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Cc1ncc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15840058__15857566
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O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1[nH]ncc1Cl s275592__15865378__15840062__15862300
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CC1COc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15840068__15859360
Cc1ccc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15840070__15859360
Cc1ncsc1COCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840072__15859360
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Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc(Cl)n1 s275592__15865378__15839960__15859360
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CSc1ccc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15839964__15859360
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O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccc([N+](=O)[O-])c1 s275592__15865378__15839974__15862300
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CN1N=C(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC1=O s275592__15865378__15839984__15862300
CN1N=C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1=O s275592__15865378__15839984__15859360
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O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1Cc2ccccc2S1 s275592__15865378__15839988__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc2cn[nH]c2c1 s275592__15865378__15839990__15862300
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Cc1noc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15839992__15862300
Cc1noc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15839992__15859360
Cc1noc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15839992__15857566
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccc1[N+](=O)[O-] s275592__15865378__15839994__15859360
COC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15841822__15862300
COC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841822__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2CC2C1 s275592__15865378__15841824__15862300
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Cc1cc([N+](=O)[O-])cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841832__15859360
O=C(Cc1cncnc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841834__15862300
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O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2[nH]nnc2cc1F s275592__15865378__15841846__15859360
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O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(Cl)[nH]c1=O s275592__15865378__15841850__15862300
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CCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc(Cl)n1 s275592__15865378__15841852__15859360
CCCCC(ON=C(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841854__15859360
CN1CCC(=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15841856__15862300
CN1CCC(=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841856__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C(F)F)CCCCC2)C1 s275592__15865378__15841858__15859360
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NC(=O)CCNC(=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841864__15862300
NC(=O)CCNC(=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841864__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC12CCC(F)(F)CC2 s275592__15865378__15841866__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2ccnn2c1O s275592__15865378__15841870__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1C(F)(F)F s275592__15865378__15841872__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1C(F)(F)F s275592__15865378__15841872__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)sn1 s275592__15865378__15841874__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)sn1 s275592__15865378__15841874__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)sn1 s275592__15865378__15841874__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc2sccc12 s275592__15865378__15841876__15859360
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Cc1cc(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)on1 s275592__15865378__15841880__15862300
Cc1cc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841880__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CCSC1 s275592__15865378__15841882__15862300
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O=C(CCCC(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841884__15862300
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O=C(CCCC(F)F)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841884__15857566
CCCCOCCNC(=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841886__15859360
O=C(Cc1ncc(Cl)s1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841890__15859360
CC1(C)CN(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15841894__15862300
CC1(C)CN(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841894__15859360
CC1(C)CN(CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15841894__15857566
Cn1cnnc1SCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841896__15862300
Cn1cnnc1SCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841896__15859360
CS(=O)(=O)NCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841898__15859360
Cc1ccc(Cl)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15841900__15862300
Cc1ccc(Cl)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841900__15859360
O=C(CCn1cccnc1=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841902__15862300
O=C(CCn1cccnc1=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841902__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(C(F)(F)F)[nH]1 s275592__15865378__15841906__15859360
O=C(CCCCN1CCCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841908__15859360
CCn1cc([N+](=O)[O-])c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841912__15859360
CSc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(O)n1 s275592__15865378__15841914__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(F)cc([N+](=O)[O-])c1 s275592__15865378__15841916__15859360
O=C(C=CC1CCCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841918__15862300
O=C(C=CC1CCCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841918__15859360
CC(O)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(F)c1 s275592__15865378__15841920__15859360
CCCC(O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841922__15862300
CCCC(O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841922__15859360
CCCC(O)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841922__15857566
Cn1ncc([N+](=O)[O-])c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841926__15862300
Cn1ncc([N+](=O)[O-])c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841926__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CSc2ccccc21 s275592__15865378__15841928__15859360
CC(O)(Cc1ccccc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841930__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(Cl)CC2)C1 s275592__15865378__15841932__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(Cl)CC2)C1 s275592__15865378__15841932__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(Cl)CC2)C1 s275592__15865378__15841932__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CCCO1 s275592__15865378__15841934__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CCCO1 s275592__15865378__15841934__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1=CCCO1 s275592__15865378__15841934__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(O)Cc3ccccc3C2)C1 s275592__15865378__15841936__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(CO)o1 s275592__15865378__15841940__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(CO)o1 s275592__15865378__15841940__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1ccc(CO)o1 s275592__15865378__15841940__15857566
CCCCCC(O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841944__15862300
CCCCCC(O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841944__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nnn2ccccc12 s275592__15865378__15843688__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nnn2ccccc12 s275592__15865378__15843688__15859360
CS(=O)(=O)c1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15843690__15859360
CN1CCOC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1=O s275592__15865378__15843692__15862300
CN1CCOC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15843692__15859360
CN1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1=O s275592__15865378__15843696__15862300
CN1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15843696__15859360
O=C(C=Cc1c(F)cccc1F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843698__15859360
O=C(C=CCOC1CCOCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843700__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccc(C(F)F)n1 s275592__15865378__15843702__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(C(F)F)n1 s275592__15865378__15843702__15859360
O=C(C=Cc1ccsc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843704__15862300
O=C(C=Cc1ccsc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843704__15859360
O=C(C=Cc1ccncn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843706__15862300
O=C(C=Cc1ccncn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843706__15859360
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)F s275592__15865378__15843708__15862300
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)F s275592__15865378__15843708__15859360
CC(=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)F s275592__15865378__15843708__15857566
CN1[C@H](C(N)=O)CC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843710__15862300
CN1[C@H](C(N)=O)CC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843710__15859360
Cc1cc(F)ncc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843714__15862300
Cc1cc(F)ncc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843714__15859360
Cc1sc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nc1O s275592__15865378__15843716__15862300
Cc1sc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc1O s275592__15865378__15843716__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC2(CC2)C1 s275592__15865378__15843720__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC2(CC2)C1 s275592__15865378__15843720__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC2(CC2)C1 s275592__15865378__15843720__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1n[nH]c2c1CCSC2 s275592__15865378__15843722__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2(CSC2)C1 s275592__15865378__15843724__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(CSC2)C1 s275592__15865378__15843724__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc2cc(O)ncc12 s275592__15865378__15843726__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc2ccnn2c1 s275592__15865378__15843728__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2ccnn2c1 s275592__15865378__15843728__15859360
CC1(O)CCN(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15843730__15862300
CC1(O)CCN(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15843730__15859360
O=C(C=Cc1ccc(F)cc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843736__15862300
O=C(C=Cc1ccc(F)cc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843736__15859360
CC(C)OC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15843738__15862300
CC(C)OC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15843738__15859360
O=C(C=Cc1ccc(Cl)s1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843740__15859360
CC1(C)CC2(CC2C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15843742__15862300
CC1(C)CC2(CC2C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15843742__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn([C@@H]2CC[C@H]2O)nn1 s275592__15865378__15843744__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCn2ncnc21 s275592__15865378__15843748__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCn2ncnc21 s275592__15865378__15843748__15859360
CCc1cccc2[nH]c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15843752__15859360
Cc1ncc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)s1 s275592__15865378__15843754__15862300
Cc1ncc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15843754__15859360
CCSc1cnccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843756__15859360
COc1nsc(OC)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843758__15859360
O=C(Cc1cc(C2CC2)on1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843760__15862300
O=C(Cc1cc(C2CC2)on1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843760__15859360
CN(C)CC=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843762__15862300
CN(C)CC=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843762__15859360
CN(C)CC=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15843762__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nccc2ncncc12 s275592__15865378__15843766__15859360
CCn1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc1=O s275592__15865378__15843768__15862300
CCn1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15843768__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(O)cc(Cl)n1 s275592__15865378__15843770__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(O)cc(Cl)n1 s275592__15865378__15843770__15859360
CC(F)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15843774__15859360
Cc1csc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15843776__15862300
Cc1csc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15843776__15859360
CCC[C@H](O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843778__15862300
CCC[C@H](O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843778__15859360
CCC[C@H](O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15843778__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCn2cnnc21 s275592__15865378__15843780__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCn2cnnc21 s275592__15865378__15843780__15859360
C#CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC=CCC1 s275592__15865378__15843782__15862300
C#CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC=CCC1 s275592__15865378__15843782__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1csc2nccn12 s275592__15865378__15843784__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1csc2nccn12 s275592__15865378__15843784__15859360
CC(C)(C)n1nccc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843788__15862300
CC(C)(C)n1nccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843788__15859360
CC1(C)C2CCC(C2)C1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843790__15862300
CC1(C)C2CCC(C2)C1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843790__15859360
CC1(C)C2CCC1(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)CC2 s275592__15865378__15843794__15862300
CC1(C)C2CCC1(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15843794__15859360
C#CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15843796__15862300
C#CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15843796__15859360
C#CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15843796__15857566
Cn1ncc2ncc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc21 s275592__15865378__15843798__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(C3CCOCC3)CC2)C1 s275592__15865378__15843800__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C3CCOCC3)CC2)C1 s275592__15865378__15843800__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(F)cc2cc[nH]c12 s275592__15865378__15843802__15859360
O=C(CC1COCCO1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843804__15862300
O=C(CC1COCCO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843804__15859360
CC(C)C1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)COC1 s275592__15865378__15843808__15862300
CC(C)C1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15843808__15859360
CC(C)C1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)COC1 s275592__15865378__15843808__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C(F)F)CC(F)(F)C2)C1 s275592__15865378__15843810__15859360
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(N=[N+]=[N-])c1 s275592__15865378__15845536__15859360
O=C(CC1CC2(CCC2)C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845538__15862300
O=C(CC1CC2(CCC2)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845538__15859360
CNC(=O)N[C@H](C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845540__15862300
CNC(=O)N[C@H](C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845540__15859360
COc1ncnc(C)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845544__15862300
COc1ncnc(C)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845544__15859360
CC(OCCN(C)C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845546__15862300
CC(OCCN(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845546__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn(O)c(=O)c1 s275592__15865378__15845548__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn(O)c(=O)c1 s275592__15865378__15845548__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc2sncc12 s275592__15865378__15845550__15859360
CC1(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15845552__15862300
CC1(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15845552__15859360
CC1(CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCO1 s275592__15865378__15845552__15857566
Cc1ncn(C)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845556__15862300
Cc1ncn(C)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845556__15859360
Cc1ncn(C)c1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845556__15857566
CC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)(CO1)C2 s275592__15865378__15845558__15862300
CC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(CO1)C2 s275592__15865378__15845558__15859360
CCn1c(C)nn(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15845560__15859360
O=C(C=Cc1c[nH]c(=O)[nH]c1=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845562__15859360
CC(CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)CC(F)(F)F s275592__15865378__15845564__15862300
CC(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)CC(F)(F)F s275592__15865378__15845564__15859360
O=C(Cc1nncs1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845568__15862300
O=C(Cc1nncs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845568__15859360
O=C(Cc1nncs1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845568__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C3CCC3)CC2(F)F)C1 s275592__15865378__15845570__15859360
CN(C)CCOCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845572__15862300
CN(C)CCOCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845572__15859360
COCCN(C)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845574__15862300
COCCN(C)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845574__15859360
CCC(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)CC(F)(F)F s275592__15865378__15845576__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(C3CC3)CCCO2)C1 s275592__15865378__15845580__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C3CC3)CCCO2)C1 s275592__15865378__15845580__15859360
Cc1ncc2ccccc2c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845584__15859360
Cn1cc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)ccc2n1 s275592__15865378__15845586__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCN(CCO)C(=O)C1 s275592__15865378__15845592__15859360
CCc1cscc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845596__15862300
CCc1cscc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845596__15859360
O=C(CC1CCCC(F)(F)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845604__15859360
Cc1n[nH]c2c1CC(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15845606__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnn1C1CC1(F)F s275592__15865378__15845608__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CC2CCC=CCCC12 s275592__15865378__15845610__15859360
CC1(C)OC2(CO)CC1(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15845612__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnn(C(F)(F)F)c1 s275592__15865378__15845614__15859360
C=C1CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)(C(F)F)C1 s275592__15865378__15845616__15862300
C=C1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)(C(F)F)C1 s275592__15865378__15845616__15859360
C#Cc1ccc(C2CC2C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15845618__15859360
CO[C@@H]1C[C@@]2(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)C[C@@H]12 s275592__15865378__15845622__15862300
CO[C@@H]1C[C@@]2(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)C[C@@H]12 s275592__15865378__15845622__15859360
CO[C@@H]1C[C@@]2(C(=O)NCC(F)=C3CN(C(=O)CSc4n[nH]c(=O)[nH]4)C3)C[C@@H]12 s275592__15865378__15845622__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc2cncnc2[nH]1 s275592__15865378__15845624__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2cncnc2[nH]1 s275592__15865378__15845624__15859360
Cc1ccc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15845626__15862300
Cc1ccc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15845626__15859360
CC1OC2(C)CC1(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)C2 s275592__15865378__15845628__15862300
CC1OC2(C)CC1(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15845628__15859360
Cn1cnnc1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845630__15862300
Cn1cnnc1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845630__15859360
Cn1cnnc1CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845630__15857566
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ncc1C(F)F s275592__15865378__15845632__15859360
CCc1nonc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845636__15862300
CCc1nonc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845636__15859360
CCc1nonc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845636__15857566
O=C(CC1(CO)CCOCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845640__15859360
O=C(Cc1cnsn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845642__15862300
O=C(Cc1cnsn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845642__15859360
O=C(Cc1cnsn1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845642__15857566
C=CCC(C)(C)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845644__15862300
C=CCC(C)(C)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845644__15859360
C=CCC(C)(C)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845644__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC(=O)N(C2CC2)C1 s275592__15865378__15845646__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(C#CC2CC2)cc1 s275592__15865378__15845648__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(C#CC2CC2)c1 s275592__15865378__15845650__15859360
COCCCCN(C)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845652__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC(c2ccccc2)O1 s275592__15865378__15845654__15859360
CC1C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)=Cc2ccccc21 s275592__15865378__15840084__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1OC1CC1 s275592__15865378__15840086__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2nccc2c1 s275592__15865378__15840088__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2nccc2c1 s275592__15865378__15840088__15859360
COc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc(C)n1 s275592__15865378__15840090__15862300
COc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc(C)n1 s275592__15865378__15840090__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(CO)c1ccc(F)cc1 s275592__15865378__15840092__15859360
CCSc1nccnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840094__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(C(F)(F)F)on1 s275592__15865378__15840096__15859360
CC(C)(C)c1nnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15840098__15859360
CCC(C)(OC)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840100__15862300
CCC(C)(OC)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840100__15859360
CCC(C)(OC)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840100__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(F)c(CO)c1 s275592__15865378__15840104__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(F)c(CO)c1 s275592__15865378__15840104__15859360
CCCC(CCCO)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840106__15862300
CCCC(CCCO)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840106__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1C[C@H]1c1cccc(F)c1 s275592__15865378__15840108__15859360
CC(O)c1ncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)s1 s275592__15865378__15840110__15862300
CC(O)c1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15840110__15859360
O=C1CC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCN1 s275592__15865378__15840112__15862300
O=C1CC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCN1 s275592__15865378__15840112__15859360
CC(C)[C@H](O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840114__15862300
CC(C)[C@H](O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840114__15859360
CC(C)[C@H](O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840114__15857566
CSC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15840116__15862300
CSC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15840116__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccccn1 s275592__15865378__15840122__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15840122__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(O)c1ccccn1 s275592__15865378__15840124__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)c1ccccn1 s275592__15865378__15840124__15859360
CC(O)(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccccn1 s275592__15865378__15840126__15862300
CC(O)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15840126__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccc(=O)n1O s275592__15865378__15840128__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(=O)n1O s275592__15865378__15840128__15859360
O=C(CCCCCn1cnnn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840130__15859360
COc1cccnc1C(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840132__15859360
Cn1ccc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)ccc21 s275592__15865378__15840134__15859360
CN(C)C1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15840136__15862300
CN(C)C1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15840136__15859360
COc1ccnc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15840138__15862300
COc1ccnc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840138__15859360
CC(CS(C)=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840140__15862300
CC(CS(C)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840140__15859360
CC(CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15840142__15862300
CC(CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15840142__15859360
O=C(C=Cc1ccncc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840144__15862300
O=C(C=Cc1ccncc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840144__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cncc(F)n1 s275592__15865378__15840146__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc(F)n1 s275592__15865378__15840146__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cncc(F)n1 s275592__15865378__15840146__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnn(C2CC2)c1 s275592__15865378__15840148__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnn(C2CC2)c1 s275592__15865378__15840148__15859360
Cc1cccc(COCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840150__15859360
O=C(CCc1nnc(C2CC2)o1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840152__15859360
CC(C)C(CO)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840154__15862300
CC(C)C(CO)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840154__15859360
CC(C)C(CO)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840154__15857566
CCOC=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840158__15862300
CCOC=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840158__15859360
CCOC=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840158__15857566
CC1c2cn[nH]c2CCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840160__15859360
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccc2[nH]ncc12 s275592__15865378__15840162__15859360
CCN1CCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840164__15862300
CCN1CCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840164__15859360
CCN1CCC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840164__15857566
Cc1nc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cs1 s275592__15865378__15840168__15862300
Cc1nc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15840168__15859360
CSc1cc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)o1 s275592__15865378__15840170__15862300
CSc1cc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15840170__15859360
O=C(CO)NCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840174__15862300
O=C(CO)NCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840174__15859360
CCC(O)Cn1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15840176__15859360
CS(=O)(=O)SCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840182__15862300
CS(=O)(=O)SCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840182__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cn2cnnc2cn1 s275592__15865378__15840186__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn2cnnc2cn1 s275592__15865378__15840186__15859360
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccs1 s275592__15865378__15840188__15862300
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccs1 s275592__15865378__15840188__15859360
CC1=C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCS1(=O)=O s275592__15865378__15840190__15859360
O=C(C=CCCc1ccccc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840194__15859360
Cc1cc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(=O)o1 s275592__15865378__15840196__15862300
Cc1cc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(=O)o1 s275592__15865378__15840196__15859360
CC(C)N1CCCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15840198__15862300
CC(C)N1CCCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15840198__15859360
COc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15840202__15859360
Cc1ccc2c(c1)C(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)C2 s275592__15865378__15840204__15862300
Cc1ccc2c(c1)C(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15840204__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCc2scnc21 s275592__15865378__15840206__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1c[nH]nc1[N+](=O)[O-] s275592__15865378__15841946__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]nc1[N+](=O)[O-] s275592__15865378__15841946__15859360
CSCCCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841948__15862300
CSCCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841948__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nc(O)n1 s275592__15865378__15841950__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc(O)n1 s275592__15865378__15841950__15859360
O=C(CC1(O)CCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841954__15862300
O=C(CC1(O)CCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841954__15859360
O=C(CC1(O)CCCC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841954__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCC1O s275592__15865378__15841956__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCC1O s275592__15865378__15841956__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCCC1O s275592__15865378__15841956__15857566
O=C(CC1(O)CCCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841958__15862300
O=C(CC1(O)CCCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841958__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(F)cnc1Cl s275592__15865378__15841960__15859360
CC(C)c1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15841962__15862300
CC(C)c1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841962__15859360
CCc1nc(C)ncc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841966__15862300
CCc1nc(C)ncc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841966__15859360
Cc1[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(C)c1C s275592__15865378__15841968__15862300
Cc1[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)c1C s275592__15865378__15841968__15859360
O=C(CN1CCCC1CO)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841970__15862300
O=C(CN1CCCC1CO)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841970__15859360
C[C@@H](O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841972__15862300
C[C@@H](O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841972__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc2ccccn2n1 s275592__15865378__15841974__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2ccccn2n1 s275592__15865378__15841974__15859360
CCCCSCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841976__15862300
CCCCSCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841976__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(OC(F)F)cn1 s275592__15865378__15841982__15859360
Cc1nn(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841984__15859360
Cc1c([N+](=O)[O-])c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841986__15859360
CCc1cnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)s1 s275592__15865378__15841992__15862300
CCc1cnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841992__15859360
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c([N+](=O)[O-])c1 s275592__15865378__15841996__15859360
CC(C)c1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc(O)n1 s275592__15865378__15841998__15859360
CSSCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842002__15862300
CSSCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842002__15859360
CSSCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842002__15857566
NC(=O)C(O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842006__15862300
NC(=O)C(O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842006__15859360
NC(=O)C(O)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842006__15857566
CCC(C)=C(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842008__15862300
CCC(C)=C(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842008__15859360
CCC(C)=C(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842008__15857566
CSC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15842010__15862300
CSC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15842010__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842012__15862300
COC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15842012__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842012__15857566
CSc1cccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15842014__15862300
CSc1cccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15842014__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1coc(Cl)n1 s275592__15865378__15842016__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1coc(Cl)n1 s275592__15865378__15842016__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2cccnc2c1 s275592__15865378__15842018__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnc(Cl)s1 s275592__15865378__15842020__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc(Cl)s1 s275592__15865378__15842020__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2(CCCCC2)C1 s275592__15865378__15842022__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(CCCCC2)C1 s275592__15865378__15842022__15859360
CC(C)(O)CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842026__15862300
CC(C)(O)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842026__15859360
CC(C)(O)CCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842026__15857566
COCCC(C)(C)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842028__15862300
COCCC(C)(C)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842028__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCC2(CCC2)CC1 s275592__15865378__15842030__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC2(CCC2)CC1 s275592__15865378__15842030__15859360
CC(C)(C)C(CO)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842032__15862300
CC(C)(C)C(CO)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842032__15859360
CS(=O)c1cccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15842036__15859360
Cc1nc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15842038__15862300
Cc1nc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15842038__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccnc2[nH]ccc12 s275592__15865378__15842040__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc2[nH]ccc12 s275592__15865378__15842040__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2CCCCN2C1 s275592__15865378__15842044__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2CCCCN2C1 s275592__15865378__15842044__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H](O)c1ccccc1 s275592__15865378__15842046__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H](O)c1ccccc1 s275592__15865378__15842046__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(O)ccn1 s275592__15865378__15842048__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(O)ccn1 s275592__15865378__15842048__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cc(O)ccn1 s275592__15865378__15842048__15857566
CC1CC(=O)NC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842050__15862300
CC1CC(=O)NC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842050__15859360
CC1CC(=O)NC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842050__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnsc1 s275592__15865378__15842058__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnsc1 s275592__15865378__15842058__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cnsc1 s275592__15865378__15842058__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cncc(Cl)n1 s275592__15865378__15842060__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc(Cl)n1 s275592__15865378__15842060__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccnc1OCCO s275592__15865378__15842064__15859360
CN1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842066__15862300
CN1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842066__15859360
Cc1nccc(Cl)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842068__15862300
Cc1nccc(Cl)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842068__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(n3cccn3)CC2)C1 s275592__15865378__15843812__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(n3cccn3)CC2)C1 s275592__15865378__15843812__15859360
CC1(C)CCC=C(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15843814__15862300
CC1(C)CCC=C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15843814__15859360
CCc1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15843816__15862300
CCc1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15843816__15859360
CCc1nc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)c[nH]1 s275592__15865378__15843816__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cn2ccncc2n1 s275592__15865378__15843818__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn2ccncc2n1 s275592__15865378__15843818__15859360
CN(C)Cc1c[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15843822__15862300
CN(C)Cc1c[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15843822__15859360
NC(=O)c1cccc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15843824__15859360
CC(C)(C)C1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15843826__15862300
CC(C)(C)C1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15843826__15859360
CCc1nnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15843828__15862300
CCc1nnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15843828__15859360
CCc1nnc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]1 s275592__15865378__15843828__15857566
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C(F)(F)C(O)C2CC2)C1 s275592__15865378__15843830__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)C(O)C2CC2)C1 s275592__15865378__15843830__15859360
C#CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCCO1 s275592__15865378__15843832__15862300
C#CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCCO1 s275592__15865378__15843832__15859360
O=C(CC1(O)CCOC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843834__15862300
O=C(CC1(O)CCOC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843834__15859360
CCOc1ccc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15843836__15859360
CSC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15843840__15862300
CSC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15843840__15859360
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COc1cn(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15843894__15859360
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C=CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15843910__15859360
C=CCC(C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)N(C)C s275592__15865378__15843910__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@]2(F)C[C@H]2c2ccccc2)C1 s275592__15865378__15843914__15859360
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CC1(C)CCCCC1=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843920__15862300
CC1(C)CCCCC1=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843920__15859360
NS(=O)(=O)C1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15843922__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2ccsc2s1 s275592__15865378__15843926__15859360
O=C(C=CCO)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843928__15862300
O=C(C=CCO)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843928__15859360
O=C(C=CCO)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15843928__15857566
CCC(O)C(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843930__15862300
CCC(O)C(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843930__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCc2ncnn21 s275592__15865378__15843932__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCc2ncnn21 s275592__15865378__15843932__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(CO)CCCO2)C1 s275592__15865378__15843934__15862300
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CCSC1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15845664__15859360
CCC(C)CC(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845666__15862300
CCC(C)CC(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845666__15859360
CCC(C)CC(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845666__15857566
O=C(CC1CCCC2(CCC2)O1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845668__15859360
C#CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCOC1 s275592__15865378__15845670__15862300
C#CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCOC1 s275592__15865378__15845670__15859360
COc1cncc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15845672__15859360
CN1CC(C)(C)CC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845674__15862300
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Cc1c(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)oc2ccccc12 s275592__15865378__15845676__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)n1cccn1 s275592__15865378__15845678__15862300
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CN(C)CCCCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845684__15862300
CN(C)CCCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845684__15859360
COc1ccnc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15845686__15862300
COc1ccnc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15845686__15859360
CC1(C)CC(=O)N(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)O1 s275592__15865378__15845688__15862300
CC1(C)CC(=O)N(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)O1 s275592__15865378__15845688__15859360
CNC(=O)N1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15845690__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=NNC(C(F)(F)F)C1 s275592__15865378__15845692__15859360
O=C(Cc1cnco1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845696__15862300
O=C(Cc1cnco1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845696__15859360
O=C(Cc1cnco1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845696__15857566
O=C(CC12CCC(CC1)C2)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845698__15862300
O=C(CC12CCC(CC1)C2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845698__15859360
O=C(C[C@@H]1CC=CCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845700__15862300
O=C(C[C@@H]1CC=CCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845700__15859360
O=C(C[C@@H]1CC=CCC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845700__15857566
CC(=Cc1cccs1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845702__15862300
CC(=Cc1cccs1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845702__15859360
COCCOCC=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845706__15862300
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O=C(CN1CC2CC2C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845708__15862300
O=C(CN1CC2CC2C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845708__15859360
O=C(CN1CC2CC2C1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845708__15857566
CCCc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nnn1CC s275592__15865378__15845712__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)n1cccn1 s275592__15865378__15845714__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)n1cccn1 s275592__15865378__15845714__15859360
Cn1nc2c(c1C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)COCC2 s275592__15865378__15845716__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@H]2C[C@H](n3ccnn3)C2)C1 s275592__15865378__15845718__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@H]2C[C@H](n3ccnn3)C2)C1 s275592__15865378__15845718__15859360
CC(C)(C)[C@@H]1CCCC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845720__15859360
O=C(CC1CC2CC2C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845722__15862300
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O=C(CC1CC2CC2C1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845722__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(CF)on1 s275592__15865378__15845728__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(CF)on1 s275592__15865378__15845728__15859360
CC(F)(F)c1ccccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845730__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn(C2CCOC2)cn1 s275592__15865378__15845736__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc2cnnn2c1 s275592__15865378__15845738__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2cnnn2c1 s275592__15865378__15845738__15859360
CCCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nn1C s275592__15865378__15840210__15862300
CCCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15840210__15859360
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O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@H]1CCc2ccccc21 s275592__15865378__15840214__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@H]1CCc2ccccc21 s275592__15865378__15840214__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCC2CC2CC1 s275592__15865378__15840224__15862300
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O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccn2ncnc12 s275592__15865378__15840226__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccn2ncnc12 s275592__15865378__15840226__15859360
O=C(C=Cc1cccc(F)c1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840228__15862300
O=C(C=Cc1cccc(F)c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840228__15859360
[N-]=[N+]=NCc1ccccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840232__15859360
CSc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc1 s275592__15865378__15840236__15862300
CSc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15840236__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)n1C1CC1 s275592__15865378__15840244__15859360
Cc1n[nH]c(C)c1SCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840246__15859360
NC(=O)NCCCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840248__15859360
Cn1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)ccc1[N+](=O)[O-] s275592__15865378__15840250__15862300
Cn1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccc1[N+](=O)[O-] s275592__15865378__15840250__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15840252__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15840252__15859360
O=C(CNC(=O)C(F)(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840254__15862300
O=C(CNC(=O)C(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840254__15859360
NC1=NC(=O)C(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)S1 s275592__15865378__15840258__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=NN(CCO)C(=O)CC1 s275592__15865378__15840264__15859360
O=C(COCC(F)(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840270__15862300
O=C(COCC(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840270__15859360
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(Cl)n1 s275592__15865378__15840272__15862300
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15840272__15859360
NC(=O)CSCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840274__15862300
NC(=O)CSCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840274__15859360
CCCCSCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840276__15862300
CCCCSCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840276__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccc(F)n1 s275592__15865378__15840278__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(F)n1 s275592__15865378__15840278__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cccc(F)n1 s275592__15865378__15840278__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)c2ccc(F)cc2)C1 s275592__15865378__15840280__15859360
COC(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840284__15862300
COC(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840284__15859360
COC(C)(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840284__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nccnc1Cl s275592__15865378__15840286__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nccnc1Cl s275592__15865378__15840286__15859360
CC1CN2CCN1C(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)C2 s275592__15865378__15840288__15862300
CC1CN2CCN1C(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15840288__15859360
CCCC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15840292__15862300
CCCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15840292__15859360
O=C(C=CC1CCOCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840294__15862300
O=C(C=CC1CCOCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840294__15859360
CSc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15840298__15859360
Cn1cc([N+](=O)[O-])c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15840300__15862300
Cn1cc([N+](=O)[O-])c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15840300__15859360
Cc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15840302__15862300
Cc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15840302__15859360
Cc1cncc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15840302__15857566
CN(C)C(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840304__15862300
CN(C)C(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840304__15859360
CN(C)C(C)(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840304__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c(-c2ccccc2)c1 s275592__15865378__15840306__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C(F)(F)CO)C1 s275592__15865378__15840310__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)CO)C1 s275592__15865378__15840310__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C(F)(F)CO)C1 s275592__15865378__15840310__15857566
Cc1nc(O)ccc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840312__15862300
Cc1nc(O)ccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840312__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c2cccc(F)c12 s275592__15865378__15840316__15859360
Cn1cc(C(F)(F)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15840318__15859360
O=C(CCCCO)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840320__15862300
O=C(CCCCO)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840320__15859360
O=C(CCCCO)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840320__15857566
Cc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1Cl s275592__15865378__15840322__15862300
Cc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15840322__15859360
CCCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15840326__15862300
CCCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15840326__15859360
O=C(Cc1c(F)cncc1Cl)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840328__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnc(F)c(F)c1 s275592__15865378__15842070__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc(F)c(F)c1 s275592__15865378__15842070__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccnc(F)c1F s275592__15865378__15842072__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc(F)c1F s275592__15865378__15842072__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@H](O)c1ccccc1 s275592__15865378__15842074__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@H](O)c1ccccc1 s275592__15865378__15842074__15859360
COc1c(F)ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1F s275592__15865378__15842076__15859360
CC1(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842082__15862300
CC1(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15842082__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCOC2(CCC2)C1 s275592__15865378__15842088__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCOC2(CCC2)C1 s275592__15865378__15842088__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc([N+](=O)[O-])[nH]n1 s275592__15865378__15842090__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc([N+](=O)[O-])[nH]n1 s275592__15865378__15842090__15859360
O=C(Cn1cnc2ccccc21)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842096__15859360
Cc1oncc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842098__15862300
Cc1oncc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842098__15859360
Cc1oncc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842098__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=Cc2ccccc2OC1 s275592__15865378__15842100__15859360
Cc1n[nH]c(SCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15842102__15862300
Cc1n[nH]c(SCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15842102__15859360
CC1CCC(=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842104__15862300
CC1CCC(=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842104__15859360
CC(OC1CCCC1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842106__15862300
CC(OC1CCCC1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842106__15859360
CCc1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)csc1C s275592__15865378__15842112__15862300
CCc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)csc1C s275592__15865378__15842112__15859360
Cc1ccnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15842114__15862300
Cc1ccnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15842114__15859360
Cc1ccnc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842114__15857566
CC(OCc1ccccc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842116__15859360
O=C1CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CN1 s275592__15865378__15842120__15862300
O=C1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15842120__15859360
O=C1CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CN1 s275592__15865378__15842120__15857566
CC1CCCC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15842122__15862300
CC1CCCC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15842122__15859360
CC(Sc1ncccn1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842126__15859360
CC(SCC1CCCO1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842130__15859360
CCCCSC(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842132__15862300
CCCCSC(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842132__15859360
NS(=O)(=O)c1c[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15842134__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cn(CCO)nn1 s275592__15865378__15842140__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn(CCO)nn1 s275592__15865378__15842140__15859360
O=C(COC(F)(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842142__15862300
O=C(COC(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842142__15859360
O=C(COC(F)(F)F)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842142__15857566
Cc1ccc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c[nH]c2c1 s275592__15865378__15842144__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c2cc(F)ccc12 s275592__15865378__15842146__15859360
O=C1NC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)N1 s275592__15865378__15842148__15862300
O=C1NC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)N1 s275592__15865378__15842148__15859360
O=C1NC[C@@H](C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)N1 s275592__15865378__15842148__15857566
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1F s275592__15865378__15842150__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cncs1 s275592__15865378__15842152__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncs1 s275592__15865378__15842152__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cncs1 s275592__15865378__15842152__15857566
Cc1nn(CCO)cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842158__15862300
Cc1nn(CCO)cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842158__15859360
CN(C)c1nc(O)cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15842160__15859360
CN(C)c1ncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)o1 s275592__15865378__15842162__15862300
CN(C)c1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15842162__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842164__15862300
COC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15842164__15859360
CC1CCC(C2(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)CC2)CC1 s275592__15865378__15842166__15859360
O=C(C=CCN1CCOCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842168__15862300
O=C(C=CCN1CCOCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842168__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1noc2ccccc12 s275592__15865378__15842170__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1noc2ccccc12 s275592__15865378__15842170__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C(F)(F)CC2CC2)C1 s275592__15865378__15842172__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)CC2CC2)C1 s275592__15865378__15842172__15859360
O=C1CSC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)=N1 s275592__15865378__15842174__15862300
O=C1CSC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)=N1 s275592__15865378__15842174__15859360
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842176__15862300
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15842176__15859360
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]1 s275592__15865378__15842176__15857566
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(Br)CC2)C1 s275592__15865378__15842178__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(Br)CC2)C1 s275592__15865378__15842178__15859360
CN1CCCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842180__15862300
CN1CCCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842180__15859360
CN1CCCCC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842180__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccnnc1Cl s275592__15865378__15842182__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnnc1Cl s275592__15865378__15842182__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)c1cccc(Cl)c1 s275592__15865378__15842184__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(=O)[nH]n1 s275592__15865378__15842186__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(=O)[nH]n1 s275592__15865378__15842186__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc2ncccc2[nH]1 s275592__15865378__15842188__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2ncccc2[nH]1 s275592__15865378__15842188__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(CO)CC2)C1 s275592__15865378__15842190__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(CO)CC2)C1 s275592__15865378__15842190__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(CO)CC2)C1 s275592__15865378__15842190__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc(O)c2ncccc12 s275592__15865378__15843938__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1n[nH]c2nc[nH]c(=O)c12 s275592__15865378__15843940__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(F)cc(F)c1 s275592__15865378__15843946__15859360
CC(C)(OCC(F)(F)F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843950__15859360
COc1cccc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15843952__15862300
COc1cccc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15843952__15859360
C=CC1(C2(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)CCC2)CCC1 s275592__15865378__15843954__15859360
CC(C)(C)c1nnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15843960__15862300
CC(C)(C)c1nnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15843960__15859360
[N-]=[N+]=NCC(F)(F)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843962__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC(F)(F)C1 s275592__15865378__15843964__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC(F)(F)C1 s275592__15865378__15843964__15859360
CCc1c[nH]cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843966__15862300
CCc1c[nH]cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843966__15859360
CCc1c[nH]cc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15843966__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1CCC[C@H]1CF s275592__15865378__15843968__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CCC[C@H]1CF s275592__15865378__15843968__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(C2CCC2)on1 s275592__15865378__15843970__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(C2CCC2)on1 s275592__15865378__15843970__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CCC[C@H]1C(F)(F)F s275592__15865378__15843972__15859360
CC(C)[C@@H](O)[C@@H](C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843976__15862300
CC(C)[C@@H](O)[C@@H](C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843976__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(F)C3CCCCC32)C1 s275592__15865378__15843978__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(F)C3CCCCC32)C1 s275592__15865378__15843978__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1onc2ccccc12 s275592__15865378__15843980__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1onc2ccccc12 s275592__15865378__15843980__15859360
CC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)(CC1)CO2 s275592__15865378__15843982__15862300
CC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(CC1)CO2 s275592__15865378__15843982__15859360
CCc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(=O)[nH]1 s275592__15865378__15843984__15862300
CCc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15843984__15859360
O=C(Cn1cc(C2CCC2)nn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843986__15859360
COc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15843988__15862300
COc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15843988__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1C[C@H]2[C@@H](C1)C2(F)F s275592__15865378__15843990__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1C[C@H]2[C@@H](C1)C2(F)F s275592__15865378__15843990__15859360
CC1(C)CC(O)(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15843992__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c2ncnc(O)c12 s275592__15865378__15843994__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1CC[C@H]2C[C@@H]1CO2 s275592__15865378__15843996__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CC[C@H]2C[C@@H]1CO2 s275592__15865378__15843996__15859360
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c2n1CCCC2 s275592__15865378__15843998__15859360
COC1(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15844000__15862300
COC1(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15844000__15859360
COC1(CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15844000__15857566
Cc1cc2[nH]c(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)cc2o1 s275592__15865378__15844004__15862300
Cc1cc2[nH]c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc2o1 s275592__15865378__15844004__15859360
Cn1ncc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844006__15862300
Cn1ncc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844006__15859360
Cn1ncc(CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15844006__15857566
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(C3CCCCO3)CC2)C1 s275592__15865378__15844010__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C3CCCCO3)CC2)C1 s275592__15865378__15844010__15859360
O=C(Cn1ncc(=O)[nH]c1=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844012__15862300
O=C(Cn1ncc(=O)[nH]c1=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844012__15859360
O=C(CC1CC1(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844014__15862300
