncccc23)s1 REAL300004040901
O=C(NCc1ncc(C(=O)O)s1)c1ccc(NC2CC2)nc1 REAL300004040902
CC(C)N1CCC(C(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040903
Cc1c(C(=O)NCc2ncc(C(=O)O)s2)nnn1Cc1ccc(F)cc1 REAL300004040904
O=C(NCc1ncc(C(=O)O)s1)c1cccc(-c2cnco2)c1 REAL300004040905
O=C(NCc1ncc(C(=O)O)s1)c1cc(O)cc(Br)c1 REAL300004040906
O=C(Cc1cc(Br)ccc1F)NCc1ncc(C(=O)O)s1 REAL300004040907
O=C(NCc1ncc(C(=O)O)s1)c1cccc(-n2ccnc2)c1 REAL300004040908
O=C(O)c1cnc(CNC(=O)c2ccncc2C(F)(F)F)s1 REAL300004040909
O=C(NCc1ncc(C(=O)O)s1)c1ccc(-c2c[nH]cn2)cc1 REAL300004040910
CC(C(=O)NCc1ncc(C(=O)O)s1)n1cnc2ccccc21 REAL300004040911
O=C(NCc1ncc(C(=O)O)s1)c1ccc(-c2ncn[nH]2)cc1 REAL300004040912
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2ccccc2F)s1 REAL300004040913
O=C(NCc1ncc(C(=O)O)s1)c1cncc(C(F)(F)F)c1 REAL300004040914
O=C(NCc1ncc(C(=O)O)s1)c1ccnc(C(F)(F)F)c1 REAL300004040915
O=C(NCc1ncc(C(=O)O)s1)c1cc2sccc2[nH]1 REAL300004040916
Cn1nc2ccccc2c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040917
O=C(NCc1ncc(C(=O)O)s1)c1cccc(Cn2ccnc2)c1 REAL300004040918
O=C(O)c1cnc(CNC(=O)c2cc(O)nc3ccc(F)cc23)s1 REAL300004040919
O=C(NCc1ncc(C(=O)O)s1)c1csc(N2CCCCC2)n1 REAL300004040920
O=C(O)c1cnc(CNC(=O)c2cccc3ccsc23)s1 REAL300004040921
O=C(NCc1ncc(C(=O)O)s1)c1cnc2ccc(F)cc2c1 REAL300004040922
Cc1nc2c(C(=O)NCc3ncc(C(=O)O)s3)cccc2[nH]1 REAL300004040923
O=C(NCc1ncc(C(=O)O)s1)c1ccn2nccc2n1 REAL300004040924
O=C(NCc1ncc(C(=O)O)s1)c1ccc2cnccc2c1 REAL300004040925
CN1CCc2cc(C(=O)NCc3ncc(C(=O)O)s3)ccc21 REAL300004040926
CCC(C)Oc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040927
O=C(O)c1cnc(CNC(=O)C(O)C2CCOCC2)s1 REAL300004040928
O=C(O)c1cnc(CNC(=O)C2CCCC3CCCCC32)s1 REAL300004040929
C=CCSc1ccccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040930
CS(=O)c1ccc(CC(=O)NCc2ncc(C(=O)O)s2)cc1 REAL300004040931
CCc1c(C(=O)NCc2ncc(C(=O)O)s2)oc2ccccc12 REAL300004040932
C#CCC1(C(=O)NCc2ncc(C(=O)O)s2)CCCCC1 REAL300004040933
CC(C)(C(=O)NCc1ncc(C(=O)O)s1)C1CCC(O)CC1 REAL300004040934
O=C(NCc1ncc(C(=O)O)s1)c1coc(C2CCCCC2)n1 REAL300004040935
CC(O)(CCc1ccccc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040936
CC(C)(C)c1ncc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040937
O=C(O)c1cnc(CNC(=O)c2ccccc2-n2ccnn2)s1 REAL300004040938
CCOc1cnc(C(=O)NCc2ncc(C(=O)O)s2)cn1 REAL300004040939
COCc1ncc(C(=O)NCc2ncc(C(=O)O)s2)s1 REAL300004040940
Cc1ccc(CCC(=O)NCc2ncc(C(=O)O)s2)s1 REAL300004040941
CC(C)(C)SCCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040942
COC1CCC(CC(=O)NCc2ncc(C(=O)O)s2)CC1 REAL300004040943
CS(=O)c1ccccc1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040944
O=C(NCc1ncc(C(=O)O)s1)c1cc(F)c(O)c(Cl)c1 REAL300004040945
Cc1nc(N)nc(C)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040946
O=C(O)c1cnc(CNC(=O)C2(O)CCSCC2)s1 REAL300004040947
CC(C)c1cc(C(=O)NCc2ncc(C(=O)O)s2)cc(O)n1 REAL300004040948
Cc1oc2ccccc2c1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040949
CC(C)Oc1ncccc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040950