O=C(CC1CC1(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844014__15859360
O=C(CC1CC1(F)F)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844014__15857566
O=C(CC1C=CS(=O)(=O)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844016__15859360
COc1cnnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15844018__15862300
COc1cnnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844018__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(C2CC2)nc1O s275592__15865378__15844022__15859360
CC(Cn1ccnc1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844024__15862300
CC(Cn1ccnc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844024__15859360
O=C(CSCCC(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844026__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c(F)ccc2[nH]ncc12 s275592__15865378__15844028__15859360
CCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1CCO s275592__15865378__15844032__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(O)ncn1 s275592__15865378__15844034__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(O)ncn1 s275592__15865378__15844034__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cc(O)ncn1 s275592__15865378__15844034__15857566
CCCn1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844036__15862300
CCCn1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844036__15859360
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nc1F s275592__15865378__15844040__15862300
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc1F s275592__15865378__15844040__15859360
Cc1cccn2c(CC(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cnc12 s275592__15865378__15844044__15859360
COc1c(Cl)cccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844046__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(CO)cn1 s275592__15865378__15844048__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(CO)cn1 s275592__15865378__15844048__15859360
CN1CC=C(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15844050__15862300
CN1CC=C(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15844050__15859360
CC[C@H](C)[C@H](O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844052__15862300
CC[C@H](C)[C@H](O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844052__15859360
CC[C@H](C)[C@H](O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844052__15857566
Cc1ncn(C)c(=O)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844054__15862300
Cc1ncn(C)c(=O)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844054__15859360
COCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15844056__15862300
COCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15844056__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2ccccc2c1F s275592__15865378__15845740__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC(=C(F)F)CC1 s275592__15865378__15845742__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1Cc2nccnc2C1 s275592__15865378__15845748__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1Cc2nccnc2C1 s275592__15865378__15845748__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23CC=CC(C2)OC3)C1 s275592__15865378__15845750__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CC=CC(C2)OC3)C1 s275592__15865378__15845750__15859360
O=C(CCCC(F)(F)CO)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845756__15862300
O=C(CCCC(F)(F)CO)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845756__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C1CC1)C1CCCO1 s275592__15865378__15845758__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C1CC1)C1CCCO1 s275592__15865378__15845758__15859360
O=C(CC1(N2CCCC2)CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845760__15862300
O=C(CC1(N2CCCC2)CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845760__15859360
CC1CCC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1C s275592__15865378__15845764__15862300
CC1CCC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1C s275592__15865378__15845764__15859360
C#CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15845766__15862300
C#CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15845766__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2cccnc12 s275592__15865378__15845768__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2cccnc12 s275592__15865378__15845768__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n(C2CCC2)n1 s275592__15865378__15845770__15859360
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C(F)F)nn1C s275592__15865378__15845772__15859360
O=C(Cc1coc(C(F)F)n1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845776__15859360
CC(C)c1ccc(F)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15845778__15859360
CC(C)(C)C(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)F s275592__15865378__15845782__15859360
CC(C)(C)n1cc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15845786__15859360
CC(=O)NC(COC(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845788__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@@]23C[C@@H](O)[C@@H]2C3)C1 s275592__15865378__15845790__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@@]23C[C@@H](O)[C@@H]2C3)C1 s275592__15865378__15845790__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)[C@@]23C[C@@H](O)[C@@H]2C3)C1 s275592__15865378__15845790__15857566
COCc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15845792__15862300
COCc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15845792__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CCCCC2C3(F)F)C1 s275592__15865378__15845794__15859360
CCCOCCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845798__15862300
CCCOCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845798__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)C1(O)CCCC1 s275592__15865378__15845800__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)C1(O)CCCC1 s275592__15865378__15845800__15859360
COc1cccc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15845802__15859360
CC1(C)COCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845804__15862300
CC1(C)COCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845804__15859360
Cc1cc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc(C)n1 s275592__15865378__15845806__15859360
Cn1ccn2ncc(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)c12 s275592__15865378__15845808__15862300
Cn1ccn2ncc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c12 s275592__15865378__15845808__15859360
O=C(C=Cc1cnc[nH]c1=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845810__15862300
O=C(C=Cc1cnc[nH]c1=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845810__15859360
C=CC1(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15845812__15862300
C=CC1(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15845812__15859360
CC1OC2(CO)CC1(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)C2 s275592__15865378__15845816__15862300
CC1OC2(CO)CC1(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15845816__15859360
Cc1n[nH]c2cnc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15845818__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCC2C1C2(F)F s275592__15865378__15845820__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(=O)[nH]c1C s275592__15865378__15845822__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(=O)[nH]c1C s275592__15865378__15845822__15859360
CC1CC1c1nocc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845826__15862300
CC1CC1c1nocc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845826__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC=Cc2ccccc21 s275592__15865378__15845828__15859360
Cc1ccnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15845832__15862300
Cc1ccnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15845832__15859360
Cc1ccnc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15845832__15857566
CCCc1ncoc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845834__15862300
CCCc1ncoc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845834__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1COc2ccc(F)cc21 s275592__15865378__15845836__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCc2ccnn2C1 s275592__15865378__15845838__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCc2ccnn2C1 s275592__15865378__15845838__15859360
O=C(CCCCCF)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845840__15862300
O=C(CCCCCF)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845840__15859360
O=C(CCCCCF)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845840__15857566
CC1(C)CCCOC1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845842__15862300
CC1(C)CCCOC1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845842__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCCC12CCC2 s275592__15865378__15845844__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCCC12CCC2 s275592__15865378__15845844__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(-c2nc[nH]n2)nc1 s275592__15865378__15845846__15859360
Cc1cccn2ncc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c12 s275592__15865378__15845848__15859360
CC(C)(C)C1CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)=NO1 s275592__15865378__15845850__15862300
CC(C)(C)C1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)=NO1 s275592__15865378__15845850__15859360
CCC(C)(C)C(C)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845852__15862300
CCC(C)(C)C(C)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845852__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(F)CCCOC2)C1 s275592__15865378__15845854__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(F)CCCOC2)C1 s275592__15865378__15845854__15859360
O=C(C=CCOCC(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845856__15859360
C#CC[C@]1(O)C[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15845858__15862300
C#CC[C@]1(O)C[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15845858__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2(C1)CC2F s275592__15865378__15845860__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(C1)CC2F s275592__15865378__15845860__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC2(C1)CC2F s275592__15865378__15845860__15857566
COC(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840334__15862300
COC(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840334__15859360
COC(F)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840334__15857566
CC(C)(C)c1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15840338__15859360
O=C(COC1C#CCCCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840340__15859360
CCc1cnoc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840342__15862300
CCc1cnoc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840342__15859360
CCc1cnoc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840342__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CN(CC(F)F)C1 s275592__15865378__15840346__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CN(CC(F)F)C1 s275592__15865378__15840346__15859360
Cc1ccsc1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840352__15862300
Cc1ccsc1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840352__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)Cc2ccccc2)C1 s275592__15865378__15840354__15859360
Cc1cc(Cl)nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15840356__15862300
Cc1cc(Cl)nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840356__15859360
CCC(C)CCC(O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840358__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc2cc(F)ccc12 s275592__15865378__15840360__15859360
COc1cccc(C)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840364__15862300
COc1cccc(C)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840364__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cn(C2CC2)nn1 s275592__15865378__15840366__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn(C2CC2)nn1 s275592__15865378__15840366__15859360
O=C(COc1ccon1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840368__15862300
O=C(COc1ccon1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840368__15859360
O=C(COc1ccon1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840368__15857566
CN1CCCC(C(C)(C)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15840370__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1snc(O)c1Cl s275592__15865378__15840372__15859360
CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC(O)CC1 s275592__15865378__15840374__15862300
CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC(O)CC1 s275592__15865378__15840374__15859360
Cc1coc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1C s275592__15865378__15840376__15862300
Cc1coc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1C s275592__15865378__15840376__15859360
Cc1coc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)c1C s275592__15865378__15840376__15857566
Cc1csc(C(C)C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15840378__15862300
Cc1csc(C(C)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15840378__15859360
CN(C)Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)o1 s275592__15865378__15840380__15862300
CN(C)Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15840380__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1occc1C1CC1 s275592__15865378__15840384__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1occc1C1CC1 s275592__15865378__15840384__15859360
Cn1cnc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15840386__15859360
O=C(CC1CC1(Cl)Cl)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840390__15862300
O=C(CC1CC1(Cl)Cl)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840390__15859360
O=C(Cc1cnccn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840392__15862300
O=C(Cc1cnccn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840392__15859360
O=C(Cc1cnccn1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840392__15857566
CN(C)Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15840394__15859360
CC(C)c1nnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)s1 s275592__15865378__15840396__15862300
CC(C)c1nnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15840396__15859360
CSc1cccc(F)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840400__15859360
Cn1cc(C(O)C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cn1 s275592__15865378__15840402__15862300
Cn1cc(C(O)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15840402__15859360
CCC1OCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840406__15862300
CCC1OCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840406__15859360
CCC1OCCC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840406__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2CC1C1C2C1(F)F s275592__15865378__15840408__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23CCC2C3)C1 s275592__15865378__15840412__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CCC2C3)C1 s275592__15865378__15840412__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C23CCC2C3)C1 s275592__15865378__15840412__15857566
CCCC(C)=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840414__15862300
CCCC(C)=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840414__15859360
CCCC(C)=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840414__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(C#CCO)c1 s275592__15865378__15840416__15859360
Cc1cc(C)c(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15840418__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nc(C2CC2)cs1 s275592__15865378__15840420__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nc(C2CC2)cs1 s275592__15865378__15840420__15859360
C=C[C@H](C)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840422__15862300
C=C[C@H](C)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840422__15859360
C=C[C@H](C)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840422__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(C2CCC2)[nH]n1 s275592__15865378__15840424__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(C2CCC2)[nH]n1 s275592__15865378__15840424__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1noc2c(F)cccc12 s275592__15865378__15840426__15859360
CCc1nn(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15840428__15859360
CS(=O)(=O)C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840432__15862300
CS(=O)(=O)C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840432__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2nccc2n1 s275592__15865378__15840436__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2nccc2n1 s275592__15865378__15840436__15859360
O=C(C=CCN1CCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840438__15862300
O=C(C=CCN1CCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840438__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nocc1-c1ccccc1 s275592__15865378__15840440__15859360
Cn1cc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cn1 s275592__15865378__15840442__15862300
Cn1cc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15840442__15859360
O=C(C=CC1CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840446__15862300
O=C(C=CC1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840446__15859360
O=C(C=CC1CC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840446__15857566
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23CCC(CC2)O3)C1 s275592__15865378__15840448__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CCC(CC2)O3)C1 s275592__15865378__15840448__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C23CCC(CC2)O3)C1 s275592__15865378__15840448__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1c[nH]c2ncncc12 s275592__15865378__15840450__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c2ncncc12 s275592__15865378__15840450__15859360
CC(C)(C)c1cncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840452__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(CO)nc1 s275592__15865378__15842194__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(CO)nc1 s275592__15865378__15842194__15859360
CSc1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842198__15862300
CSc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15842198__15859360
CCC1=C(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15842200__15862300
CCC1=C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15842200__15859360
Cc1cnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842202__15862300
Cc1cnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15842202__15859360
CC=C(CC)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842206__15862300
CC=C(CC)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842206__15859360
CC=C(CC)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842206__15857566
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23CCCC2CCC3)C1 s275592__15865378__15842210__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CCCC2CCC3)C1 s275592__15865378__15842210__15859360
Cc1[nH]nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1F s275592__15865378__15842214__15862300
Cc1[nH]nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1F s275592__15865378__15842214__15859360
Cc1[nH]nc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)c1F s275592__15865378__15842214__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)C2=CCOCC2)C1 s275592__15865378__15842216__15859360
O=C(CC12CC(C1)C2)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842218__15862300
O=C(CC12CC(C1)C2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842218__15859360
O=C(CC12CC(C1)C2)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842218__15857566
CC1(Br)CC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842220__15859360
O=C(C=C1CCOc2ccccc21)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842222__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cncc(F)c1O s275592__15865378__15842224__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc(F)c1O s275592__15865378__15842224__15859360
Cc1cccn2nc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15842226__15859360
C#CCC(CC#C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842228__15862300
C#CCC(CC#C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842228__15859360
C#CCC(CC#C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842228__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)c2cnccn2)C1 s275592__15865378__15842230__15859360
CCC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)O s275592__15865378__15842232__15862300
CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)O s275592__15865378__15842232__15859360
CCC(C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)O s275592__15865378__15842232__15857566
CCC(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842234__15862300
CCC(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842234__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(c1)N=S=N2 s275592__15865378__15842238__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1C[C@H]1C(F)(F)F s275592__15865378__15842242__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1C[C@H]1C(F)(F)F s275592__15865378__15842242__15859360
CC1(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1(Cl)Cl s275592__15865378__15842244__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCN(C2CC2)CC1 s275592__15865378__15842246__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCN(C2CC2)CC1 s275592__15865378__15842246__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(CO)CCOCC2)C1 s275592__15865378__15842248__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(CO)CCOCC2)C1 s275592__15865378__15842248__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)S(N)(=O)=O s275592__15865378__15842250__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)S(N)(=O)=O s275592__15865378__15842250__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1C[C@H]1c1ccccc1 s275592__15865378__15842252__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1C[C@H]1c1ccccc1 s275592__15865378__15842252__15859360
CS(=O)(=O)N1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15842256__15859360
NS(=O)(=O)C1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842262__15862300
NS(=O)(=O)C1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842262__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1coc(CO)c1 s275592__15865378__15842264__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1coc(CO)c1 s275592__15865378__15842264__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1coc(CO)c1 s275592__15865378__15842264__15857566
CC(C)[C@H]1CC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842268__15862300
CC(C)[C@H]1CC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842268__15859360
Cn1nnc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15842270__15859360
Cc1onc(CO)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842272__15862300
Cc1onc(CO)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842272__15859360
COCn1nccc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842274__15862300
COCn1nccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842274__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1Cc2ccccc2C1 s275592__15865378__15842276__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1Cc2ccccc2C1 s275592__15865378__15842276__15859360
COc1nscc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842278__15862300
COc1nscc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842278__15859360
Cc1ccc2ncc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc2c1 s275592__15865378__15842280__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CC2(c2ccccc2)C3)C1 s275592__15865378__15842282__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1Cc2cccnc2C1 s275592__15865378__15842286__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1Cc2cccnc2C1 s275592__15865378__15842286__15859360
COc1cnc(F)cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842288__15862300
COc1cnc(F)cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842288__15859360
C=CC(C)(O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842290__15862300
C=CC(C)(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842290__15859360
C=CC(C)(O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842290__15857566
O=C(CCC1(O)CCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842292__15862300
O=C(CCC1(O)CCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842292__15859360
O=C(CCC1(O)CCC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842292__15857566
CCc1nnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)s1 s275592__15865378__15842294__15862300
CCc1nnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15842294__15859360
CC(C)(C)c1ccncc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842296__15859360
CCC(C)(CO)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842298__15862300
CCC(C)(CO)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842298__15859360
CCC(C)(CO)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842298__15857566
Cn1c(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc2ccccc21 s275592__15865378__15842302__15859360
CN(C)C1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842304__15862300
CN(C)C1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842304__15859360
CN(C)C1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842304__15857566
O=C(CS(=O)(=O)C1CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842308__15862300
O=C(CS(=O)(=O)C1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842308__15859360
O=C(CCN1CCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842312__15862300
O=C(CCN1CCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842312__15859360
O=C(CCN1CCCC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842312__15857566
CCCC(NC(C)=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842314__15862300
CCCC(NC(C)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842314__15859360
CCCn1cccc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842316__15862300
CCCn1cccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842316__15859360
CC(C)CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)COC1 s275592__15865378__15844060__15862300
CC(C)CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15844060__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CCO[C@H]1C(F)(F)F s275592__15865378__15844062__15859360
O=C(C=Cc1ccc(F)nc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844066__15862300
O=C(C=Cc1ccc(F)nc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844066__15859360
CC(C)CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15844068__15862300
CC(C)CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15844068__15859360
O=C(CCC(O)C(F)(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844070__15862300
O=C(CCC(O)C(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844070__15859360
O=C(CCc1n[nH]c2ccccc12)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844072__15859360
Cn1cnc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15844076__15862300
Cn1cnc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844076__15859360
Cc1cc(C2CC2)ncc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844078__15859360
O=C(Cc1n[nH]c(C2CC2)n1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844080__15862300
O=C(Cc1n[nH]c(C2CC2)n1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844080__15859360
CC1(C)CC1CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844082__15862300
CC1(C)CC1CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844082__15859360
CC1(C)CC1CCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844082__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1C[C@H]1C1CCCO1 s275592__15865378__15844084__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1C[C@H]1C1CCCO1 s275592__15865378__15844084__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCS1(=O)=O s275592__15865378__15844086__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCS1(=O)=O s275592__15865378__15844086__15859360
O=C(C=CC1CCCO1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844088__15862300
O=C(C=CC1CCCO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844088__15859360
O=C(C=CC1CCCO1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844088__15857566
O=C(C#CC1CCCCO1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844090__15862300
O=C(C#CC1CCCCO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844090__15859360
Cc1ccc2cccnc2c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844092__15859360
CCOCCOCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844094__15862300
CCOCCOCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844094__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1CCC[C@H]1C1CC1 s275592__15865378__15844096__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CCC[C@H]1C1CC1 s275592__15865378__15844096__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccnc1CO s275592__15865378__15844098__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccnc1CO s275592__15865378__15844098__15859360
CC1(C)CC2(CC(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)C2)C1 s275592__15865378__15844100__15862300
CC1(C)CC2(CC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)C2)C1 s275592__15865378__15844100__15859360
C=CCn1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cn1 s275592__15865378__15844104__15862300
C=CCn1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15844104__15859360
Cn1ccc(C(C)(C)C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844110__15862300
Cn1ccc(C(C)(C)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844110__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(n3ccnn3)CC2)C1 s275592__15865378__15844114__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(n3ccnn3)CC2)C1 s275592__15865378__15844114__15859360
CC12COC(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)(C1)C2 s275592__15865378__15844118__15862300
CC12COC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(C1)C2 s275592__15865378__15844118__15859360
CC12COC(C(=O)NCC(F)=C3CN(C(=O)CSc4n[nH]c(=O)[nH]4)C3)(C1)C2 s275592__15865378__15844118__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc2n(c1)CCOC2 s275592__15865378__15844122__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2n(c1)CCOC2 s275592__15865378__15844122__15859360
C#CC1(O)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15844130__15862300
C#CC1(O)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15844130__15859360
C#CC1(O)CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15844130__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c(F)ccc2[nH]cnc12 s275592__15865378__15844138__15859360
C[C@@H]1C[C@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC(C)(C)C1 s275592__15865378__15844142__15862300
C[C@@H]1C[C@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC(C)(C)C1 s275592__15865378__15844142__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]c1C s275592__15865378__15844144__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]c1C s275592__15865378__15844144__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]c1C s275592__15865378__15844144__15857566
Cc1cnc2ccccc2c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844146__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(C2CC2)n[nH]c1=O s275592__15865378__15844148__15859360
COCc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15844150__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCc2[nH]cnc21 s275592__15865378__15844152__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCc2[nH]cnc21 s275592__15865378__15844152__15859360
CC1(C)C(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1(C)C s275592__15865378__15844154__15862300
CC1(C)C(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15844154__15859360
NC(=O)c1cnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cn1 s275592__15865378__15844156__15862300
NC(=O)c1cnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15844156__15859360
Cc1oc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)[nH]c2c1C s275592__15865378__15844158__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C3(O)CCOCC3)CC2)C1 s275592__15865378__15844160__15859360
O=C(CC(O)C1CCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844166__15862300
O=C(CC(O)C1CCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844166__15859360
CC1(C)COCC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)O1 s275592__15865378__15844170__15859360
O=C(CCC1CC(F)(F)C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844172__15862300
O=C(CCC1CC(F)(F)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844172__15859360
O=C(C=Cc1cccc(Cl)c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844174__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c(F)ccc2ccoc12 s275592__15865378__15844176__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2CCCC21 s275592__15865378__15844178__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2CCCC21 s275592__15865378__15844178__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC2CCCC21 s275592__15865378__15844178__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CN2CCN1CC2 s275592__15865378__15845864__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CN2CCN1CC2 s275592__15865378__15845864__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCc2nncn21 s275592__15865378__15845866__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCc2nncn21 s275592__15865378__15845866__15859360
C=CCCC(CC(C)C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845868__15862300
C=CCCC(CC(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845868__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCC2(C1)CC2(F)F s275592__15865378__15845870__15859360
CCC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCOCC1 s275592__15865378__15845872__15862300
CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCOCC1 s275592__15865378__15845872__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23CC(CO2)C3)C1 s275592__15865378__15845874__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CC(CO2)C3)C1 s275592__15865378__15845874__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C23CC(CO2)C3)C1 s275592__15865378__15845874__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCc2ccnn21 s275592__15865378__15845876__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCc2ccnn21 s275592__15865378__15845876__15859360
O=C(CC1CCC(O)C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845878__15862300
O=C(CC1CCC(O)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845878__15859360
O=C(CC1CCC(O)C1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845878__15857566
C[C@@H](C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)(C)O s275592__15865378__15845880__15862300
C[C@@H](C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)(C)O s275592__15865378__15845880__15859360
C[C@@H](C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)(C)O s275592__15865378__15845880__15857566
CC(C)N(C)C(=O)CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845882__15862300
CC(C)N(C)C(=O)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845882__15859360
CN1c2ccccc2CC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845884__15859360
CN1CC2CC1(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)C2 s275592__15865378__15845886__15862300
CN1CC2CC1(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15845886__15859360
CN1CC2CC1(C(=O)NCC(F)=C1CN(C(=O)CSc3n[nH]c(=O)[nH]3)C1)C2 s275592__15865378__15845886__15857566
Cn1ncc(C(F)F)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845888__15859360
Cc1cc(=O)[nH]nc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845890__15862300
Cc1cc(=O)[nH]nc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845890__15859360
CC1(C)CCCC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)O1 s275592__15865378__15845898__15862300
CC1(C)CCCC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)O1 s275592__15865378__15845898__15859360
O=C(CC12CNC(=O)C(C1)C2)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845900__15862300
O=C(CC12CNC(=O)C(C1)C2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845900__15859360
Cc1cnccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845902__15862300
Cc1cnccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845902__15859360
COc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15845904__15859360
Cn1nncc1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845906__15862300
Cn1nncc1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845906__15859360
Cn1nncc1CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845906__15857566
Cc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nc1 s275592__15865378__15845908__15862300
Cc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15845908__15859360
Cc1nnc2n1CC(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)C2 s275592__15865378__15845910__15862300
Cc1nnc2n1CC(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15845910__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23COC(C2)C3)C1 s275592__15865378__15845912__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23COC(C2)C3)C1 s275592__15865378__15845912__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C23COC(C2)C3)C1 s275592__15865378__15845912__15857566
CC(O)C1CC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845914__15862300
CC(O)C1CC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845914__15859360
CC(O)C1CC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845914__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc[nH]c1C1CCCC1 s275592__15865378__15845916__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2ccnc(O)c2n1 s275592__15865378__15845920__15859360
CCCCn1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nn1 s275592__15865378__15845922__15862300
CCCCn1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15845922__15859360
O=C(CN1CC2CCC1C2)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845924__15862300
O=C(CN1CC2CCC1C2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845924__15859360
O=C1C[C@@H]2OCC[C@]2(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15845928__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccc(CF)c1 s275592__15865378__15845932__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(CF)c1 s275592__15865378__15845932__15859360
COCC(NC(C)=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845934__15862300
COCC(NC(C)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845934__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCc2[nH]c(O)nc2C1 s275592__15865378__15845936__15859360
CC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)(C1)OC2 s275592__15865378__15845938__15862300
CC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(C1)OC2 s275592__15865378__15845938__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc(-n2ccnc2)n1 s275592__15865378__15845940__15859360
CCC1(C)CCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)O1 s275592__15865378__15845942__15862300
CCC1(C)CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)O1 s275592__15865378__15845942__15859360
O=C(C#CC1(C(F)(F)F)CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845944__15859360
Cc1nc(=O)c(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15845946__15859360
C[C@@H]1C[C@@]2(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)C[C@@H]12 s275592__15865378__15845952__15862300
C[C@@H]1C[C@@]2(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)C[C@@H]12 s275592__15865378__15845952__15859360
C[C@@H]1C[C@@]2(C(=O)NCC(F)=C3CN(C(=O)CSc4n[nH]c(=O)[nH]4)C3)C[C@@H]12 s275592__15865378__15845952__15857566
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CO1 s275592__15865378__15845956__15862300
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15845956__15859360
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CO1 s275592__15865378__15845956__15857566
CC(C)N1CCC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15845962__15859360
O=C(Cn1cncn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845964__15862300
O=C(Cn1cncn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845964__15859360
O=C(Cn1cncn1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845964__15857566
O=C(C=C1CCCCCC1(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845968__15859360
C=C(C)[C@@H]1OCCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845970__15862300
C=C(C)[C@@H]1OCCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845970__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCc2ncccc21 s275592__15865378__15845972__15859360
[N-]=[N+]=NC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(CC1)C2 s275592__15865378__15845974__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc2nn[nH]c12 s275592__15865378__15845976__15859360
CN(C)c1ccc(F)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15845978__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCC2(CCC2)O1 s275592__15865378__15845982__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC2(CCC2)O1 s275592__15865378__15845982__15859360
CN(C)C(=O)C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840454__15862300
CN(C)C(=O)C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840454__15859360
CN(C)C(=O)C=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840454__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccc(=O)o1 s275592__15865378__15840456__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(=O)o1 s275592__15865378__15840456__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cccc(=O)o1 s275592__15865378__15840456__15857566
Cc1cc(F)ccc1C(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840458__15859360
O=C(C=Cc1nccs1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840460__15862300
O=C(C=Cc1nccs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840460__15859360
CC1(C#CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15840462__15862300
CC1(C#CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15840462__15859360
CC1(C#CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15840462__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(F)CCS(=O)(=O)C2)C1 s275592__15865378__15840464__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1OCCn2ccnc21 s275592__15865378__15840466__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1OCCn2ccnc21 s275592__15865378__15840466__15859360
CCc1nc(O)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15840470__15859360
O=C(C=Cc1ccc2[nH]ccc2c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840474__15859360
COc1ccc(OC)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15840476__15859360
C=CC1(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15840478__15862300
C=CC1(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15840478__15859360
C=CC1(CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15840478__15857566
Cc1ncsc1C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840480__15862300
Cc1ncsc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840480__15859360
[N-]=[N+]=N[C@@H]1C=CC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15840484__15862300
[N-]=[N+]=N[C@@H]1C=CC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15840484__15859360
CC(C)CSCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840486__15862300
CC(C)CSCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840486__15859360
CC(=O)N1CCCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840490__15862300
CC(=O)N1CCCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840490__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(=O)[nH]c(=O)[nH]1 s275592__15865378__15840492__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(=O)[nH]c(=O)[nH]1 s275592__15865378__15840492__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)n1ccnc1 s275592__15865378__15840496__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)n1ccnc1 s275592__15865378__15840496__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)n1ccnc1 s275592__15865378__15840496__15857566
O=C(CSc1ncn[nH]1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840500__15862300
O=C(CSc1ncn[nH]1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840500__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccnc1O s275592__15865378__15840502__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccnc1O s275592__15865378__15840502__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cccnc1O s275592__15865378__15840502__15857566
Cc1oncc1C(=O)NCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840504__15859360
O=C(CNC(=O)CC(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840506__15859360
CC(C)CSCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840508__15862300
CC(C)CSCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840508__15859360
O=C(CCSC1CCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840510__15859360
Cc1ccc(SCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15840512__15859360
O=C(CSC(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840514__15862300
O=C(CSC(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840514__15859360
O=C(CSC(F)F)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840514__15857566
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15840516__15862300
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15840516__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc(O)n1 s275592__15865378__15840518__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc(O)n1 s275592__15865378__15840518__15859360
Cc1cc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15840520__15859360
Cc1nc(O)nc(C)c1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840522__15859360
Cc1ncc([N+](=O)[O-])cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840524__15859360
CS(=O)c1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15840528__15859360
CC1CCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15840530__15862300
CC1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15840530__15859360
CC1CCC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15840530__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccc[n+]1[O-] s275592__15865378__15840532__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc[n+]1[O-] s275592__15865378__15840532__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cccc[n+]1[O-] s275592__15865378__15840532__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CCC1 s275592__15865378__15840534__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CCC1 s275592__15865378__15840534__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1=CCC1 s275592__15865378__15840534__15857566
C=CCC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15840536__15862300
C=CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15840536__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc2c1C(=O)NC2 s275592__15865378__15840538__15859360
NC(=O)c1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)on1 s275592__15865378__15840540__15862300
NC(=O)c1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)on1 s275592__15865378__15840540__15859360
COc1cc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)on1 s275592__15865378__15840544__15862300
COc1cc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)on1 s275592__15865378__15840544__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc(OC(F)F)c1 s275592__15865378__15840546__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(O)Cc1ccccc1 s275592__15865378__15840548__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)Cc1ccccc1 s275592__15865378__15840548__15859360
Cc1ccnc(O)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840550__15862300
Cc1ccnc(O)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840550__15859360
O=C(C=C1CN2CCC1CC2)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840552__15862300
O=C(C=C1CN2CCC1CC2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840552__15859360
CCCC(CCC)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840554__15862300
CCCC(CCC)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840554__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(F)o1 s275592__15865378__15840556__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(F)o1 s275592__15865378__15840556__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1ccc(F)o1 s275592__15865378__15840556__15857566
CCCC(=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)CCC s275592__15865378__15840558__15862300
CCCC(=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)CCC s275592__15865378__15840558__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc2nc(O)ccc12 s275592__15865378__15840560__15859360
Cc1cc(=O)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15840562__15862300
Cc1cc(=O)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15840562__15859360
O=C(C=C1CCSCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840564__15862300
O=C(C=C1CCSCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840564__15859360
CON=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840566__15862300
CON=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840566__15859360
CON=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840566__15857566
C#CCC(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840568__15862300
C#CCC(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840568__15859360
C#CCC(C)(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840568__15857566
CCSc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15840570__15859360
O=C(C[C@@H](O)c1ccccc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840572__15862300
O=C(C[C@@H](O)c1ccccc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840572__15859360
Cc1ncnc(C)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840576__15862300
Cc1ncnc(C)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840576__15859360
O=C(CN1CC2C=CC1C2)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842318__15862300
O=C(CN1CC2C=CC1C2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842318__15859360
O=C(CSC(F)(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842320__15862300
O=C(CSC(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842320__15859360
O=C(CCSC(F)(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842322__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc([N+](=O)[O-])[nH]1 s275592__15865378__15842324__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc([N+](=O)[O-])[nH]1 s275592__15865378__15842324__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1OC(F)F s275592__15865378__15842326__15859360
CC1=NOC(=O)C1CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842330__15862300
CC1=NOC(=O)C1CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842330__15859360
CC(=O)Nc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15842332__15859360
Cn1cc([N+](=O)[O-])cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842334__15862300
Cn1cc([N+](=O)[O-])cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842334__15859360
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cnc2ncnn12 s275592__15865378__15842336__15859360
CN(CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(N)=O s275592__15865378__15842342__15862300
CN(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(N)=O s275592__15865378__15842342__15859360
CN(CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(N)=O s275592__15865378__15842342__15857566
CC1=NOC(=O)C1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842348__15862300
CC1=NOC(=O)C1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842348__15859360
O=C(CSc1cccs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842350__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nc(=O)[nH][nH]1 s275592__15865378__15842352__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nc(=O)[nH][nH]1 s275592__15865378__15842352__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1nc(=O)[nH][nH]1 s275592__15865378__15842352__15857566
O=C(CSc1nccs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842354__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(F)CC2)C1 s275592__15865378__15842358__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(F)CC2)C1 s275592__15865378__15842358__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(F)CC2)C1 s275592__15865378__15842358__15857566
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc([N+](=O)[O-])c1 s275592__15865378__15842360__15859360
CC(C)CCSCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842366__15862300
CC(C)CCSCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842366__15859360
CC(C)CCCOCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842368__15862300
CC(C)CCCOCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842368__15859360
CCOC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842374__15862300
CCOC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15842374__15859360
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842376__15862300
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15842376__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C(F)(F)C2CC2)C1 s275592__15865378__15842378__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)C2CC2)C1 s275592__15865378__15842378__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C(F)(F)C2CC2)C1 s275592__15865378__15842378__15857566
CCOc1oc(C)nc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842380__15862300
CCOc1oc(C)nc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842380__15859360
CCCCC[C@H](O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842384__15862300
CCCCC[C@H](O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842384__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2c(c1)CCCC2 s275592__15865378__15842386__15859360
O=C(COCCO)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842396__15862300
O=C(COCCO)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842396__15859360
O=C(COCCO)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842396__15857566
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)=NO1 s275592__15865378__15842400__15862300
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)=NO1 s275592__15865378__15842400__15859360
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)=NO1 s275592__15865378__15842400__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ncc(F)cn1 s275592__15865378__15842402__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ncc(F)cn1 s275592__15865378__15842402__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1ncc(F)cn1 s275592__15865378__15842402__15857566
CC(C)(CF)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842404__15862300
CC(C)(CF)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842404__15859360
CC(C)(CF)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842404__15857566
CC(C)[C@@H](O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842406__15862300
CC(C)[C@@H](O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842406__15859360
CC(C)[C@@H](O)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842406__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2sccc2c1 s275592__15865378__15842408__15859360
CSC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842410__15862300
CSC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842410__15859360
CSC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842410__15857566
Cc1cc(Cl)cc(C)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842414__15859360
Cc1cccc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cnc12 s275592__15865378__15842416__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(C(F)F)no1 s275592__15865378__15842418__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(C(F)F)no1 s275592__15865378__15842418__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=NOCC1 s275592__15865378__15842420__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=NOCC1 s275592__15865378__15842420__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1=NOCC1 s275592__15865378__15842420__15857566
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(CCO)CC2)C1 s275592__15865378__15842424__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(CCO)CC2)C1 s275592__15865378__15842424__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(CCO)CC2)C1 s275592__15865378__15842424__15857566
CC(C)C(C)(O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842430__15862300
CC(C)C(C)(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842430__15859360
CC(C)C(C)(O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842430__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc(O)c([N+](=O)[O-])c1 s275592__15865378__15842432__15859360
CCN1CCN(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842434__15862300
CCN1CCN(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842434__15859360
CCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn(C)c1=O s275592__15865378__15842436__15859360
CCSCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)no1 s275592__15865378__15842438__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(c1)COCC2 s275592__15865378__15844180__15859360
CCc1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cs1 s275592__15865378__15844182__15862300
CCc1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15844182__15859360
CCN1C(=O)CCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844184__15862300
CCN1C(=O)CCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844184__15859360
O=C(CC1=CSC2=NCCN12)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844186__15859360
CC1(C)CC(C)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15844194__15862300
CC1(C)CC(C)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15844194__15859360
CC1(C)CC(C)(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15844194__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@@]2(F)C[C@@H]2c2ccccc2)C1 s275592__15865378__15844196__15859360
Cn1nccc1C(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844198__15859360
Cc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)o1 s275592__15865378__15844200__15862300
Cc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15844200__15859360
COCc1ccoc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844202__15862300
COCc1ccoc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844202__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CS(=O)(=O)CCC1 s275592__15865378__15844204__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc2cn[nH]c2s1 s275592__15865378__15844206__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2cn[nH]c2s1 s275592__15865378__15844206__15859360
O=C(C=Cc1ccccc1Cl)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844208__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(-n2ccnc2)nc1 s275592__15865378__15844210__15859360
CC1CCSC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844214__15862300
CC1CCSC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844214__15859360
O=C(COc1ccccn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844216__15862300
O=C(COc1ccccn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844216__15859360
CCC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)n1ccnc1 s275592__15865378__15844220__15862300
CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)n1ccnc1 s275592__15865378__15844220__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn2cc[nH]c(=O)c2n1 s275592__15865378__15844222__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nc(C2CC2)n[nH]1 s275592__15865378__15844224__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nc(C2CC2)n[nH]1 s275592__15865378__15844224__15859360
O=C(COc1ccc(F)cn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844226__15862300
O=C(COc1ccc(F)cn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844226__15859360
CC1CC(C)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC(C)O1 s275592__15865378__15844228__15862300
CC1CC(C)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC(C)O1 s275592__15865378__15844228__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc(OC2CC2)c1 s275592__15865378__15844230__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCCCC1 s275592__15865378__15844232__15862300
COC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCCCC1 s275592__15865378__15844232__15859360
CC(CN(C)C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844234__15862300
CC(CN(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844234__15859360
CC(CN(C)C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844234__15857566
COCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCCO1 s275592__15865378__15844238__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCc2cn[nH]c21 s275592__15865378__15844240__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCc2cn[nH]c21 s275592__15865378__15844240__15859360
COc1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)ccnc1F s275592__15865378__15844244__15862300
COc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccnc1F s275592__15865378__15844244__15859360
O=C(CC1CCCOCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844246__15862300
O=C(CC1CCCOCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844246__15859360
O=C(Cn1nnc2ccccc21)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844248__15859360
Cn1cc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nn1 s275592__15865378__15844250__15862300
Cn1cc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15844250__15859360
Cn1cc(CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)nn1 s275592__15865378__15844250__15857566
O=C(CC1(O)CCCOC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844252__15862300
O=C(CC1(O)CCCOC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844252__15859360
Cc1c(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15844254__15862300
Cc1c(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15844254__15859360
O=C(C=Cc1cccc(CO)c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844258__15859360
CC(C)c1nnc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15844260__15859360
CCn1nccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844262__15862300
CCn1nccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844262__15859360
Cc1coc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844264__15862300
Cc1coc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844264__15859360
Cc1cc(C)cc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844266__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nncs1 s275592__15865378__15844270__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nncs1 s275592__15865378__15844270__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1nncs1 s275592__15865378__15844270__15857566
CC(=O)N[C@@H](C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15844272__15862300
CC(=O)N[C@@H](C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15844272__15859360
O=C(C#CC1CCCOC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844274__15862300
O=C(C#CC1CCCOC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844274__15859360
O=C(CC1CCC=CCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844276__15862300
O=C(CC1CCC=CCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844276__15859360
Cc1cc(C)n2ccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c2n1 s275592__15865378__15844282__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c2c(n[nH]c1=O)CCC2 s275592__15865378__15844284__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1[C@H]2CCCO[C@H]21 s275592__15865378__15844286__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1[C@H]2CCCO[C@H]21 s275592__15865378__15844286__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)[C@@H]1[C@H]2CCCO[C@H]21 s275592__15865378__15844286__15857566
CCCCc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15844288__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(c3cccs3)CC2)C1 s275592__15865378__15844290__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(c3cccs3)CC2)C1 s275592__15865378__15844290__15859360
CCC(C)(C)CCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844292__15862300
CCC(C)(C)CCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844292__15859360
O=C(CC(C(F)F)n1ccnc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844296__15859360
O=C(COC1CCCCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844300__15862300
O=C(COC1CCCCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844300__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(C3CCCO3)CC2)C1 s275592__15865378__15844302__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C3CCCO3)CC2)C1 s275592__15865378__15844302__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC(n2ccnc2)C1 s275592__15865378__15845984__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC(n2ccnc2)C1 s275592__15865378__15845984__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)C1CCOCC1 s275592__15865378__15845986__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)C1CCOCC1 s275592__15865378__15845986__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCC12CCC2 s275592__15865378__15845988__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCC12CCC2 s275592__15865378__15845988__15859360
NC(=O)c1cc(F)cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15845990__15859360
Cc1oc(Cl)nc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845992__15862300
Cc1oc(Cl)nc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845992__15859360
Cc1cnsc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15845996__15862300
Cc1cnsc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15845996__15859360
Cc1cnsc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15845996__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CC2CCCCCCC12 s275592__15865378__15845998__15859360
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O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H](O)Cc1c[nH]cn1 s275592__15865378__15846002__15859360
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccn1CC1CC1 s275592__15865378__15846004__15859360
CCc1onc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1C s275592__15865378__15846006__15862300
CCc1onc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1C s275592__15865378__15846006__15859360
Cn1cc(SCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cn1 s275592__15865378__15846008__15862300
Cn1cc(SCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15846008__15859360
CC(C)CC(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846010__15862300
CC(C)CC(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846010__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)C1CCC1 s275592__15865378__15846012__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)C1CCC1 s275592__15865378__15846012__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)C1CCC1 s275592__15865378__15846012__15857566
CC(OC(F)F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846014__15862300
CC(OC(F)F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846014__15859360
CC(OC(F)F)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15846014__15857566
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)O1 s275592__15865378__15846016__15862300
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)O1 s275592__15865378__15846016__15859360
CC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)O1 s275592__15865378__15846016__15857566
O=C(COc1ccc(Cl)cn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846018__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2nncc2c1 s275592__15865378__15846020__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2nncc2c1 s275592__15865378__15846020__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCCNC1=O s275592__15865378__15846022__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCCNC1=O s275592__15865378__15846022__15859360
CC1CC(C)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15846024__15862300
CC1CC(C)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15846024__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2(CCCC2)CO1 s275592__15865378__15846026__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(CCCC2)CO1 s275592__15865378__15846026__15859360
O=C(CC1CC2(CC2)CO1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846028__15862300
O=C(CC1CC2(CC2)CO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846028__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2oc(Cl)cc2[nH]1 s275592__15865378__15846030__15859360
Cn1cnc2c1CCCC2C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846032__15859360
CC(C)(F)C(C)(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846034__15862300
CC(C)(F)C(C)(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846034__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@]23COC[C@H]2C3(F)F)C1 s275592__15865378__15846036__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@]23COC[C@H]2C3(F)F)C1 s275592__15865378__15846036__15859360
Cc1cn(C(C)C)cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846040__15862300
Cc1cn(C(C)C)cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846040__15859360
CC1CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCS1 s275592__15865378__15846042__15862300
CC1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCS1 s275592__15865378__15846042__15859360
CC12CC(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)(CCO1)C2 s275592__15865378__15846044__15862300
CC12CC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(CCO1)C2 s275592__15865378__15846044__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC2(CC1)CC(O)C2 s275592__15865378__15846046__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1C[C@@H]2CCCCC[C@@H]21 s275592__15865378__15846048__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1C[C@@H]2CCCCC[C@@H]21 s275592__15865378__15846048__15859360
CC1=NOC2(C1)CC(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)C2 s275592__15865378__15846050__15862300
CC1=NOC2(C1)CC(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15846050__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(Cl)nc1C s275592__15865378__15846056__15859360
C#Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)o1 s275592__15865378__15846058__15862300
C#Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15846058__15859360
C#Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15846058__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc2c(=O)[nH]ccc12 s275592__15865378__15846060__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2n(n1)CC1(CC1)C2 s275592__15865378__15846064__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nnc2n1CCCCC2 s275592__15865378__15846068__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(-c2cc[nH]n2)c1 s275592__15865378__15846070__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1-c1ncn[nH]1 s275592__15865378__15846074__15859360
CC1(C)CC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CO1 s275592__15865378__15846076__15862300
CC1(C)CC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15846076__15859360
CC(C)C[C@H](CNC=O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846078__15859360
O=C(CC1CCCCC1(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846084__15859360
O=C(CC1CCC(=O)NC1=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846086__15862300
O=C(CC1CCC(=O)NC1=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846086__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2(CCC2)CO1 s275592__15865378__15846088__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(CCC2)CO1 s275592__15865378__15846088__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(CC2CCC2)c[nH]1 s275592__15865378__15846090__15859360
Cc1csc2ncc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)n12 s275592__15865378__15846094__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc2nc[nH]c12 s275592__15865378__15846096__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@H]2C[C@@](F)(CO)C2)C1 s275592__15865378__15846098__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@H]2C[C@@](F)(CO)C2)C1 s275592__15865378__15846098__15859360
CC1CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)=NO1 s275592__15865378__15846100__15862300
CC1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)=NO1 s275592__15865378__15846100__15859360
CC1CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)=NO1 s275592__15865378__15846100__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1snc2ccccc12 s275592__15865378__15846102__15859360
CC(C)C1=NOC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15846104__15862300
CC(C)C1=NOC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15846104__15859360
CC(C)(CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)N=[N+]=[N-] s275592__15865378__15840582__15862300
CC(C)(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)N=[N+]=[N-] s275592__15865378__15840582__15859360
CC(C)(CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)N=[N+]=[N-] s275592__15865378__15840582__15857566
CC1(F)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15840584__15862300
CC1(F)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15840584__15859360
CC1(F)CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15840584__15857566
CCSc1cccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840586__15859360
Cc1cnc(Cl)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15840588__15862300
Cc1cnc(Cl)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840588__15859360
CSC(C)CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840590__15862300
CSC(C)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840590__15859360
O=C(CC(=O)NC1CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840592__15862300
O=C(CC(=O)NC1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840592__15859360
O=C(CC(=O)NC1CC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840592__15857566
CC(O)(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15840594__15859360
COCC(O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840596__15862300
COCC(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840596__15859360
COCC(O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840596__15857566
CC1CCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)S1 s275592__15865378__15840598__15862300
CC1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)S1 s275592__15865378__15840598__15859360
CC(O)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15840600__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(O)CCSC2)C1 s275592__15865378__15840602__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(O)CCSC2)C1 s275592__15865378__15840602__15859360
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccccn1 s275592__15865378__15840606__15862300
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15840606__15859360
C#CC(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840608__15862300
C#CC(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840608__15859360
C#CC(C)(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840608__15857566
CSC1CCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840610__15862300
CSC1CCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840610__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c(C(F)(F)F)c1 s275592__15865378__15840612__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H](O)Cc1ccccc1 s275592__15865378__15840614__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H](O)Cc1ccccc1 s275592__15865378__15840614__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=COc2ccccc2O1 s275592__15865378__15840616__15859360
CN(C)C(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncn1C s275592__15865378__15840618__15859360
CN1CCCCC1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840620__15862300
CN1CCCCC1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840620__15859360
Cn1cncc1C(O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840622__15862300
Cn1cncc1C(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840622__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1conc1-c1ccccc1 s275592__15865378__15840624__15859360
O=C(Cc1nccc2ccccc12)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840626__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(F)cc2[nH]nnc12 s275592__15865378__15840628__15859360
CCOc1ccc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15840630__15859360
O=C(C=CC1CCOC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840632__15862300
O=C(C=CC1CCOC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840632__15859360
O=C(C=CC1CCOC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840632__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c(F)ccnc1Cl s275592__15865378__15840634__15859360
COc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15840636__15862300
COc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15840636__15859360
CC(C)n1ncnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840638__15862300
CC(C)n1ncnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840638__15859360
CC(C)C(O)C(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840640__15862300
CC(C)C(O)C(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840640__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nccc(Cl)c1F s275592__15865378__15840642__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2ncnc2c1 s275592__15865378__15840644__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2ncnc2c1 s275592__15865378__15840644__15859360
Cc1cc(O)nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15840646__15862300
Cc1cc(O)nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840646__15859360
COC(C)C(O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840648__15862300
COC(C)C(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840648__15859360
COC(C)C(O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840648__15857566
O=C1NC[C@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)N1 s275592__15865378__15840650__15862300
O=C1NC[C@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)N1 s275592__15865378__15840650__15859360
O=C1NC[C@H](C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)N1 s275592__15865378__15840650__15857566
CC(C)(CS(N)(=O)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840652__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cn2c(n1)SCC2 s275592__15865378__15840654__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn2c(n1)SCC2 s275592__15865378__15840654__15859360
O=C(Cc1ccnc(F)c1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840656__15862300
O=C(Cc1ccnc(F)c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840656__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnc(C=NO)s1 s275592__15865378__15840658__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc(C=NO)s1 s275592__15865378__15840658__15859360
CCSC(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840662__15862300
CCSC(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840662__15859360
CCSC(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840662__15857566
CCSc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15840664__15859360
Cc1ncn2ccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15840666__15859360
CC1CN(C(C)C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15840668__15862300
CC1CN(C(C)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15840668__15859360
CC1CN(C(C)C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15840668__15857566
CC(=O)NCCNC(=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840670__15859360
CC1(C)CCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CO1 s275592__15865378__15840674__15862300
CC1(C)CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15840674__15859360
CSCc1cccnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840676__15859360
CC1CCN1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840678__15862300
CC1CCN1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840678__15859360
CC1CCN1CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840678__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(-c2ccco2)[nH]1 s275592__15865378__15840680__15859360
O=C(CC(O)Cc1ccccc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840682__15859360
COC(C)(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15840684__15862300
COC(C)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15840684__15859360
COC(C)(C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15840684__15857566
Cn1ccc2[nH]c(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)cc21 s275592__15865378__15840688__15862300
Cn1ccc2[nH]c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc21 s275592__15865378__15840688__15859360
CN(C)CC(O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840692__15862300
CN(C)CC(O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840692__15859360
COc1cc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cn1 s275592__15865378__15840694__15862300
COc1cc(C)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15840694__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CCC(CO)(CC2)CC3)C1 s275592__15865378__15840696__15859360
O=C(COC1CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840698__15862300
O=C(COC1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840698__15859360
O=C(COC1CC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840698__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2n(n1)CCCC2O s275592__15865378__15840700__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ncc[nH]1 s275592__15865378__15840702__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ncc[nH]1 s275592__15865378__15840702__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1ncc[nH]1 s275592__15865378__15840702__15857566
O=C(C=CC1CCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840704__15862300
O=C(C=CC1CCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840704__15859360
O=C(C=CC1CCC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840704__15857566
COc1nc(O)cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15842442__15862300
COc1nc(O)cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15842442__15859360
Cc1sc(Cl)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1C s275592__15865378__15842444__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842446__15862300
COC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15842446__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15842446__15857566
CC(C)(O)C(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842448__15862300
CC(C)(O)C(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842448__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(O)c1cccnc1 s275592__15865378__15842450__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)c1cccnc1 s275592__15865378__15842450__15859360
CC(C)(OCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15842452__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2ccsc2c1 s275592__15865378__15842456__15859360
Cn1nc(O)cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842458__15862300
Cn1nc(O)cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842458__15859360
Cn1nc(O)cc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842458__15857566
CCc1c[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15842462__15862300
CCc1c[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15842462__15859360
CCc1c[nH]c(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842462__15857566
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1(F)Cl s275592__15865378__15842466__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1(F)Cl s275592__15865378__15842466__15859360
Cc1cccc2ncc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)n12 s275592__15865378__15842470__15859360
CCCC=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842472__15862300
CCCC=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842472__15859360
CCCC=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842472__15857566
CC=C(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842474__15862300
CC=C(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842474__15859360
CC=C(F)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842474__15857566
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccc2ccccc12 s275592__15865378__15842476__15859360
CSc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842478__15862300
CSc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15842478__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2(C1)CC2(F)F s275592__15865378__15842480__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(C1)CC2(F)F s275592__15865378__15842480__15859360
O=C(NCC(F)=C1CN(C(=O)CC2CC2)C1)c1nsnc1O s275592__15865378__15842482__13186218
CC(C)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186220
CC(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186222
COCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186224
O=C(NCC(F)=C1CN(C(=O)c2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__13186226
O=C(NCC(F)=C1CN(C(=O)c2ccncc2)C1)c1nsnc1O s275592__15865378__15842482__13186228
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cc2)C1)c1nsnc1O s275592__15865378__15842482__13186230
CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186232
O=C(NCC(F)=C1CN(C(=O)c2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__13186234
O=C(NCC(F)=C1CN(C(=O)Cc2cccs2)C1)c1nsnc1O s275592__15865378__15842482__13186236
O=C(NCC(F)=C1CN(C(=O)c2ccco2)C1)c1nsnc1O s275592__15865378__15842482__13186238
CC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186240
Cc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186242
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__13186244
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccco2)C1)c1nsnc1O s275592__15865378__15842482__13186246
O=C(NCC(F)=C1CN(C(=O)c2ccccc2F)C1)c1nsnc1O s275592__15865378__15842482__13186248
O=C(NCC(F)=C1CN(C(=O)c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__13186250
CC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186252
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186254
O=C(NCC(F)=C1CN(C(=O)c2cnccn2)C1)c1nsnc1O s275592__15865378__15842482__13186256
Cc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186258
O=C(NCC(F)=C1CN(C(=O)CC2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186260
O=C(NCC(F)=C1CN(C(=O)CCC2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186262
O=C(NCC(F)=C1CN(C(=O)c2cccc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__13186264
O=C(NCC(F)=C1CN(C(=O)c2cccs2)C1)c1nsnc1O s275592__15865378__15842482__13186266
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__13186268
O=C(NCC(F)=C1CN(C(=O)Cc2ccsc2)C1)c1nsnc1O s275592__15865378__15842482__13186270
CC1CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186272
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__13186274
CCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186276
CC(C)=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186278
O=C(NCC(F)=C1CN(C(=O)C2=COCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186280
O=C(NCC(F)=C1CN(C(=O)c2cc[n+]([O-])cc2)C1)c1nsnc1O s275592__15865378__15842482__13186282
O=C(NCC(F)=C1CN(C(=O)C2CC3C=CC2C3)C1)c1nsnc1O s275592__15865378__15842482__13186284
CC(=O)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186286
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)[nH]n2)C1)c1nsnc1O s275592__15865378__15842482__13186288
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__13186290
O=C(NCC(F)=C1CN(C(=O)CC2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186292
O=C(NCC(F)=C1CN(C(=O)C2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186294
CSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186296
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__13186298
CSCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186300
CC(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186302
O=C(NCC(F)=C1CN(C(=O)c2ccsc2)C1)c1nsnc1O s275592__15865378__15842482__13186306
Cc1occc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186308
O=C(NCC(F)=C1CN(C(=O)CC2C=CCC2)C1)c1nsnc1O s275592__15865378__15842482__13186310
O=C(NCC(F)=C1CN(C(=O)Cn2cnnn2)C1)c1nsnc1O s275592__15865378__15842482__13186312
O=C(NCC(F)=C1CN(C(=O)CN2CCCC2=O)C1)c1nsnc1O s275592__15865378__15842482__13186314
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__13186316
Cc1noc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186318
Cc1nnsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186320
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842482__13186322
O=C(NCC(F)=C1CN(C(=O)C2CC=CCC2)C1)c1nsnc1O s275592__15865378__15842482__13186324
O=C(NCC(F)=C1CN(C(=O)CCc2ccco2)C1)c1nsnc1O s275592__15865378__15842482__13186326
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__13186328
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CC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186334
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1C s275592__15865378__15842482__13186336
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Cc1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186342
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Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__13186348
CCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186350
CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186352
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__13186354
Cn1cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186356
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CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186362
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__13186364
CC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186366
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O=C(NCC(F)=C1CN(C(=O)c2ccccc2O)C1)c1nsnc1O s275592__15865378__15842482__13186370
CCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186372
CC(C)SCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186374
N#CCSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186376
CC(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186378
CCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186380
CC(C)OCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186382
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15842482__13186384
O=C(NCC(F)=C1CN(C(=O)CCC2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186386
O=C(NCC(F)=C1CN(C(=O)C2COCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186388
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]n2)C1)c1nsnc1O s275592__15865378__15842482__13186390
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cccn1 s275592__15865378__15842482__13186392
CCCCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186394
CSC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186396
CCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186398
CC(C)COCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186400
CCOCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186402
O=C(NCC(F)=C1CN(C(=O)COCC2CC2)C1)c1nsnc1O s275592__15865378__15842482__13186404
O=C(NCC(F)=C1CN(C(=O)CC2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186406
Cc1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186408
O=C(NCC(F)=C1CN(C(=O)c2cn[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__13186410
O=C(NCC(F)=C1CN(C(=O)CNC(=O)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__13186412
COCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186414
O=C(NCC(F)=C1CN(C(=O)COC2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186416
Cc1ncncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186418
CCSCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186420
CCOC1CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186422
O=C(NCC(F)=C1CN(C(=O)c2cnsn2)C1)c1nsnc1O s275592__15865378__15842482__13186424
O=C(NCC(F)=C1CN(C(=O)c2cnns2)C1)c1nsnc1O s275592__15865378__15842482__13186426
COC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186428
O=C(NCC(F)=C1CN(C(=O)c2ccon2)C1)c1nsnc1O s275592__15865378__15842482__13186430
CCCSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186432
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__13186434
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15842482__13186436
O=C(NCC(F)=C1CN(C(=O)c2cncs2)C1)c1nsnc1O s275592__15865378__15842482__13186438
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15842482__13186440
Cc1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__13186446
CC(C)COC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186448
CCCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186450
CCC=C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186452
CS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186454
O=C(NCC(F)=C1CN(C(=O)C=C2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186456
Cc1ocnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186458
CCOC(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186460
O=C(NCC(F)=C1CN(C(=O)CC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__13186462
COC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186464
CC(C)OCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186466
CC(OCC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186468
CCCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186470
CCCCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186472
C=CCCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186474
O=C(NCC(F)=C1CN(C(=O)C2CCOC2)C1)c1nsnc1O s275592__15865378__15842482__13186476
O=C(NCC(F)=C1CN(C(=O)c2ccnc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__13186478
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__13186480
Cn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186482
CCC(OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186484
COCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186486
CCCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186488
COC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186490
Cn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__13186492
O=C(NCC(F)=C1CN(C(=O)C2CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186494
C=CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186496
O=C(NCC(F)=C1CN(C(=O)C2=COCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186498
COC(=O)C1CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186500
O=C(NCC(F)=C1CN(C(=O)C2CCCOC2)C1)c1nsnc1O s275592__15865378__15842482__13186504
CCOCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186506
CCNC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186508
O=C(NCC(F)=C1CN(C(=O)c2cscn2)C1)c1nsnc1O s275592__15865378__15842482__13186510
COCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186512
CC(C)(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186514
C=CCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186516
O=C(NCC(F)=C1CN(C(=O)c2cocn2)C1)c1nsnc1O s275592__15865378__15842482__13186518
O=C1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__13186520
O=C(NCC(F)=C1CN(C(=O)CC2=CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186522
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__13186524
CSCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186526
CN1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186528
CCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186530
CC(C)(C)/C=C/C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186532
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)nc2)C1)c1nsnc1O s275592__15865378__15842482__13186534
CC(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186536
COCCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186538
CCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186540
Cc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186542
CC(C)(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186544
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC2O3)C1)c1nsnc1O s275592__15865378__15842482__13186546
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__13186548
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__13186550
Nc1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186552
O=C(NCC(F)=C1CN(C(=O)CCC2CC2)C1)c1nsnc1O s275592__15865378__15842482__13186554
Cc1[nH]nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__13186556
O=C(NCC(F)=C1CN(C(=O)CC2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__13186558
CCCCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186560
O=C(NCC(F)=C1CN(C(=O)Cc2ccon2)C1)c1nsnc1O s275592__15865378__15842482__13186562
CCc1ocnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186566
O=C(NCC(F)=C1CN(C(=O)CC2CCOC2)C1)c1nsnc1O s275592__15865378__15842482__13186568
O=C(NCC(F)=C1CN(C(=O)C2CC=CC2)C1)c1nsnc1O s275592__15865378__15842482__13186570
O=C(NCC(F)=C1CN(C(=O)Cc2ccn[nH]2)C1)c1nsnc1O s275592__15865378__15842482__13186572
O=C(NCC(F)=C1CN(C(=O)c2ccncc2F)C1)c1nsnc1O s275592__15865378__15842482__13186574
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nnn1C s275592__15865378__15842482__13186576
Cc1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186578
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__13186580
CN1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__13186582
Cc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__13186584
O=C(NCC(F)=C1CN(C(=O)CCC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__13186586
C=CCOCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186588
O=C(NCC(F)=C1CN(C(=O)CC2CCC2)C1)c1nsnc1O s275592__15865378__15842482__13186592
O=C(NCC(F)=C1CN(C(=O)c2cccc(=O)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__13186596
CC1(C)C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1(C)C s275592__15865378__15842482__13186598
Cc1ncoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186600
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__13186602
O=C(NCC(F)=C1CN(C(=O)C2C3CCCC32)C1)c1nsnc1O s275592__15865378__15842482__13186604
N#Cc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__13186606
Cc1cscc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186608
O=C(NCC(F)=C1CN(C(=O)CCC2CCC2)C1)c1nsnc1O s275592__15865378__15842482__13186610
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__13186612
O=C(NCC(F)=C1CN(C(=O)CCc2nnc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__13186614
Cc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186616
Cc1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186618
CC=C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186620
O=C(NCC(F)=C1CN(C(=O)CCC2CCOC2)C1)c1nsnc1O s275592__15865378__15842482__13186622
O=C(NCC(F)=C1CN(C(=O)CCc2ccoc2)C1)c1nsnc1O s275592__15865378__15842482__13186624
O=C(NCC(F)=C1CN(C(=O)C2CC(F)(F)C2)C1)c1nsnc1O s275592__15865378__15842482__13186626
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__13186628
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)=C1CCCC1 s275592__15865378__15842482__13186630
O=C(NCC(F)=C1CN(C(=O)CC2CCCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186632
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__13186634
O=C(NCC(F)=C1CN(C(=O)C=C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__13186636
O=C(NCC(F)=C1CN(C(=O)c2cncc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__13186638
CCC(=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CC s275592__15865378__15842482__13186640
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c(=O)c2)C1)c1nsnc1O s275592__15865378__15842482__13186642
CC(C)=C(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186644
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCN1 s275592__15865378__15842482__13186646
O=C(NCC(F)=C1CN(C(=O)C2=CCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186648
O=C(NCC(F)=C1CN(C(=O)C(F)=C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186650
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__13186652
Cn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__13186654
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__13186656
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)oc1C s275592__15865378__15842482__13186658
O=C(NCC(F)=C1CN(C(=O)Cc2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__13186660
O=C(NCC(F)=C1CN(C(=O)C2CCCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186662
Cc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1O s275592__15865378__15842482__13186664
CCC(SC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186666
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cccc1 s275592__15865378__15842482__13186668
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ncn1 s275592__15865378__15842482__13186670
CC1(C)CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186672
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__13186674
CCC(C)OCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186676
CC1(C)C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186678
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__13186680
CC(O)(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__13186682
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15842482__13186684
CSC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186686
O=C(NCC(F)=C1CN(C(=O)CN2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__13186688
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186690
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cncn1 s275592__15865378__15842482__13186692
NC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__13186694
CN1CCOCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186696
Cc1nscc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186698
C#CCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186700
CC(C)(C)OCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186702
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__13186704
C#CCNC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186706
CCNC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186708
CNC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186710
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__13186714
COC(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186716
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__13186718
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cn2)C1)c1nsnc1O s275592__15865378__15842482__13186720
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__13186722
O=C(NCC(F)=C1CN(C(=O)c2cncnc2)C1)c1nsnc1O s275592__15865378__15842482__13186724
O=C(NCC(F)=C1CN(C(=O)c2ncccc2O)C1)c1nsnc1O s275592__15865378__15842482__13186726
O=C(NCC(F)=C1CN(C(=O)C2=CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__13186730
O=C(NCC(F)=C1CN(C(=O)Cc2ccoc2)C1)c1nsnc1O s275592__15865378__15842482__13186732
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__13186736
O=C(NCC(F)=C1CN(C(=O)C2=CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186740
C[C@H](NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186742
O=C(NCC(F)=C1CN(C(=O)CC2OCCCO2)C1)c1nsnc1O s275592__15865378__15842482__13186744
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__13186746
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__13186748
Cc1ccn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186750
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1 s275592__15865378__15842482__13186752
O=C(NCC(F)=C1CN(C(=O)CCn2ccnn2)C1)c1nsnc1O s275592__15865378__15842482__13186754
CC(=O)N1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__13186756
Cn1oc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1=O s275592__15865378__15842482__13186758
CCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186760
COC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__13186762
CC1OCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186764
C#CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186766
O=C(NCC(F)=C1CN(C(=O)c2ccoc2Cl)C1)c1nsnc1O s275592__15865378__15842482__13186768
C=CC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186770
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ns1 s275592__15865378__15842482__13186772
CCn1ccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186778
O=C(NCC(F)=C1CN(C(=O)C2CCCOCC2)C1)c1nsnc1O s275592__15865378__15842482__13186780
O=C(NCC(F)=C1CN(C(=O)CCc2ncc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__13186782
O=C(NCC(F)=C1CN(C(=O)C2CCC(O)CC2)C1)c1nsnc1O s275592__15865378__15842482__13186784
CC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186786
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__13186788
COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__13186790
CCc1occc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186792
Cc1cc[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186794
Cn1nncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186796
O=C1NC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__13186798
CCCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186800
CC1CC(C)C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__13186802
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@@H]2C(F)F)C1)c1nsnc1O s275592__15865378__15842482__13186804
Cc1coc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186806
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__13186810
CCc1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186812
CC(C)[C@@H](O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186814
CCOC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__13186816
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__13186818
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__13186820
Cc1nnc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__13186822
Cn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__13186824
CNC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186826
O=C(NCC(F)=C1CN(C(=O)c2sccc2F)C1)c1nsnc1O s275592__15865378__15842482__13186828
CCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__13186830
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__13186832
CCn1nncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186834
Cc1csc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__13186836
O=C(NCC(F)=C1CN(C(=O)C2CC2(F)F)C1)c1nsnc1O s275592__15865378__15842482__13186838
CCC(C)=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186840
Cc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186842
CC(C)C#CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186846
Cc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186848
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCC2)C1)c1nsnc1O s275592__15865378__15842482__13186850
Cc1c[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186852
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)=C1CCC1 s275592__15865378__15842482__13186854
O=C(NCC(F)=C1CN(C(=O)C#CC2CC2)C1)c1nsnc1O s275592__15865378__15842482__13186856
CC(C)(C)C#CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186858
Cc1n[nH]c(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__13186860
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__13186862
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2[N+](=O)[O-])C1)c1nsnc1O s275592__15865378__15842482__13186864
Cc1cn(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186866
O=C(NCC(F)=C1CN(C(=O)C2CCCC(F)C2)C1)c1nsnc1O s275592__15865378__15842482__13186868
Cn1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__13186870
COCC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__13186872
CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186202
COCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__13186204
O=C(NCC(F)=C1CN(C(=O)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__13186210
O=C(NCC(F)=C1CN(C(=O)C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__13186212
O=C(NCC(F)=C1CN(C(=O)C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__13186214
O=C(NCC(F)=C1CN(C(=O)C2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__13186216
C=CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__14130358
O=C(NCC(F)=C1CN(C(=O)CCNC(=O)C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__14130362
CC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__14130366
CS(=O)(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130370
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)COC3)C1)c1nsnc1O s275592__15865378__15842482__14130372
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCCC1 s275592__15865378__15842482__14130376
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__14130378
CCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14130382
O=C(NCC(F)=C1CN(C(=O)c2ccc3nncn3c2)C1)c1nsnc1O s275592__15865378__15842482__14130392
O=C(NCC(F)=C1CN(C(=O)c2cccn3ccnc23)C1)c1nsnc1O s275592__15865378__15842482__14130396
CNC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14130398
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14130402
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(=O)N1 s275592__15865378__15842482__14130406
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14130412
O=C(NCC(F)=C1CN(C(=O)c2cncc(Cl)c2)C1)c1nsnc1O s275592__15865378__15842482__14130420
Cc1nccn1CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130432
Cc1noc(C)c1C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130434
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842482__14130436
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__14130442
O=C(NCC(F)=C1CN(C(=O)CCN2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__14130454
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCOCC1 s275592__15865378__15842482__14130458
O=C(NCC(F)=C1CN(C(=O)COc2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__14130462
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__14130464
Cc1cc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842482__14130466
CC(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__14130470
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)cc2)C1)c1nsnc1O s275592__15865378__15842482__14130478
CC(C)CCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130492
CCn1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14130498
CC(C)CC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130504
CCCCCCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130510
O=C(NCC(F)=C1CN(C(=O)c2ccc3nccn3c2)C1)c1nsnc1O s275592__15865378__15842482__14130514
O=C(NCC(F)=C1CN(C(=O)CN2CCCCC2=O)C1)c1nsnc1O s275592__15865378__15842482__14135180
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1=O s275592__15865378__15842482__14135184
COCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135188
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__14135190
CCCc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__14135192
O=C(NCC(F)=C1CN(C(=O)CN2CCCNC2=O)C1)c1nsnc1O s275592__15865378__15842482__14135202
O=C(Nc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135206
O=C(NCC(F)=C1CN(C(=O)c2cn3cccnc3n2)C1)c1nsnc1O s275592__15865378__15842482__14135214
O=C(NCC(F)=C1CN(C(=O)C23CCCN2CCC3)C1)c1nsnc1O s275592__15865378__15842482__14135218
CCc1ccc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135228
O=C(NCC(F)=C1CN(C(=O)c2cccn3nccc23)C1)c1nsnc1O s275592__15865378__15842482__14135230
O=C(NCC(F)=C1CN(C(=O)c2cccnc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14135238
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2OCCC3)C1)c1nsnc1O s275592__15865378__15842482__14135244
CCOc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__14135248
O=C(NCC(F)=C1CN(C(=O)c2ncnc3[nH]ccc23)C1)c1nsnc1O s275592__15865378__15842482__14135252
O=C(NCC(F)=C1CN(C(=O)c2cc3cnccc3o2)C1)c1nsnc1O s275592__15865378__15842482__14135260
O=C(NCC(F)=C1CN(C(=O)c2ccn3cncc3c2)C1)c1nsnc1O s275592__15865378__15842482__14135262
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c(=O)[nH]c2=O)C1)c1nsnc1O s275592__15865378__15842482__14135264
Cc1nnccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135266
O=C(NCC(F)=C1CN(C(=O)c2ccnc(C3CC3)c2)C1)c1nsnc1O s275592__15865378__15842482__14135268
COCc1csc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14135272
CC(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14135274
Cn1cc(C(N)=O)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135280
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCOCC1 s275592__15865378__15842482__14135288
O=C1CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__14135292
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14135296
Cc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1C s275592__15865378__15842482__14135300
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1Cl s275592__15865378__15842482__14135302
Cc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__14135306
CCCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135308
COc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__14135310
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1C s275592__15865378__15842482__14135312
O=C(NCC(F)=C1CN(C(=O)c2cccnc2C(F)F)C1)c1nsnc1O s275592__15865378__15842482__14135316
Cc1cncc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14135318
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__14135320
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14135324
O=C(NCC(F)=C1CN(C(=O)C2CCCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14135328
COCCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14135336
Cn1ccc(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14135338
Cc1cnc(COCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14135340
O=C(NCC(F)=C1CN(C(=O)c2ccnc3nn[nH]c23)C1)c1nsnc1O s275592__15865378__15842482__14135342
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15842482__14130526
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(F)(F)C1 s275592__15865378__15842482__14130528
O=C(NCC(F)=C1CN(C(=O)c2cc3c([nH]2)CCC3)C1)c1nsnc1O s275592__15865378__15842482__14130530
CC(C)c1scnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130534
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(Cl)n1 s275592__15865378__15842482__14130536
COCc1nocc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130550
CC(C)n1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14130552
Cc1nn(C(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130554
CCc1oc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842482__14130562
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCCC1=O s275592__15865378__15842482__14130564
Cn1nc2c(c1C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)CCC2 s275592__15865378__15842482__14130568
CN1CCCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1=O s275592__15865378__15842482__14130570
CN1C(=O)CN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1=O s275592__15865378__15842482__14130578
O=C(NCC(F)=C1CN(C(=O)C2CCc3[nH]ncc3C2)C1)c1nsnc1O s275592__15865378__15842482__14130580
CCCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__14130588
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCOCC3)C2)C1)c1nsnc1O s275592__15865378__15842482__14130592
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)s2)C1)c1nsnc1O s275592__15865378__15842482__14130594
COCc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130596
CCCc1occc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130598
Cc1ccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14130600
CC(CCC(C)(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130608
CCCCCCC(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130610
CN(C)C1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14130622
CC1(C)CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14130628
CN1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14130638
Cn1cncc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130640
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3cccnc23)C1)c1nsnc1O s275592__15865378__15842482__14130644
O=C(NCC(F)=C1CN(C(=O)COc2ccsc2)C1)c1nsnc1O s275592__15865378__15842482__14130646
CCCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14130648
CCc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14130652
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)oc1CC s275592__15865378__15842482__14130658
COc1cc[nH]c(=O)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130664
CC(C)Cc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14130666
CCn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14130668
CN(C)c1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130670
CCC(CC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130674
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccco1 s275592__15865378__15842482__14130678
CC(Oc1ccccn1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130680
CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__14130682
O=C(NCC(F)=C1CN(C(=O)c2ccn3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__14135346
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCCO3)C1)c1nsnc1O s275592__15865378__15842482__14135354
COc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14135356
CC(C)(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14135370
O=C(NCC(F)=C1CN(C(=O)C2CC3CC2C2CC32)C1)c1nsnc1O s275592__15865378__15842482__14135372
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C(C)O1 s275592__15865378__15842482__14135374
O=C(NCC(F)=C1CN(C(=O)C23CCCCC2OCC3)C1)c1nsnc1O s275592__15865378__15842482__14135378
CC(C)(C)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135380
O=C(NCC(F)=C1CN(C(=O)[C@]23CCC[C@H]2OCC3)C1)c1nsnc1O s275592__15865378__15842482__14135382
CC1CC1C1CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135384
CC1(C)COC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14135388
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__14135394
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CC(F)F s275592__15865378__15842482__14135402
O=C(NCC(F)=C1CN(C(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)C1)c1nsnc1O s275592__15865378__15842482__14135406
CC1(C)CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)OC1 s275592__15865378__15842482__14135408
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3O[C@H]2[C@H]2C[C@@H]32)C1)c1nsnc1O s275592__15865378__15842482__14135418
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2C[C@H]2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14135422
CC1COC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14135424
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ncc1=O s275592__15865378__15842482__14135430
Cc1nc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14135432
O=C(NCC(F)=C1CN(C(=O)[C@@]23CCC[C@@H]2C3)C1)c1nsnc1O s275592__15865378__15842482__14135434
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15842482__14135436
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCO[C@H]2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14135438
CC(C)n1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14135442
CC[C@@H]1OCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135448
O=C(NCC(F)=C1CN(C(=O)CC2CCC(C3CC3)O2)C1)c1nsnc1O s275592__15865378__15842482__14135452
CCc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15842482__14135458
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)c1 s275592__15865378__15842482__14135460
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842482__14135462
O=C(NCC(F)=C1CN(C(=O)c2nccc3occc23)C1)c1nsnc1O s275592__15865378__15842482__14135466
O=C(NCC(F)=C1CN(C(=O)C2CC[C@H]3C[C@H]3CC2)C1)c1nsnc1O s275592__15865378__15842482__14135470
CCn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14135476
Cn1nccc1[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135478
CC1CC2CC2CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135480
O=C(NCC(F)=C1CN(C(=O)[C@@H]2OC[C@@H]3COCC[C@@H]32)C1)c1nsnc1O s275592__15865378__15842482__14135486
Cn1ccnc1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135492
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3CCCC[C@@H]32)C1)c1nsnc1O s275592__15865378__15842482__14135494
C[C@H](CC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135498
C[C@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__14130686
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14130688
CN(C)C(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130706
CCNC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130708
CCCNC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130710
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccnc1 s275592__15865378__15842482__14130714
CCCNC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130716
CC(C)NC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130718
Cc1ccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14130730
Cn1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1=O s275592__15865378__15842482__14130734
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14130744
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14130746
CN(C)CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130748
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__14130750
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14130752
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cccc1 s275592__15865378__15842482__14130754
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14130762
CO[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__14130764
O=C1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__14130766
CC(=O)N1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130768
COc1cc(C)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130770
CC(=O)N[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14130772
CC(=O)N[C@@H](CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130776
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__14130778
CC(=O)N[C@H](CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130780
C[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14130782
CC[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14130784
O=C(NCC(F)=C1CN(C(=O)c2ncccc2Cl)C1)c1nsnc1O s275592__15865378__15842482__14130786
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)cn2)C1)c1nsnc1O s275592__15865378__15842482__14130788
Cc1cc(F)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130790
Cc1ccc(F)c(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14130794
Cc1ccc(=O)n(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14130802
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__14130804
O=C(NCC(F)=C1CN(C(=O)c2cccc(C(F)F)c2)C1)c1nsnc1O s275592__15865378__15842482__14130806
CCCN(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130808
O=C(NCC(F)=C1CN(C(=O)CCCc2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__14130814
O=C(NCC(F)=C1CN(C(=O)c2cnc(C3CC3)s2)C1)c1nsnc1O s275592__15865378__15842482__14130816
CNC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14130818
COc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130822
CCCN(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130824
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15842482__14130832
COc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130834
CCCCCCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130836
O=C(NCC(F)=C1CN(C(=O)c2cnn3cc[nH]c23)C1)c1nsnc1O s275592__15865378__15842482__14130840
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCO1 s275592__15865378__15842482__14130842
O=C(NCC(F)=C1CN(C(=O)c2occ3c2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14130844
CC1(C)COC(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14130846
COCCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14130850
CCC[C@@H](NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130854
O=C1CCCCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__14130858
C#Cc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130860
Cc1[nH]cnc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130862
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCCC3)CC2)C1)c1nsnc1O s275592__15865378__15842482__14130864
O=C(NCC(F)=C1CN(C(=O)c2cc3[nH]ccc3s2)C1)c1nsnc1O s275592__15865378__15842482__14130866
O=C(NCC(F)=C1CN(C(=O)Cn2c(=O)[nH][nH]c2=O)C1)c1nsnc1O s275592__15865378__15842482__14130872
O=C(NCC(F)=C1CN(C(=O)COCc2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__14130878
O=C(NCC(F)=C1CN(C(=O)C2Cc3cccnc3C2)C1)c1nsnc1O s275592__15865378__15842482__14130880
COc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__14130882
CC(F)(F)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130884
O=C(NCC(F)=C1CN(C(=O)C23CCCN(CC2)C3)C1)c1nsnc1O s275592__15865378__15842482__14130890
CC(=O)N(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130896
COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCC1 s275592__15865378__15842482__14130900
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__14130910
COCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14130918
Cc1nn(C)c(F)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130926
C[C@H](CC1CCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130928
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)o2)C1)c1nsnc1O s275592__15865378__15842482__14130934
Cc1cc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14130940
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(F)(F)F s275592__15865378__15842482__14130942
CCc1nc[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130946
CN(C)S(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130948
CN1C(=O)CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130954
O=C(NCC(F)=C1CN(C(=O)C2CCC(C3CC3)CC2)C1)c1nsnc1O s275592__15865378__15842482__14130962
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)cn2)C1)c1nsnc1O s275592__15865378__15842482__14130968
O=C(NCC(F)=C1CN(C(=O)c2cncnc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14130970
CC(=O)N1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14130976
Cn1cncc1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130982
Cc1nn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)n1C s275592__15865378__15842482__14130984
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__14130992
Cc1n[nH]c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131000
Cc1n[nH]c(C)c1C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131002
CCCCCCN(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131004
O=C(NCC(F)=C1CN(C(=O)c2cnn3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__14131014
O=C(NCC(F)=C1CN(C(=O)c2nccn3ccnc23)C1)c1nsnc1O s275592__15865378__15842482__14131024
CCN(CC)C(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14131032
CCn1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1=O s275592__15865378__15842482__14131038
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15842482__14131042
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1F s275592__15865378__15842482__14131048
Cc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131050
O=C(NCC(F)=C1CN(C(=O)c2ccc3cccnc3c2)C1)c1nsnc1O s275592__15865378__15842482__14131052
Cc1ccc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131054
CC(C)CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131056
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1Cl s275592__15865378__15842482__14131066
CC(C)(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131068
O=C(NCC(F)=C1CN(C(=O)c2ccncn2)C1)c1nsnc1O s275592__15865378__15842482__14131070
O=C(NCC(F)=C1CN(C(=O)c2nc3ncccn3n2)C1)c1nsnc1O s275592__15865378__15842482__14131074
CCCCCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131076
O=C(NCC(F)=C1CN(C(=O)CCc2ncccn2)C1)c1nsnc1O s275592__15865378__15842482__14131082
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842482__14131084
O=C(NCC(F)=C1CN(C(=O)c2cc3ncccn3n2)C1)c1nsnc1O s275592__15865378__15842482__14131088
O=C(NCC(F)=C1CN(C(=O)Cc2ccco2)C1)c1nsnc1O s275592__15865378__15842482__14131092
O=C(NCC(F)=C1CN(C(=O)c2ncccn2)C1)c1nsnc1O s275592__15865378__15842482__14131098
CCC(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131100
CC(C)c1nnsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131108
O=C(NCC(F)=C1CN(C(=O)c2cccc3[nH]cnc23)C1)c1nsnc1O s275592__15865378__15842482__14131110
O=C(NCC(F)=C1CN(C(=O)c2cccnn2)C1)c1nsnc1O s275592__15865378__15842482__14131112
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1F s275592__15865378__15842482__14131114
CCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14131120
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14131126
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842482__14131130
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15842482__14131134
O=C(NCC(F)=C1CN(C(=O)CCn2cnnn2)C1)c1nsnc1O s275592__15865378__15842482__14131136
CC1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14131138
CCCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14131144
CCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15842482__14131146
O=C(NCC(F)=C1CN(C(=O)c2ncccc2F)C1)c1nsnc1O s275592__15865378__15842482__14131150
CC(C)[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14131156
O=C(NCC(F)=C1CN(C(=O)COCc2ccncc2)C1)c1nsnc1O s275592__15865378__15842482__14131162
CC1OCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131176
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOC1 s275592__15865378__15842482__14131178
O=C(NCC(F)=C1CN(C(=O)c2cnn(C(F)F)c2)C1)c1nsnc1O s275592__15865378__15842482__14131180
CC(C)Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14131182
NC(=O)c1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14131190
CCC(CC)(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131192
CCCC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__14131196
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__14131198
CCCC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131200
CCC(CC)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131202
CCC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131204
CCCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131208
O=C(NCC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131216
O=C(NCC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131218
O=C(NCC(F)=C1CN(C(=O)CCCc2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__14131224
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__14131228
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCOC1 s275592__15865378__15842482__14131230
CN1CCC(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14131232
O=C(NCC(F)=C1CN(C(=O)c2cn(CC3CC3)nn2)C1)c1nsnc1O s275592__15865378__15842482__14131234
CCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14131236
CC(C)n1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14131238
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nnn1C(C)C s275592__15865378__15842482__14131240
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14131246
CC(Cc1cnn(C)c1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131252
O=C(NCC(F)=C1CN(C(=O)CCC2CCCOC2)C1)c1nsnc1O s275592__15865378__15842482__14131254
O=C(NCC(F)=C1CN(C(=O)CCn2cnccc2=O)C1)c1nsnc1O s275592__15865378__15842482__14131258
COCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__14131266
O=C(NCC(F)=C1CN(C(=O)c2coc(CC3CC3)n2)C1)c1nsnc1O s275592__15865378__15842482__14131268
Cc1oc(C2CC2)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131270
O=C(NCC(F)=C1CN(C(=O)C2CC2C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14131274
O=C(NCC(F)=C1CN(C(=O)c2c[nH]cc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14131278
CCC1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131282
CCC1(C(C)C)CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131284
CCC1(C)CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131286
CC(C)C1(C)CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131290
Cn1cc(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14131294
COCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131300
CCc1c[nH]c(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14131304
COCCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131314
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__14131318
Cc1nonc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131322
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14131330
Cc1ncsc1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131332
Cc1oc(C(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131346
O=C(NCC(F)=C1CN(C(=O)c2cccc3ccncc23)C1)c1nsnc1O s275592__15865378__15842482__14131348
C=CCCOCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131852
O=C(NCC(F)=C1CN(C(=O)COC2CCOC2)C1)c1nsnc1O s275592__15865378__15842482__14131856
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)NC(N)=O s275592__15865378__15842482__14131860
CC(C)(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__14131864
Cc1oc(C(C)C)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131866
Cc1cccn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1=O s275592__15865378__15842482__14131868