Cc1cccc2c1OC(C(=O)NCc1ncc(C(=O)O)s1)C2 REAL300004040951
NS(=O)(=O)CCCCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040952
CC1(C(=O)NCc2ncc(C(=O)O)s2)CCc2ccccc2C1 REAL300004040953
CC(C)Oc1cc(C(=O)NCc2ncc(C(=O)O)s2)ccn1 REAL300004040954
CC(C)c1scnc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040955
COC1(C(=O)NCc2ncc(C(=O)O)s2)CCOCC1 REAL300004040956
O=C(O)c1cnc(CNC(=O)C2CCc3[nH]ncc3C2)s1 REAL300004040957
COc1c(C(=O)NCc2ncc(C(=O)O)s2)[nH]c(=O)[nH]c1=O REAL300004040958
O=C(O)c1cnc(CNC(=O)c2ccc(C3CC3)s2)s1 REAL300004040959
CCCc1cc(C(=O)NCc2ncc(C(=O)O)s2)ccc1Cl REAL300004040960
Cc1ccc(C(=O)NCc2ncc(C(=O)O)s2)c(Cl)c1C REAL300004040961
CC(C)(CC(=O)NCc1ncc(C(=O)O)s1)C1CCCCC1 REAL300004040962
O=C(NCc1ncc(C(=O)O)s1)c1cccc(C2CCC2)c1 REAL300004040963
CC1CCC(C)(C=CC(=O)NCc2ncc(C(=O)O)s2)C1(C)C REAL300004040964
O=C(O)c1cnc(CNC(=O)c2c[nH]c3cccnc23)s1 REAL300004040965
CCCc1nc(C)c(C(=O)NCc2ncc(C(=O)O)s2)o1 REAL300004040966
CC(Oc1ccccn1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040967
O=C(Cc1ccc2c(c1)COC2)NCc1ncc(C(=O)O)s1 REAL300004040968
O=C(O)c1cnc(CNC(=O)C2(Nc3ccccc3)CC2)s1 REAL300004040969
O=C(NCc1ncc(C(=O)O)s1)c1ccc(CO)c(F)c1 REAL300004040970
CCCCS(=O)(=O)NCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040971
Cn1nnc2ccc(C(=O)NCc3ncc(C(=O)O)s3)cc21 REAL300004040972
Cc1ccsc1CCCC(=O)NCc1ncc(C(=O)O)s1 REAL300004040973
CNc1ccc(C(=O)NCc2ncc(C(=O)O)s2)cc1F REAL300004040974
CC(OCc1ccc(F)cc1)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040975
CC(C)c1ccc2occ(C(=O)NCc3ncc(C(=O)O)s3)c2c1 REAL300004040976
Cc1nc(CC2CC2)oc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040977
CCOCc1nc(C)c(C(=O)NCc2ncc(C(=O)O)s2)s1 REAL300004040978
O=C(O)c1cnc(CNC(=O)C(O)Cc2cccc(C(F)(F)F)c2)s1 REAL300004040979
COc1cc(C(=O)NCc2ncc(C(=O)O)s2)sc1S(N)(=O)=O REAL300004040980
Cc1nc2ccccc2cc1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040981
O=C(O)c1cnc(CNC(=O)C2(Cc3ccc(F)cc3)CCOCC2)s1 REAL300004040982
O=C(O)c1cnc(CNC(=O)C2(Cc3cccc(F)c3)CCOCC2)s1 REAL300004040983
COCc1nc(C(=O)NCc2ncc(C(=O)O)s2)c(-c2ccccc2)s1 REAL300004040984
CC(C)(C)Oc1cccc(CCC(=O)NCc2ncc(C(=O)O)s2)n1 REAL300004040985
O=C(O)c1cnc(CNC(=O)C2CCCN2c2ccccc2)s1 REAL300004040986
Cc1nsc(NC2CC2)c1C(=O)NCc1ncc(C(=O)O)s1 REAL300004040987
CCn1ncc2cc(C(=O)NCc3ncc(C(=O)O)s3)c(C)nc21 REAL300004040988
O=C(O)c1cnc(CNC(=O)c2c[nH]nc2-c2ccccn2)s1 REAL300004040989
O=C(O)c1cnc(CNC(=O)c2ocnc2-c2ccccc2)s1 REAL300004040990
O=C(O)c1cnc(CNC(=O)C2CC(O)(c3cccc(Cl)c3)C2)s1 REAL300004040991
O=C(Cn1ccc(C(F)F)n1)NCc1ncc(C(=O)O)s1 REAL300004040992
CC(C(=O)NCc1ncc(C(=O)O)s1)n1nnnc1C(C)(C)C REAL300004040993
O=C(O)c1cnc(CNC(=O)c2nc3ccccc3s2)s1 REAL300004040994
O=C(Cc1nc(-c2ccc(F)cc2)cs1)NCc1ncc(C(=O)O)s1 REAL300004040995
O=C(Cn1cnc2ccccc21)NCc1ncc(C(=O)O)s1 REAL300004040996
CCc1nc2ccccc2n1CC(=O)NCc1ncc(C(=O)O)s1 REAL300004040997
CC(C)C(NS(C)(=O)=O)C(=O)NCc1ncc(C(=O)O)s1 REAL300004040998
CC(C(=O)NCc1ncc(C(=O)O)s1)N1CCc2ccccc21 REAL300004040999
Cn1ncc(C(=O)NCc2ncc(C(=O)O)s2)c1-n1cnnc1 REAL300004041000