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CC2)C1)c1nsnc1O s275592__15865378__15842482__14131884
O=C(NCC(F)=C1CN(C(=O)C2CCCC3(CC3)C2)C1)c1nsnc1O s275592__15865378__15842482__14131886
O=C(NCC(F)=C1CN(C(=O)C2(c3ccccn3)CC2)C1)c1nsnc1O s275592__15865378__15842482__14131888
O=C(NCC(F)=C1CN(C(=O)c2cnn(C3CCC3)c2)C1)c1nsnc1O s275592__15865378__15842482__14131890
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCCN3C2)C1)c1nsnc1O s275592__15865378__15842482__14131894
CC(C)Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__14131902
CN(C)c1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14131906
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)C2)C1)c1nsnc1O s275592__15865378__15842482__14133584
NC(=O)Cc1occc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133586
Cn1cc(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14133590
O=C(NCC(F)=C1CN(C(=O)C(C2CCC2)C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__14133592
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(C)n1 s275592__15865378__15842482__14133594
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14133596
CN(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133608
O=C(NCC(F)=C1CN(C(=O)C2CCCc3[nH]nnc32)C1)c1nsnc1O s275592__15865378__15842482__14133612
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]ncc3c2)C1)c1nsnc1O s275592__15865378__15842482__14133614
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)cn2)C1)c1nsnc1O s275592__15865378__15842482__14133618
O=C(NCC(F)=C1CN(C(=O)c2nccc3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__14133620
CCCC(CCC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133626
CCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133628
O=C(NCC(F)=C1CN(C(=O)Cc2cc(F)ccc2F)C1)c1nsnc1O s275592__15865378__15842482__14133630
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)c(F)c2)C1)c1nsnc1O s275592__15865378__15842482__14133632
O=C(NCC(F)=C1CN(C(=O)c2cccc(F)c2F)C1)c1nsnc1O s275592__15865378__15842482__14133634
CC(C)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14131352
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14131354
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15842482__14131360
O=C(NCC(F)=C1CN(C(=O)c2cnoc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14131364
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14131366
CC(C)c1oncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131368
CC1(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14131376
Cc1cnoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131378
COc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14131388
Cc1cc(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__14131390
O=C(NCC(F)=C1CN(C(=O)c2cc3sccc3[nH]2)C1)c1nsnc1O s275592__15865378__15842482__14131406
CC(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14131412
O=C(NCC(F)=C1CN(C(=O)C2(F)CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14131416
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14131426
O=C(NCC(F)=C1CN(C(=O)c2ncoc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14131428
CCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14131430
CCN(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131434
O=C(NCC(F)=C1CN(C(=O)C2CC23CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14131436
O=C(NCC(F)=C1CN(C(=O)CCc2cnccn2)C1)c1nsnc1O s275592__15865378__15842482__14131440
CC(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__14131446
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14131448
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccncc3c2)C1)c1nsnc1O s275592__15865378__15842482__14131452
O=C(NCC(F)=C1CN(C(=O)CCCn2cncn2)C1)c1nsnc1O s275592__15865378__15842482__14131454
O=C(NCC(F)=C1CN(C(=O)c2ccc3cnccc3c2)C1)c1nsnc1O s275592__15865378__15842482__14131456
O=C(NCC(F)=C1CN(C(=O)c2csc(Cl)n2)C1)c1nsnc1O s275592__15865378__15842482__14131458
CC(C)(CC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131460
Cc1conc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131468
CC(C)c1ocnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131470
O=C1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C(=O)N1 s275592__15865378__15842482__14131474
O=C(NCC(F)=C1CN(C(=O)c2cc3c([nH]2)CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14131478
CCC(=O)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14131484
COC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(F)(F)F s275592__15865378__15842482__14131490
O=C(NCC(F)=C1CN(C(=O)c2cnn(CC3CC3)c2)C1)c1nsnc1O s275592__15865378__15842482__14131496
CCC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__14131504
CCC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__14131506
O=C(NCC(F)=C1CN(C(=O)C2CCc3[nH]cnc3C2)C1)c1nsnc1O s275592__15865378__15842482__14131508
CC(=O)N1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14131510
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCCCC1 s275592__15865378__15842482__14131922
O=C(NCC(F)=C1CN(C(=O)C2CCCc3[nH]ncc32)C1)c1nsnc1O s275592__15865378__15842482__14131926
CCOCCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14131944
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__14131956
O=C(NCC(F)=C1CN(C(=O)CCOCC(F)F)C1)c1nsnc1O s275592__15865378__15842482__14131962
O=C(NCC(F)=C1CN(C(=O)Cn2ncnn2)C1)c1nsnc1O s275592__15865378__15842482__14131964
Cn1ncc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131966
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ncn1 s275592__15865378__15842482__14131968
O=C(NCC(F)=C1CN(C(=O)C2CN3CCC2CC3)C1)c1nsnc1O s275592__15865378__15842482__14131970
CCCC[C@@H](C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131972
CCc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14131974
O=C(NCC(F)=C1CN(C(=O)c2cccc3nn[nH]c23)C1)c1nsnc1O s275592__15865378__15842482__14131978
CC1=C(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14131980
CC(C)(C)CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131982
C=CCC(CC=C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131996
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC=CCC1 s275592__15865378__15842482__14132000
Cn1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14132002
O=C(NCC(F)=C1CN(C(=O)C2CS(=O)(=O)C2)C1)c1nsnc1O s275592__15865378__15842482__14132004
Cc1scc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14132006
CCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132012
CCCC(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132014
CCC(C)CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132016
CC(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132018
Cc1ccn(CC(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14132026
O=C(NCC(F)=C1CN(C(=O)c2cccn3nnnc23)C1)c1nsnc1O s275592__15865378__15842482__14132032
C=C(Cl)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132034
CC(C)n1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132036
O=C(NCC(F)=C1CN(C(=O)c2ccn(C(F)F)n2)C1)c1nsnc1O s275592__15865378__15842482__14132040
O=C(NCC(F)=C1CN(C(=O)c2ccnn2C(F)F)C1)c1nsnc1O s275592__15865378__15842482__14132042
C=CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132044
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(C)n1 s275592__15865378__15842482__14132050
O=C(NCC(F)=C1CN(C(=O)Cn2nccn2)C1)c1nsnc1O s275592__15865378__15842482__14132056
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14132060
CCCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132068
CCCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14132070
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C2CC2)n1 s275592__15865378__15842482__14132072
Cc1c(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__14132076
COc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__14132082
O=C(NCC(F)=C1CN(C(=O)Cc2c(F)cccc2F)C1)c1nsnc1O s275592__15865378__15842482__14133638
CC1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133642
CC1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133644
COC1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133648
COC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133650
CCCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14133652
Cc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133662
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc32)C1)c1nsnc1O s275592__15865378__15842482__14133672
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]ccc3c2)C1)c1nsnc1O s275592__15865378__15842482__14133676
C=CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133684
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1F s275592__15865378__15842482__14133686
NS(=O)(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133688
CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133690
CCCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133692
Cc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133694
NC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133696
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)c1 s275592__15865378__15842482__14133698
NC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133704
O=C(NCC(F)=C1CN(C(=O)c2ccc3nonc3c2)C1)c1nsnc1O s275592__15865378__15842482__14133706
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(Cl)c2)C1)c1nsnc1O s275592__15865378__15842482__14133708
O=C(NCC(F)=C1CN(C(=O)CCCc2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14133716
Cc1nocc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133720
Cc1cc(C)cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133724
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1Cl s275592__15865378__15842482__14133730
Cc1cc(Cl)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133732
O=C(NCC(F)=C1CN(C(=O)c2ccc3ncccc3c2)C1)c1nsnc1O s275592__15865378__15842482__14133738
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1Cl s275592__15865378__15842482__14133740
CC(CC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133742
COc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133744
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__14133746
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133750
Cc1ccc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133756
Cc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1F s275592__15865378__15842482__14133764
Cc1cccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133766
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC=CC1 s275592__15865378__15842482__14133772
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]c1=O s275592__15865378__15842482__14133774
COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14133776
CC1CC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133778
CCCCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133780
C=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133782
C=CCCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133784
C=CC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133786
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)CC2)C1)c1nsnc1O s275592__15865378__15842482__14133788
O=C(NCC(F)=C1CN(C(=O)C[C@H]2CCOC2)C1)c1nsnc1O s275592__15865378__15842482__14133790
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14133792
O=C(NCC(F)=C1CN(C(=O)CC2=CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__14133794
CCc1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133796
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133798
CC(C)[C@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__14133800
CCC1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133804
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)no2)C1)c1nsnc1O s275592__15865378__15842482__14128902
CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14128908
O=C(NCC(F)=C1CN(C(=O)c2ccccc2Cl)C1)c1nsnc1O s275592__15865378__15842482__14128910
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)cc2)C1)c1nsnc1O s275592__15865378__15842482__14128916
CCCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14128918
COc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14128920
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccccc3n2)C1)c1nsnc1O s275592__15865378__15842482__14128922
O=C(NCC(F)=C1CN(C(=O)c2cccc(Cl)c2)C1)c1nsnc1O s275592__15865378__15842482__14128934
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14128938
CCCCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14128948
O=C(NCC(F)=C1CN(C(=O)CCc2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14128950
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14128954
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14128958
O=C(NCC(F)=C1CN(C(=O)COc2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14128960
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccccc3c2)C1)c1nsnc1O s275592__15865378__15842482__14128962
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14128964
COc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14128966
O=C(NCC(F)=C1CN(C(=O)c2c(F)cccc2F)C1)c1nsnc1O s275592__15865378__15842482__14128982
CN(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14128992
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14128994
Cc1ccc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14128996
Cc1cc(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14128998
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(Cl)cc2)C1)c1nsnc1O s275592__15865378__15842482__14129002
CCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14129006
CCOc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129008
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cc2)C1)c1nsnc1O s275592__15865378__15842482__14129010
CCOc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129012
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cc2F)C1)c1nsnc1O s275592__15865378__15842482__14129014
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14129016
O=C(NCC(F)=C1CN(C(=O)C2CC23CCOC3)C1)c1nsnc1O s275592__15865378__15842482__14131518
CCC1CCCN1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131524
COCCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131526
CCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131528
CCCCCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14131530
COCCCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131536
COCCCOCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131538
CC(C)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131540
O=C(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)NCC1CC1 s275592__15865378__15842482__14131542
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cccn1 s275592__15865378__15842482__14131546
O=C(NCC(F)=C1CN(C(=O)c2coc(C3CCC3)n2)C1)c1nsnc1O s275592__15865378__15842482__14131548
Cc1n[nH]c(C(C)C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131556
NC(=O)CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131560
CC1CCN(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14131570
O=C(NCC(F)=C1CN(C(=O)C(C2CC2)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14131574
O=C(NCC(F)=C1CN(C(=O)Cc2nc[nH]n2)C1)c1nsnc1O s275592__15865378__15842482__14131602
CN(C)C(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14131610
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C(C)C s275592__15865378__15842482__14131614
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCC1 s275592__15865378__15842482__14131618
NC(=O)N1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131622
CC(C)(C)c1n[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131624
CCn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14131638
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cnn(C)c1 s275592__15865378__15842482__14131640
CCCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14131642
O=C(NCC(F)=C1CN(C(=O)CCC2CCCCO2)C1)c1nsnc1O s275592__15865378__15842482__14131644
CCC(OC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131652
COc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)nn1C s275592__15865378__15842482__14131656
CC(C)n1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14131658
CN(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842482__14131660
NC(=O)C1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14131666
CC1CCCC(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14131672
O=C(NCC(F)=C1CN(C(=O)c2ccnc(C3CC3)n2)C1)c1nsnc1O s275592__15865378__15842482__14131674
O=C(NCC(F)=C1CN(C(=O)c2csc3cncn23)C1)c1nsnc1O s275592__15865378__15842482__14131678
CC1CCCCC1OCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131680
O=C(NCC(F)=C1CN(C(=O)COC2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__14131682
O=C(NCC(F)=C1CN(C(=O)c2ccnc3[nH]cnc23)C1)c1nsnc1O s275592__15865378__15842482__14132086
Cc1cccc(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132088
O=C(NCC(F)=C1CN(C(=O)C2C=CC=CC=C2)C1)c1nsnc1O s275592__15865378__15842482__14132090
C=C(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132092
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]cnc3c2)C1)c1nsnc1O s275592__15865378__15842482__14132094
O=C(NCC(F)=C1CN(C(=O)CCc2ccncn2)C1)c1nsnc1O s275592__15865378__15842482__14132098
CC(C)Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14132100
CCC(C)n1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132104
CC(C)Cn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132106
Cn1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14132110
Cn1nccc1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132112
Cn1nc(C2CC2)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132114
O=C(NCC(F)=C1CN(C(=O)c2cc3occc3[nH]2)C1)c1nsnc1O s275592__15865378__15842482__14132116
O=C(NCC(F)=C1CN(C(=O)c2ccns2)C1)c1nsnc1O s275592__15865378__15842482__14132118
C=C(C)C(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)OCC s275592__15865378__15842482__14132122
CCN(CC)CC(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132124
CCC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__14132128
O=C(NCC(F)=C1CN(C(=O)c2cn3c(n2)CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14132136
Cc1n[nH]c(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132142
COCCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14132154
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14132156
Cc1c(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__14132160
O=C(NCC(F)=C1CN(C(=O)c2[nH]ccc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14132164
Cc1cnc(CCCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14132172
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__14132176
COC1CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14132180
COCC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132182
CCC(CC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132184
CC(C)(CC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132188
Cn1ncc(C2CC2)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132192
O=C(NCC(F)=C1CN(C(=O)c2cc3c(o2)CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14132196
O=C(NCC(F)=C1CN(C(=O)CC2(C(F)(F)F)CC2)C1)c1nsnc1O s275592__15865378__15842482__14132214
O=C(NCC(F)=C1CN(C(=O)c2cc3c([nH]2)CCOC3)C1)c1nsnc1O s275592__15865378__15842482__14132216
O=C(NCC(F)=C1CN(C(=O)Cc2cc(C3CC3)no2)C1)c1nsnc1O s275592__15865378__15842482__14132218
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ccnn23)C1)c1nsnc1O s275592__15865378__15842482__14132220
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CN1 s275592__15865378__15842482__14132222
O=C(NCC(F)=C1CN(C(=O)CC2CC3CCC2O3)C1)c1nsnc1O s275592__15865378__15842482__14132224
CCn1nnc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132226
CC(C)c1nocc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132228
O=C(NCC(F)=C1CN(C(=O)CC2CCNC2=O)C1)c1nsnc1O s275592__15865378__15842482__14132230
Cc1ncc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14132232
CC(C)CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14132236
CCOC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14132238
O=C(NCC(F)=C1CN(C(=O)Cn2cc(C3CC3)nn2)C1)c1nsnc1O s275592__15865378__15842482__14132242
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14132244
CC1CCCC1(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133806
CC(F)(F)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133808
COC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133810
CCCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133812
C[C@@]1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(=O)N1 s275592__15865378__15842482__14133814
CCc1nocc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133818
CC1COCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133820
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1C s275592__15865378__15842482__14133822
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__14133824
COCC(OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133826
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133828
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCO1 s275592__15865378__15842482__14133830
CCC[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133832
O=C(NCC(F)=C1CN(C(=O)C23CCCCC2C3)C1)c1nsnc1O s275592__15865378__15842482__14133834
CC(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14133836
C=C1CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133838
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(F)F s275592__15865378__15842482__14133840
Cc1ccoc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133842
CCc1ncoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133844
C#Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133846
CCOc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842482__14133852
CC(Oc1cccnc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133864
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cccc1=O s275592__15865378__15842482__14133870
O=C(NCC(F)=C1CN(C(=O)C2(CF)CC2)C1)c1nsnc1O s275592__15865378__15842482__14133872
O=C(NCC(F)=C1CN(C(=O)C2CC3(CC3)C2)C1)c1nsnc1O s275592__15865378__15842482__14133874
Cc1cc(=O)[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133876
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)F)[nH]n2)C1)c1nsnc1O s275592__15865378__15842482__14133880
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14133882
O=C(NCC(F)=C1CN(C(=O)c2conc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14133884
CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(CC)CC s275592__15865378__15842482__14133888
NC(=O)c1coc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133902
O=C(NCC(F)=C1CN(C(=O)C2CCCC(F)(F)C2)C1)c1nsnc1O s275592__15865378__15842482__14133904
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccsc1 s275592__15865378__15842482__14133912
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccs1 s275592__15865378__15842482__14133914
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccco1 s275592__15865378__15842482__14133916
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nnn1CC s275592__15865378__15842482__14133922
O=C(NCC(F)=C1CN(C(=O)c2cc3occc3s2)C1)c1nsnc1O s275592__15865378__15842482__14133932
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCNC1=O s275592__15865378__15842482__14133934
NC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__14133942
O=C(NCC(F)=C1CN(C(=O)c2ncsc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14133944
CCOC1CC2(C1)CC2C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133946
Cc1ncccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133950
O=C(NCC(F)=C1CN(C(=O)c2ocnc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14133952
CC(C)(C)n1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14133958
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c2C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__14133962
CC1CCCN1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133964
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__14133966
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1C s275592__15865378__15842482__14133970
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14129024
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__14129026
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)c1 s275592__15865378__15842482__14129028
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2F)C1)c1nsnc1O s275592__15865378__15842482__14129030
Cc1ccccc1OCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129032
O=C(NCC(F)=C1CN(C(=O)c2cccc3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__14129034
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842482__14129038
O=C(NCC(F)=C1CN(C(=O)CC2CC3CCC2C3)C1)c1nsnc1O s275592__15865378__15842482__14129044
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__14129048
CC(Oc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129050
COc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14129052
O=C(NCC(F)=C1CN(C(=O)CCC2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14129054
CCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129058
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccco1 s275592__15865378__15842482__14129088
O=C(NCC(F)=C1CN(C(=O)c2cn3ccccc3n2)C1)c1nsnc1O s275592__15865378__15842482__14129090
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)s2)C1)c1nsnc1O s275592__15865378__15842482__14129106
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3o2)C1)c1nsnc1O s275592__15865378__15842482__14129114
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__14129120
O=C(NCC(F)=C1CN(C(=O)CCCC2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14129124
O=C(NCC(F)=C1CN(C(=O)c2cc3c(s2)CCC3)C1)c1nsnc1O s275592__15865378__15842482__14129132
O=C(NCC(F)=C1CN(C(=O)c2sccc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14129140
CC(=O)NCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129154
O=C(NCC(F)=C1CN(C(=O)C2(c3ccccc3)CC2)C1)c1nsnc1O s275592__15865378__15842482__14129156
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__14129160
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2Cl)C1)c1nsnc1O s275592__15865378__15842482__14129164
Cc1ccc(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14129172
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1=O s275592__15865378__15842482__14129174
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__14129178
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)c1 s275592__15865378__15842482__14129180
COc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129182
O=C(NCC(F)=C1CN(C(=O)COCC2CCOC2)C1)c1nsnc1O s275592__15865378__15842482__14131684
CC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131690
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)S(C)(=O)=O s275592__15865378__15842482__14131696
CC(CC1CCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131700
CC(CC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131708
CCC(CC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131710
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccn3c2)C1)c1nsnc1O s275592__15865378__15842482__14131718
Cc1nc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__14131726
Cc1nn(C)cc1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131728
O=C(NCC(F)=C1CN(C(=O)CCC2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__14131736
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccnc1 s275592__15865378__15842482__14131738
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14131742
COc1cc(C)sc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131748
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCCCCC1 s275592__15865378__15842482__14131750
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__14131752
CC(C)N1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131756
CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14131758
C[C@H]1CC[C@@](C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1(C)C s275592__15865378__15842482__14131764
CC(C)CCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131768
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)cs2)C1)c1nsnc1O s275592__15865378__15842482__14131772
O=C(NCC(F)=C1CN(C(=O)c2csc(Cl)c2)C1)c1nsnc1O s275592__15865378__15842482__14131774
O=C(NCC(F)=C1CN(C(=O)c2ccsc2Cl)C1)c1nsnc1O s275592__15865378__15842482__14131780
C=C(C)CC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131784
CCCCCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131788
Cc1ncc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14131790
COc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14131794
Cc1sccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131800
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1C s275592__15865378__15842482__14131808
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14131812
O=C(NCC(F)=C1CN(C(=O)CNC(=O)N2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14131822
C#CCOCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131824
COCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14131826
C#CCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131828
CC(C)N1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131832
O=C(NCC(F)=C1CN(C(=O)CCOCC2CC2)C1)c1nsnc1O s275592__15865378__15842482__14131836
CNS(=O)(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131840
CC1CC1c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14131844
CCCc1onc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14131846
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14132268
CC(C)N1CCCC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132270
O=C(NCC(F)=C1CN(C(=O)CCc2ccsc2)C1)c1nsnc1O s275592__15865378__15842482__14132292
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(F)c2)C1)c1nsnc1O s275592__15865378__15842482__14132300
O=C(NCC(F)=C1CN(C(=O)c2cc(F)ccc2F)C1)c1nsnc1O s275592__15865378__15842482__14132302
Cc1cc(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14132312
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1F s275592__15865378__15842482__14132314
Cc1noc(C(C)C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132318
O=C(NCC(F)=C1CN(C(=O)c2snnc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14132324
Cc1c(Cl)cncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132328
CC(C)(C(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132330
CC(C)[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__14132338
Cc1ncn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132342
Cc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1F s275592__15865378__15842482__14132344
O=C(NCC(F)=C1CN(C(=O)CCCc2ccsc2)C1)c1nsnc1O s275592__15865378__15842482__14132346
O=C(NCC(F)=C1CN(C(=O)c2ccc3cc[nH]c3n2)C1)c1nsnc1O s275592__15865378__15842482__14132348
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]ccc3c2)C1)c1nsnc1O s275592__15865378__15842482__14132350
O=C(NCC(F)=C1CN(C(=O)Cc2cncs2)C1)c1nsnc1O s275592__15865378__15842482__14132352
Cc1cc(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1C s275592__15865378__15842482__14132354
O=C(NCC(F)=C1CN(C(=O)c2cn[nH]c(=O)c2)C1)c1nsnc1O s275592__15865378__15842482__14132362
Cc1[nH]c(=O)[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132366
O=C(NCC(F)=C1CN(C(=O)c2cscc2Cl)C1)c1nsnc1O s275592__15865378__15842482__14132378
CCc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132384
O=C(NCC(F)=C1CN(C(=O)C2(C3CC3)CC2)C1)c1nsnc1O s275592__15865378__15842482__14132386
COC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14132390
O=C1CCC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__14132392
Cn1ccnc1COCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132394
CN1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1=O s275592__15865378__15842482__14132396
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14132400
CC1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133972
O=C(NCC(F)=C1CN(C(=O)C2(CF)CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__14133976
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccncc3C2)C1)c1nsnc1O s275592__15865378__15842482__14133986
O=C(NCC(F)=C1CN(C(=O)CC(F)(F)C(F)F)C1)c1nsnc1O s275592__15865378__15842482__14133994
CC1(C)CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133996
CN(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CC(C)(C)C s275592__15865378__15842482__14133998
O=C(NCC(F)=C1CN(C(=O)CCc2cncs2)C1)c1nsnc1O s275592__15865378__15842482__14134002
NC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14134006
NC(=O)[C@@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134008
O=C(NCC(F)=C1CN(C(=O)c2ocnc2C(F)F)C1)c1nsnc1O s275592__15865378__15842482__14134012
Cn1ncc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14134014
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__14134016
CC(F)(F)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14134018
CC[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__14134026
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)(F)F s275592__15865378__15842482__14134028
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)[nH]1 s275592__15865378__15842482__14134034
O=C(NCC(F)=C1CN(C(=O)c2nccn3ccnc23)C1)c1nsnc1O s275592__15865378__15842482__14134036
Cc1ccn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14134040
O=C(NCC(F)=C1CN(C(=O)c2nccc3[nH]ccc23)C1)c1nsnc1O s275592__15865378__15842482__14134042
COc1cc(=O)[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134046
Cn1cncc1[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134052
O=C(NCC(F)=C1CN(C(=O)CCc2c[nH]nn2)C1)c1nsnc1O s275592__15865378__15842482__14134054
O=C(NCC(F)=C1CN(C(=O)C2(CF)CCC2)C1)c1nsnc1O s275592__15865378__15842482__14134056
C=C[C@@H]1OCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134058
CC(C)C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134062
CC[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134064
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]3CC[C@@H]2O3)C1)c1nsnc1O s275592__15865378__15842482__14134076
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCC(=O)N1 s275592__15865378__15842482__14134082
Cn1cc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14134086
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccco2)C1)c1nsnc1O s275592__15865378__15842482__14134088
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__14134090
O=C(NCC(F)=C1CN(C(=O)c2cccc3cc[nH]c23)C1)c1nsnc1O s275592__15865378__15842482__14134096
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__14134100
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(Cl)c1 s275592__15865378__15842482__14134104
CCC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134108
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1F s275592__15865378__15842482__14134112
O=C(NCC(F)=C1CN(C(=O)c2cccc3[nH]ccc23)C1)c1nsnc1O s275592__15865378__15842482__14134114
CC(C)=CCCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134116
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1F s275592__15865378__15842482__14134118
C=Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14134120
CC(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134122
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2OCC3)C1)c1nsnc1O s275592__15865378__15842482__14134124
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCO3)C1)c1nsnc1O s275592__15865378__15842482__14134126
O=C(NCC(F)=C1CN(C(=O)C2(C(F)(F)F)CC2)C1)c1nsnc1O s275592__15865378__15842482__14134130
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842482__14129202
O=C(NCC(F)=C1CN(C(=O)Cn2cncn2)C1)c1nsnc1O s275592__15865378__15842482__14129210
Cc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__14129214
O=C(NCC(F)=C1CN(C(=O)CCCc2cccs2)C1)c1nsnc1O s275592__15865378__15842482__14129218
CCc1sc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842482__14129222
O=C(NCC(F)=C1CN(C(=O)CN2C(=O)CNC2=O)C1)c1nsnc1O s275592__15865378__15842482__14129228
CN1CC(=O)N(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1=O s275592__15865378__15842482__14129230
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3[nH]2)C1)c1nsnc1O s275592__15865378__15842482__14129232
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)sc1C s275592__15865378__15842482__14129234
O=C(NCC(F)=C1CN(C(=O)CN2CCCCCC2=O)C1)c1nsnc1O s275592__15865378__15842482__14129238
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)sc1C s275592__15865378__15842482__14129240
Cc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14129242
O=C1NC(=O)C(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__14129246
NC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129250
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__14129252
NC(=O)c1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129254
O=C(NCC(F)=C1CN(C(=O)CN2C(=O)CCC2=O)C1)c1nsnc1O s275592__15865378__15842482__14129268
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)n1C s275592__15865378__15842482__14129270
NC(=O)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14129274
CC(=O)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14129276
Cc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129282
O=C(NCC(F)=C1CN(C(=O)CCc2cccs2)C1)c1nsnc1O s275592__15865378__15842482__14129292
O=C(NCC(F)=C1CN(C(=O)Cn2ccccc2=O)C1)c1nsnc1O s275592__15865378__15842482__14129296
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCC3)C1)c1nsnc1O s275592__15865378__15842482__14129300
Cc1noc(C)c1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129302
COCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14129304
CCc1onc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129316
O=C(NCC(F)=C1CN(C(=O)COc2ccc(F)cc2)C1)c1nsnc1O s275592__15865378__15842482__14129326
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]nnc3c2)C1)c1nsnc1O s275592__15865378__15842482__14129330
Cc1n[nH]c(C)c1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129340
O=C(NCC(F)=C1CN(C(=O)COCc2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14129344
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14129348
O=C(NCC(F)=C1CN(C(=O)CCc2ccccc2F)C1)c1nsnc1O s275592__15865378__15842482__14129354
Cc1csc(=O)n1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129356
COCCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132420
Cc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132428
O=C(NCC(F)=C1CN(C(=O)c2cnc3cc[nH]c3c2)C1)c1nsnc1O s275592__15865378__15842482__14132434
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]ncc3c2)C1)c1nsnc1O s275592__15865378__15842482__14132436
O=C(NCC(F)=C1CN(C(=O)C2CCC2(F)F)C1)c1nsnc1O s275592__15865378__15842482__14132438
O=C(NCC(F)=C1CN(C(=O)c2ccsn2)C1)c1nsnc1O s275592__15865378__15842482__14132440
CCOc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__14132442
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)cc1F s275592__15865378__15842482__14132444
Cc1cc(COCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14132448
Cc1cc(COCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__14132450
Cn1nccc1COCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132452
O=C(NCC(F)=C1CN(C(=O)c2ccc3nc[nH]c3n2)C1)c1nsnc1O s275592__15865378__15842482__14132454
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]c1C s275592__15865378__15842482__14132456
O=C(NCC(F)=C1CN(C(=O)c2cc3cccn3cn2)C1)c1nsnc1O s275592__15865378__15842482__14132460
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)s1 s275592__15865378__15842482__14132464
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCC1 s275592__15865378__15842482__14132466
CCc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132468
O=C(NCC(F)=C1CN(C(=O)CC2C=CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14132470
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cn2)C1)c1nsnc1O s275592__15865378__15842482__14132474
CCc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14132478
O=C(NCC(F)=C1CN(C(=O)C2CCn3cncc3C2)C1)c1nsnc1O s275592__15865378__15842482__14132480
CCOCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14132486
O=C(NCC(F)=C1CN(C(=O)CC2CC(F)(F)C2)C1)c1nsnc1O s275592__15865378__15842482__14132496
COCc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132504
CCc1nnc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132508
O=C(NCC(F)=C1CN(C(=O)C2CC3C=CC2O3)C1)c1nsnc1O s275592__15865378__15842482__14132520
CCCCC(C)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132522
O=C(NCC(F)=C1CN(C(=O)C2CCc3nccn3C2)C1)c1nsnc1O s275592__15865378__15842482__14132524
O=C(NCC(F)=C1CN(C(=O)C2CCn3ccnc3C2)C1)c1nsnc1O s275592__15865378__15842482__14132526
O=C(NCC(F)=C1CN(C(=O)C2CCc3cncn3C2)C1)c1nsnc1O s275592__15865378__15842482__14132528
COC1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132536
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__14132538
O=C(NCC(F)=C1CN(C(=O)C2CCCC3CC32)C1)c1nsnc1O s275592__15865378__15842482__14132540
O=C(NCC(F)=C1CN(C(=O)CC2CCC3CC23)C1)c1nsnc1O s275592__15865378__15842482__14132542
O=C(NCC(F)=C1CN(C(=O)C2CCC3CC3C2)C1)c1nsnc1O s275592__15865378__15842482__14132544
CCC(C)C(OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132546
COC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14132548
CN1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1=O s275592__15865378__15842482__14132550
O=C(NCC(F)=C1CN(C(=O)Cn2cc(C3CC3)cn2)C1)c1nsnc1O s275592__15865378__15842482__14132560
CCCC1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132564
CCC(CC)C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132570
O=C(NCC(F)=C1CN(C(=O)CC2CS(=O)(=O)C2)C1)c1nsnc1O s275592__15865378__15842482__14132572
Cn1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1=O s275592__15865378__15842482__14132578
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)[nH]n2)C1)c1nsnc1O s275592__15865378__15842482__14134134
O=C(NCC(F)=C1CN(C(=O)CCCC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__14134136
Cc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14134142
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CC(C)(C)C s275592__15865378__15842482__14134146
CCn1nc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134148
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3C2)C1)c1nsnc1O s275592__15865378__15842482__14134150
O=C(NCC(F)=C1CN(C(=O)c2noc3c2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14134154
O=C(NCC(F)=C1CN(C(=O)c2ccncc2Cl)C1)c1nsnc1O s275592__15865378__15842482__14134160
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__14134166
Cc1ccccc1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134168
O=C(NCC(F)=C1CN(C(=O)C2C3CCCCCCC32)C1)c1nsnc1O s275592__15865378__15842482__14134172
O=C(NCC(F)=C1CN(C(=O)C2CC23CC3)C1)c1nsnc1O s275592__15865378__15842482__14134174
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)(F)CC2)C1)c1nsnc1O s275592__15865378__15842482__14134184
Cc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14134198
CC(NS(C)(=O)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134200
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]1 s275592__15865378__15842482__14134206
O=C(NCC(F)=C1CN(C(=O)c2cnc3ccccc3c2)C1)c1nsnc1O s275592__15865378__15842482__14134208
O=C(NCC(F)=C1CN(C(=O)c2ccc3cc[nH]c3c2)C1)c1nsnc1O s275592__15865378__15842482__14134212
CCOc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14134214
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14134216
O=C(NCC(F)=C1CN(C(=O)Cc2cnc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__14134222
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(F)c2F)C1)c1nsnc1O s275592__15865378__15842482__14134224
O=C(NCC(F)=C1CN(C(=O)CC2CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14134228
C=CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134236
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)[nH]1 s275592__15865378__15842482__14134240
O=C(NCC(F)=C1CN(C(=O)C(F)c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14134242
O=C(NCC(F)=C1CN(C(=O)C2CC23CCC3)C1)c1nsnc1O s275592__15865378__15842482__14134246
O=C1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)NC(=O)N1 s275592__15865378__15842482__14134252
Cc1cccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14134262
O=C(NCC(F)=C1CN(C(=O)Cn2cc(Cl)cn2)C1)c1nsnc1O s275592__15865378__15842482__14134270
Cc1cccc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134132
CCc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14134278
CCCN1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1=O s275592__15865378__15842482__14134280
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1ccnc1 s275592__15865378__15842482__14134282
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15842482__14134284
Cc1ccnn1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134288
CCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14134294
Cc1ccn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)c1 s275592__15865378__15842482__14134298
Cc1noc(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129364
Cc1n[nH]c(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129366
CC(C)(C)C(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129370
CCc1noc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129372
Cc1cccc(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14129384
O=C(NCC(F)=C1CN(C(=O)COc2cccc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__14129390
O=C(NCC(F)=C1CN(C(=O)CCOc2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14129398
O=C(NCC(F)=C1CN(C(=O)COc2ccccc2F)C1)c1nsnc1O s275592__15865378__15842482__14129404
Cc1noc(CCCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14129410
Cc1cc(NC(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14129416
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]c1=O s275592__15865378__15842482__14129420
CC(C)c1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129426
CN(C)c1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129436
Cc1c[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129438
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14129446
O=C(NCC(F)=C1CN(C(=O)c2cccc3cnccc23)C1)c1nsnc1O s275592__15865378__15842482__14129448
Cc1nccn1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129462
CC(CN1CCOCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129466
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14129468
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__14129474
CCn1cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129478
CC(C)n1cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129480
O=C(NCC(F)=C1CN(C(=O)c2scnc2Cl)C1)c1nsnc1O s275592__15865378__15842482__14129488
CCn1cc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129492
CCc1ncncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129494
CC(C)c1ncncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129496
O=C(NCC(F)=C1CN(C(=O)CC2CCCOC2)C1)c1nsnc1O s275592__15865378__15842482__14129500
O=C(NCC(F)=C1CN(C(=O)C2CCC=CCC2)C1)c1nsnc1O s275592__15865378__15842482__14129502
NC(=O)c1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14129504
O=C(NCC(F)=C1CN(C(=O)C2CCS(=O)(=O)N2)C1)c1nsnc1O s275592__15865378__15842482__14129506
Cc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14129508
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(C)c1F s275592__15865378__15842482__14129510
O=C(NCC(F)=C1CN(C(=O)CCCN2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14129514
CCC(C)C(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129516
O=C(NCC(F)=C1CN(C(=O)CCN2CCCC2=O)C1)c1nsnc1O s275592__15865378__15842482__14129518
CNS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129522
CCCS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129526
CC(C)S(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129528
O=C(NCC(F)=C1CN(C(=O)c2cnc3ccccn23)C1)c1nsnc1O s275592__15865378__15842482__14132582
CCc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132598
CCN1CCOCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132600
O=C(NCC(F)=C1CN(C(=O)C2(F)CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14132604
CCc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132606
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccnc1 s275592__15865378__15842482__14132610
CN(C)Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14132620
O=C(NCC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132628
O=C(NCC(F)=C1CN(C(=O)c2cnn(CCF)c2)C1)c1nsnc1O s275592__15865378__15842482__14132634
Cc1cc(C)nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14132636
O=C(NCC(F)=C1CN(C(=O)c2cccc3ncnn23)C1)c1nsnc1O s275592__15865378__15842482__14132642
Cn1cncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132644
O=C(NCC(F)=C1CN(C(=O)c2cccc3cccnc23)C1)c1nsnc1O s275592__15865378__15842482__14132646
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(F)cc2)C1)c1nsnc1O s275592__15865378__15842482__14132650
O=C(NCC(F)=C1CN(C(=O)CCc2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__14132654
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__14132656
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__14132666
O=C(NCC(F)=C1CN(C(=O)Cn2ccc(=O)[nH]c2=O)C1)c1nsnc1O s275592__15865378__15842482__14132678
COCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14132680
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)s1 s275592__15865378__15842482__14132688
NC(=O)NCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132694
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14132698
CCn1c(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14132702
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14132704
CCc1nnsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132706
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__14132708
COc1ccc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132712
O=C(NCC(F)=C1CN(C(=O)CCN2C(=O)CCC2=O)C1)c1nsnc1O s275592__15865378__15842482__14132734
O=C(NCC(F)=C1CN(C(=O)C2CCS(=O)(=O)C2)C1)c1nsnc1O s275592__15865378__15842482__14132736
CC(=O)N1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14132740
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3O2)C1)c1nsnc1O s275592__15865378__15842482__14132744
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)no2)C1)c1nsnc1O s275592__15865378__15842482__14134302
CCc1oncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134304
CC(Cc1cccs1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134306
CC(C)c1nccn1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134308
O=C(NCC(F)=C1CN(C(=O)c2cnc(C3CC3)nc2)C1)c1nsnc1O s275592__15865378__15842482__14134314
O=C(NCC(F)=C1CN(C(=O)Cc2cscn2)C1)c1nsnc1O s275592__15865378__15842482__14134318
CC1CCN(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14134322
CC1CCCN(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14134324
COc1nc(C)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134326
O=C(NCC(F)=C1CN(C(=O)c2coc(C3CC3)n2)C1)c1nsnc1O s275592__15865378__15842482__14134328
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@@H]2c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14134330
COCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14134338
O=C(NCC(F)=C1CN(C(=O)c2ccc3cccnn23)C1)c1nsnc1O s275592__15865378__15842482__14134352
O=C(NCC(F)=C1CN(C(=O)c2cnc3cccnn23)C1)c1nsnc1O s275592__15865378__15842482__14134356
CN(C)C(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134358
Cc1ccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14134366
CCC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__14134372
CC1(C)C2CCC1(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)CC2 s275592__15865378__15842482__14134380
C=CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14134384
CC(C)c1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134388
O=C(NCC(F)=C1CN(C(=O)c2scnc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14134392
COCc1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134394
CC(C)c1nnnn1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134396
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCCC1 s275592__15865378__15842482__14134398
Cc1nc(C2CC2)oc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134406
Cc1nc(C(C)C)oc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134408
O=C(NCC(F)=C1CN(C(=O)CCc2cn[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__14134428
CC(Cc1cnc[nH]1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134436
C=CCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14134438
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14134440
O=C(NCC(F)=C1CN(C(=O)C2CCCC3CCCN32)C1)c1nsnc1O s275592__15865378__15842482__14134444
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__14134448
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ncccc23)C1)c1nsnc1O s275592__15865378__15842482__14129530
O=C(NCC(F)=C1CN(C(=O)CCCn2cccn2)C1)c1nsnc1O s275592__15865378__15842482__14129540
CC(C)(C)CC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129552
O=C(NCC(F)=C1CN(C(=O)CCc2nccs2)C1)c1nsnc1O s275592__15865378__15842482__14129558
COCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129568
CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCCC1=O s275592__15865378__15842482__14129572
CC1OC(C)C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1C s275592__15865378__15842482__14129578
CCC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129596
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccc(F)c1 s275592__15865378__15842482__14129606
O=C(NCC(F)=C1CN(C(=O)C2CCCS2(=O)=O)C1)c1nsnc1O s275592__15865378__15842482__14129618
O=C(NCC(F)=C1CN(C(=O)c2noc3c2COCC3)C1)c1nsnc1O s275592__15865378__15842482__14129620
O=C(NCC(F)=C1CN(C(=O)C2CCc3cn[nH]c3C2)C1)c1nsnc1O s275592__15865378__15842482__14129624
CCN1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14129634
CC1CCC(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__14129640
Cc1cc(=O)[nH]c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129644
C[C@@H](Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129646
C[C@H](Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129648
O=C(NCC(F)=C1CN(C(=O)C23CCC(CC2)CC3)C1)c1nsnc1O s275592__15865378__15842482__14129652
CCCCCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129660
CC[C@H](C)[C@H](NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129666
CCCCCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129668
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)cc2)C1)c1nsnc1O s275592__15865378__15842482__14129672
CC1=CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14129676
CC(C)(C)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129682
NC(=O)N1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14132748
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1F s275592__15865378__15842482__14132750
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1C s275592__15865378__15842482__14132754
Cc1oc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14132776
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14132778
Cc1cc(C)n(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14132786
COCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14132792
Cc1cc(=O)oc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132794
Cn1cc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132796
CC(C)=CC1C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1(C)C s275592__15865378__15842482__14132798
Cc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14132806
O=C(NCC(F)=C1CN(C(=O)c2ccn3ccnc3c2)C1)c1nsnc1O s275592__15865378__15842482__14132830
O=C(NCC(F)=C1CN(C(=O)c2cccc3nccn23)C1)c1nsnc1O s275592__15865378__15842482__14132832
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]ccc3n2)C1)c1nsnc1O s275592__15865378__15842482__14132834
O=C(NCC(F)=C1CN(C(=O)c2ccc3nnnn3c2)C1)c1nsnc1O s275592__15865378__15842482__14132836
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15842482__14132840
O=C(NCC(F)=C1CN(C(=O)c2ncc(Cl)s2)C1)c1nsnc1O s275592__15865378__15842482__14132846
O=C(NCC(F)=C1CN(C(=O)c2ncc3ccccn23)C1)c1nsnc1O s275592__15865378__15842482__14132852
O=C(NCC(F)=C1CN(C(=O)c2onc3c2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14132856
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14132860
COCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132862
O=C(NCC(F)=C1CN(C(=O)c2cnc3nccn3c2)C1)c1nsnc1O s275592__15865378__15842482__14132876
O=C(NCC(F)=C1CN(C(=O)CCc2ccon2)C1)c1nsnc1O s275592__15865378__15842482__14132878
O=C(NCC(F)=C1CN(C(=O)CCc2cncnc2)C1)c1nsnc1O s275592__15865378__15842482__14132880
COc1coc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1=O s275592__15865378__15842482__14132886
COc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1=O s275592__15865378__15842482__14132888
Cc1cc(Cl)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14132890
O=C(NCC(F)=C1CN(C(=O)c2ccc3cncn3c2)C1)c1nsnc1O s275592__15865378__15842482__14132894
CCc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14132896
Cc1csc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14132898
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1C s275592__15865378__15842482__14132902
Cc1cncn1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132904
C=C(C)[C@@H]1OCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134470
O=C(NCC(F)=C1CN(C(=O)c2cn(C3CCC3)nn2)C1)c1nsnc1O s275592__15865378__15842482__14134480
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCCO1 s275592__15865378__15842482__14134488
O=C(NCC(F)=C1CN(C(=O)c2ccnn2C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__14134490
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccnn1C s275592__15865378__15842482__14134508
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)sn1 s275592__15865378__15842482__14134518
O=C(NCC(F)=C1CN(C(=O)c2cn3c(n2)CCC3)C1)c1nsnc1O s275592__15865378__15842482__14134522
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccncc2)C1)c1nsnc1O s275592__15865378__15842482__14134524
C[C@@H]1[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCN1C s275592__15865378__15842482__14134526
CC(C)(C)c1nc[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134528
CC(C)(C)C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134532
NC(=O)c1ncn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14134538
CC[C@@H]1[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCN1C s275592__15865378__15842482__14134540
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3C=C[C@H]2CC3)C1)c1nsnc1O s275592__15865378__15842482__14134544
CCN(CC)C(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129696
C=CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__14129700
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__14129704
Cc1ccccc1C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129710
O=C(NCC(F)=C1CN(C(=O)C(F)Cc2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__14129716
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__14129720
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15842482__14129730
CC(C)c1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129748
CCc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129752
CC1CCC(C)N1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129754
O=C(NCC(F)=C1CN(C(=O)C2CCc3nncn3C2)C1)c1nsnc1O s275592__15865378__15842482__14129756
CCOCCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129772
O=C(NCC(F)=C1CN(C(=O)c2cncc3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__14129774
Cn1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14129776
O=C(NCC(F)=C1CN(C(=O)CCCN2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14129778
Cc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14129792
CNC(=O)NC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129794
CCc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__14129798
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14129802
C#CCN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14129804
O=C(NCC(F)=C1CN(C(=O)CCN2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14129808
Cc1ccc(C)n1C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129810
Cc1cnn(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14129814
CCS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129820
NC(=O)Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14129832
CCN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129844
O=C(NCC(F)=C1CN(C(=O)[C@H]2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__14129852
O=C(NCC(F)=C1CN(C(=O)CCC(F)F)C1)c1nsnc1O s275592__15865378__15842482__14132916
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(=O)[nH]1 s275592__15865378__15842482__14132928
CCOc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__14132934
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CC2)CC3)C1)c1nsnc1O s275592__15865378__15842482__14132936
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14132938
O=C(NCC(F)=C1CN(C(=O)CCC2CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14132942
Cc1onc(C2CC2)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132946
Cc1noc(C2CC2)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132948
O=C(NCC(F)=C1CN(C(=O)c2cc3ncccc3o2)C1)c1nsnc1O s275592__15865378__15842482__14132950
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(=O)[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__14132952
CC(CC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132954
O=C(NCC(F)=C1CN(C(=O)c2cc(F)c[nH]2)C1)c1nsnc1O s275592__15865378__15842482__14132964
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14132968
CCCCC(CC)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14132972
CCC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(=O)N1 s275592__15865378__15842482__14132974
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CNC(=O)C1 s275592__15865378__15842482__14132976
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC2CC2C1 s275592__15865378__15842482__14132994
O=C(NCC(F)=C1CN(C(=O)C2(CCF)CC2)C1)c1nsnc1O s275592__15865378__15842482__14132998
COCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133000
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cnn(C)c1 s275592__15865378__15842482__14133004
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14133006
Cc1nccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14133020
Cn1cnn(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1=O s275592__15865378__15842482__14133022
O=C(NCC(F)=C1CN(C(=O)COCC(F)F)C1)c1nsnc1O s275592__15865378__15842482__14133024
O=C(NCC(F)=C1CN(C(=O)CCCCc2c[nH]nn2)C1)c1nsnc1O s275592__15865378__15842482__14133030
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__14133032
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)nn1 s275592__15865378__15842482__14133040
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2(F)F)C1)c1nsnc1O s275592__15865378__15842482__14133046
O=C(NCC(F)=C1CN(C(=O)C2(C3CC3)CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__14133048
CC(C)n1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133050
CN(C)C1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__14133066
CNS(=O)(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133068
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCN1 s275592__15865378__15842482__14133072
O=C(NCC(F)=C1CN(C(=O)c2occ3c2CCC3)C1)c1nsnc1O s275592__15865378__15842482__14133076
O=C(NCC(F)=C1CN(C(=O)c2occ3c2CCOC3)C1)c1nsnc1O s275592__15865378__15842482__14133078
Cc1cncc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133080
CCn1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14134546
O=C(NCC(F)=C1CN(C(=O)[C@@]23COC[C@@H]2C3)C1)c1nsnc1O s275592__15865378__15842482__14134550
O=C(NCC(F)=C1CN(C(=O)c2cncc3nc[nH]c23)C1)c1nsnc1O s275592__15865378__15842482__14134554
CC(C)(C)n1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14134564
O=C(NCC(F)=C1CN(C(=O)C(F)C(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__14134568
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cc2F)C1)c1nsnc1O s275592__15865378__15842482__14134572
Cc1c(F)cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134574
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14134582
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1F s275592__15865378__15842482__14134584
Cc1c(Cl)cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134588
O=C(NCC(F)=C1CN(C(=O)c2sccc2Cl)C1)c1nsnc1O s275592__15865378__15842482__14134590
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__14134596
CC1CCCC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134598
COc1cccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134600
O=C(NCC(F)=C1CN(C(=O)CNC(=O)C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14134602
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccoc1 s275592__15865378__15842482__14134606
CCC(=O)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134614
CC(C)C(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134634
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CS(=O)(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134638
CN(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)S(C)(=O)=O s275592__15865378__15842482__14134640
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COCC(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134646
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CCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14134694
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CCCCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14129904
CC(C)CC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129906
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Cc1nsc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129922
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CC1CC(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14129942
CC(=O)N1CCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129950
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14129952
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__14129956
CC1(C)CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14129958
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14129962
NC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14129964
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CCCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129976
CC(=O)NC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__14129978
CC1(C)CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14129984
CC1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14129986
CC(C)(C)C12CC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(C1)C2 s275592__15865378__15842482__14130002
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COCCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__14130012
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__14130014
CC(CC1CCCO1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130016
CC(C)c1occc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130018
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COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cnn(C)c1 s275592__15865378__15842482__14133086
COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCOC1 s275592__15865378__15842482__14133090
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCC1 s275592__15865378__15842482__14133094
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOC1 s275592__15865378__15842482__14133100
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COc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__14133112
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCC1 s275592__15865378__15842482__14133122
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COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCC1 s275592__15865378__15842482__14133132
Cc1cccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133136
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CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__14133144
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CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__14133160
Cc1ccc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133168
Cc1nn(C)c(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133172
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Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]1 s275592__15865378__15842482__14133180
Cc1nn(C)c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133182
Cc1cc(C)n(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14133194
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COc1ccc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133216
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Cc1noc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14133230
CC(NC(=O)C(C)(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133240
CC(C)(C)C(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133242
CNC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134714
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__14134736
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__14134738
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CC1CC2(CCO1)CC2C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134744
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C1CC1 s275592__15865378__15842482__14134748
CC(C)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134750
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]nnc3n2)C1)c1nsnc1O s275592__15865378__15842482__14134754
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCC3)C1)c1nsnc1O s275592__15865378__15842482__14134762
CCc1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134764
COc1nc(C)ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134768
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2CCC3)C1)c1nsnc1O s275592__15865378__15842482__14134772
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COc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__14134778
CC(C)(C)n1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14134782
O=C(NCC(F)=C1CN(C(=O)C2(F)CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__14134790
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O=C(NCC(F)=C1CN(C(=O)CC2CCC(F)(F)C2)C1)c1nsnc1O s275592__15865378__15842482__14134794
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)nc2)C1)c1nsnc1O s275592__15865378__15842482__14134800
C=CCn1cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134804
CN(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCC1 s275592__15865378__15842482__14134810
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O=C(NCC(F)=C1CN(C(=O)CN2CCOCC2=O)C1)c1nsnc1O s275592__15865378__15842482__14134824
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]nnc3c2)C1)c1nsnc1O s275592__15865378__15842482__14134826
CCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14134828
O=C(NCC(F)=C1CN(C(=O)c2cnn3ncccc23)C1)c1nsnc1O s275592__15865378__15842482__14134830
Cc1nn(C)cc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134832
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCC1 s275592__15865378__15842482__14134842
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCCC1 s275592__15865378__15842482__14134852
COc1cc(C)cnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134858
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CCOCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130024
CNC(=O)CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130026
CC(C)(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14130034
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1C s275592__15865378__15842482__14130036
COC1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130038
CC1CCC(C)N1C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130046
C=CCCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130048
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CCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14130066
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CC1CCCCC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130076
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CN(C)c1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14130100
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COCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__14130108
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CC1CCC(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14130116
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CC(C)OCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130132
NC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130134
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14130138
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14130144
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Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C1CC1 s275592__15865378__15842482__14130150
NC(=O)N1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130162
CC(C)CC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130170
Cc1cccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130176
Cc1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133250
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15842482__14133268
O=C(NCC(F)=C1CN(C(=O)c2cccc3[nH]ncc23)C1)c1nsnc1O s275592__15865378__15842482__14133272
O=C(NCC(F)=C1CN(C(=O)c2cccc3cn[nH]c23)C1)c1nsnc1O s275592__15865378__15842482__14133282
Cc1n[nH]c(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14133286
O=C(NCC(F)=C1CN(C(=O)c2cnn3cccnc23)C1)c1nsnc1O s275592__15865378__15842482__14133294
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__14133296
Cc1n[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133302
COc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133304
Cc1cc(F)cc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133306
COc1csc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133314
CN1C(=O)CCC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133316
O=C(NCC(F)=C1CN(C(=O)CCc2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__14133320
O=C(NCC(F)=C1CN(C(=O)c2ccn3nnnc3c2)C1)c1nsnc1O s275592__15865378__15842482__14133326
COc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133328
CCCC(OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133336
C=C(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133340
Cc1ccn(C(C)CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14133344
O=C1CN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCN1 s275592__15865378__15842482__14133348
CCCCCCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133358
CC(CC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133366
NC(=O)C1CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133368
O=C(NCC(F)=C1CN(C(=O)C2CCNC2=O)C1)c1nsnc1O s275592__15865378__15842482__14133374
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]c1=O s275592__15865378__15842482__14133376
CN1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)NC1=O s275592__15865378__15842482__14133378
C=CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133380
C#CCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133382
CN1CCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133386
C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133388
O=C(NCC(F)=C1CN(C(=O)CC2CC=CCC2)C1)c1nsnc1O s275592__15865378__15842482__14133390
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14133392
CCC(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133394
O=C(NCC(F)=C1CN(C(=O)CCCF)C1)c1nsnc1O s275592__15865378__15842482__14133398
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(F)(F)F s275592__15865378__15842482__14133400
Cc1cocc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133402
C[C@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133404
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C=CCC1 s275592__15865378__15842482__14133406
CN1C(=O)CC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133410
Cn1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14133412
CC1(C)CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133414
O=C(NCC(F)=C1CN(C(=O)c2ccn3c2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14134876
O=C(NCC(F)=C1CN(C(=O)COCC2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14134878
O=C(NCC(F)=C1CN(C(=O)c2cnc(C3CC3)o2)C1)c1nsnc1O s275592__15865378__15842482__14134890
O=C1NC(=O)[C@H](CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__14134892
COCc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14134898
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCC3)C1)c1nsnc1O s275592__15865378__15842482__14134900
C#CCN1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134902
Cc1ccncc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134906
C[C@@H]1OCCO[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134914
Cn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1=O s275592__15865378__15842482__14134916
CCc1cnc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__14134918
CN1CCCC1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134932
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCNC1=O s275592__15865378__15842482__14134940
CC[C@@H]1CCO[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134946
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2c[nH]cn2)C1)c1nsnc1O s275592__15865378__15842482__14134954
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCOC3)C1)c1nsnc1O s275592__15865378__15842482__14134958
O=C(NCC(F)=C1CN(C(=O)C2CCC=CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14134964
Cc1cn(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14134968
O=C(NCC(F)=C1CN(C(=O)C23CCCN(CCC2)C3)C1)c1nsnc1O s275592__15865378__15842482__14134972
COc1ccncc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14134980
CC1C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1C1CC1 s275592__15865378__15842482__14134986
O=C(NCC(F)=C1CN(C(=O)C2CCC3CCCCN32)C1)c1nsnc1O s275592__15865378__15842482__14134990
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccncc1 s275592__15865378__15842482__14134994
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCNC(=O)C1 s275592__15865378__15842482__14134998
O=C(NCC(F)=C1CN(C(=O)C2CCCC23CC3)C1)c1nsnc1O s275592__15865378__15842482__14135000
O=C(NCC(F)=C1CN(C(=O)COCC2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__14130200
CC(NC(=O)C1CCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130204
CC(=O)N[C@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15842482__14130212
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1C s275592__15865378__15842482__14130216
CCOc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14130220
CCn1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__14130222
O=C(NCC(F)=C1CN(C(=O)CCc2cncc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__14130226
Cn1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__14130228
COCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14130230
Cc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14130232
CC(C)CC(C(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130234
COC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14130240
CC1(C)C(C)(C)C1(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130242
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__14130244
CC1(C)CCCCC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130256
Cc1[nH]cnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130258
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCOCC1 s275592__15865378__15842482__14130264
O=C(NCC(F)=C1CN(C(=O)C2CC23CCOCC3)C1)c1nsnc1O s275592__15865378__15842482__14130274
CC1(C)CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__14130276
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCOCC1 s275592__15865378__15842482__14130278
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C(=O)N1 s275592__15865378__15842482__14130282
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1C(C)C s275592__15865378__15842482__14130284
CC1(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(=O)N1 s275592__15865378__15842482__14130294
CCOc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130296
O=C(NCC(F)=C1CN(C(=O)c2cc3n(c2)CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14130300
NC(=O)c1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14130302
CC(C)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__14130306
CCC(CC)C(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130310
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC2CCC1C2 s275592__15865378__15842482__14130314
COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCCCC1 s275592__15865378__15842482__14130324
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842482__14130342
CC(=O)NCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130350
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C(C)(C)C s275592__15865378__15842482__14130352
CC(Cc1ccco1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14130354
CC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133416
Cc1cnn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133420
CC(C)C(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133422
CCCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14133424
C=CC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133426
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__14133428
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCC3)C2)C1)c1nsnc1O s275592__15865378__15842482__14133430
CC#CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133432
O=C(NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3COC[C@H]32)C1)c1nsnc1O s275592__15865378__15842482__14133434
O=C(NCC(F)=C1CN(C(=O)CCCC2CC2)C1)c1nsnc1O s275592__15865378__15842482__14133436
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1=O s275592__15865378__15842482__14133438
CCCC(OCC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133440
CC1(C)CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133442
Cc1coc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14133444
O=C(NCC(F)=C1CN(C(=O)c2csc(=O)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__14133446
C=CC(CC)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133450
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__14133452
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3C[C@@H]3C2)C1)c1nsnc1O s275592__15865378__15842482__14133454
CCCc1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133460
CC(C)c1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133462
Cc1nc[nH]c(=O)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133464
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(=O)NC1 s275592__15865378__15842482__14133466
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1C(C)C s275592__15865378__15842482__14133470
CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14133476
CCCN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133480
O=C(NCC(F)=C1CN(C(=O)C2(c3cccnc3)CC2)C1)c1nsnc1O s275592__15865378__15842482__14133482
CCOC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133484
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)s1 s275592__15865378__15842482__14133488
O=C(NCC(F)=C1CN(C(=O)Cc2cnoc2)C1)c1nsnc1O s275592__15865378__15842482__14133490
CN1C(=O)CC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133492
CC1(C)CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133496
CC(C)c1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133502
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14133508
CC(C)N1C(=O)CC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14133512
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CCC2)C1)c1nsnc1O s275592__15865378__15842482__14133516
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CCCC2)C1)c1nsnc1O s275592__15865378__15842482__14133518
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cncnc1 s275592__15865378__15842482__14133520
Cc1cc(C2(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)CC2)on1 s275592__15865378__15842482__14133530
CC(C)N1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__14133534
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(=O)[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__14133536
O=C(NCC(F)=C1CN(C(=O)C2(F)CCOC2)C1)c1nsnc1O s275592__15865378__15842482__14133542
COc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__14133544
O=C(NCC(F)=C1CN(C(=O)c2nc(Cl)cs2)C1)c1nsnc1O s275592__15865378__15842482__14133546
O=C(NCC(F)=C1CN(C(=O)CC2CCCC2(F)F)C1)c1nsnc1O s275592__15865378__15842482__14133548
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1C s275592__15865378__15842482__14133554
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cn2)C1)c1nsnc1O s275592__15865378__15842482__14133564
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccc(F)cc32)C1)c1nsnc1O s275592__15865378__15842482__14133568
O=C(NCC(F)=C1CN(C(=O)c2ccoc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__14133578
O=C(NCC(F)=C1CN(C(=O)c2coc(C(F)F)c2)C1)c1nsnc1O s275592__15865378__15842482__14133580
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccsc2)C1)c1nsnc1O s275592__15865378__15842482__14135026
COc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__14135032
O=C(NCC(F)=C1CN(C(=O)c2cn3c(n2)COCC3)C1)c1nsnc1O s275592__15865378__15842482__14135036
COCc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135042
CCC1CCCC1(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135044
O=C(NCC(F)=C1CN(C(=O)c2cc3cnccc3[nH]2)C1)c1nsnc1O s275592__15865378__15842482__14135046
Cc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)s1 s275592__15865378__15842482__14135052
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15842482__14135056
O=C(NCC(F)=C1CN(C(=O)C23CCC(CC2)C3)C1)c1nsnc1O s275592__15865378__15842482__14135064
CN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135066
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1Cl s275592__15865378__15842482__14135068
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__14135072
O=C(NCC(F)=C1CN(C(=O)C2(C(F)(F)F)CCC2)C1)c1nsnc1O s275592__15865378__15842482__14135076
O=C(NCC(F)=C1CN(C(=O)c2ncc(F)cc2F)C1)c1nsnc1O s275592__15865378__15842482__14135078
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)S(C)(=O)=O s275592__15865378__15842482__14135080
CS(=O)(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135082
O=C(NCC(F)=C1CN(C(=O)Cc2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__14135094
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__14135100
NC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__14135102
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1=O s275592__15865378__15842482__14135104
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1=O s275592__15865378__15842482__14135110
CC(F)(F)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135120
O=C(NCC(F)=C1CN(C(=O)COC2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__14135126
O=C(NCC(F)=C1CN(C(=O)CCOCC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__14135128
O=C(NCC(F)=C1CN(C(=O)CCc2ccncc2)C1)c1nsnc1O s275592__15865378__15842482__14135138
CC(C)(C)n1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14135140
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CN1 s275592__15865378__15842482__14135142
CC(C)CN1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135146
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842482__14135148
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__14135150
CCCc1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135154
CCc1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135156
CC(C)c1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__14135158
CC(C)(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15842482__14135160
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2CCC3)C1)c1nsnc1O s275592__15865378__15842482__14135164
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__14135168
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nn2)C1)c1nsnc1O s275592__15865378__15842482__14135174
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1C s275592__15865378__15842482__15278136
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1 s275592__15865378__15842482__15585620
Cc1sc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__15855922
O=C(NCC(F)=C1CN(C(=O)CN2CCC(CO)CC2)C1)c1nsnc1O s275592__15865378__15842482__15855930
O=C(NCC(F)=C1CN(C(=O)c2ccccc2O)C1)c1nsnc1O s275592__15865378__15842482__15855932
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1Cl s275592__15865378__15842482__15855944
O=C(NCC(F)=C1CN(C(=O)CSc2ccncc2)C1)c1nsnc1O s275592__15865378__15842482__15855950
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1O s275592__15865378__15842482__15855954
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]cnc3c2)C1)c1nsnc1O s275592__15865378__15842482__15855960
O=C(NCC(F)=C1CN(C(=O)C2CSCCS2)C1)c1nsnc1O s275592__15865378__15842482__15855966
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)ccn2)C1)c1nsnc1O s275592__15865378__15842482__15855968
O=C(NCC(F)=C1CN(C(=O)CO)C1)c1nsnc1O s275592__15865378__15842482__15855972
O=C(NCC(F)=C1CN(C(=O)c2cccc(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15855974
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)ccc2O)C1)c1nsnc1O s275592__15865378__15842482__15855976
CCOC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855978
O=C(NCC(F)=C1CN(C(=O)COc2ccccc2O)C1)c1nsnc1O s275592__15865378__15842482__15855980
CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__15855984
NC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855986
Nc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855988
Nc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__15855990
O=C(NCC(F)=C1CN(C(=O)c2ccc[n+]([O-])c2)C1)c1nsnc1O s275592__15865378__15842482__15855992
CNc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855994
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1N s275592__15865378__15842482__15855996
COC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856004
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ncn2)C1)c1nsnc1O s275592__15865378__15842482__15856006
C#CCSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856008
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2NCC3)C1)c1nsnc1O s275592__15865378__15842482__15857750
CSC=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857758
O=C(NCC(F)=C1CN(C(=O)c2cnccc2O)C1)c1nsnc1O s275592__15865378__15842482__15857774
CC1=NC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CS1 s275592__15865378__15842482__15857776
O=C(NCC(F)=C1CN(C(=O)C(=O)C(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15857778
CCC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15857780
Cc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1Cl s275592__15865378__15842482__15857782
O=C(NCC(F)=C1CN(C(=O)C2(CO)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15857784
Cc1ccc(C#N)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857788
Nc1ccn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15857790
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnc1N s275592__15865378__15842482__15857794
N#Cc1cc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857796
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2O)C1)c1nsnc1O s275592__15865378__15842482__15857798
Cn1ccnc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857800
CC(C)(CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)[N+](=O)[O-] s275592__15865378__15842482__15857802
CN1C(=O)CSC1=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857804
COC1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15857810
CC1C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCN1C s275592__15865378__15842482__15857814
O=C(NCC(F)=C1CN(C(=O)c2cncc(O)n2)C1)c1nsnc1O s275592__15865378__15842482__15857816
CN1CCCCC1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857822
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)s2)C1)c1nsnc1O s275592__15865378__15842482__15857824
CCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15857826
NC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857828
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15857832
O=C(NCC(F)=C1CN(C(=O)COC(F)F)C1)c1nsnc1O s275592__15865378__15842482__15857834
Cc1c(C#N)cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857844
Cc1nc(=O)[nH]c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857850
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(=O)N1 s275592__15865378__15842482__15857868
Cc1csc(NCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15859740
O=C(NCC(F)=C1CN(C(=O)CSCc2ncc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15859744
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCSCC1 s275592__15865378__15842482__15859748
O=C(NCC(F)=C1CN(C(=O)C2=CCCS2)C1)c1nsnc1O s275592__15865378__15842482__15859750
CC1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859752
O=C(NC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859754
O=C(NCC(F)=C1CN(C(=O)c2ncc(Cl)cn2)C1)c1nsnc1O s275592__15865378__15842482__15859760
CCC1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859762
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccoc3c2)C1)c1nsnc1O s275592__15865378__15842482__15859766
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15842482__15859768
Cc1noc(COCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15859772
O=C(NCC(F)=C1CN(C(=O)C2CCSC2)C1)c1nsnc1O s275592__15865378__15842482__15859774
O=C(NCC(F)=C1CN(C(=O)C2CCO2)C1)c1nsnc1O s275592__15865378__15842482__15859778
CCNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15859784
O=C(NCC(F)=C1CN(C(=O)C=CC2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15859790
CCCC(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859794
Cn1ncc([N+](=O)[O-])c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859798
CC(C)(CC#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859806
O=C(NCC(F)=C1CN(C(=O)C2(Cl)CC2)C1)c1nsnc1O s275592__15865378__15842482__15859808
O=C(NCC(F)=C1CN(C(=O)C2=CCCO2)C1)c1nsnc1O s275592__15865378__15842482__15859810
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)o2)C1)c1nsnc1O s275592__15865378__15842482__15859816
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1O s275592__15865378__15842482__15859822
COc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15859828
O=C(NCC(F)=C1CN(C(=O)C2(CO)COC2)C1)c1nsnc1O s275592__15865378__15842482__15859830
CC1CC(C#N)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859834
CC(C)=CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859836
CC=C(C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CC s275592__15865378__15842482__15859838
O=C(NCC(F)=C1CN(C(=O)C2COC2)C1)c1nsnc1O s275592__15865378__15842482__15859842
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(N)n1 s275592__15865378__15842482__15859846
O=C(NCC(F)=C1CN(C(=O)C=CC2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15859850
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)c(F)c2)C1)c1nsnc1O s275592__15865378__15842482__15859852
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859854
O=C(NCC(F)=C1CN(C(=O)C23CCC(F)(CC2)CC3)C1)c1nsnc1O s275592__15865378__15842482__15859856
N#CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15859858
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(C3CC3)n2)C1)c1nsnc1O s275592__15865378__15842482__15859860
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15859862
CNc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15859864
Cc1nccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861706
O=C(NCC(F)=C1CN(C(=O)c2cnc(F)c(F)c2)C1)c1nsnc1O s275592__15865378__15842482__15861708
O=C(NCC(F)=C1CN(C(=O)c2ccnc(F)c2F)C1)c1nsnc1O s275592__15865378__15842482__15861710
O=C(NCC(F)=C1CN(C(=O)[C@H](O)c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15861712
Nc1c[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861720
O=C(NCC(F)=C1CN(C(=O)COc2ccc(O)cc2)C1)c1nsnc1O s275592__15865378__15842482__15861736
CC1(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__15861738
O=C(NCC(F)=C1CN(C(=O)C2CCOC3(CCC3)C2)C1)c1nsnc1O s275592__15865378__15842482__15861746
CC(C)(C)OC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861748
O=C(NCC(F)=C1CN(C(=O)c2cc([N+](=O)[O-])[nH]n2)C1)c1nsnc1O s275592__15865378__15842482__15861750
O=C(NCC(F)=C1CN(C(=O)C=CCO)C1)c1nsnc1O s275592__15865378__15842482__15861754
CCC(O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861758
O=C(NCC(F)=C1CN(C(=O)C2CCCc3ncnn32)C1)c1nsnc1O s275592__15865378__15842482__15861762
O=C(NCC(F)=C1CN(C(=O)C2(CO)CCCO2)C1)c1nsnc1O s275592__15865378__15842482__15861764
COc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15861782
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)c1=O s275592__15865378__15842482__15861786
CC(C)(C)c1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__15861796
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15861798
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(F)(F)C1 s275592__15865378__15842482__15861802
CCc1c[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861804
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCC[C@H]2CF)C1)c1nsnc1O s275592__15865378__15842482__15861806
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CCC3)on2)C1)c1nsnc1O s275592__15865378__15842482__15861810
CC(C)[C@@H](O)[C@@H](C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861816
O=C(NCC(F)=C1CN(C(=O)C2(F)C3CCCCC32)C1)c1nsnc1O s275592__15865378__15842482__15861818
O=C(NCC(F)=C1CN(C(=O)c2onc3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__15861820
CC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(CC1)CO2 s275592__15865378__15842482__15861822
CCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]1 s275592__15865378__15842482__15861824
CC(C)(Cc1cnn[nH]1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863542
O=C(NCC(F)=C1CN(C(=O)C2(C(=O)C3CC3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15863548
O=CN1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863550
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__15863554
CC(C)(C)N1CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863556
O=C(NCC(F)=C1CN(C(=O)CCC2CC2(F)F)C1)c1nsnc1O s275592__15865378__15842482__15863560
O=C(NCC(F)=C1CN(C(=O)CCCC(=O)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15863562
Cc1c(F)ccc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863566
Nc1ccn(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15863568
Cc1nnc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15863572
Cc1cnnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15863576
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__15863578
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cccc1 s275592__15865378__15842482__15863580
CSCC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15863582
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__15863584
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]2C(F)F)C1)c1nsnc1O s275592__15865378__15842482__15863586
CCn1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnc1O s275592__15865378__15842482__15863594
O=C(NCC(F)=C1CN(C(=O)c2coc(=O)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15863596
CC=CC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863598
O=C(NCC(F)=C1CN(C(=O)c2cc3cccnc3[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15863602
CCCC[C@H](C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863606
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1F s275592__15865378__15842482__15863610
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__15863612
CCC=C(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863618
O=C(NCC(F)=C1CN(C(=O)C2C3(CC3)C23CC3)C1)c1nsnc1O s275592__15865378__15842482__15863620
CCC=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863622
Cn1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15863624
CCC(F)(F)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863628
Cc1nocc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863636
O=C(NCC(F)=C1CN(C(=O)Cc2csnn2)C1)c1nsnc1O s275592__15865378__15842482__15863642
CC(=Cc1cccnc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863644
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__15863656
COCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__15863658
O=C1N[C@@H](CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__15863662
CC(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864230
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnc1C#N s275592__15865378__15842482__15864234
C=CCC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__15864238
CC1CCOC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864240
O=C(NCC(F)=C1CN(C(=O)C2=C(Cl)CCOC2)C1)c1nsnc1O s275592__15865378__15842482__15864244
Nc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15856020
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CN1 s275592__15865378__15842482__15856024
CC1CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15856026
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C(=O)OC1(C)C s275592__15865378__15842482__15856034
CCCCSC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856038
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1N s275592__15865378__15842482__15856044
CC(=O)CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856046
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3N2)C1)c1nsnc1O s275592__15865378__15842482__15856050
Nc1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856052
CCc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856058
Nc1nonc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856062
O=C(NCC(F)=C1CN(C(=O)c2cn(CCO)nn2)C1)c1nsnc1O s275592__15865378__15842482__15856064
O=C(NCC(F)=C1CN(C(=O)COC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15856066
O=C1NC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__15856072
O=C(NCC(F)=C1CN(C(=O)c2cncs2)C1)c1nsnc1O s275592__15865378__15842482__15856078
Nc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15856084
Cc1nn(CCO)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856096
O=C(NCC(F)=C1CN(C(=O)CCN2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15856100
CCCC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856102
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1C#N s275592__15865378__15842482__15856104
Cc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15856106
O=C(NCC(F)=C1CN(C(=O)c2c(O)cc(O)cc2O)C1)c1nsnc1O s275592__15865378__15842482__15856108
[N-]=[N+]=NCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856110
O=C(NCC(F)=C1CN(C(=O)Cn2cc(CO)nn2)C1)c1nsnc1O s275592__15865378__15842482__15856114
C#CCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856116
O=C(NCC(F)=C1CN(C(=O)Cc2nnco2)C1)c1nsnc1O s275592__15865378__15842482__15856118
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)SCCO1 s275592__15865378__15842482__15856120
CN(CCO)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856124
O=C(NCC(F)=C1CN(C(=O)c2cnc(Cl)cn2)C1)c1nsnc1O s275592__15865378__15842482__15856126
O=C(NCC(F)=C1CN(C(=O)C2CCCS2)C1)c1nsnc1O s275592__15865378__15842482__15856128
COC(=O)CC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856132
COC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857874
Cc1cc(F)c(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857880
O=C(NCC(F)=C1CN(C(=O)CC2CCCC(O)C2)C1)c1nsnc1O s275592__15865378__15842482__15857884
CC(O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857888
CC1(C)CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__15857894
Cn1cccc1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857900
CCS(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857902
CC(=O)c1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857906
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)cc2)C1)c1nsnc1O s275592__15865378__15842482__15857910
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1[N+](=O)[O-] s275592__15865378__15842482__15857912
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__15857914
O=C(NCC(F)=C1CN(C(=O)CNC(=O)C(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15857916
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1O s275592__15865378__15842482__15857932
O=C(NCC(F)=C1CN(C(=O)COCC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15857934
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(Cl)n1 s275592__15865378__15842482__15857936
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1F s275592__15865378__15842482__15857938
NC(=O)CSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857940
CCCCSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857942
Nc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857944
Cc1ccc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15857946
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__15857952
CC(C)CSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857954
CC(=O)N1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857958
O=C(NCC(F)=C1CN(C(=O)c2cc(=O)[nH]c(=O)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15857960
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccnc2F)C1)c1nsnc1O s275592__15865378__15842482__15857964
O=C(NCC(F)=C1CN(C(=O)C2CN3CCCN2CC3)C1)c1nsnc1O s275592__15865378__15842482__15857974
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1O s275592__15865378__15842482__15857980
O=C(NCC(F)=C1CN(C(=O)Cn2cccc2)C1)c1nsnc1O s275592__15865378__15842482__15857988
O=C(NCC(F)=C1CN(C(=O)C2CCCCS2)C1)c1nsnc1O s275592__15865378__15842482__15859866
O=C(NCC(F)=C1CN(C(=O)C2SCCS2)C1)c1nsnc1O s275592__15865378__15842482__15859868
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842482__15859870
CC1=NOC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859874
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)cc2F)C1)c1nsnc1O s275592__15865378__15842482__15859884
O=C(NCC(F)=C1CN(C(=O)c2ccn(CO)n2)C1)c1nsnc1O s275592__15865378__15842482__15859886
O=C(NCC(F)=C1CN(C(=O)c2cccc3ncoc23)C1)c1nsnc1O s275592__15865378__15842482__15859896
C#CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859904
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1Cl s275592__15865378__15842482__15859912
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1CO s275592__15865378__15842482__15859914
O=C(NCC(F)=C1CN(C(=O)c2cc(O)cc(=O)o2)C1)c1nsnc1O s275592__15865378__15842482__15859916
Nc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1N s275592__15865378__15842482__15859924
Cc1c(F)ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15859932
COc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859934
O=C(NCC(F)=C1CN(C(=O)C(O)CC2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15859936
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2C(F)F)C1)c1nsnc1O s275592__15865378__15842482__15859938
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N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC12CCC2 s275592__15865378__15842482__15861850
CNc1c(N)cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861852
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COc1cnnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861870
CC(Cn1ccnc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861876
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ncn2)C1)c1nsnc1O s275592__15865378__15842482__15861886
CCCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15861890
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1F s275592__15865378__15842482__15861896
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)cn2)C1)c1nsnc1O s275592__15865378__15842482__15861904
CN1CC=C(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15861906
CC[C@H](C)[C@H](O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861908
Cc1ncn(C)c(=O)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861912
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15842482__15861914
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)COC1 s275592__15865378__15842482__15861920
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(F)nc2)C1)c1nsnc1O s275592__15865378__15842482__15861926
CC(C)CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__15861928
O=C(NCC(F)=C1CN(C(=O)CCC(O)C(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15861930
Cn1cnc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861936
O=C(NCC(F)=C1CN(C(=O)Cc2n[nH]c(C3CC3)n2)C1)c1nsnc1O s275592__15865378__15842482__15861940
CC1(C)CC1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861942
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__15861944
O=C(NCC(F)=C1CN(C(=O)C2CCS2(=O)=O)C1)c1nsnc1O s275592__15865378__15842482__15861946
O=C(NCC(F)=C1CN(C(=O)c2cc3nc[nH]c3cn2)C1)c1nsnc1O s275592__15865378__15842482__15864246
C[S+](C)CCC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864248
N#CC1CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864250
CC(C)(C)C(O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864254
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15864260
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)F)on2)C1)c1nsnc1O s275592__15865378__15842482__15864262
O=C(NCC(F)=C1CN(C(=O)C(O)c2c[nH]cn2)C1)c1nsnc1O s275592__15865378__15842482__15864266
O=C(NCC(F)=C1CN(C(=O)C=CC=C(Cl)Cl)C1)c1nsnc1O s275592__15865378__15842482__15864272
CCC(C)(C)C(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864274
CCC(C)(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864276
Nc1ncc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864278
CC(=O)N1CC2CC2(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864282
O=C(NCC(F)=C1CN(C(=O)CC2CCC3(CCC3)O2)C1)c1nsnc1O s275592__15865378__15842482__15864286
O=C(NCC(F)=C1CN(C(=O)c2[nH]cc3c2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__15864290
O=C(NCC(F)=C1CN(C(=O)c2ccnn2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15864292
Nc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15864294
C#CC1CC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15864296
CSc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15864306
CC=CC=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864312
CN1CC(O)CC1(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864316
COCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15864318
C[C@@H]1[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[C@@H](O)C(=O)N1C s275592__15865378__15842482__15864324
Cn1ncnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864328
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@@H](O)C2)C1)c1nsnc1O s275592__15865378__15842482__15864330
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CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C(C)(C)O1 s275592__15865378__15842482__15864340
Cn1c(Cl)cnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864342
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC=CCC2)C1)c1nsnc1O s275592__15865378__15842482__15864344
COCC=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864348
CN1CCN(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864354
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCCC(O)C1 s275592__15865378__15842482__15864356
O=C(NCC(F)=C1CN(C(=O)c2cccc3nonc23)C1)c1nsnc1O s275592__15865378__15842482__15864358
O=C(NCC(F)=C1CN(C(=O)CCOC2COC2)C1)c1nsnc1O s275592__15865378__15842482__15864360
[N-]=[N+]=N[C@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864362
CC(=O)C(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864364
Cc1ccc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856136
COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__15856138
O=C(NCC(F)=C1CN(C(=O)C2CC3CC3C2)C1)c1nsnc1O s275592__15865378__15842482__15856140
O=C(NCC(F)=C1CN(C(=O)Cc2cncnc2)C1)c1nsnc1O s275592__15865378__15842482__15856158
Cc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15856160
O=C(NCC(F)=C1CN(C(=O)CCc2nc(=O)[nH][nH]2)C1)c1nsnc1O s275592__15865378__15842482__15856168
O=C1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15856170
O=C(NCC(F)=C1CN(C(=O)C2C3CCC(=O)C32)C1)c1nsnc1O s275592__15865378__15842482__15856176
COC(=O)C12CC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(C1)C2 s275592__15865378__15842482__15856182
Cc1ccncc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856186
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)[nH]c2=O)C1)c1nsnc1O s275592__15865378__15842482__15856188
CNc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15856190
CS(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856194
O=C(NCC(F)=C1CN(C(=O)C(=O)C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15856196
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)n1 s275592__15865378__15842482__15856198
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cnn(C)c1 s275592__15865378__15842482__15856202
Nc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1F s275592__15865378__15842482__15856208
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1F s275592__15865378__15842482__15856210
O=NN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856224
O=C(NCC(F)=C1CN(C(=O)C=C(Cl)Cl)C1)c1nsnc1O s275592__15865378__15842482__15856226
CSc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15856230
O=C(NCC(F)=C1CN(C(=O)c2cnncc2O)C1)c1nsnc1O s275592__15865378__15842482__15856232
CN1CCCC(O)(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15856236
Cc1[nH]c(C#N)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856238
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__15856240
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(C)(C)C1 s275592__15865378__15842482__15856244
CC1CN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15856250
CCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857998
COc1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858000
Cc1cccc(O)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858002
O=C(NCC(F)=C1CN(C(=O)c2cccc(F)c2O)C1)c1nsnc1O s275592__15865378__15842482__15858004
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15858006
CCN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15858008
CC1CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15858032
CC(OC1CCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858036
CN(C)C(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858038
C#CCC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858040
O=C(NCC(F)=C1CN(C(=O)c2cncc(Cl)c2O)C1)c1nsnc1O s275592__15865378__15842482__15858042
Nc1ncccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858044
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC12CCCC2 s275592__15865378__15842482__15858046
O=C(NCC(F)=C1CN(C(=O)c2cc(O)cc(Cl)c2)C1)c1nsnc1O s275592__15865378__15842482__15858052
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15858058
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15858064
C=CC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858068
[N-]=[N+]=NCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858070
Cc1ccc(C)n1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858072
Cc1cccnc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858074
CC(O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858076
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CC1(C)COC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858080
CSCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858082
Cc1c(N)ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__15858084
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(Cl)cn2)C1)c1nsnc1O s275592__15865378__15842482__15858086
COC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__15858088
Cn1nncc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858092
O=C(NCC(F)=C1CN(C(=O)Cc2cnccc2O)C1)c1nsnc1O s275592__15865378__15842482__15858096
O=C(NCC(F)=C1CN(C(=O)CCCc2cncs2)C1)c1nsnc1O s275592__15865378__15842482__15858098
[N-]=[N+]=Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15858100
[N-]=[N+]=Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15858102
[N-]=[N+]=Nc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858104
COC(=O)COCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858110
O=C(NCC(F)=C1CN(C(=O)CC2CCCCC2F)C1)c1nsnc1O s275592__15865378__15842482__15858112
N#Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15858114
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCO1 s275592__15865378__15842482__15859990
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCOC3)C1)c1nsnc1O s275592__15865378__15842482__15859998
CCC(CC)(CO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860000
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15860002
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)cc2)C1)c1nsnc1O s275592__15865378__15842482__15860004
CSc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860006
Cc1ccc(NCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15860008
O=C(NCC(F)=C1CN(C(=O)C2CCC3CC3CC2)C1)c1nsnc1O s275592__15865378__15842482__15860022
O=C(NCC(F)=C1CN(C(=O)c2cccn3ncnc23)C1)c1nsnc1O s275592__15865378__15842482__15860024
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__15860026
CC1(CCCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N=N1 s275592__15865378__15842482__15860034
Nc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15860038
O=C(NCC(F)=C1CN(C(=O)C23CCC2C3)C1)c1nsnc1O s275592__15865378__15842482__15860044
CCCC(C)=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860050
O=C(NCC(F)=C1CN(C(=O)c2nc(C3CC3)cs2)C1)c1nsnc1O s275592__15865378__15842482__15860056
O=C(NCC(F)=C1CN(C(=O)C(=O)C2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15860058
C=C[C@H](C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860060
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CCC3)[nH]n2)C1)c1nsnc1O s275592__15865378__15842482__15860064
CS(=O)(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860076
O=C(NCC(F)=C1CN(C(=O)c2ccn3nccc3n2)C1)c1nsnc1O s275592__15865378__15842482__15860082
O=C(NCC(F)=C1CN(C(=O)C=CCN2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15860084
Cn1cc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15860088
O=C(NCC(F)=C1CN(C(=O)C=CC2CC2)C1)c1nsnc1O s275592__15865378__15842482__15860092
O=C(NCC(F)=C1CN(C(=O)C23CCC(CC2)O3)C1)c1nsnc1O s275592__15865378__15842482__15860096
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ncncc23)C1)c1nsnc1O s275592__15865378__15842482__15860100
O=C(NCC(F)=C1CN(C(=O)CCc2cccc(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15860102
N#Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15860110
O=C(NCC(F)=C1CN(C(=O)C=CC2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__15861948
O=C(NCC(F)=C1CN(C(=O)C#CC2CCCCO2)C1)c1nsnc1O s275592__15865378__15842482__15861950
Cc1oncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861960
CC(C)CC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861966
O=C(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861968
CCC(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861972
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2O)C1)c1nsnc1O s275592__15865378__15842482__15861974
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15861976
O=C(NCC(F)=C1CN(C(=O)CCNc2nccs2)C1)c1nsnc1O s275592__15865378__15842482__15861980
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15861986
CC1CC1(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861988
O=C(NCC(F)=C1CN(C(=O)C2CCN(C3CC3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15861992
CCC(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861996
O=C(NCC(F)=C1CN(C(=O)C2(CO)CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15861998
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)S(N)(=O)=O s275592__15865378__15842482__15862000
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15862002
NS(=O)(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15862012
O=C(NCC(F)=C1CN(C(=O)c2coc(CO)c2)C1)c1nsnc1O s275592__15865378__15842482__15862014
CC(C)[C@H]1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15862018
O=C1NC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15862020
Cn1cc(NCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15862022
Cc1onc(CO)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862026
COCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862028
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3C2)C1)c1nsnc1O s275592__15865378__15842482__15862030
COc1nscc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862032
O=C(NCC(F)=C1CN(C(=O)c2cccc(O)c2F)C1)c1nsnc1O s275592__15865378__15842482__15862040
CCOCCOCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862046
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCC[C@H]2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15862050
O=C(NCC(F)=C1CN(C(=O)c2cccnc2CO)C1)c1nsnc1O s275592__15865378__15842482__15862054
CC1(C)CC2(CC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)C2)C1 s275592__15865378__15842482__15862056
C=CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15862060
Cn1ccc(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15862066
O=C(NCC(F)=C1CN(C(=O)C2(n3ccnn3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15862070
[N-]=[N+]=NC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864374
O=C(NCC(F)=C1CN(C(=O)C23CCC(CO2)C3)C1)c1nsnc1O s275592__15865378__15842482__15864376
O=C(NCC(F)=C1CN(C(=O)C2C3CCC32)C1)c1nsnc1O s275592__15865378__15842482__15864378
CC1(C)CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15864382
COC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1C s275592__15865378__15842482__15864384
CC(C)(C)C(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864386
C=C1CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864388
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@H]3CC[C@H]2O3)C1)c1nsnc1O s275592__15865378__15842482__15864390
C[C@@H]1C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[C@@H]1C s275592__15865378__15842482__15864392
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15842482__15864394
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CCC3)OC2)C1)c1nsnc1O s275592__15865378__15842482__15864398
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(F)c2O)C1)c1nsnc1O s275592__15865378__15842482__15864400
Cc1nnn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15864412
CC(C)n1cncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864416
Cc1nnc2n1C(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)CC2 s275592__15865378__15842482__15864422
CCN(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864424
Nc1cc(O)nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15864426
O=C(NCC(F)=C1CN(C(=O)c2cccn3cnnc23)C1)c1nsnc1O s275592__15865378__15842482__15864432
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC2C=CC1C2 s275592__15865378__15842482__15864434
COC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1(C)C s275592__15865378__15842482__15864436
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1nc[nH]n1 s275592__15865378__15842482__15864442
O=C(NCC(F)=C1CN(C(=O)c2[nH]ncc2C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15864448
O=C(NCC(F)=C1CN(C(=O)C2CCC3C2C3(F)F)C1)c1nsnc1O s275592__15865378__15842482__15864450
O=C(NCC(F)=C1CN(C(=O)C(F)OC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15864456
C=C1CC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15864458
O=C(NCC(F)=C1CN(C(=O)C2=Cc3ccccc3C2)C1)c1nsnc1O s275592__15865378__15842482__15864472
COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccnc1 s275592__15865378__15842482__15864474
CCC1(C#CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)COC1 s275592__15865378__15842482__15864476
COc1ccc(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864478
O=C(NCC(F)=C1CN(C(=O)C2=C[C@@H]3CCCC[C@H]23)C1)c1nsnc1O s275592__15865378__15842482__15864482
CC1(C)CC1(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864484
CC(C)c1c[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864486
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)N=N3)C1)c1nsnc1O s275592__15865378__15842482__15856264
O=C(NCC(F)=C1CN(C(=O)Cc2cncc(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15856274
NC(=O)CCNC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856276
Nc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15856282
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1C(F)(F)F s275592__15865378__15842482__15856286
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)sn1 s275592__15865378__15842482__15856288
CC1(C)C(=O)CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856290
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__15856292
O=C(NCC(F)=C1CN(C(=O)c2cccnc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15856296
Nc1cc(N)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856298
CC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)c(O)c(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15856316
O=C(NCC(F)=C1CN(C(=O)C(O)c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15856318
CCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856320
CC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856322
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15856328
Cc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856330
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15856332
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])cc2)C1)c1nsnc1O s275592__15865378__15842482__15856334
COC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856336
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1O s275592__15865378__15842482__15856338
Nc1cc(F)c(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856340
CCCCOC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856348
Nc1n[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856354
CC(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856356
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])s2)C1)c1nsnc1O s275592__15865378__15842482__15856364
CCCn1cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856370
CCOC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856372
O=C(NCC(F)=C1CN(C(=O)CN2CC3C=CC2C3)C1)c1nsnc1O s275592__15865378__15842482__15856374
O=C(NCC(F)=C1CN(C(=O)CSC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15856376
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842482__15856380
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15856382
O=C(NCC(F)=C1CN(C(=O)C2CCCC23OCCO3)C1)c1nsnc1O s275592__15865378__15842482__15858122
CCCCCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858124
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(=O)CC1 s275592__15865378__15842482__15858128
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ncccc1F s275592__15865378__15842482__15858134
CCc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858136
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C#N s275592__15865378__15842482__15858138
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1ccnc1 s275592__15865378__15842482__15858144
O=C(NCC(F)=C1CN(C(=O)CSc2ncn[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15858148
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]c(=O)[nH]c1=O s275592__15865378__15842482__15858150
O=C(NCC(F)=C1CN(C(=O)c2cccnc2O)C1)c1nsnc1O s275592__15865378__15842482__15858152
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15858154
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(Cl)c1 s275592__15865378__15842482__15858160
CC(C)CSCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858164
Nc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858168
Nc1c(F)cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858172
O=C(NCC(F)=C1CN(C(=O)CSC(F)F)C1)c1nsnc1O s275592__15865378__15842482__15858176
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__15858178
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(O)n1 s275592__15865378__15842482__15858180
Cc1noc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858188
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(O)cc2)C1)c1nsnc1O s275592__15865378__15842482__15858196
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15858198
O=C(NCC(F)=C1CN(C(=O)c2cccc[n+]2[O-])C1)c1nsnc1O s275592__15865378__15842482__15858200
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15858204
Cc1ccc(C)n1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858206
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)=NN1 s275592__15865378__15842482__15858220
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__15858222
O=C1CCC(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__15858226
COCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858228
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15858230
CC(=O)c1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15858232
CP(C)(=O)C(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858236
N#CCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858238
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15858240
C=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15858242
CC1(C)CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15858244
CN1N=C(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1=O s275592__15865378__15842482__15858246
CN(C)C(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860112
O=C(NCC(F)=C1CN(C(=O)[C@@]23C[C@@H](O)[C@@H]2C3)C1)c1nsnc1O s275592__15865378__15842482__15860130
COCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__15860132
O=C(Cc1ccsc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860136
CCCOCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860140
O=C(NCC(F)=C1CN(C(=O)C(F)C2(O)CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15860142
CC1(C)COCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860146
C=C1CCC1(C(=O)OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860148
Cn1ccn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)c12 s275592__15865378__15842482__15860152
O=C(NCC(F)=C1CN(C(=O)C=Cc2cnc[nH]c2=O)C1)c1nsnc1O s275592__15865378__15842482__15860154
C=CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__15860156
CC1OC2(CO)CC1(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15860160
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]c1C s275592__15865378__15842482__15860166
CC1CC1c1nocc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860172
N#C[C@]1(O)C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15860176
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15860180
CCCc1ncoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860182
O=C(NCC(F)=C1CN(C(=O)C2CCc3ccnn3C2)C1)c1nsnc1O s275592__15865378__15842482__15860188
O=C(NCC(F)=C1CN(C(=O)CCCCCF)C1)c1nsnc1O s275592__15865378__15842482__15860190
N#CC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15860192
CC1(C)CCCOC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860194
O=C(NCC(F)=C1CN(C(=O)C2CCCCC23CCC3)C1)c1nsnc1O s275592__15865378__15842482__15860196
CC(C)(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)=NO1 s275592__15865378__15842482__15860204
CCC(C)(C)C(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860206
O=C(NCC(F)=C1CN(C(=O)C2(F)CCCOC2)C1)c1nsnc1O s275592__15865378__15842482__15860208
C#CC[C@]1(O)C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15860212
O=C(NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3CCCC(=O)[C@H]32)C1)c1nsnc1O s275592__15865378__15842482__15860214
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CC3F)C1)c1nsnc1O s275592__15865378__15842482__15860216
O=C(NCC(F)=C1CN(C(=O)C2CN3CCN2CC3)C1)c1nsnc1O s275592__15865378__15842482__15860220
O=C(NCC(F)=C1CN(C(=O)C2CCCc3nncn32)C1)c1nsnc1O s275592__15865378__15842482__15860222
C=CCCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860224
CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCOCC1 s275592__15865378__15842482__15860228
O=C(NCC(F)=C1CN(C(=O)C23CC(CO2)C3)C1)c1nsnc1O s275592__15865378__15842482__15860230
O=C(NCC(F)=C1CN(C(=O)C2CCCc3ccnn32)C1)c1nsnc1O s275592__15865378__15842482__15860232
CC12COC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(C1)C2 s275592__15865378__15842482__15862074
O=C(NCC(F)=C1CN(C(=O)c2cc3n(c2)CCOC3)C1)c1nsnc1O s275592__15865378__15842482__15862080
CC(=O)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862082
C#CC1(O)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15862092
C[C@@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(C)(C)C1 s275592__15865378__15842482__15862106
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]c1C s275592__15865378__15842482__15862108
O=C(NCC(F)=C1CN(C(=O)C2CCCc3[nH]cnc32)C1)c1nsnc1O s275592__15865378__15842482__15862116
CC1(C)C(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1(C)C s275592__15865378__15842482__15862118
NC(=O)c1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15862120
CCOC(=O)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862126
O=C(NCC(F)=C1CN(C(=O)CC(O)C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15862132
O=C(NCC(F)=C1CN(C(=O)CCC2CC(F)(F)C2)C1)c1nsnc1O s275592__15865378__15842482__15862140
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCC32)C1)c1nsnc1O s275592__15865378__15842482__15862146
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CCN3)C1)c1nsnc1O s275592__15865378__15842482__15862150
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15862154
CCN1C(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862156
CC1(C)CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15862166
Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15862172
COCc1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862174
O=C(NCC(F)=C1CN(C(=O)c2cc3cn[nH]c3s2)C1)c1nsnc1O s275592__15865378__15842482__15862178
CC1CCSC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862188
O=C1CC2CC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)CC2C1 s275592__15865378__15842482__15862190
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2nc[nH]n2)C1)c1nsnc1O s275592__15865378__15842482__15864490
O=C(NCC(F)=C1CN(C(=O)c2cnoc2C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15864492
CC(C)(F)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864494
COC1CC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15864496
Cc1ncccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864500
O=C(NCC(F)=C1CN(C(=O)C23CCCCN2CCC3)C1)c1nsnc1O s275592__15865378__15842482__15864504
O=C(NCC(F)=C1CN(C(=O)CC2CC(C(F)F)C2)C1)c1nsnc1O s275592__15865378__15842482__15864506
Cc1c(N)cc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864508
O=C(NCC(F)=C1CN(C(=O)c2cncc3[nH]ccc23)C1)c1nsnc1O s275592__15865378__15842482__15864512
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2C[C@H]2C[C@@H]32)C1)c1nsnc1O s275592__15865378__15842482__15864514
Cc1cccc([C@@H](C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15864516
O=C(NCC(F)=C1CN(C(=O)C23CC=CCN2CCC3)C1)c1nsnc1O s275592__15865378__15842482__15864528
CC(C)C(C)C(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864532
Cn1nccc1C(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864534
CC[C@H](CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__15864540
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCCO3)C2)C1)c1nsnc1O s275592__15865378__15842482__15864544
CCC=CC=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864546
O=C(NCC(F)=C1CN(C(=O)CC2CC3(CCC3)C2)C1)c1nsnc1O s275592__15865378__15842482__15864552
CNC(=O)N[C@H](C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864554
COc1ncnc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864558
CC(OCCN(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864560
O=C(NCC(F)=C1CN(C(=O)c2ccn(O)c(=O)c2)C1)c1nsnc1O s275592__15865378__15842482__15864562
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15842482__15864566
Cc1ncn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864570
CC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(CO1)C2 s275592__15865378__15842482__15864572
Cc1nc(C#N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864576
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CC(F)(F)F s275592__15865378__15842482__15864580
O=C(NCC(F)=C1CN(C(=O)Cc2nncs2)C1)c1nsnc1O s275592__15865378__15842482__15864586
CN(C)CCOCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864590
Cc1cc(N)cnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864592
COCCN(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864594
O=C(NCC(F)=C1CN(C(=O)C2CN(C3CCOC3)C2)C1)c1nsnc1O s275592__15865378__15842482__15864600
COc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1O s275592__15865378__15842482__15864604
O=C(NCC(F)=C1CN(C(=O)CCCc2c[nH]nn2)C1)c1nsnc1O s275592__15865378__15842482__15864606
CC(=C(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__15864610
CC(CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__15864612
O=C(NCC(F)=C1CN(C(=O)CCCN2CCOC2=O)C1)c1nsnc1O s275592__15865378__15842482__15856390
CC1=NOC(=O)C1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856392
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCN3)C1)c1nsnc1O s275592__15865378__15842482__15856398
Cn1cc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856400
Nc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856406
CN(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(N)=O s275592__15865378__15842482__15856410
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15856412
CC1=NOC(=O)C1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856418
O=C(NCC(F)=C1CN(C(=O)c2nc(=O)[nH][nH]2)C1)c1nsnc1O s275592__15865378__15842482__15856424
O=C(NCC(F)=C1CN(C(=O)C2(F)CC2)C1)c1nsnc1O s275592__15865378__15842482__15856434
O=C(NCC(F)=C1CN(C(=O)c2c(O)cccc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15856438
CC(C)CCSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856444
CC(C)CCCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856446
CN1CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15856454
O=C(NCC(F)=C1CN(C(=O)c2cccn(O)c2=O)C1)c1nsnc1O s275592__15865378__15842482__15856462
Nc1ncncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856466
Nc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__15856468
Cc1nc(N)ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856474
CC(C)n1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15858252
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15858256
CCN(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__15858258
CCOC(=O)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858262
O=C(NCC(F)=C1CN(C(=O)C=C(C2CC2)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15858264
CC(O)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__15858266
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15858272
O=C(NCC(F)=C1CN(C(=O)c2[nH]ncc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15858278
Cc1scnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858282
Nc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15858284
Nc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15858286
O=C(NCC(F)=C1CN(C(=O)c2cccc(F)n2)C1)c1nsnc1O s275592__15865378__15842482__15858288
COC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858294
O=C(NCC(F)=C1CN(C(=O)c2nccnc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15858296
CCOC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15858298
CC1CN2CCN1C(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15858300
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(F)F s275592__15865378__15842482__15858302
O=C(NCC(F)=C1CN(C(=O)C(F)=CC2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15858304
Cc1cccnc1C(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858306
CC(CC#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858308
CC1C(=O)CCC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858316
O=C(NCC(F)=C1CN(C(=O)c2ccnn2CC2CC2)C1)c1nsnc1O s275592__15865378__15842482__15858318
CS(=O)(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15858322
O=C(NCC(F)=C1CN(C(=O)C[C@H]2CCCC[C@@H]2O)C1)c1nsnc1O s275592__15865378__15842482__15858336
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__15858338
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cnnn1 s275592__15865378__15842482__15858340
O=C(NCC(F)=C1CN(C(=O)c2cnnc(Cl)c2)C1)c1nsnc1O s275592__15865378__15842482__15858342
Cn1cc(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15858350
O=NN1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858354
O=C(NCC(F)=C1CN(C(=O)CCCc2nccs2)C1)c1nsnc1O s275592__15865378__15842482__15858360
CCC1CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858366
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]3C[C@@H]2CC3=O)C1)c1nsnc1O s275592__15865378__15842482__15860234
O=C(NCC(F)=C1CN(C(=O)CC2CCC(O)C2)C1)c1nsnc1O s275592__15865378__15842482__15860236
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)(C)O s275592__15865378__15842482__15860240
CC(C)N(C)C(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860242
Cc1scc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15860246
CN1CC2CC1(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15860250
Cc1cc(=O)[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860254
O=C1OCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15860258
CC1(C)CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15860264
O=C(NCC(F)=C1CN(C(=O)CC23CNC(=O)C(C2)C3)C1)c1nsnc1O s275592__15865378__15842482__15860266
Cc1cnccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860268
Cn1nncc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860272
Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__15860276
Cc1nnc2n1CC(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15860280
O=C(NCC(F)=C1CN(C(=O)C23COC(C2)C3)C1)c1nsnc1O s275592__15865378__15842482__15860284
CC(O)C1CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860286
O=C(NCC(F)=C1CN(C(=O)C2C3CC4C(C3=O)C42)C1)c1nsnc1O s275592__15865378__15842482__15860288
CCCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__15860296
O=C(NCC(F)=C1CN(C(=O)CN2CC3CCC2C3)C1)c1nsnc1O s275592__15865378__15842482__15860298
O=C(NCC(F)=C1CN(C(=O)c2cccc(CF)c2)C1)c1nsnc1O s275592__15865378__15842482__15860310
COCC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860312
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1N s275592__15865378__15842482__15860314
CC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(C1)OC2 s275592__15865378__15842482__15860318
CCC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15860322
C[C@@H]1C[C@@]2(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)C[C@@H]12 s275592__15865378__15842482__15860334
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__15860338
O=C(NCC(F)=C1CN(C(=O)Cn2cncn2)C1)c1nsnc1O s275592__15865378__15842482__15860346
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2CCCN3)C1)c1nsnc1O s275592__15865378__15842482__15860350
O=C(NCC(F)=C1CN(C(=O)c2cccc(=O)o2)C1)c1nsnc1O s275592__15865378__15842482__15860352
Cc1cc(O)ccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860354
O=C(NCC(F)=C1CN(C(=O)COc2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__15862196
CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1ccnc1 s275592__15865378__15842482__15862200
O=C(NCC(F)=C1CN(C(=O)c2nc(C3CC3)n[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15862204
O=C(NCC(F)=C1CN(C(=O)COc2ccc(F)cn2)C1)c1nsnc1O s275592__15865378__15842482__15862206
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CC2)N=N3)C1)c1nsnc1O s275592__15865378__15842482__15862208
CC1CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(C)O1 s275592__15865378__15842482__15862210
COC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCCC1 s275592__15865378__15842482__15862214
CC(CN(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862216
O=C(NCC(F)=C1CN(C(=O)C2CCCc3cn[nH]c32)C1)c1nsnc1O s275592__15865378__15842482__15862224
CNc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15862226
COc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccnc1F s275592__15865378__15842482__15862230
O=C(NCC(F)=C1CN(C(=O)CC2CCCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15862232
Cn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__15862236
CC1(C)C(C#N)C1(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862238
O=C(NCC(F)=C1CN(C(=O)C2Cc3cccnc3C2)C1)c1nsnc1O s275592__15865378__15842482__15862240
COc1cnc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862242
C=CC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862244
O=C(NCC(F)=C1CN(C(=O)CCC2(O)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15862246
CCc1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15862248
CCC(C)(CO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862252
Nc1nc(Cl)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15862260
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15862262
O=C(NCC(F)=C1CN(C(=O)CS(=O)(=O)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15862266
Cn1nc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862272
CCc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15862276
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1(F)Cl s275592__15865378__15842482__15862280
CCCC=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862286
CC=C(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862288
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842482__15862292
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOC1 s275592__15865378__15842482__15862294
O=C(NCC(F)=C1CN(C(=O)C(=O)C2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15862296
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CC3(F)F)C1)c1nsnc1O s275592__15865378__15842482__15862298
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nsnc1O s275592__15865378__15842482__15862300
CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__15862302
CC(C)Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__15862306
CCS(=O)(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862312
CC(O)CCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862314
O=C(NCC(F)=C1CN(C(=O)c2ncn3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__15862316
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccncc2)C1)c1nsnc1O s275592__15865378__15842482__15864614
CCNc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864616
O=C(NCC(F)=C1CN(C(=O)c2cncc(F)n2)C1)c1nsnc1O s275592__15865378__15842482__15864618
O=C(NCC(F)=C1CN(C(=O)c2cnn(C3CC3)c2)C1)c1nsnc1O s275592__15865378__15842482__15864620
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__15864622
Nc1cc(O)nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15864626
C[C@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__15864628
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccc(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15864634
CC(C)C(CO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864638
CCOC=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864642
Nc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15864644
O=C(NCC(F)=C1CN(C(=O)Cc2cc(F)ccc2O)C1)c1nsnc1O s275592__15865378__15842482__15864646
CCN1CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864656
Cc1nc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15864662
CSc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15864664
O=C(CO)NCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864668
CS(=O)(=O)SCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864678
O=C(NCC(F)=C1CN(C(=O)c2cn3cnnc3cn2)C1)c1nsnc1O s275592__15865378__15842482__15864684
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccs1 s275592__15865378__15842482__15864686
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)o1 s275592__15865378__15842482__15864694
O=C1CCC(C#CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15864696
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC2CCC1C2 s275592__15865378__15842482__15864698
CC(C)N1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864700
Cc1ccc2c(c1)C(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15864710
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1C s275592__15865378__15842482__15864716
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@H]2C(F)F)C1)c1nsnc1O s275592__15865378__15842482__15864718
O=C(NCC(F)=C1CN(C(=O)[C@H]2CCc3ccccc32)C1)c1nsnc1O s275592__15865378__15842482__15864720
O=C(NCC(F)=C1CN(C(=O)C2(C3CC3)CCCO2)C1)c1nsnc1O s275592__15865378__15842482__15864730
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(N)cc1F s275592__15865378__15842482__15856492
CCc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15856494
N#Cc1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856502
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1Cl s275592__15865378__15842482__15856504
CCC(C)(C)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856508
CSSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856512
CCOC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15856516
NC(=O)C(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856518
CCC(C)=C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856520
Nc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842482__15856522
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2NCC3)C1)c1nsnc1O s275592__15865378__15842482__15856526
CSC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15842482__15856528
COC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15856530
CSc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856532
O=C(NCC(F)=C1CN(C(=O)c2coc(Cl)n2)C1)c1nsnc1O s275592__15865378__15842482__15856534
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(O)cc2)C1)c1nsnc1O s275592__15865378__15842482__15856540
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)=NN1 s275592__15865378__15842482__15856546
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)c1 s275592__15865378__15842482__15856552
CC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15856554
N#Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856556
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(Cl)c2)C1)c1nsnc1O s275592__15865378__15842482__15856560
O=C(NCC(F)=C1CN(C(=O)CNc2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15856566
Nc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856572
Nc1ccc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856576
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1O s275592__15865378__15842482__15856578
O=C(NCC(F)=C1CN(C(=O)c2cc(F)ccc2O)C1)c1nsnc1O s275592__15865378__15842482__15856580
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)c1 s275592__15865378__15842482__15856582
NC(=O)NCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856586
O=C(NCC(F)=C1CN(C(=O)CNc2ccc(O)cc2)C1)c1nsnc1O s275592__15865378__15842482__15856588
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15856592
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1Cl s275592__15865378__15842482__15856604
CS(C)(=O)=NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858372
[N-]=[N+]=NCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858376
C=CCCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858382
CC(C)C(=O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858384
CC(O)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858388
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__15858392
CC(C)(C)OCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858396
CC(C)Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15842482__15858404
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1CCO s275592__15865378__15842482__15858406
CC(=O)OCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858408
C#CCN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858412
CNc1nc(C)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858420
Nc1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858424
CC(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858426
Nc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858428
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(N)c1 s275592__15865378__15842482__15858430
O=C(NCC(F)=C1CN(C(=O)Cn2cccnc2=O)C1)c1nsnc1O s275592__15865378__15842482__15858432
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1N s275592__15865378__15842482__15858434
CC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858440
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)NC1CC1 s275592__15865378__15842482__15858444
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15858448
CCCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__15858458
O=C(NCC(F)=C1CN(C(=O)C=CC2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15858460
Nc1ccc(Cl)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858462
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15858468
Cn1cc([N+](=O)[O-])c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15858472
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15858474
Cc1onc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C#N s275592__15865378__15842482__15858476
CN(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858478
O=C(NCC(F)=C1CN(C(=O)C(F)(F)CO)C1)c1nsnc1O s275592__15865378__15842482__15858486
Cc1nc(O)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858488
N#CCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860358
O=C(NCC(F)=C1CN(C(=O)C=Cc2nccs2)C1)c1nsnc1O s275592__15865378__15842482__15860360
CC1(C#CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15860362
O=C(NCC(F)=C1CN(C(=O)C2OCCn3ccnc32)C1)c1nsnc1O s275592__15865378__15842482__15860366
C=CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15860378
CC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860380
Cc1ncsc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860382
[N-]=[N+]=N[C@@H]1C=CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15860386
O=C(NCC(F)=C1CN(C(=O)COC2CC2)C1)c1nsnc1O s275592__15865378__15842482__15860388
Nc1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15860392
O=C(NCC(F)=C1CN(C(=O)c2ncc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15860394
O=C(NCC(F)=C1CN(C(=O)C=CC2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15860398
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1nccs1 s275592__15865378__15842482__15860400
O=C(NCC(F)=C1CN(C(=O)C=CBr)C1)c1nsnc1O s275592__15865378__15842482__15860402
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccccc2F)C1)c1nsnc1O s275592__15865378__15842482__15860404
CC(CCN(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860406
O=C1CC(C#CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15860408
CSc1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860410
CC1(C)OC[C@H](C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15860414
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__15860420
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__15860424
O=C(NCC(F)=C1CN(C(=O)C2CC(C3CC3)C2)C1)c1nsnc1O s275592__15865378__15842482__15860432
O=C(NCC(F)=C1CN(C(=O)c2cn(C3CC3)cn2)C1)c1nsnc1O s275592__15865378__15842482__15860434
Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15860440
CC(C)[C@H](NC=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860442
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1O s275592__15865378__15842482__15860450
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cncnc1 s275592__15865378__15842482__15860458
O=C(NCC(F)=C1CN(C(=O)c2ccn3c2CCC3)C1)c1nsnc1O s275592__15865378__15842482__15860462
C=C(C)[C@@H]1OCCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860466
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nnc1C s275592__15865378__15842482__15860474
CC1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15860476
Cn1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1=O s275592__15865378__15842482__15862326
CSC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862328
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccc(N)cn1 s275592__15865378__15842482__15862330
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCCOC2)C1)c1nsnc1O s275592__15865378__15842482__15862332
N#Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15862334
Cc1c(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__15862338
Nc1cccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15862342
CCn1nccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862348
Cc1coc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15862350
O=C(NCC(F)=C1CN(C(=O)c2nncs2)C1)c1nsnc1O s275592__15865378__15842482__15862356
CC(=O)N[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15842482__15862358
O=C(NCC(F)=C1CN(C(=O)C#CC2CCCOC2)C1)c1nsnc1O s275592__15865378__15842482__15862360
O=C(NCC(F)=C1CN(C(=O)CC2CCC=CCC2)C1)c1nsnc1O s275592__15865378__15842482__15862364
O=C(NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3CCCO[C@H]32)C1)c1nsnc1O s275592__15865378__15842482__15862374
O=C(NCC(F)=C1CN(C(=O)C2(c3cccs3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15862378
CCC(C)(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862380
O=C(NCC(F)=C1CN(C(=O)COC2CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15862388
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCO3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15862390
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccc(F)cc1 s275592__15865378__15842482__15862392
CC1(C)CC(=O)NCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862402
O=C(NCC(F)=C1CN(C(=O)c2cnn(CCO)c2)C1)c1nsnc1O s275592__15865378__15842482__15862406
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@@H](OC(F)F)C2)C1)c1nsnc1O s275592__15865378__15842482__15862408
O=C(NCC(F)=C1CN(C(=O)c2cccn3nncc23)C1)c1nsnc1O s275592__15865378__15842482__15862412
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)no1 s275592__15865378__15842482__15862416
O=C(NCC(F)=C1CN(C(=O)c2csc3cncn23)C1)c1nsnc1O s275592__15865378__15842482__15862424
CC(C)(C)c1noc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15862426
C=C(F)C1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15862428
O=C1COC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15862436
CC12CC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(C1)C(C)(C)O2 s275592__15865378__15842482__15863670
O=C(NCC(F)=C1CN(C(=O)c2coc(C(F)F)n2)C1)c1nsnc1O s275592__15865378__15842482__15863672
O=C(C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)NC1CC1 s275592__15865378__15842482__15863674
CC(C)NC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863680
C=C(Cl)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863686
CC(C)(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__15863690
CCC(CCOC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863692
O=C(NCC(F)=C1CN(C(=O)C2CC3C=CCC(C3)C2)C1)c1nsnc1O s275592__15865378__15842482__15863694
Cc1nc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)oc1C s275592__15865378__15842482__15863696
Cc1coc(C)c1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863698
O=C(NCC(F)=C1CN(C(=O)C23CC(CN2C2CC2)C3)C1)c1nsnc1O s275592__15865378__15842482__15863700
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__15863704
C=Cn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863714
Cc1coc(C(C)C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863716
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15863720
Cn1ccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863724
CC(=O)OCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863732
Cc1nc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]c1C s275592__15865378__15842482__15863736
CCc1oc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863738
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC=CC1 s275592__15865378__15842482__15863740
O=C(NCC(F)=C1CN(C(=O)CCNc2cncnc2)C1)c1nsnc1O s275592__15865378__15842482__15864740
CCc1cscc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864748
O=C1CSC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864760
C=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)(C(F)F)C1 s275592__15865378__15842482__15864772
CO[C@@H]1C[C@@]2(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)C[C@@H]12 s275592__15865378__15842482__15864778
O=C(NCC(F)=C1CN(C(=O)c2cc3cncnc3[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15864780
Cc1ccc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15864782
CC1OC2(C)CC1(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15864784
Cn1cnnc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864786
CCc1nonc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864792
O=C(NCC(F)=C1CN(C(=O)Cc2cnsn2)C1)c1nsnc1O s275592__15865378__15842482__15864798
C=CCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864800
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ncc1N s275592__15865378__15842482__15864814
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1O s275592__15865378__15842482__15864818
CC(C)(C)O[C@H]1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15864826
CCC(C)CC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15864832
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOC1 s275592__15865378__15842482__15864836
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COc1ccnc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15864856
CC1(C)CC(=O)N(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15864858
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O=C(NCC(F)=C1CN(C(=O)CCN2CCC(O)CC2)C1)c1nsnc1O s275592__15865378__15842482__15856612
Cc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15856614
O=C(NCC(F)=C1CN(C(=O)CCOc2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__15856620
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15856622
CCCN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856624
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(Cl)c1 s275592__15865378__15842482__15856628
Cc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15856632
CC(C)CCOCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856634
O=C(NCC(F)=C1CN(C(=O)COCc2ccco2)C1)c1nsnc1O s275592__15865378__15842482__15856638
CC(CO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856640
Cc1ccc(F)c(N)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856646
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Nc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15856652
CN1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15856658
Nc1c(F)cc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858498
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CCOC(=O)C(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858502
O=C(NCC(F)=C1CN(C(=O)C(=O)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15858504
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1Cl s275592__15865378__15842482__15858508
CCCCCCCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858514
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15842482__15858516
O=C1N[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__15858518
O=C(NCC(F)=C1CN(C(=O)c2cncc(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15858522
COc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15858524
O=C(NCC(F)=C1CN(C(=O)Cc2cnccc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15858526
O=C(NCC(F)=C1CN(C(=O)CC2(O)CC2)C1)c1nsnc1O s275592__15865378__15842482__15858528
O=C(NCC(F)=C1CN(C(=O)CCCCC(F)(F)F)C1)c1nsnc1O s275592__15865378__15842482__15858536
O=C(NCC(F)=C1CN(C(=O)Cc2ccn[nH]c2=O)C1)c1nsnc1O s275592__15865378__15842482__15858540
Cc1oc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858544
COC(=O)CC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858548
Cc1nc(CO)sc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858554
O=C(NCC(F)=C1CN(C(=O)c2cccc(=S)n2O)C1)c1nsnc1O s275592__15865378__15842482__15858556
CNc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15858566
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)ccn2)C1)c1nsnc1O s275592__15865378__15842482__15858572
O=C(NCC(F)=C1CN(C(=O)C2CCC2F)C1)c1nsnc1O s275592__15865378__15842482__15858574
N#CCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858576
O=C(NCC(F)=C1CN(C(=O)C2C(F)(F)C23CCC3)C1)c1nsnc1O s275592__15865378__15842482__15858582
O=C(NCC(F)=C1CN(C(=O)c2ccn3nccc3c2)C1)c1nsnc1O s275592__15865378__15842482__15858596
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(C)n1 s275592__15865378__15842482__15858598
Nc1c(F)ccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858602
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cnc(C#N)n1 s275592__15865378__15842482__15858610
CCOC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858618
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CCC3)O2)C1)c1nsnc1O s275592__15865378__15842482__15860482
O=C(NCC(F)=C1CN(C(=O)C2CC(n3ccnc3)C2)C1)c1nsnc1O s275592__15865378__15842482__15860488
O=C(NCC(F)=C1CN(C(=O)C(F)C2CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15860490
O=C(NCC(F)=C1CN(C(=O)C2CCCC23CCC3)C1)c1nsnc1O s275592__15865378__15842482__15860492
Cc1oc(Cl)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860498
Cc1cnsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860502
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]ccc3n2)C1)c1nsnc1O s275592__15865378__15842482__15860506
O=C(NCC(F)=C1CN(C(=O)[C@@H](O)Cc2c[nH]cn2)C1)c1nsnc1O s275592__15865378__15842482__15860508
CCc1onc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__15860512
Cn1cc(SCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15860514
CC(C)CC(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860516
O=C(NCC(F)=C1CN(C(=O)C(F)C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15860518
CC(OC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860520
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15860522
O=C(NCC(F)=C1CN(C(=O)c2ccn3nncc3c2)C1)c1nsnc1O s275592__15865378__15842482__15860526
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCNC1=O s275592__15865378__15842482__15860528
CC1CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__15860530
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCCC3)CO2)C1)c1nsnc1O s275592__15865378__15842482__15860532
O=C(NCC(F)=C1CN(C(=O)CC2CC3(CC3)CO2)C1)c1nsnc1O s275592__15865378__15842482__15860534
CC(C)(F)C(C)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860542
O=C(NCC(F)=C1CN(C(=O)[C@]23COC[C@H]2C3(F)F)C1)c1nsnc1O s275592__15865378__15842482__15860544
O=C1CCC(F)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15860546
Cc1cn(C(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860550
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCS1 s275592__15865378__15842482__15860552
CC12CC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(CCO1)C2 s275592__15865378__15842482__15860554
CC(C)(CCC#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860558
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3CCCCC[C@@H]32)C1)c1nsnc1O s275592__15865378__15842482__15860560
CC1=NOC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15860562
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15860570
CC1(C)CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__15860588
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C(=O)N1 s275592__15865378__15842482__15860600
O=C(NCC(F)=C1CN(C(=O)CC2CCC3CC3C2)C1)c1nsnc1O s275592__15865378__15842482__15862442
Cc1ccsc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862452
Cc1ccccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862454
Cn1cccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862458
O=C(NCC(F)=C1CN(C(=O)C=Cc2c[nH]cn2)C1)c1nsnc1O s275592__15865378__15842482__15862464
Cc1csc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15862468
O=C(NCC(F)=C1CN(C(=O)C=Cc2cncs2)C1)c1nsnc1O s275592__15865378__15842482__15862474
O=C(NCC(F)=C1CN(C(=O)C=Cc2ncc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15862484
Cn1cc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__15862486
O=C(NCC(F)=C1CN(C(=O)[C@]23C[C@H]2COC32CCC2)C1)c1nsnc1O s275592__15865378__15842482__15862490
CCC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)COC1 s275592__15865378__15842482__15862492
Cn1nccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862498
O=C(NCC(F)=C1CN(C(=O)C=Cc2cn[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__15862500
CCc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15862504
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15842482__15862508
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(N)s1 s275592__15865378__15842482__15862518
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2CF)C1)c1nsnc1O s275592__15865378__15842482__15862520
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCS3)C1)c1nsnc1O s275592__15865378__15842482__15862524
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__15862526
CC1CN(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15862530
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccncc1 s275592__15865378__15842482__15862534
O=C(NCC(F)=C1CN(C(=O)CNc2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__15862540
NC(=O)[C@@H]1CCCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862544
O=C(NCC(F)=C1CN(C(=O)Cc2cnns2)C1)c1nsnc1O s275592__15865378__15842482__15862548
Cc1oc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1CO s275592__15865378__15842482__15862550
O=C(NCC(F)=C1CN(C(=O)C(F)=C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15862554
CCC(CO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862556
CC(C)(O)C(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862558
CON1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15862560
O=C(NCC(F)=C1CN(C(=O)c2cn(C3COC3)nn2)C1)c1nsnc1O s275592__15865378__15842482__15863744
O=C(NCC(F)=C1CN(C(=O)c2ccc3ncnn3c2)C1)c1nsnc1O s275592__15865378__15842482__15863746
O=C(NCC(F)=C1CN(C(=O)c2cccc3oncc23)C1)c1nsnc1O s275592__15865378__15842482__15863748
O=C(NCC(F)=C1CN(C(=O)CC(O)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15863750
Cc1c(O)ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__15863760
O=C(NCC(F)=C1CN(C(=O)COC2CCCOC2)C1)c1nsnc1O s275592__15865378__15842482__15863764
CC(C)CC(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863770
CC1(C#CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)COC1 s275592__15865378__15842482__15863772
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)c1 s275592__15865378__15842482__15863776
CC(=CC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863786
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1nc[nH]n1 s275592__15865378__15842482__15863788
O=C1CC2(CC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)C2)N1 s275592__15865378__15842482__15863790
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(Cl)n1 s275592__15865378__15842482__15863792
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(CO)c2)C1)c1nsnc1O s275592__15865378__15842482__15863794
CC1(C)C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1(F)F s275592__15865378__15842482__15863800
N#C[C@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863804
CC(=O)c1cn(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863810
O=C(NCC(F)=C1CN(C(=O)C2(O)CC3CCC2C3)C1)c1nsnc1O s275592__15865378__15842482__15863812
CCC1CCCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863814
O=C(NCC(F)=C1CN(C(=O)C=Cc2cocn2)C1)c1nsnc1O s275592__15865378__15842482__15863816
CC(=Cn1ccnn1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863820
CC(C)n1cnnc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863824
O=C(NCC(F)=C1CN(C(=O)CC2(CO)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15863830
O=C(NCC(F)=C1CN(C(=O)c2coc3c2CCCC3)C1)c1nsnc1O s275592__15865378__15842482__15863832
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCO3)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15863834
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(N)c1O s275592__15865378__15842482__15863836
CN(C)Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__15863838
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O=C(NCC(F)=C1CN(C(=O)CC2(CO)CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15863844
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C=CCn1ccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858694
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Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1O s275592__15865378__15842482__15858732
COc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__15858734
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CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)=NO1 s275592__15865378__15842482__15860614
CC(C)C1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15860618
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CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C=CCCC1 s275592__15865378__15842482__15860644
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CCCN1C(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860662
Cc1ccc(F)c(O)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860664
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CC1CCCC(O)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15860668
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1C s275592__15865378__15842482__15860672
CC12CC(CC(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(CO1)C2 s275592__15865378__15842482__15860676
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CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1F s275592__15865378__15842482__15862600
CCC(F)(F)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862606
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CC(=Cc1ccncc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862620
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Cc1cc(F)sc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862664
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COC1C[C@@H]2CC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)C[C@H]12 s275592__15865378__15842482__15863868
O=C(NCC(F)=C1CN(C(=O)C2C3CCOCC32)C1)c1nsnc1O s275592__15865378__15842482__15863872
Cc1cnn(C(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15863874
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cnnc1 s275592__15865378__15842482__15863876
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(F)nc2)C1)c1nsnc1O s275592__15865378__15842482__15863878
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC2CC2C1 s275592__15865378__15842482__15863882
O=C(NCC(F)=C1CN(C(=O)C=CCF)C1)c1nsnc1O s275592__15865378__15842482__15863884
O=C(NCC(F)=C1CN(C(=O)C2(CC(F)F)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15863888
O=C(NCC(F)=C1CN(C(=O)C(F)CC2CC2)C1)c1nsnc1O s275592__15865378__15842482__15863892
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__15863894
Cc1c(O)cc(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863896
CC(C)CCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863902
CN1CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863906
O=C(NCC(F)=C1CN(C(=O)c2ccnc3c2CCC3)C1)c1nsnc1O s275592__15865378__15842482__15863910
O=C(NCC(F)=C1CN(C(=O)C=CCn2cncn2)C1)c1nsnc1O s275592__15865378__15842482__15863914
O=C(NCC(F)=C1CN(C(=O)C=CC2CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15863918
CSc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15863920
O=C(NCC(F)=C1CN(C(=O)CNc2ccncc2)C1)c1nsnc1O s275592__15865378__15842482__15863922
N#Cc1ccccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863926
Cc1nnc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15863928
CC(C)(C)O[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863930
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccc(N)c1 s275592__15865378__15842482__15863938
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]c1C s275592__15865378__15842482__15863940
CCOC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15863948
Cc1cc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__15863956
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)sn1 s275592__15865378__15842482__15863960
O=C(NCC(F)=C1CN(C(=O)c2ncoc2C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15863962
O=C1N[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__15863964
COC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863966
CC(O)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863968
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccco1 s275592__15865378__15842482__15863970
Cc1nn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)o1 s275592__15865378__15842482__15863972
N#CCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863976
O=C(NCC(F)=C1CN(C(=O)c2cnn3ccsc23)C1)c1nsnc1O s275592__15865378__15842482__15863978
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cnc2O)C1)c1nsnc1O s275592__15865378__15842482__15863982
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]n1 s275592__15865378__15842482__15856786
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C#N s275592__15865378__15842482__15856788
O=C(NCC(F)=C1CN(C(=O)c2cc3ncccc3[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15856790
O=C(NCC(F)=C1CN(C(=O)C2(CO)CC2)C1)c1nsnc1O s275592__15865378__15842482__15856792
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)c1 s275592__15865378__15842482__15856796
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)nc2)C1)c1nsnc1O s275592__15865378__15842482__15856800
CSc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__15856806
CCC1=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15842482__15856808
O=C(NCC(F)=C1CN(C(=O)c2csc([N+](=O)[O-])c2)C1)c1nsnc1O s275592__15865378__15842482__15856816
O=C(NCC(F)=C1CN(C(=O)c2cc([N+](=O)[O-])c[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15856822
Cc1cc(C)c(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856824
O=C(NCC(F)=C1CN(C(=O)c2cccc(Cl)c2O)C1)c1nsnc1O s275592__15865378__15842482__15856826
O=C(NCC(F)=C1CN(C(=O)c2ccno2)C1)c1nsnc1O s275592__15865378__15842482__15856830
O=C(NCC(F)=C1CN(C(=O)[C@@H]2Cc3ccccc3N2)C1)c1nsnc1O s275592__15865378__15842482__15856836
CNc1snc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856838
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1F s275592__15865378__15842482__15856842
O=C(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__15856844
Nc1c(Cl)cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856846
Nc1cc(F)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856854
Cc1nsc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856856
CC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15856862
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15856868
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15856870
O=C(NCC(F)=C1CN(C(=O)c2c(O)cccc2O)C1)c1nsnc1O s275592__15865378__15842482__15856872
[N-]=[N+]=NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856874
Cc1c(N)cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856876
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__15856878
O=C(NCC(F)=C1CN(C(=O)C2=CCCSC2)C1)c1nsnc1O s275592__15865378__15842482__15856886
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]1 s275592__15865378__15842482__15856890
C[C@H](O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15856892
Cc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)sc1C s275592__15865378__15842482__15856894
CCN1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15856896
C[C@@](O)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842482__15856898
O=C(NCC(F)=C1CN(C(=O)C2(O)CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15856902
O=C(NCC(F)=C1CN(C(=O)C=C2CN3CCC2CC3)C1)c1nsnc1O s275592__15865378__15842482__15858744
CCCC(CCC)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858748
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__15858750
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)o2)C1)c1nsnc1O s275592__15865378__15842482__15858752
CCCC(=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CCC s275592__15865378__15842482__15858754
Cc1cc(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__15858758
O=C(NCC(F)=C1CN(C(=O)C=C2CCSCC2)C1)c1nsnc1O s275592__15865378__15842482__15858760
CON=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858762
C#CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858766
O=C(NCC(F)=C1CN(C(=O)C[C@@H](O)c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15858774
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnc1Cl s275592__15865378__15842482__15858782
Cc1ncnc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858784
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1F s275592__15865378__15842482__15858790
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N=[N+]=[N-] s275592__15865378__15842482__15858792
CC1(F)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15858798
Cn1ncc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858800
CCC(C)(OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858808
Nc1cc(F)cc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858810
CC(C)(C)CCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858812
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(CO)c2)C1)c1nsnc1O s275592__15865378__15842482__15858816
CCCC(CCCO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858820
CC(O)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15858826
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCN1 s275592__15865378__15842482__15858828
CC(C)[C@H](O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15858830
CSC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15858832
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cccc(O)c1 s275592__15865378__15842482__15858834
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccn1 s275592__15865378__15842482__15858840
O=C(NCC(F)=C1CN(C(=O)C(O)c2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__15858844
CC(O)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccn1 s275592__15865378__15842482__15858846
O=C(NCC(F)=C1CN(C(=O)c2cccc(=O)n2O)C1)c1nsnc1O s275592__15865378__15842482__15858848
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)cn2)C1)c1nsnc1O s275592__15865378__15842482__15858852
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1N s275592__15865378__15842482__15858858
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__15858866
O=C(NCC(F)=C1CN(C(=O)c2ccnn2CCF)C1)c1nsnc1O s275592__15865378__15842482__15860726
N#Cc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860740
N#Cc1ccnc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15860746
O=C(NCC(F)=C1CN(C(=O)CC=C(Cl)Cl)C1)c1nsnc1O s275592__15865378__15842482__15860748
CN(C)C(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860752
C#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15860756
O=C(NCC(F)=C1CN(C(=O)c2ccnc(CO)c2)C1)c1nsnc1O s275592__15865378__15842482__15860758
CN(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)[C@@H]1CCC[C@H]1O s275592__15865378__15842482__15860762
CC(C)(C)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15860770
N#Cc1cncc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15860772
CCC1CN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15860778
O=C1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15860782
Cc1cn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860784
O=C(NCC(F)=C1CN(C(=O)C2(N3CCCC3)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15860792
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)c1 s275592__15865378__15842482__15860798
CC(=O)CCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860800
C=CC=CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860802
COC(=O)[C@@H]1C[C@]1(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860804
C=CCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860806
O=C(NCC(F)=C1CN(C(=O)COCc2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__15860808
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(=O)[nH]1 s275592__15865378__15842482__15860810
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC(C2)S3)C1)c1nsnc1O s275592__15865378__15842482__15860814
O=C(NCC(F)=C1CN(C(=O)C=Cc2cncc(F)c2)C1)c1nsnc1O s275592__15865378__15842482__15860822
C#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15860826
CN1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860828
CCCC=CC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860832
O=C(NCC(F)=C1CN(C(=O)C2CC=CCO2)C1)c1nsnc1O s275592__15865378__15842482__15860842
O=C(NCC(F)=C1CN(C(=O)C23CCOC2CCOC3)C1)c1nsnc1O s275592__15865378__15842482__15860844
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(c2)CCC3)C1)c1nsnc1O s275592__15865378__15842482__15862692
CCCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15862698
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC(C3)C2)C1)c1nsnc1O s275592__15865378__15842482__15862700
O=C(NCC(F)=C1CN(C(=O)C=Cc2ncco2)C1)c1nsnc1O s275592__15865378__15842482__15862704
COC(=O)C(OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862708
O=C(NCC(F)=C1CN(C(=O)C2(F)C#CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15862716
CC(CC1CCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862718
Cc1nsc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15862722
O=C(NCC(F)=C1CN(C(=O)C2CCC3(C2)N=N3)C1)c1nsnc1O s275592__15865378__15842482__15862724
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CC(C)[C@@H](NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860908
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CN(C)[C@H]1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15860942
CN1CC=CCC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860944
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CC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C(C)O1 s275592__15865378__15842482__15860968
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CCCC(CC)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862808
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C=C(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862818
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CC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)(CC1)OC2 s275592__15865378__15842482__15864152
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CCCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__15864170
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COCc1noc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15864190
O=C(NCC(F)=C1CN(C(=O)CC2CC(O)C23CCC3)C1)c1nsnc1O s275592__15865378__15842482__15864194
[N-]=[N+]=N[C@@H]1C[C@@]2(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)C[C@@H]12 s275592__15865378__15842482__15864196
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CCOc1oc(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857022
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CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)=NO1 s275592__15865378__15842482__15857048
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CC(C)(CO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857066
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Cc1cccc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857098
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NC(=O)NC(CO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857112
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CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)COC(=O)OC1 s275592__15865378__15842482__15859010
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CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1=O s275592__15865378__15842482__15859040
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CC1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859060
CC1CCC(O)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15859062
CC1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859064
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CC1(C)CCC(O)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15859070
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CCOC(=O)C(CC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859084
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Cc1cc(Cl)nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15859102
Cc1oc(C#N)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859104
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CCNc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15860974
CCOc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860978
O=C(NCC(F)=C1CN(C(=O)C2C3CC4C(C3)C42)C1)c1nsnc1O s275592__15865378__15842482__15860980
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)noc1C1CC1 s275592__15865378__15842482__15860984
Cn1c([N+](=O)[O-])cnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860986
O=C(NCC(F)=C1CN(C(=O)[C@@H](O)C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15860990
CC1(C)CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15860992
COC(=O)[C@@H]1[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1(C)C s275592__15865378__15842482__15860996
COCC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15860998
C[C@]1(C(F)(F)F)C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861002
CC(Cc1ccncc1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861004
COC1CC(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861010
CC(F)(F)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861014
O=C(NCC(F)=C1CN(C(=O)c2nnc3ccccn23)C1)c1nsnc1O s275592__15865378__15842482__15861018
N#Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861020
O=C(NCC(F)=C1CN(C(=O)[C@]23C[C@@H]4C[C@@H]2C3[C@H]4O)C1)c1nsnc1O s275592__15865378__15842482__15861022
C[C@@H](OCCN(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861032
CNC(=O)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861040
O=C(NCC(F)=C1CN(C(=O)C23COC(CCO2)C3)C1)c1nsnc1O s275592__15865378__15842482__15861048
CCn1cnnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861050
O=C(NCC(F)=C1CN(C(=O)C2(C3CCC3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15861058
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@@H]3C[C@@H]32)C1)c1nsnc1O s275592__15865378__15842482__15861066
CC1(C)C(C)(C)C1(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861068
CC(C)[C@@H]1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861072
O=C(NCC(F)=C1CN(C(=O)c2ccn(CCF)n2)C1)c1nsnc1O s275592__15865378__15842482__15861086
O=C(NCC(F)=C1CN(C(=O)c2cnc3cn[nH]c3c2)C1)c1nsnc1O s275592__15865378__15842482__15862930
CC(=Cc1ccccn1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862946
CC(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__15862950
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(F)C1 s275592__15865378__15842482__15862956
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__15862958
O=C(NCC(F)=C1CN(C(=O)c2nc(=O)[nH]c(=O)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15862962
CCc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15862970
O=C(NCC(F)=C1CN(C(=O)C#CC2CCCO2)C1)c1nsnc1O s275592__15865378__15842482__15862984
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC=CC1 s275592__15865378__15842482__15862988
O=C(NCC(F)=C1CN(C(=O)C23CCCC(C2)OC3)C1)c1nsnc1O s275592__15865378__15842482__15862990
CC1OCCC1(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15862992
Cc1ncc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15863006
CCc1scnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863008
Cc1cccc(C(O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15863018
C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863036
CC(=O)NC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__15857138
Nc1ccc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857140
O=C(NCC(F)=C1CN(C(=O)CCc2ccccc2O)C1)c1nsnc1O s275592__15865378__15842482__15857146
CC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857148
Cc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857154
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842482__15857162
O=C(NCC(F)=C1CN(C(=O)CCN2CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15857164
Cc1nc(C)n(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15857168
N#CCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857172
O=C(NCC(F)=C1CN(C(=O)CN2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15857176
O=C(NCC(F)=C1CN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1)c1nsnc1O s275592__15865378__15842482__15857178
CN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15857180
O=C(NCC(F)=C1CN(C(=O)CN2CCC(CO)CC2)C1)c1nsnc1O s275592__15865378__15842482__15857184
O=C(NCC(F)=C1CN(C(=O)CN2CCCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15857196
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCOCC1 s275592__15865378__15842482__15857200
O=C(NCC(F)=C1CN(C(=O)CCNc2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__15857204
Cc1cnc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857206
CCCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15857208
Cn1cc[n+](CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857214
COC(=O)[C@H]1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15857216
CNc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15857224
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1F s275592__15865378__15842482__15857226
Cc1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857228
CSC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15857232
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)F)no2)C1)c1nsnc1O s275592__15865378__15842482__15857242
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)co1 s275592__15865378__15842482__15857244
O=C(NCC(F)=C1CN(C(=O)C2=NOCC2)C1)c1nsnc1O s275592__15865378__15842482__15857252
COc1cccc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859116
O=C(NCC(F)=C1CN(C(=O)c2cn(C3CC3)nn2)C1)c1nsnc1O s275592__15865378__15842482__15859120
O=C(NCC(F)=C1CN(C(=O)COc2ccon2)C1)c1nsnc1O s275592__15865378__15842482__15859122
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(O)CC1 s275592__15865378__15842482__15859132
Cc1coc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__15859134
Cc1csc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15859136
CN(C)Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15859138
O=C(NCC(F)=C1CN(C(=O)c2occc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15859150
O=C(NCC(F)=C1CN(C(=O)CC2CC2(Cl)Cl)C1)c1nsnc1O s275592__15865378__15842482__15859156
O=C(NCC(F)=C1CN(C(=O)Cc2cnccn2)C1)c1nsnc1O s275592__15865378__15842482__15859158
CC(C#N)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859162
CC(C)c1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15859164
COC(=O)c1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859166
Nc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15859176
Cn1cc(C(O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15859178
CCC1OCCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859182
COc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15859186
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)n1 s275592__15865378__15842482__15859190
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1ccccn1 s275592__15865378__15842482__15859194
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2OCO3)C1)c1nsnc1O s275592__15865378__15842482__15859198
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)nn2)C1)c1nsnc1O s275592__15865378__15842482__15859208
O=C(NCC(F)=C1CN(C(=O)CN2CCC(O)CC2)C1)c1nsnc1O s275592__15865378__15842482__15859210
CCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1O s275592__15865378__15842482__15859214
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)c1O s275592__15865378__15842482__15859216
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(N)c1 s275592__15865378__15842482__15859218
CN(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__15859226
Cn1cccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859228
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCN(C)CC1 s275592__15865378__15842482__15859230
O=C(NCC(F)=C1CN(C(=O)COc2ccsn2)C1)c1nsnc1O s275592__15865378__15842482__15861094
O=C(NCC(F)=C1CN(C(=O)CCN2CCC(F)C2)C1)c1nsnc1O s275592__15865378__15842482__15861098
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(=O)[nH]1 s275592__15865378__15842482__15861100
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC2(CC2)C1 s275592__15865378__15842482__15861106
CN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1=O s275592__15865378__15842482__15861108
O=C(NCC(F)=C1CN(C(=O)CCOC2CC2)C1)c1nsnc1O s275592__15865378__15842482__15861110
Cn1cncc1C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861118
Cc1cccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861120
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)c1cnccn1 s275592__15865378__15842482__15861122
CCCCC(O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861126
COC1CN(C)C(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861136
O=C(NCC(F)=C1CN(C(=O)CCCCCO)C1)c1nsnc1O s275592__15865378__15842482__15861138
O=C(NCC(F)=C1CN(C(=O)C2=CS(=O)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15861142
NS(=O)(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861146
COC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCSC1 s275592__15865378__15842482__15861148
O=C(NCC(F)=C1CN(C(=O)c2csnc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15861150
COC(=O)[C@@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861166
Cc1conc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861172
CCOCC(N=[N+]=[N-])C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861174
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)(F)CO2)C1)c1nsnc1O s275592__15865378__15842482__15861176
C#Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861178
CCOC(=O)[C@@H]1CC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861180
N#Cc1cccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861190
Cc1cc(C#N)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15861192
CCc1noc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15861194
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CN(C)C s275592__15865378__15842482__15861196
Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15861202
N#CCc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861206
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCc3ccccc32)C1)c1nsnc1O s275592__15865378__15842482__15861212
Nc1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15863050
CC(CCO)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863056
O=C(NCC(F)=C1CN(C(=O)C(F)=CC2CC2)C1)c1nsnc1O s275592__15865378__15842482__15863058
CC(C)(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__15863072
O=C(NCC(F)=C1CN(C(=O)CC2CC(F)C2)C1)c1nsnc1O s275592__15865378__15842482__15863076
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc(C)n1 s275592__15865378__15842482__15863078
O=C(NCC(F)=C1CN(C(=O)C(F)CC2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15863080
COc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ncc1F s275592__15865378__15842482__15863082
O=C(NCC(F)=C1CN(C(=O)C2CCN3CCOCC23)C1)c1nsnc1O s275592__15865378__15842482__15863086
O=C(NCC(F)=C1CN(C(=O)C(F)CC2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15863090
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CC3(F)F)C1)c1nsnc1O s275592__15865378__15842482__15863094
O=C(NCC(F)=C1CN(C(=O)c2ncccc2CO)C1)c1nsnc1O s275592__15865378__15842482__15863096
O=C(NCC(F)=C1CN(C(=O)C(F)=Cc2cnc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15863098
CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cccn1 s275592__15865378__15842482__15863110
O=C1CCC(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CN1 s275592__15865378__15842482__15863120
O=C(NCC(F)=C1CN(C(=O)[C@H](O)CF)C1)c1nsnc1O s275592__15865378__15842482__15863130
O=C(NCC(F)=C1CN(C(=O)C2=CC3(CCOC3)C2)C1)c1nsnc1O s275592__15865378__15842482__15863132
CCC1(C)C=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863134
CCC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863136
Cc1nnc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1C s275592__15865378__15842482__15863138
O=C(NCC(F)=C1CN(C(=O)c2coc3c2COC3)C1)c1nsnc1O s275592__15865378__15842482__15863146
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@H](n3cnnc3)C2)C1)c1nsnc1O s275592__15865378__15842482__15863148
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CC(F)C3)C1)c1nsnc1O s275592__15865378__15842482__15863152
CCn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15863154
CN1CCOCC1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863160
CCCC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863166
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Nc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1O s275592__15865378__15842482__15857270
CC(C)C(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857276
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(O)c2F)C1)c1nsnc1O s275592__15865378__15842482__15857284
CCN1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15857286
COc1nc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15857294
COC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15857302
COC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__15857304
CC(C)(O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857306
O=C(NCC(F)=C1CN(C(=O)C(O)c2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__15857308
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15857310
Cc1c(N)cnn1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857316
CNc1nnc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15857320
COC(=O)CSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857326
O=C(NCC(F)=C1CN(C(=O)c2nccc(Cl)c2O)C1)c1nsnc1O s275592__15865378__15842482__15857328
N#CC1CC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15857330
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ccc2O)C1)c1nsnc1O s275592__15865378__15842482__15857336
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n(C)c1 s275592__15865378__15842482__15857340
Nc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857346
Nc1ccc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857348
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1N s275592__15865378__15842482__15857354
Cc1oc(CO)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857358
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ncnn23)C1)c1nsnc1O s275592__15865378__15842482__15857362
CC(O)(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(F)(F)F s275592__15865378__15842482__15857366
Cc1csc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15857370
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15857372
O=C(NCC(F)=C1CN(C(=O)Cc2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__15857374
CC(=O)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857376
O=C(NCC(F)=C1CN(C(=O)c2ccnc(Cl)c2)C1)c1nsnc1O s275592__15865378__15842482__15857378
O=C(NCC(F)=C1CN(C(=O)C2(O)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15859240
O=C(NCC(F)=C1CN(C(=O)C(O)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15859246
O=C(NCC(F)=C1CN(C(=O)c2ccccc2CO)C1)c1nsnc1O s275592__15865378__15842482__15859248
O=C(NCC(F)=C1CN(C(=O)c2nc3n(n2)CCCN3)C1)c1nsnc1O s275592__15865378__15842482__15859254
NC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15859256
O=C(NCC(F)=C1CN(C(=O)Cn2cnnc2)C1)c1nsnc1O s275592__15865378__15842482__15859258
O=C(NCC(F)=C1CN(C(=O)C2CCc3ccccc32)C1)c1nsnc1O s275592__15865378__15842482__15859260
CSc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15859266
O=C(NCC(F)=C1CN(C(=O)C2(C(=O)NC3CC3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15859268
CC(=O)CCCCCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859278
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1O s275592__15865378__15842482__15859280
C=C(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859282
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2ccccn2)C1)c1nsnc1O s275592__15865378__15842482__15859286
CC(C)(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859288
O=C(NCC(F)=C1CN(C(=O)c2cccc(O)c2O)C1)c1nsnc1O s275592__15865378__15842482__15859290
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1CC s275592__15865378__15842482__15859292
CCCn1nc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859296
CC1=CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15859298
CCSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859302
CC(=O)OCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859304
CC(C)=C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859306
Cc1c(O)cccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859308
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccc1O s275592__15865378__15842482__15859310
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)c(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15859314
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C(F)F)C1)c1nsnc1O s275592__15865378__15842482__15859322
Cc1cc(N)ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859324
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1ccnc1 s275592__15865378__15842482__15859326
COc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15859328
Nc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15859330
Nc1c(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1F s275592__15865378__15842482__15859332
Cc1sncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859338
O=C(NCC(F)=C1CN(C(=O)c2ccncc2O)C1)c1nsnc1O s275592__15865378__15842482__15859340
CC(=O)CSCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859342
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ccc2F)C1)c1nsnc1O s275592__15865378__15842482__15859346
CCNc1scnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859352
N#Cc1csc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15859354
CC1(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N=N1 s275592__15865378__15842482__15859356
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nsnc1O s275592__15865378__15842482__15859360
O=C(NCC(F)=C1CN(C(=O)COC2COC2)C1)c1nsnc1O s275592__15865378__15842482__15861226
C[C@@H]1C[C@]2(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)C[C@H]12 s275592__15865378__15842482__15861228
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1CCO s275592__15865378__15842482__15861230
Cc1ccnc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861234
O=C(NCC(F)=C1CN(C(=O)[C@@H]2NC(=O)[C@H]3CC[C@H]32)C1)c1nsnc1O s275592__15865378__15842482__15861236
CCc1nsc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861238
CNC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861240
CC(OC1COC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861248
COC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCOC1 s275592__15865378__15842482__15861260
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2COC3)C1)c1nsnc1O s275592__15865378__15842482__15861268
O=C(NCC(F)=C1CN(C(=O)c2nnn3ccccc23)C1)c1nsnc1O s275592__15865378__15842482__15861270
CN1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1=O s275592__15865378__15842482__15861276
Cc1ccnc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861284
CN1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1=O s275592__15865378__15842482__15861286
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(F)c1O s275592__15865378__15842482__15861288
O=C(NCC(F)=C1CN(C(=O)c2cccc(C(F)F)n2)C1)c1nsnc1O s275592__15865378__15842482__15861296
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccsc2)C1)c1nsnc1O s275592__15865378__15842482__15861298
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccncn2)C1)c1nsnc1O s275592__15865378__15842482__15861300
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(F)F s275592__15865378__15842482__15861304
CN1[C@H](C(N)=O)CC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861306
Cc1cc(F)ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861310
Cc1sc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1O s275592__15865378__15842482__15861312
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC2(CC2)C1 s275592__15865378__15842482__15861316
O=C(NCC(F)=C1CN(C(=O)C2CC3(CSC3)C2)C1)c1nsnc1O s275592__15865378__15842482__15861320
CCOC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861322
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccnn3c2)C1)c1nsnc1O s275592__15865378__15842482__15861328
CC1(O)CCN(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861330
C=CCOC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863174
O=C(NCC(F)=C1CN(C(=O)C2CCCSS2)C1)c1nsnc1O s275592__15865378__15842482__15863176
Cn1cnnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863182
O=C(NCC(F)=C1CN(C(=O)CC2C[C@@H]3COC[C@H]23)C1)c1nsnc1O s275592__15865378__15842482__15863184
N#CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15863188
O=C(NCC(F)=C1CN(C(=O)c2ccccc2C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15863194
Cc1cc(N)n(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15863198
Nc1ncn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15863202
CC(=O)[C@@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1(C)C s275592__15865378__15842482__15863208
CC(=O)NC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863210
O=C(NCC(F)=C1CN(C(=O)C2=CCCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15863212
C[C@@H]1OCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863214
Cn1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15863218
O=C(NCC(F)=C1CN(C(=O)C2CC(F)C2)C1)c1nsnc1O s275592__15865378__15842482__15863220
O=C(NCC(F)=C1CN(C(=O)C2C[C@H]3CC(=O)[C@@H]2C3)C1)c1nsnc1O s275592__15865378__15842482__15863228
CCC(O)C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863232
O=C(NCC(F)=C1CN(C(=O)c2ncnc3nc[nH]c23)C1)c1nsnc1O s275592__15865378__15842482__15863234
CN(C)c1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863236
O=C(NCC(F)=C1CN(C(=O)c2ncn3cccnc23)C1)c1nsnc1O s275592__15865378__15842482__15863240
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ncc1C#N s275592__15865378__15842482__15863244
Cc1cnc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863246
O=C(NCC(F)=C1CN(C(=O)c2csc(CO)n2)C1)c1nsnc1O s275592__15865378__15842482__15863250
CCC(C)(C)OCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863252
CC(=O)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15863254
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__15863258
Cn1ccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15863260
Cc1ncc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15863262
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15863264
O=C1NC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842482__15863266
CCC1(CC)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863270
CN1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863276
O=C(NCC(F)=C1CN(C(=O)c2cccc3nnoc23)C1)c1nsnc1O s275592__15865378__15842482__15863280
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnc1F s275592__15865378__15842482__15863282
Cc1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15863286
O=C(NCC(F)=C1CN(C(=O)C2CCN2C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15863288
CC1(O)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863290
CCCCCC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863294
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15855626
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)cc2)C1)c1nsnc1O s275592__15865378__15842482__15855632
C=CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855634
O=C(NCC(F)=C1CN(C(=O)c2cc(=O)[nH]c(=O)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15855636
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)OCO3)C1)c1nsnc1O s275592__15865378__15842482__15855638
CN(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855640
Nc1ccc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855642
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CCOC1C(C)C1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857420
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CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC(=O)C1 s275592__15865378__15842482__15857496
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Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(N)c1C s275592__15865378__15842482__15859414
COc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15842482__15859418
CC(C)n1ncnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859420
CC(C)C(O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859422
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COC(C)C(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859432
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CC1CN(C(C)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859468
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__15859476
Nc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1F s275592__15865378__15842482__15859478
CC1CCN1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859482
COC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CC1 s275592__15865378__15842482__15859488
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(F)cc2)C1)c1nsnc1O s275592__15865378__15842482__15861336
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1N s275592__15865378__15842482__15861338
CC(C)OC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15861340
Cc1ccc(N)c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861344
CC1(C)CC2(CC2C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861346
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CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(C#N)C1 s275592__15865378__15842482__15861388
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Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__15861396
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Cn1cnnc1SCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861412
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Cc1ccc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861422
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CCc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861426
Nc1nc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15861442
O=C(NCC(F)=C1CN(C(=O)C2(n3cncn3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15863296
Cn1cccc1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863298
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Cn1c(C#N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863302
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Cc1nc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]c1C s275592__15865378__15842482__15863316
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)n1cnnn1 s275592__15865378__15842482__15863326
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CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842482__15863336
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CC1(C#CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15842482__15863376
CC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(F)F s275592__15865378__15842482__15863380
CC(C)(C)C1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15863382
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1C s275592__15865378__15842482__15863388
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CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842482__15863398
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COC(=O)[C@@H]1CCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863406
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CC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855680
CCCCCC(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855684
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Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc(O)n1 s275592__15865378__15842482__15855692
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CCc1nc(C)ncc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855714
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Cc1[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)c1C s275592__15865378__15842482__15855718
O=C(NCC(F)=C1CN(C(=O)CN2CCCC2CO)C1)c1nsnc1O s275592__15865378__15842482__15855720
C[C@@H](O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855722
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccn3n2)C1)c1nsnc1O s275592__15865378__15842482__15855724
CCCCSCCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855726
CCN(CC)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855728
Cc1n[nH]c(SCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15855730
CC1CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15855732
CC(OC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855734
CNc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855738
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)csc1C s275592__15865378__15842482__15855742
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15855744
CCOC=C(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855752
CC(C)(C#N)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855756
CCn1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1O s275592__15865378__15842482__15855758
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__15855764
O=C(NCC(F)=C1CN(C(=O)CN2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15855766
CC(C)C(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855768
Nc1cc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15855770
COc1noc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855772
O=C(NCC(F)=C1CN(C(=O)C2=C(Cl)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15855780
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)SC s275592__15865378__15842482__15855784
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CO1 s275592__15865378__15842482__15855790
CC(=O)CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855792
CC1CC=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15857504
CC(O)C(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857506
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCOCC2)C1)c1nsnc1O s275592__15865378__15842482__15857508
Cc1ccnc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857510
Cc1cc(CO)oc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857514
O=C(NCC(F)=C1CN(C(=O)C2(O)CCOC2)C1)c1nsnc1O s275592__15865378__15842482__15857516
CCC(C)(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857522
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1O s275592__15865378__15842482__15857524
COc1ccc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857526
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)on2)C1)c1nsnc1O s275592__15865378__15842482__15857530
O=C(NCC(F)=C1CN(C(=O)C2SCCCS2)C1)c1nsnc1O s275592__15865378__15842482__15857532
O=C(NCC(F)=C1CN(C(=O)C2CC23CCSCC3)C1)c1nsnc1O s275592__15865378__15842482__15857534
C=C1CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857536
O=C(NCC(F)=C1CN(C(=O)CC2CC=CC2)C1)c1nsnc1O s275592__15865378__15842482__15857548
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)o2)C1)c1nsnc1O s275592__15865378__15842482__15857552
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2CO)C1)c1nsnc1O s275592__15865378__15842482__15857558
CC(=O)OC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857560
O=C(NCC(F)=C1CN(C(=O)CC2OCCO2)C1)c1nsnc1O s275592__15865378__15842482__15857568
COC(OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857572
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnc1S s275592__15865378__15842482__15857574
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)c(F)c2)C1)c1nsnc1O s275592__15865378__15842482__15857576
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC=CC1 s275592__15865378__15842482__15857578
O=C(NCC(F)=C1CN(C(=O)CCC[N+](=O)[O-])C1)c1nsnc1O s275592__15865378__15842482__15857582
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2cccnc2)C1)c1nsnc1O s275592__15865378__15842482__15857584
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15857586
[N-]=[N+]=Nc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15857588
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(Cl)n1 s275592__15865378__15842482__15857600
Nc1cccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857602
O=C(NCC(F)=C1CN(C(=O)c2cccc(Cl)n2)C1)c1nsnc1O s275592__15865378__15842482__15857612
COC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857614
O=C(NCC(F)=C1CN(C(=O)c2cccc([N+](=O)[O-])c2)C1)c1nsnc1O s275592__15865378__15842482__15857622
CCN(CC)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857624
COC(=O)C1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859490
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(Cl)nc2)C1)c1nsnc1O s275592__15865378__15842482__15859500
O=C(NCC(F)=C1CN(C(=O)C2=CCCOC2)C1)c1nsnc1O s275592__15865378__15842482__15859502
N#Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15859504
CCn1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842482__15859508
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC(C2)C3=O)C1)c1nsnc1O s275592__15865378__15842482__15859512
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1(F)F s275592__15865378__15842482__15859514
Nc1nnn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15859516
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__15859520
CC(C)(C)C(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859522
CCCCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859528
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15842482__15859530
O=C(NCC(F)=C1CN(C(=O)C2CCSCC2)C1)c1nsnc1O s275592__15865378__15842482__15859532
Nc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__15859534
COCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15859536
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)NCC3)C1)c1nsnc1O s275592__15865378__15842482__15859540
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15859546
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)COC1 s275592__15865378__15842482__15859548
Cc1nc(Cl)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859550
Cc1cc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15859552
Cn1nc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859556
O=C(NCC(F)=C1CN(C(=O)C2=CCCCO2)C1)c1nsnc1O s275592__15865378__15842482__15859558
Cn1cc(C#N)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859560
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15842482__15859562
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__15859564
O=C(NCC(F)=C1CN(C(=O)c2cc(CO)on2)C1)c1nsnc1O s275592__15865378__15842482__15859574
CCNc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cs1 s275592__15865378__15842482__15859576
CC1CC(=O)NCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859578
CSCCC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859580
O=C1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__15859582
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2COCC3)C1)c1nsnc1O s275592__15865378__15842482__15859586
CCNc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15859592
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]ncc3n2)C1)c1nsnc1O s275592__15865378__15842482__15859596
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCS1 s275592__15865378__15842482__15859604
O=C(NCC(F)=C1CN(C(=O)C2=CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15859608
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(N)n1 s275592__15865378__15842482__15859612
Cc1csc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861462
CCC[C@H](O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861464
O=C(NCC(F)=C1CN(C(=O)C2CCCn3cnnc32)C1)c1nsnc1O s275592__15865378__15842482__15861466
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC=CCC1 s275592__15865378__15842482__15861470
O=C(NCC(F)=C1CN(C(=O)c2csc3nccn23)C1)c1nsnc1O s275592__15865378__15842482__15861472
Cn1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861476
CC(C)(C)n1nccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861480
CC1(C)C2CCC(C2)C1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861482
CC1(C)C2CCC1(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)CC2 s275592__15865378__15842482__15861486
C#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__15861488
O=C(NCC(F)=C1CN(C(=O)C2(C3CCOCC3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15861492
O=C(NCC(F)=C1CN(C(=O)CC2COCCO2)C1)c1nsnc1O s275592__15865378__15842482__15861498
CC(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)COC1 s275592__15865378__15842482__15861502
Cn1ncc(N)c1CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861508
O=C(NCC(F)=C1CN(C(=O)C2(n3cccn3)CC2)C1)c1nsnc1O s275592__15865378__15842482__15861510
Nc1ccnn1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861512
CC1(C)CCC=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861514
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c[nH]1 s275592__15865378__15842482__15861516
O=C(NCC(F)=C1CN(C(=O)c2cn3ccncc3n2)C1)c1nsnc1O s275592__15865378__15842482__15861518
CN(C)Cc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861522
CC(C)(C)C1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861526
CCc1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__15861528
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C(O)C2CC2)C1)c1nsnc1O s275592__15865378__15842482__15861530
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCO1 s275592__15865378__15842482__15861532
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCOC2)C1)c1nsnc1O s275592__15865378__15842482__15861534
CSC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842482__15861540
C#CCCC1(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N=N1 s275592__15865378__15842482__15861546
Nc1cc(O)c(O)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15861548
CC1(O)CCC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15861552
COC1(C#N)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861554
CC1CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861556
[N-]=[N+]=NCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15861558
Cn1ncnc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861562
O=C1CSC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__15861570
C[C@H]1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C[C@@H](C)O1 s275592__15865378__15842482__15861572
CC(C)n1ccnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861574
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCC(O)CC1 s275592__15865378__15842482__15861576
CC1(OCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__15861580
O=C(NCC(F)=C1CN(C(=O)c2coc3c2CSC3)C1)c1nsnc1O s275592__15865378__15842482__15863420
CCc1occ(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863422
O=C(NCC(F)=C1CN(C(=O)C2CC3COCCN3C2)C1)c1nsnc1O s275592__15865378__15842482__15863430
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)cn1 s275592__15865378__15842482__15863434
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CCCO2)C1)c1nsnc1O s275592__15865378__15842482__15863436
CC(=O)N1C[C@H](O)C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863438
CC(C)(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15863444
Cc1c[nH]c(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15863448
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__15863454
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15842482__15863462
COc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1F s275592__15865378__15842482__15863464
CC1(C)[C@H]2C[C@H](C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)C[C@H]21 s275592__15865378__15842482__15863468
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]1 s275592__15865378__15842482__15863472
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N1CCC1 s275592__15865378__15842482__15863476
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15863478
O=C(NCC(F)=C1CN(C(=O)[C@H](O)Cc2c[nH]cn2)C1)c1nsnc1O s275592__15865378__15842482__15863486
O=C(NCC(F)=C1CN(C(=O)C#CC2CCCCC2)C1)c1nsnc1O s275592__15865378__15842482__15863488
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCOC3)C2)C1)c1nsnc1O s275592__15865378__15842482__15863502
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)CN(C)C s275592__15865378__15842482__15863504
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n[nH]c1=O s275592__15865378__15842482__15863506
O=C(NCC(F)=C1CN(C(=O)[C@H]2CC2(F)F)C1)c1nsnc1O s275592__15865378__15842482__15863508
CC(C)c1cnn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863512
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C=CCC1 s275592__15865378__15842482__15863516
O=C(NCC(F)=C1CN(C(=O)Cc2cn[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__15863518
COCC1(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCC1 s275592__15865378__15842482__15863520
Nc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15863522
CN(C)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15863524
O=C(NCC(F)=C1CN(C(=O)C(F)c2ccc(F)cc2)C1)c1nsnc1O s275592__15865378__15842482__15863532
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CS(=O)(=O)C1 s275592__15865378__15842482__15863534
O=C(NCC(F)=C1CN(C(=O)c2cn(CCCF)nn2)C1)c1nsnc1O s275592__15865378__15842482__15863538
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842482__15855796
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)=NN1 s275592__15865378__15842482__15855798
CCc1csc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15855800
CC(C)(C)CC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855802
CC(=O)C(C)(C)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855804
O=C(NCC(F)=C1CN(C(=O)c2cnc(F)cc2F)C1)c1nsnc1O s275592__15865378__15842482__15855810
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(F)c2)C1)c1nsnc1O s275592__15865378__15842482__15855812
CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(=O)C1 s275592__15865378__15842482__15855814
O=C(NCC(F)=C1CN(C(=O)Cc2cc[nH]c2)C1)c1nsnc1O s275592__15865378__15842482__15855816
CCc1nc(N)sc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855828
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C2(O)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15855830
O=C(NCC(F)=C1CN(C(=O)c2cc3ccncc3[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15855832
CCCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855836
CCOC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855838
O=C(NCC(F)=C1CN(C(=O)Cc2cccnc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15855842
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3cn2)C1)c1nsnc1O s275592__15865378__15842482__15855846
COC(=O)C(C)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855852
O=C(NCC(F)=C1CN(C(=O)CC2CCSCC2)C1)c1nsnc1O s275592__15865378__15842482__15855854
O=C(NCC(F)=C1CN(C(=O)C(CO)c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15855856
Cc1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15855858
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]2c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15855862
CC(O)(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C1CCC1 s275592__15865378__15842482__15855864
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)O1 s275592__15865378__15842482__15855868
Nc1cccn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1=O s275592__15865378__15842482__15855870
CC(=O)CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15855876
CC(O)c1cn(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1 s275592__15865378__15842482__15855878
Cn1nccc1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855880
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15855882
O=C(NCC(F)=C1CN(C(=O)CC2CSC2)C1)c1nsnc1O s275592__15865378__15842482__15855884
Cc1[nH]nc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1[N+](=O)[O-] s275592__15865378__15842482__15855886
O=C(NCC(F)=C1CN(C(=O)c2cnc3ncccn23)C1)c1nsnc1O s275592__15865378__15842482__15855888
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)oc1C s275592__15865378__15842482__15855890
COCCNC(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855892
O=C(NCC(F)=C1CN(C(=O)C2(F)CCC2)C1)c1nsnc1O s275592__15865378__15842482__15855898
Cn1cc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15855902
CC(C)c1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cnn1C s275592__15865378__15842482__15855904
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCCCC1 s275592__15865378__15842482__15855906
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc(Cl)n1 s275592__15865378__15842482__15855908
CN1N=C(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1=O s275592__15865378__15842482__15857632
O=C(NCC(F)=C1CN(C(=O)c2cnc[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15857636
O=C(NCC(F)=C1CN(C(=O)c2ccc3cn[nH]c3c2)C1)c1nsnc1O s275592__15865378__15842482__15857640
Cc1noc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15857642
CCOC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857644
CCc1noc(CCC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15857652
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15857654
CSc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15857656
O=C(NCC(F)=C1CN(C(=O)Cn2ccnn2)C1)c1nsnc1O s275592__15865378__15842482__15857670
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1N s275592__15865378__15842482__15857672
CN1CCCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857674
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__15857678
O=C(NCC(F)=C1CN(C(=O)CCc2ncc(F)cn2)C1)c1nsnc1O s275592__15865378__15842482__15857682
C=CC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15842482__15857684
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15857686
O=C(NCC(F)=C1CN(C(=O)c2ccnc(Cl)c2O)C1)c1nsnc1O s275592__15865378__15842482__15857688
O=C(NCC(F)=C1CN(C(=O)C2(O)COC2)C1)c1nsnc1O s275592__15865378__15842482__15857690
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(F)c1 s275592__15865378__15842482__15857692
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)nc2F)C1)c1nsnc1O s275592__15865378__15842482__15857694
CCC(C)C(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857696
O=C(NCC(F)=C1CN(C(=O)c2ncncc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15857702
COc1cc(N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857704
CC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)=C1CC1 s275592__15865378__15842482__15857712
CC1CN2CCN1CC2C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857714
Cc1cc(N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857726
CC1CC(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857728
CCn1cc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15857730
COC(=O)N[C@@H](C)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857732
Cc1c(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)nn1C s275592__15865378__15842482__15857734
N#CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1 s275592__15865378__15842482__15857738
CC1=NN(C)C(=O)C1CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857742
N#Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15857744
CC1=CC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857746
CN(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15857748
O=C(NCC(F)=C1CN(C(=O)CN2CCCOC2=O)C1)c1nsnc1O s275592__15865378__15842482__15859618
O=C(NCC(F)=C1CN(C(=O)c2cccc3occc23)C1)c1nsnc1O s275592__15865378__15842482__15859624
CC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15859626
Cc1cnc(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)s1 s275592__15865378__15842482__15859640
Nc1cnc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15859642
CCc1cc(N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859644
CCc1sc(N)nc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859646
Cn1ccc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4nsnc4O)C3)cc21 s275592__15865378__15842482__15859656
O=C1CCCCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859658
CN(C)CC(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859662
O=C1CCCCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15859666
CN1C2CCC1CC(C(=O)N1CC(=C(F)CNC(=O)c3nsnc3O)C1)C2 s275592__15865378__15842482__15859670
CCCC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859672
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15842482__15859674
CCCCC(O)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859676
O=C(NCC(F)=C1CN(C(=O)Cc2ncncc2Cl)C1)c1nsnc1O s275592__15865378__15842482__15859678
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15842482__15859680
Cc1cc(C#N)cnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859686
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC(=O)N1 s275592__15865378__15842482__15859688
COC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)C(C)O s275592__15865378__15842482__15859690
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)ccn1C1CC1 s275592__15865378__15842482__15859694
O=C(NCC(F)=C1CN(C(=O)CSC2CC2)C1)c1nsnc1O s275592__15865378__15842482__15859698
O=C(NCC(F)=C1CN(C(=O)CCCC2CCC2)C1)c1nsnc1O s275592__15865378__15842482__15859702
CC(C)(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)on1 s275592__15865378__15842482__15859704
O=C(NCC(F)=C1CN(C(=O)c2cncc(C(F)F)c2)C1)c1nsnc1O s275592__15865378__15842482__15859708
CCC(O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859710
CCCCC[C@@H](O)CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859716
Cc1cc(N)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15859718
CN1C(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15859720
O=C(NCC(F)=C1CN(C(=O)c2ccn3ccsc23)C1)c1nsnc1O s275592__15865378__15842482__15859726
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2CCCC[C@H]2O)C1)c1nsnc1O s275592__15865378__15842482__15859730
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c(O)c1 s275592__15865378__15842482__15859732
Nc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1F s275592__15865378__15842482__15859734
CCn1nnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1C s275592__15865378__15842482__15859736
N#Cc1cn[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861586
O=C(NCC(F)=C1CN(C(=O)C2CCc3cn[nH]c32)C1)c1nsnc1O s275592__15865378__15842482__15861590
CNC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861592
COC(=O)C1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861598
O=C(NCC(F)=C1CN(C(=O)CCc2cnoc2)C1)c1nsnc1O s275592__15865378__15842482__15861604
O=C(NCC(F)=C1CN(C(=O)Cc2cnsc2)C1)c1nsnc1O s275592__15865378__15842482__15861610
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2CCCN3)C1)c1nsnc1O s275592__15865378__15842482__15861620
C=CCC(C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1)N(C)C s275592__15865378__15842482__15861626
CCCC(C(=O)OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861644
O=C(NCC(F)=C1CN(C(=O)CCCCF)C1)c1nsnc1O s275592__15865378__15842482__15861646
CC1(C)CCCCC1=CC(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861648
CCC1CC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CCC1=O s275592__15865378__15842482__15861652
O=C(NCC(F)=C1CN(C(=O)c2ccnc3[nH]ccc23)C1)c1nsnc1O s275592__15865378__15842482__15861660
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCCN3C2)C1)c1nsnc1O s275592__15865378__15842482__15861664
O=C(NCC(F)=C1CN(C(=O)[C@@H](O)c2ccccc2)C1)c1nsnc1O s275592__15865378__15842482__15861666
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ccn2)C1)c1nsnc1O s275592__15865378__15842482__15861668
O=C(NCC(F)=C1CN(C(=O)c2cc(O)cs2)C1)c1nsnc1O s275592__15865378__15842482__15861670
Cc1cc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1C s275592__15865378__15842482__15861672
CC1CC(=O)NC1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861676
O=C(NCC(F)=C1CN(C(=O)c2cnsc2)C1)c1nsnc1O s275592__15865378__15842482__15861686
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cc1Cl s275592__15865378__15842482__15861688
O=C(NCC(F)=C1CN(C(=O)c2cncc(Cl)n2)C1)c1nsnc1O s275592__15865378__15842482__15861692
Cn1nc(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15861694
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)C1 s275592__15865378__15842482__15861700
CN1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15861704
O=C(NCC(F)=C1CN(C(=O)c2ccccc2[N+](=O)[O-])C1)c1nsnc1O s275592__15865378__15842482__15855502
CN1CCC(O)(CC(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15855514
O=C(NCC(F)=C1CN(C(=O)C2CCCSC2)C1)c1nsnc1O s275592__15865378__15842482__15855516
O=C1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)N1 s275592__15865378__15842482__15855518
Cc1cccc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)c1 s275592__15865378__15842482__15855522
Cc1ncc(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855524
Cn1cc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)n1 s275592__15865378__15842482__15855526
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)n(O)c2)C1)c1nsnc1O s275592__15865378__15842482__15855528
CC(C)C=C(C#N)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855536
Nc1csnc1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855538
O=C(NCC(F)=C1CN(C(=O)Cn2cncn2)C1)c1nsnc1O s275592__15865378__15842482__15855544
COC1(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842482__15855548
CCC(C(=O)OC)C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855550
O=C(NCC(F)=C1CN(C(=O)C2CSC2)C1)c1nsnc1O s275592__15865378__15842482__15855552
O=C(NCC(F)=C1CN(C(=O)c2cnc3sccn23)C1)c1nsnc1O s275592__15865378__15842482__15855556
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)o1 s275592__15865378__15842482__15855558
O=C(NCC(F)=C1CN(C(=O)CC2(CO)CC2)C1)c1nsnc1O s275592__15865378__15842482__15855560
N#Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3nsnc3O)C2)cn1 s275592__15865378__15842482__15855572
O=C(NCC(F)=C1CN(C(=O)Cc2nccs2)C1)c1nsnc1O s275592__15865378__15842482__15855582
O=C(NCC(F)=C1CN(C(=O)C2CCC=CO2)C1)c1nsnc1O s275592__15865378__15842482__15855594
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2NCCC3)C1)c1nsnc1O s275592__15865378__15842482__15855604
O=C(NCC(F)=C1CN(C(=O)Cc2cc(=O)[nH]c(=O)[nH]2)C1)c1nsnc1O s275592__15865378__15842482__15855608
O=C(NCC(F)=C1CN(C(=O)C2(O)CCCC2)C1)c1nsnc1O s275592__15865378__15842482__15855622
Nc1cccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2nsnc2O)C1 s275592__15865378__15842482__15855624
CCC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842484__15862300
CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15842484__15859360
CCC(C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)C s275592__15865378__15842484__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(=O)n(C2CC2)c1 s275592__15865378__15842486__15859360
CC(C)Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)no1 s275592__15865378__15842488__15862300
CC(C)Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)no1 s275592__15865378__15842488__15859360
Cc1nc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)ccc2n1C s275592__15865378__15842490__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(-n2cncn2)c1 s275592__15865378__15842492__15859360
CCS(=O)(=O)C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842494__15862300
CCS(=O)(=O)C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842494__15859360
CC(O)CCCCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842496__15862300
CC(O)CCCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842496__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ncn2ccccc12 s275592__15865378__15842498__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ncn2ccccc12 s275592__15865378__15842498__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC2C(C1)C2(F)F s275592__15865378__15842500__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCOC1C(F)(F)F s275592__15865378__15842504__15859360
Cn1cncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1=O s275592__15865378__15842506__15862300
Cn1cncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15842506__15859360
CSC(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842508__15862300
CSC(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842508__15859360
CSC(C)(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842508__15857566
CC1CN(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)O1 s275592__15865378__15842512__15862300
CC1CN(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)O1 s275592__15865378__15842512__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccncc1 s275592__15865378__15842516__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccncc1 s275592__15865378__15842516__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(Cl)ncc1F s275592__15865378__15842520__15859360
NC(=O)[C@@H]1CCCC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842524__15862300
NC(=O)[C@@H]1CCCC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842524__15859360
O=C(Cc1cnns1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842528__15862300
O=C(Cc1cnns1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842528__15859360
O=C(Cc1cnns1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842528__15857566
Cc1oc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc1CO s275592__15865378__15842530__15862300
Cc1oc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1CO s275592__15865378__15842530__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)=C1CCC1 s275592__15865378__15842534__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)=C1CCC1 s275592__15865378__15842534__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)=C1CCC1 s275592__15865378__15842534__15857566
CCC(CO)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842536__15862300
CCC(CO)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842536__15859360
CCC(CO)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842536__15857566
CC(C)(O)C(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842538__15862300
CC(C)(O)C(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842538__15859360
CC(C)(O)C(F)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842538__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1OCCO s275592__15865378__15842540__15859360
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)CCc1ccccc1 s275592__15865378__15842542__15859360
CCSc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15842544__15859360
O=C(CCN1CCC(O)CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842546__15862300
O=C(CCN1CCC(O)CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842546__15859360
Cn1ccnc1SCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842548__15859360
O=C(CCOc1cccnc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842550__15862300
O=C(CCOc1cccnc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842550__15859360
CCCN1CCCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842552__15862300
CCCN1CCCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842552__15859360
CC(C)CCOCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842556__15862300
CC(C)CCOCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842556__15859360
O=C(COCc1ccco1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842558__15862300
O=C(COCc1ccco1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842558__15859360
CC(CO)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842560__15862300
CC(CO)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842560__15859360
CC(CO)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842560__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2sccc2cn1 s275592__15865378__15842562__15859360
CCN1CCN(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842564__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnoc1 s275592__15865378__15842566__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnoc1 s275592__15865378__15842566__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cnoc1 s275592__15865378__15842566__15857566
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(F)cc1 s275592__15865378__15844304__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15844304__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CCCN2CCCC[C@H]12 s275592__15865378__15844306__15859360
CC(C)COC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15844308__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@@]23CCCCC[C@H]2OCC3)C1 s275592__15865378__15844310__15859360
O=C(Cc1ccc2ocnc2c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844312__15859360
CC1(C)CC(=O)NCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844314__15862300
CC1(C)CC(=O)NCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844314__15859360
CN(C)C(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cscn1 s275592__15865378__15844316__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnn(CCO)c1 s275592__15865378__15844318__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnn(CCO)c1 s275592__15865378__15844318__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@H]2C[C@@H](OC(F)F)C2)C1 s275592__15865378__15844320__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@H]2C[C@@H](OC(F)F)C2)C1 s275592__15865378__15844320__15859360
CCc1[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc1Cl s275592__15865378__15844322__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccn2nncc12 s275592__15865378__15844324__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccn2nncc12 s275592__15865378__15844324__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c2cnccc2c1 s275592__15865378__15844326__15859360
CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1(O)CCCCC1 s275592__15865378__15844328__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)c2cscn2)C1 s275592__15865378__15844332__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1csc2cncn12 s275592__15865378__15844334__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1csc2cncn12 s275592__15865378__15844334__15859360
CC(C)(C)c1noc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844336__15862300
CC(C)(C)c1noc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844336__15859360
C=C(F)C1(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15844338__15862300
C=C(F)C1(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15844338__15859360
Cc1cccc(NC(=O)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844340__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(=O)[nH][nH]c2c1 s275592__15865378__15844342__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC2CCC(C1)S2 s275592__15865378__15844344__15859360
CC1(c2cccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c2)CC1 s275592__15865378__15844346__15859360
O=C(CC1CCC2CC2C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844348__15862300
O=C(CC1CCC2CC2C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844348__15859360
Cn1ncc2ccnc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c21 s275592__15865378__15844350__15859360
CC1(OCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15844352__15859360
CC(C)n1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15844354__15859360
Cc1ccsc1C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844358__15862300
Cc1ccsc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844358__15859360
Cc1ccccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844360__15862300
Cc1ccccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844360__15859360
CCc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15844364__15859360
O=C(C=Cc1ccc2c(c1)CCO2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844366__15859360
O=C(C=Cc1c[nH]cn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844368__15862300
O=C(C=Cc1c[nH]cn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844368__15859360
O=C(C=Cc1c[nH]cn1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844368__15857566
Cc1csc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844372__15862300
Cc1csc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844372__15859360
O=C(C=Cc1ccc(F)c(F)c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844374__15859360
O=C(C=Cc1cncs1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844376__15862300
O=C(C=Cc1cncs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844376__15859360
Cc1cc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15844380__15859360
O=C(C=Cc1ccc(C2CC2)cc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844382__15859360
O=C(C=Cc1ncc[nH]1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844384__15862300
O=C(C=Cc1ncc[nH]1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844384__15859360
O=C(C=Cc1ncc[nH]1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844384__15857566
Cn1cc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nn1 s275592__15865378__15844386__15862300
Cn1cc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15844386__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@]23C[C@H]2COC32CCC2)C1 s275592__15865378__15844388__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@]23C[C@H]2COC32CCC2)C1 s275592__15865378__15844388__15859360
CCC1(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)COC1 s275592__15865378__15844390__15862300
CCC1(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15844390__15859360
CCC1(CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)COC1 s275592__15865378__15844390__15857566
Cn1nccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844396__15862300
Cn1nccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844396__15859360
O=C(C=Cc1cn[nH]c1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844398__15862300
O=C(C=Cc1cn[nH]c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844398__15859360
O=C(C=Cc1cn[nH]c1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844398__15857566
CCc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)o1 s275592__15865378__15844402__15862300
CCc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15844402__15859360
Cc1cc(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15844404__15862300
Cc1cc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15844404__15859360
O=C(C=Cc1nc2ccccc2o1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844408__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CS(=O)(=O)C1 s275592__15865378__15844412__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1C[C@H]1CF s275592__15865378__15844414__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1C[C@H]1CF s275592__15865378__15844414__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)[C@@H]1C[C@H]1CF s275592__15865378__15844414__15857566
CC(C)CN1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15844416__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnc2n1CCS2 s275592__15865378__15844418__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2n1CCS2 s275592__15865378__15844418__15859360
COc1ccccc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844420__15859360
O=C(C=Cc1cc(F)ccc1F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844422__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1CO[C@@H]2CCCC[C@H]12 s275592__15865378__15844424__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CO[C@@H]2CCCC[C@H]12 s275592__15865378__15844424__15859360
C=CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCOCC1 s275592__15865378__15846106__15862300
C=CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15846106__15859360
Cc1cccc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)nn12 s275592__15865378__15846110__15859360
O=C(CC1CC2(CCC2)CO1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846112__15862300
O=C(CC1CC2(CCC2)CO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846112__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CC2CCCCCC12 s275592__15865378__15846114__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CC2CCCCCC12 s275592__15865378__15846114__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnn2c1C(=O)NCC2 s275592__15865378__15846116__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nnc2n1CCCC2 s275592__15865378__15846120__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nnc2n1CCCC2 s275592__15865378__15846120__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1CCCC[C@H]1O s275592__15865378__15846122__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CCCC[C@H]1O s275592__15865378__15846122__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)[C@@H]1CCCC[C@H]1O s275592__15865378__15846122__15857566
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C=CCCC1 s275592__15865378__15846124__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C=CCCC1 s275592__15865378__15846124__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C=CCCC1 s275592__15865378__15846124__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CNc2ncnn2C1 s275592__15865378__15846126__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CNc2ncnn2C1 s275592__15865378__15846126__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2c(F)cccn12 s275592__15865378__15846128__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2ccnc2n1 s275592__15865378__15846130__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2ccnc2n1 s275592__15865378__15846130__15859360
O=C(CC1CC2(CC2)C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846134__15862300
O=C(CC1CC2(CC2)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846134__15859360
O=C(CC1CC2(CC2)C1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15846134__15857566
CCCN1C(=O)CCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846142__15862300
CCCN1C(=O)CCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846142__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnccc1C(F)F s275592__15865378__15846144__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnccc1C(F)F s275592__15865378__15846144__15859360
CC1CCCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15846146__15862300
CC1CCCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15846146__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cn1C s275592__15865378__15846148__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1C s275592__15865378__15846148__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1C s275592__15865378__15846148__15857566
CC12CC(CC(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)(CO1)C2 s275592__15865378__15846152__15862300
CC12CC(CC(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(CO1)C2 s275592__15865378__15846152__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(F)CC3(CCC3)C2)C1 s275592__15865378__15846154__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(F)CC3(CCC3)C2)C1 s275592__15865378__15846154__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCn2nccc2C1 s275592__15865378__15846160__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCn2nccc2C1 s275592__15865378__15846160__15859360
CC1CCCc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)nn21 s275592__15865378__15846162__15859360
CN(C)C1CCN(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15846164__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2sncc2c1 s275592__15865378__15846166__15859360
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]c2c1CCCC2 s275592__15865378__15846170__15859360
CCc1[nH]c(C)nc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846172__15862300
CCc1[nH]c(C)nc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846172__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2(CC(O)C2)C1 s275592__15865378__15846174__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(CC(O)C2)C1 s275592__15865378__15846174__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(CCF)cc1 s275592__15865378__15846176__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(CCF)cc1 s275592__15865378__15846176__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23COC(CF)(C2)C3)C1 s275592__15865378__15846178__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23COC(CF)(C2)C3)C1 s275592__15865378__15846178__15859360
Cn1nnc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15846180__15859360
NC(=O)c1cccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1F s275592__15865378__15846186__15859360
Cc1cc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15846188__15862300
Cc1cc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15846188__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCOC1 s275592__15865378__15846190__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCOC1 s275592__15865378__15846190__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCOC1 s275592__15865378__15846190__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2nc[nH]c(=O)c2c1 s275592__15865378__15846192__15859360
Cc1cn2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cnc2s1 s275592__15865378__15846194__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(c3ccncc3)CC2)C1 s275592__15865378__15846196__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(c3ccncc3)CC2)C1 s275592__15865378__15846196__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1coc(Cl)c1 s275592__15865378__15846200__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1coc(Cl)c1 s275592__15865378__15846200__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCc2cnnn2C1 s275592__15865378__15846204__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCc2cnnn2C1 s275592__15865378__15846204__15859360
CCOc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)oc(=O)c1 s275592__15865378__15846206__15859360
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c2cc[nH]c2n1 s275592__15865378__15846208__15859360
O=C(Cc1c[nH]c2cccnc12)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846210__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nnc1C s275592__15865378__15846212__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nnc1C s275592__15865378__15846212__15859360
CC1CCCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15846214__15862300
CC1CCCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15846214__15859360
CN(C)[C@H]1C[C@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15846216__15862300
CN(C)[C@H]1C[C@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15846216__15859360
CN(C)[C@H]1C[C@H](C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15846216__15857566
CSc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15846218__15859360
O=C1NCCCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846222__15862300
O=C1NCCCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846222__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nncn1C1CC1 s275592__15865378__15846224__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nncn1C1CC1 s275592__15865378__15846224__15859360
CC1(C)[C@@H](C(F)F)[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846228__15862300
CC1(C)[C@@H](C(F)F)[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846228__15859360
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nccs1 s275592__15865378__15840706__15862300
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nccs1 s275592__15865378__15840706__15859360
O=C(C=CBr)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840708__15862300
O=C(C=CBr)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840708__15859360
O=C(C=Cc1ccccc1F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840710__15862300
O=C(C=Cc1ccccc1F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840710__15859360
CC(CCN(C)C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840712__15862300
CC(CCN(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840712__15859360
CSc1nccnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840714__15862300
CSc1nccnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840714__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=Cc2ccccc2C1O s275592__15865378__15840716__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c(-c2ccncc2)n1 s275592__15865378__15840718__15859360
O=C(C=Cc1cccnc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840720__15862300
O=C(C=Cc1cccnc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840720__15859360
NC(=O)c1ccc(F)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840724__15859360
O=C(C=Cc1ccc(F)cc1F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840728__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC(C2CC2)C1 s275592__15865378__15840730__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC(C2CC2)C1 s275592__15865378__15840730__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC(C2CC2)C1 s275592__15865378__15840730__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cn(C2CC2)cn1 s275592__15865378__15840732__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn(C2CC2)cn1 s275592__15865378__15840732__15859360
Cc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc1 s275592__15865378__15840734__15862300
Cc1ccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15840734__15859360
CC(C)[C@H](NC=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840736__15862300
CC(C)[C@H](NC=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840736__15859360
Cc1cc(C)c(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15840738__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc2ncccc12 s275592__15865378__15840740__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cnc1C(F)F s275592__15865378__15840742__15859360
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cncnc1 s275592__15865378__15840746__15862300
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncnc1 s275592__15865378__15840746__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23OC4C5COCC4C2C53)C1 s275592__15865378__15840748__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2c1CCC2 s275592__15865378__15840750__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2c1CCC2 s275592__15865378__15840750__15859360
CCSC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15840754__15862300
CCSC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15840754__15859360
CCn1ccnc1C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840756__15862300
CCn1ccnc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840756__15859360
CCC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)n1cncn1 s275592__15865378__15840758__15862300
CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)n1cncn1 s275592__15865378__15840758__15859360
Cc1[nH]c(C(C)(C)C)cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840760__15859360
COc1ncc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15840762__15859360
CCCCCCC(O)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840766__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccnn1CCF s275592__15865378__15840768__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnn1CCF s275592__15865378__15840768__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(F)c(CO)c(F)c1 s275592__15865378__15840772__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc2nc[nH]c(=O)c12 s275592__15865378__15840776__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc(F)c(Cl)c1 s275592__15865378__15840778__15859360
CC1=NS(=O)(=O)NC=C1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840780__15859360
O=C(CC=C(Cl)Cl)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840782__15862300
O=C(CC=C(Cl)Cl)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840782__15859360
CN(C)C(=O)C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840786__15862300
CN(C)C(=O)C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840786__15859360
CN(C)C(=O)C=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840786__15857566
C#CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15840788__15862300
C#CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15840788__15859360
C#CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15840788__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccnc(CO)c1 s275592__15865378__15840790__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc(CO)c1 s275592__15865378__15840790__15859360
COc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(OC)n1 s275592__15865378__15840792__15859360
CN(CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1CCC[C@H]1O s275592__15865378__15840794__15862300
CN(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CCC[C@H]1O s275592__15865378__15840794__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(F)C(F)(F)C2(F)F)C1 s275592__15865378__15840796__15859360
CC(C)(C)c1ncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)o1 s275592__15865378__15840798__15862300
CC(C)(C)c1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15840798__15859360
C[C@H]1c2cn[nH]c2CC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840800__15859360
CC(=O)Nc1cnccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840802__15859360
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cs1 s275592__15865378__15840806__15862300
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15840806__15859360
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)cs1 s275592__15865378__15840806__15857566
CC(C)Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]n1 s275592__15865378__15840810__15862300
CC(C)Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15840810__15859360
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cnn1CCO s275592__15865378__15840812__15862300
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cnn1CCO s275592__15865378__15840812__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)CCc1ccccc1 s275592__15865378__15840814__15859360
C#CCN1CCCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840816__15862300
C#CCN1CCCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840816__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(OC(F)F)c1 s275592__15865378__15840818__15859360
Cc1cccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1[N+](=O)[O-] s275592__15865378__15840820__15859360
CC(Cc1ccccc1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840824__15862300
CC(Cc1ccccc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840824__15859360
O=C(Cn1cccnc1=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840826__15862300
O=C(Cn1cccnc1=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840826__15859360
O=C(CSCC1CCCCO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842568__15859360
CN1CCN(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842572__15862300
CN1CCN(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842572__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=COCC1 s275592__15865378__15842576__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=COCC1 s275592__15865378__15842576__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1=COCC1 s275592__15865378__15842576__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc2c(c1)OCC2 s275592__15865378__15842580__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(c1)OCC2 s275592__15865378__15842580__15859360
CSc1ccsc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842582__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nc(Cl)ccc1F s275592__15865378__15842588__15859360
Cc1nn(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1[N+](=O)[O-] s275592__15865378__15842590__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CCCSC1 s275592__15865378__15842592__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CCCSC1 s275592__15865378__15842592__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1=CCCSC1 s275592__15865378__15842592__15857566
Cc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(=O)[nH]1 s275592__15865378__15842596__15862300
Cc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15842596__15859360
C[C@H](O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842598__15862300
C[C@H](O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842598__15857566
Cc1nc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)sc1C s275592__15865378__15842600__15862300
Cc1nc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)sc1C s275592__15865378__15842600__15859360
CCN1CCN(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842602__15862300
CCN1CCN(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842602__15859360
C[C@@](O)(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccccc1 s275592__15865378__15842604__15862300
C[C@@](O)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15842604__15859360
CC1(c2ccccc2)CC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842606__15859360
COc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nc1 s275592__15865378__15842610__15862300
COc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15842610__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(F)n[nH]1 s275592__15865378__15842612__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(F)n[nH]1 s275592__15865378__15842612__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cc(F)n[nH]1 s275592__15865378__15842612__15857566
CC1(C)CC=C(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842616__15862300
CC1(C)CC=C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842616__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1C=CCC1 s275592__15865378__15842618__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1C=CCC1 s275592__15865378__15842618__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1C=CCC1 s275592__15865378__15842618__15857566
CC(C)(C)c1cccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15842620__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCC(O)C1 s275592__15865378__15842622__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCC(O)C1 s275592__15865378__15842622__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCCC(O)C1 s275592__15865378__15842622__15857566
CC1CC=C(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842624__15862300
CC1CC=C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842624__15859360
CC1CC=C(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842624__15857566
CC(O)C(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842626__15862300
CC(O)C(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842626__15859360
CC(O)C(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842626__15857566
O=C(CC1(O)CCOCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842628__15862300
O=C(CC1(O)CCOCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842628__15859360
Cc1ccnc(Cl)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842630__15862300
Cc1ccnc(Cl)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842630__15859360
Cc1cc(CO)oc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842632__15862300
Cc1cc(CO)oc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842632__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(O)CCOC2)C1 s275592__15865378__15842634__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(O)CCOC2)C1 s275592__15865378__15842634__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(O)CCOC2)C1 s275592__15865378__15842634__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(c1)C(=O)NC2 s275592__15865378__15842636__15859360
Cn1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc1O s275592__15865378__15842638__15862300
Cn1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15842638__15859360
Cn1nc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)cc1O s275592__15865378__15842638__15857566
COc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15842640__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(Cl)on1 s275592__15865378__15842642__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(Cl)on1 s275592__15865378__15842642__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC12CCSCC2 s275592__15865378__15842644__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC12CCSCC2 s275592__15865378__15842644__15859360
C=C1CC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842646__15862300
C=C1CC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842646__15859360
C=C1CC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842646__15857566
O=C(COc1cncc(Cl)n1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842648__15859360
O=C(CC1CC=CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842654__15862300
O=C(CC1CC=CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842654__15859360
O=C(CC1CC=CC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842654__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnoc1-c1ccoc1 s275592__15865378__15842656__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(C2CC2)o1 s275592__15865378__15842658__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(C2CC2)o1 s275592__15865378__15842658__15859360
COc1cc(CO)ccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842660__15859360
O=C(Cc1ccccc1CO)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842664__15862300
O=C(Cc1ccccc1CO)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842664__15859360
CN(C)c1noc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15842668__15859360
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CC2)C1 s275592__15865378__15842670__13186218
CC(C)(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186220
CC(F)(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186222
COCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186224
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccccn2)C1 s275592__15865378__15842670__13186226
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccncc2)C1 s275592__15865378__15842670__13186228
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(F)cc2)C1 s275592__15865378__15842670__13186230
CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186232
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccnc2)C1 s275592__15865378__15842670__13186234
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cccs2)C1 s275592__15865378__15842670__13186236
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccco2)C1 s275592__15865378__15842670__13186238
CC(=O)NCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186240
Cc1ccsc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186242
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)s1 s275592__15865378__15842670__13186244
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2ccco2)C1 s275592__15865378__15842670__13186246
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccccc2F)C1 s275592__15865378__15842670__13186248
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccccc2)C1 s275592__15865378__15842670__13186250
CC(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186252
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCCC2)C1 s275592__15865378__15842670__13186254
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnccn2)C1 s275592__15865378__15842670__13186256
Cc1ccccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186258
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCCC2)C1 s275592__15865378__15842670__13186260
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC2CCCC2)C1 s275592__15865378__15842670__13186262
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccc(F)c2)C1 s275592__15865378__15842670__13186264
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccs2)C1 s275592__15865378__15842670__13186266
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1 s275592__15865378__15842670__13186268
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2ccsc2)C1 s275592__15865378__15842670__13186270
CC1CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186272
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__13186274
CCOCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186276
CC(C)=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186278
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=COCCO2)C1 s275592__15865378__15842670__13186280
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc[n+]([O-])cc2)C1 s275592__15865378__15842670__13186282
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3C=CC2C3)C1 s275592__15865378__15842670__13186284
CC(=O)NC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186286
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(=O)[nH]n2)C1 s275592__15865378__15842670__13186288
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__13186290
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCCCC2)C1 s275592__15865378__15842670__13186292
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCO2)C1 s275592__15865378__15842670__13186294
CSCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186296
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)no1 s275592__15865378__15842670__13186298
CSCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186300
CC(C)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186302
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccsc2)C1 s275592__15865378__15842670__13186306
Cc1occc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186308
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2C=CCC2)C1 s275592__15865378__15842670__13186310
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2cnnn2)C1 s275592__15865378__15842670__13186312
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CN2CCCC2=O)C1 s275592__15865378__15842670__13186314
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1 s275592__15865378__15842670__13186316
Cc1noc(C)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186318
Cc1nnsc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186320
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c(C)o1 s275592__15865378__15842670__13186322
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC=CCC2)C1 s275592__15865378__15842670__13186324
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2ccco2)C1 s275592__15865378__15842670__13186326
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)on1 s275592__15865378__15842670__13186328
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc[nH]2)C1 s275592__15865378__15842670__13186330
CC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186334
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1C s275592__15865378__15842670__13186336
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccoc2)C1 s275592__15865378__15842670__13186338
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2cccn2)C1 s275592__15865378__15842670__13186340
Cc1ccoc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186342
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3CCC2C3)C1 s275592__15865378__15842670__13186344
Cc1c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cnn1C s275592__15865378__15842670__13186348
CCCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186350
CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186352
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1 s275592__15865378__15842670__13186354
Cn1cccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186356
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCn2cncn2)C1 s275592__15865378__15842670__13186358
CCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186362
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__13186364
CC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186366
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCn2cccn2)C1 s275592__15865378__15842670__13186368
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccccc2O)C1 s275592__15865378__15842670__13186370
CCC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186372
CC(C)SCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186374
N#CCSCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186376
CC(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186378
CCC(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186380
CC(C)OCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186382
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]n1 s275592__15865378__15842670__13186384
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC2CCCO2)C1 s275592__15865378__15842670__13186386
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2COCCO2)C1 s275592__15865378__15842670__13186388
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc[nH]n2)C1 s275592__15865378__15842670__13186390
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)n1cccn1 s275592__15865378__15842670__13186392
CCCCC(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186394
CSC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186396
CCOC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186398
CCOCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186402
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COCC2CC2)C1 s275592__15865378__15842670__13186404
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCCO2)C1 s275592__15865378__15842670__13186406
Cc1ncsc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186408
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cn[nH]c2)C1 s275592__15865378__15842670__13186410
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CNC(=O)C2CC2)C1 s275592__15865378__15842670__13186412
COCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186414
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COC2CCCC2)C1 s275592__15865378__15842670__13186416
Cc1ncncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186418
CCSCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186420
CCOC1CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186422
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnsn2)C1 s275592__15865378__15842670__13186424
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnns2)C1 s275592__15865378__15842670__13186426
COC(=O)NCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186428
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccon2)C1 s275592__15865378__15842670__13186430
CCCSCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186432
CC(=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__13186434
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]n1 s275592__15865378__15842670__13186436
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cncs2)C1 s275592__15865378__15842670__13186438
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n(C)n1 s275592__15865378__15842670__13186440
Cc1cnn(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__13186446
CCC=C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186452
CS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186454
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=C2CCCCC2)C1 s275592__15865378__15842670__13186456
Cc1ocnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186458
CCOC(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186460
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC(F)(F)F)C1 s275592__15865378__15842670__13186462
COC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186464
CC(C)OCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186466
CC(OCC1CC1)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186468
CCCOCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186470
C=CCCOC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186474
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCOC2)C1 s275592__15865378__15842670__13186476
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccnc(F)c2)C1 s275592__15865378__15842670__13186478
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)s1 s275592__15865378__15842670__13186480
Cn1nccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186482
CCC(OC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186484
COCCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186486
CCCC(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186488
COC(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186490
Cn1cc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1 s275592__15865378__15842670__13186492
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCCCC2)C1 s275592__15865378__15842670__13186494
C=CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186496
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=COCCC2)C1 s275592__15865378__15842670__13186498
COC(=O)C1CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186500
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCOC2)C1 s275592__15865378__15842670__13186504
CCOCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186506
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cscn2)C1 s275592__15865378__15842670__13186510
COCC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186512
CC(C)(C)CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186514
C=CCOCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186516
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cocn2)C1 s275592__15865378__15842670__13186518
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2CCC(=O)N2)C1 s275592__15865378__15842670__13186520
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2=CCCCC2)C1 s275592__15865378__15842670__13186522
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c[nH]1 s275592__15865378__15842670__13186524
CSCC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186526
CN1CCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186528
CCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186530
CC(C)(C)/C=C/C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186532
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(F)nc2)C1 s275592__15865378__15842670__13186534
CC(C#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186536
COCCOCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186538
CCCC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186540
Cc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186542
CC(C)(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186544
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3CCC2O3)C1 s275592__15865378__15842670__13186546
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)no1 s275592__15865378__15842670__13186548
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1 s275592__15865378__15842670__13186550
Nc1nccnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186552
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC2CC2)C1 s275592__15865378__15842670__13186554
Cc1[nH]nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1C s275592__15865378__15842670__13186556
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCOCC2)C1 s275592__15865378__15842670__13186558
CCCCOCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186560
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2ccon2)C1 s275592__15865378__15842670__13186562
CCc1ocnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186566
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCOC2)C1 s275592__15865378__15842670__13186568
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC=CC2)C1 s275592__15865378__15842670__13186570
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2ccn[nH]2)C1 s275592__15865378__15842670__13186572
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccncc2F)C1 s275592__15865378__15842670__13186574
Cc1c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nnn1C s275592__15865378__15842670__13186576
Cc1ccncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186578
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__13186580
Cc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__13186584
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC(F)(F)F)C1 s275592__15865378__15842670__13186586
C=CCOCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186588
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCC2)C1 s275592__15865378__15842670__13186592
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccc(=O)[nH]2)C1 s275592__15865378__15842670__13186596
CC1(C)C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1(C)C s275592__15865378__15842670__13186598
Cc1ncoc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186600
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__13186602
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2C3CCCC32)C1 s275592__15865378__15842670__13186604
N#Cc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__13186606
Cc1cscc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186608
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC2CCC2)C1 s275592__15865378__15842670__13186610
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__13186612
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2nnc[nH]2)C1 s275592__15865378__15842670__13186614
Cc1cccnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186616
Cc1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186618
CC=C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186620
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC2CCOC2)C1 s275592__15865378__15842670__13186622
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2ccoc2)C1 s275592__15865378__15842670__13186624
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC(F)(F)C2)C1 s275592__15865378__15842670__13186626
CC1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__13186628
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)=C1CCCC1 s275592__15865378__15842670__13186630
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCCCO2)C1 s275592__15865378__15842670__13186632
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n[nH]1 s275592__15865378__15842670__13186634
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=C2CCC2)C1 s275592__15865378__15842670__13186636
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cncc(F)c2)C1 s275592__15865378__15842670__13186638
CCC(=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)CC s275592__15865378__15842670__13186640
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc[nH]c(=O)c2)C1 s275592__15865378__15842670__13186642
CC(C)=C(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186644
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCNC(=O)C2)C1 s275592__15865378__15842670__13186646
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCC2)C1 s275592__15865378__15842670__13186648
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(F)=C2CCCC2)C1 s275592__15865378__15842670__13186650
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__13186652
Cn1cnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__13186654
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2COC(=O)C2)C1 s275592__15865378__15842670__13186656
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)oc1C s275592__15865378__15842670__13186658
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cccnc2)C1 s275592__15865378__15842670__13186660
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCCO2)C1 s275592__15865378__15842670__13186662
Cc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1O s275592__15865378__15842670__13186664
CCC(SC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186666
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)n1cccc1 s275592__15865378__15842670__13186668
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)ncn1 s275592__15865378__15842670__13186670
CC1(C)CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186672
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]1 s275592__15865378__15842670__13186674
CCC(C)OCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186676
CC1(C)C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186678
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__13186680
CC(O)(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__13186682
CC1=C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCO1 s275592__15865378__15842670__13186684
CSC(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186686
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CCCO2)C1 s275592__15865378__15842670__13186690
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)n1cncn1 s275592__15865378__15842670__13186692
NC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__13186694
Cc1nscc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186698
C#CCCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186700
CC(C)(C)OCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186702
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c[nH]1 s275592__15865378__15842670__13186704
C#CCNC(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186706
CCNC(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186708
COc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)on1 s275592__15865378__15842670__13186714
COC(C)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186716
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)co1 s275592__15865378__15842670__13186718
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(F)cn2)C1 s275592__15865378__15842670__13186720
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1N s275592__15865378__15842670__13186722
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cncnc2)C1 s275592__15865378__15842670__13186724
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ncccc2O)C1 s275592__15865378__15842670__13186726
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCOCC2)C1 s275592__15865378__15842670__13186730
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2ccoc2)C1 s275592__15865378__15842670__13186732
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)co1 s275592__15865378__15842670__13186736
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCCCC2)C1 s275592__15865378__15842670__13186740
C[C@H](NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186742
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)co1 s275592__15865378__15842670__13186746
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2ccc[nH]2)C1 s275592__15865378__15842670__13186748
Cc1ccn(C)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186750
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cnn1 s275592__15865378__15842670__13186752
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCn2ccnn2)C1 s275592__15865378__15842670__13186754
CC(=O)N1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__13186756
Cn1oc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cc1=O s275592__15865378__15842670__13186758
CCC(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186760
COC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__13186762
CC1OCCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186764
C#CCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186766
C=CC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186770
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)ns1 s275592__15865378__15842670__13186772
CCn1ccnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186778
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCOCC2)C1 s275592__15865378__15842670__13186780
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2ncc[nH]2)C1 s275592__15865378__15842670__13186782
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC(O)CC2)C1 s275592__15865378__15842670__13186784
CC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186786
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__13186788
COC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__13186790
CCc1occc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186792
Cc1cc[nH]c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186794
Cn1nncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186796
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2COC(=O)N2)C1 s275592__15865378__15842670__13186798
CCCCC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186800
CC1CC(C)C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)O1 s275592__15865378__15842670__13186802
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2C[C@@H]2C(F)F)C1 s275592__15865378__15842670__13186804
Cc1coc(C)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186806
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__13186810
CCc1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186812
CC(C)[C@@H](O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186814
CCOC1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__13186816
CC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15842670__13186818
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nn1 s275592__15865378__15842670__13186820
Cc1nnc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__13186822
Cn1cnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__13186824
CCn1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__13186830
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__13186832
CCn1nncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186834
Cc1csc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__13186836
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC2(F)F)C1 s275592__15865378__15842670__13186838
CCC(C)=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186840
Cc1cnccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186842
CC(C)C#CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186846
Cc1sccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186848
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2(O)CCC2)C1 s275592__15865378__15842670__13186850
Cc1c[nH]nc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186852
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)=C1CCC1 s275592__15865378__15842670__13186854
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C#CC2CC2)C1 s275592__15865378__15842670__13186856
CC(C)(C)C#CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186858
Cc1n[nH]c(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__13186860
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nn1 s275592__15865378__15842670__13186862
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2[N+](=O)[O-])C1 s275592__15865378__15842670__13186864
Cc1cn(C)nc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186866
Cn1ccc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__13186870
COCC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__13186872
CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186202
COCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186204
CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__13186206
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC2)C1 s275592__15865378__15842670__13186210
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC2)C1 s275592__15865378__15842670__13186212
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCC2)C1 s275592__15865378__15842670__13186214
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCOCC2)C1 s275592__15865378__15842670__13186216
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCC(=O)N2)C1 s275592__15865378__15842670__14130378
CNC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14130398
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__14130412
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cs1 s275592__15865378__15842670__14130442
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCOCC1 s275592__15865378__15842670__14130464
CC(C)CC(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130504
Cc1nnccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14135266
CN1CCC(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14130638
Cn1cncc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130640
CCn1cnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__14130668
CCC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)N(C)C s275592__15865378__15842670__14130682
CC1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C(C)O1 s275592__15865378__15842670__14135374
CC(C)(C)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14135380
CC1CC1C1CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14135384
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C[C@@H]2C[C@H]2C2CC2)C1 s275592__15865378__15842670__14135422
CC1COC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14135424
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@]23CCC[C@@H]2C3)C1 s275592__15865378__15842670__14135434
CC[C@@H]1OCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14135448
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)no1 s275592__15865378__15842670__14130744
CCC(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)C s275592__15865378__15842670__14130746
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CCC(=O)N2)C1 s275592__15865378__15842670__14130766
C[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14130782
CCCN(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130824
CC(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)(C)C s275592__15865378__15842670__14130832
Cc1[nH]cnc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130862
CCc1nc[nH]c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130946
Cc1n[nH]c(C)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131000
Cc1ncccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131050
CC(C)CCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131056
CC(C)(C)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131068
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccncn2)C1 s275592__15865378__15842670__14131070
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)ccn1 s275592__15865378__15842670__14131084
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2ccco2)C1 s275592__15865378__15842670__14131092
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ncccn2)C1 s275592__15865378__15842670__14131098
CCC(C)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131100
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccnn2)C1 s275592__15865378__15842670__14131112
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__14131126
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c(C)o1 s275592__15865378__15842670__14131130
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCn2cnnn2)C1 s275592__15865378__15842670__14131136
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ncccc2F)C1 s275592__15865378__15842670__14131150
CC1OCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131176
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCOC1 s275592__15865378__15842670__14131178
CCC(CC)(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131192
CC1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCO1 s275592__15865378__15842670__14131198
CCCC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131200
CCC(CC)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131202
CCC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131204
CCCC(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131208
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(=O)NCC2CC2)C1 s275592__15865378__15842670__14131216
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCOC1 s275592__15865378__15842670__14131230
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nn1 s275592__15865378__15842670__14131246
CCC1(C)CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131286
CC(C)C1(C)CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131290
COCC(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131300
CCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15842670__14131318
Cc1nonc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131322
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(C(F)F)CC2)C1 s275592__15865378__15842670__14131884
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC(F)C2)C1 s275592__15865378__15842670__14133584
CN(C)CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133608
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2c[nH]c(=O)cn2)C1 s275592__15865378__15842670__14133618
CCCC(CCC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133626
CC1(CCC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14131376
Cc1cnoc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131378
CCN(C)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131434
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC23CCCC3)C1 s275592__15865378__15842670__14131436
Cc1conc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131468
CCOC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__14131956
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2ncnn2)C1 s275592__15865378__15842670__14131964
CCCC[C@@H](C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131972
C=CCC(CC=C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131996
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC=CCC1 s275592__15865378__15842670__14132000
CCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132012
CC(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132018
C=CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132044
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2nccn2)C1 s275592__15865378__15842670__14132056
CC1CCCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133642
CC1CCCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14133644
Cc1ncccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133662
C=CCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133684
CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133690
CCCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133692
NC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133696
NC(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133704
Cc1nocc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133720
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCCC1 s275592__15865378__15842670__14133746
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133750
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC=CC1 s275592__15865378__15842670__14133772
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]c1=O s275592__15865378__15842670__14133774
COC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)C s275592__15865378__15842670__14133776
CC1CC1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133778
CCCCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133780
C=C1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133782
C=CCCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133784
C=CC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133786
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C[C@H]2CCOC2)C1 s275592__15865378__15842670__14133790
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__14133792
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2=CCOCC2)C1 s275592__15865378__15842670__14133794
CCc1ccoc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133796
CCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133798
CCC1CCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133804
CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14128908
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cc1 s275592__15865378__15842670__14128958
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC23CCOC3)C1 s275592__15865378__15842670__14131518
CCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131528
CC(C)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131540
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(C2CC2)C2CC2)C1 s275592__15865378__15842670__14131574
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2nc[nH]n2)C1 s275592__15865378__15842670__14131602
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCCC1 s275592__15865378__15842670__14131618
CCCC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)C s275592__15865378__15842670__14131642
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2C=CC=CC=C2)C1 s275592__15865378__15842670__14132090
C=C(C)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132092
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccns2)C1 s275592__15865378__15842670__14132118
CCC1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)O1 s275592__15865378__15842670__14132128
COCCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14132154
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14132156
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCNC2=O)C1 s275592__15865378__15842670__14132230
Cc1ncc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__14132232
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__14132244
CC1CCCC1(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133806
CC(F)(F)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133808
CCCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133812
C[C@@]1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC(=O)N1 s275592__15865378__15842670__14133814
CCc1nocc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133818
CC1COCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133820
Cc1c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)ccn1C s275592__15865378__15842670__14133822
COCC(OC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133826
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14133828
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCCO1 s275592__15865378__15842670__14133830
CCC[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133832
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C23CCCCC2C3)C1 s275592__15865378__15842670__14133834
CC(C)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14133836
C=C1CC(C)(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14133838
CC(C)(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)F s275592__15865378__15842670__14133840
Cc1ccoc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133842
CCc1ncoc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133844
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(CF)CC2)C1 s275592__15865378__15842670__14133872
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3(CC3)C2)C1 s275592__15865378__15842670__14133874
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)c1ccco1 s275592__15865378__15842670__14133916
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCNC1=O s275592__15865378__15842670__14133934
CC1CCCN1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133964
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(=O)[nH]c2)C1 s275592__15865378__15842670__14129048
CCCCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14129058
CC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131690
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14131742
CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__14131758
C#CCOCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131824
C#CCOC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14131828
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCOCC2CC2)C1 s275592__15865378__15842670__14131836
CC(C)(C(N)=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132330
Cc1ncn(C)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132342
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cncs2)C1 s275592__15865378__15842670__14132352
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cn[nH]c(=O)c2)C1 s275592__15865378__15842670__14132362
Cc1[nH]c(=O)[nH]c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132366
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(C3CC3)CC2)C1 s275592__15865378__15842670__14132386
COC1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14132390
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2CCCC(=O)N2)C1 s275592__15865378__15842670__14132392
CC1CCN(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14133972
NC(=O)[C@@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134008
CC[C@@H](C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)N(C)C s275592__15865378__15842670__14134026
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)(F)F s275592__15865378__15842670__14134028
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c(C)[nH]1 s275592__15865378__15842670__14134034
Cc1ccn(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__14134040
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2c[nH]nn2)C1 s275592__15865378__15842670__14134054
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(CF)CCC2)C1 s275592__15865378__15842670__14134056
C=C[C@@H]1OCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134058
CC(C)C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134062
CC[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134064
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]3CC[C@@H]2O3)C1 s275592__15865378__15842670__14134076
CC(C)CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134122
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2cncn2)C1 s275592__15865378__15842670__14129210
NC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14129250
Cc1cnccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132428
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC2(F)F)C1 s275592__15865378__15842670__14132438
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccsn2)C1 s275592__15865378__15842670__14132440
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCC1 s275592__15865378__15842670__14132466
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2C=CCCC2)C1 s275592__15865378__15842670__14132470
CCOCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14132486
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3C=CC2O3)C1 s275592__15865378__15842670__14132520
COC1CCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132536
CC1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CO1 s275592__15865378__15842670__14132538
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCC3CC32)C1 s275592__15865378__15842670__14132540
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCC3CC23)C1 s275592__15865378__15842670__14132542
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC3CC3C2)C1 s275592__15865378__15842670__14132544
COC1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14132548
CCC(CC)C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132570
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC23CC3)C1 s275592__15865378__15842670__14134174
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cnc[nH]2)C1 s275592__15865378__15842670__14134222
C=CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134236
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c(C)[nH]1 s275592__15865378__15842670__14134240
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC23CCC3)C1 s275592__15865378__15842670__14134246
Cc1ccnn1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134288
Cc1c[nH]cc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14129438
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__14129446
Cc1nccn1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14129462
CCn1cccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14129478
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCCOC2)C1 s275592__15865378__15842670__14129500
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC=CCC2)C1 s275592__15865378__15842670__14129502
Cc1nccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__14129508
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(F)CCCC2)C1 s275592__15865378__15842670__14132604
Cn1cncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132644
CCc1oncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134304
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cscn2)C1 s275592__15865378__15842670__14134318
CN(C)C(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134358
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2cn[nH]c2)C1 s275592__15865378__15842670__14134428
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CC2)C1 s275592__15865378__15842670__14134440
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CCC2)C1 s275592__15865378__15842670__14134448
COCCC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14129568
CCC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14129596
COCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14132860
COCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132862
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2ccon2)C1 s275592__15865378__15842670__14132878
Cc1cncn1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132904
C[C@@H]1[C@H](C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCN1C s275592__15865378__15842670__14134526
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2CCCO2)C1 s275592__15865378__15842670__14129852
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC(F)F)C1 s275592__15865378__15842670__14132916
COCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__14132938
CC(CC(F)F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14132954
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(F)c[nH]2)C1 s275592__15865378__15842670__14132964
CC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14132968
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CNC(=O)C1 s275592__15865378__15842670__14132976
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC2CC2C1 s275592__15865378__15842670__14132994
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(CCF)CC2)C1 s275592__15865378__15842670__14132998
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COCC(F)F)C1 s275592__15865378__15842670__14133024
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@]23COC[C@@H]2C3)C1 s275592__15865378__15842670__14134550
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14134582
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc[nH]c2)C1 s275592__15865378__15842670__14134596
CC1CCCC1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134598
CN1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1=O s275592__15865378__15842670__14134658
CC(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__14129880
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(C3CC3)CCC2)C1 s275592__15865378__15842670__14133108
COc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)co1 s275592__15865378__15842670__14133112
CC(C)(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCC1 s275592__15865378__15842670__14133122
COC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCC1 s275592__15865378__15842670__14133132
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2csnn2)C1 s275592__15865378__15842670__14133140
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15842670__14133160
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnco2)C1 s275592__15865378__15842670__14133174
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCn2ccnc2)C1 s275592__15865378__15842670__14133200
CNC(=O)NCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134714
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2c[nH]cn2)C1 s275592__15865378__15842670__14134792
CN(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCC1 s275592__15865378__15842670__14134810
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(F)cn2)C1 s275592__15865378__15842670__14134866
C=CCCOCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130048
C=CCOC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130050
NC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130134
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__14130138
Cc1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133250
Cc1n[nH]nc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133302
CCCC(OC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133336
C=C(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133340
CC(CC(N)=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133366
NC(=O)C1CCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133368
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCNC2=O)C1 s275592__15865378__15842670__14133374
Cn1c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c[nH]c1=O s275592__15865378__15842670__14133376
CN1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)NC1=O s275592__15865378__15842670__14133378
C=CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133380
C#CCCCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133382
CN1CCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133386
C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133388
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CC=CCC2)C1 s275592__15865378__15842670__14133390
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__14133392
CCC(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133394
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCCF)C1 s275592__15865378__15842670__14133398
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)(F)F s275592__15865378__15842670__14133400
Cc1cocc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133402
C[C@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133404
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C=CCC1 s275592__15865378__15842670__14133406
CN1C(=O)CC[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133410
Cn1nnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__14133412
CC1(C)CCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133414
CC[C@@H]1CCO[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14134946
CC1C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1C1CC1 s275592__15865378__15842670__14134986
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCC23CC3)C1 s275592__15865378__15842670__14135000
Cc1[nH]cnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14130258
CC1CCC(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14133416
Cc1cnn(C)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133420
CC(C)C(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133422
CCCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__14133424
C=CC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133426
CCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__14133428
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3(CCC3)C2)C1 s275592__15865378__15842670__14133430
CC#CCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133432
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3COC[C@H]32)C1 s275592__15865378__15842670__14133434
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCCC2CC2)C1 s275592__15865378__15842670__14133436
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1=O s275592__15865378__15842670__14133438
CC1(C)CCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133442
Cc1coc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__14133444
C=CC(CC)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133450
CC(C)(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__14133452
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3C[C@@H]3C2)C1 s275592__15865378__15842670__14133454
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cnoc2)C1 s275592__15865378__15842670__14133490
CN1C(=O)CC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14133492
CC1(C)CC(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__14133496
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(F)CCOC2)C1 s275592__15865378__15842670__14133542
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1C s275592__15865378__15842670__14133554
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)(C)C s275592__15865378__15842670__14135056
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C23CCC(CC2)C3)C1 s275592__15865378__15842670__14135064
CN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14135066
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]1 s275592__15865378__15842670__14135072
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cccnc2)C1 s275592__15865378__15842670__14135094
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__14135100
CC(F)(F)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14135120
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CN1 s275592__15865378__15842670__14135142
CCc1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__14135156
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2c[nH]nn2)C1 s275592__15865378__15842670__14135174
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nn1C s275592__15865378__15842670__15278136
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cnn1 s275592__15865378__15842670__15585620
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccccc2O)C1 s275592__15865378__15842670__15855932
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CO)C1 s275592__15865378__15842670__15855972
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccc(O)c2)C1 s275592__15865378__15842670__15855974
NC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855986
Nc1ncccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855988
Nc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n[nH]1 s275592__15865378__15842670__15855990
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc[n+]([O-])c2)C1 s275592__15865378__15842670__15855992
COC(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856004
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(O)ncn2)C1 s275592__15865378__15842670__15856006
C#CCSCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856008
CSC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857758
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnccc2O)C1 s275592__15865378__15842670__15857774
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(=O)C(F)(F)F)C1 s275592__15865378__15842670__15857778
CCC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15857780
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(CO)CCC2)C1 s275592__15865378__15842670__15857784
Nc1ccn(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15857790
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCCC2O)C1 s275592__15865378__15842670__15857798
Cn1ccnc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857800
CC1C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCN1C s275592__15865378__15842670__15857814
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cncc(O)n2)C1 s275592__15865378__15842670__15857816
NC(=O)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857828
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15857832
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COC(F)F)C1 s275592__15865378__15842670__15857834
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC(=O)N1 s275592__15865378__15842670__15857868
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCS2)C1 s275592__15865378__15842670__15859750
CC1=NOC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15859752
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(=O)NC2CC2)C1 s275592__15865378__15842670__15859754
CCC1=NOC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15859762
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]n1 s275592__15865378__15842670__15859768
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCSC2)C1 s275592__15865378__15842670__15859774
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCO2)C1 s275592__15865378__15842670__15859778
CCCC(O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859794
CC(C)(CC#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859806
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(Cl)CC2)C1 s275592__15865378__15842670__15859808
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCO2)C1 s275592__15865378__15842670__15859810
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(CO)o2)C1 s275592__15865378__15842670__15859816
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(CO)COC2)C1 s275592__15865378__15842670__15859830
CC1CC(C#N)(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15859834
CC(C)=CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859836
CC=C(C=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)CC s275592__15865378__15842670__15859838
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2COC2)C1 s275592__15865378__15842670__15859842
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=CC2CCCC2)C1 s275592__15865378__15842670__15859850
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15859854
N#CC1=C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15859858
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)O1 s275592__15865378__15842670__15859862
Nc1c[nH]nc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861720
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=CCO)C1 s275592__15865378__15842670__15861754
CCc1c[nH]cc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861804
O=CN1CCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863550
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n[nH]1 s275592__15865378__15842670__15863554
Cc1cnnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15863576
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]2C(F)F)C1 s275592__15865378__15842670__15863586
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2coc(=O)[nH]2)C1 s275592__15865378__15842670__15863596
CC=CC(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863598
CCCC[C@H](C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863606
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)N(C)C s275592__15865378__15842670__15863612
CCC=C(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863618
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2C3(CC3)C23CC3)C1 s275592__15865378__15842670__15863620
CCC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863622
Cn1nnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1N s275592__15865378__15842670__15863624
CCC(F)(F)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863628
Cc1nocc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863636
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2csnn2)C1 s275592__15865378__15842670__15863642
CC1=C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15842670__15863656
CC(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15864230
CC1CCOC1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864240
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CNC(=O)C2)C1 s275592__15865378__15842670__15856024
Nc1cnn(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15856052
Nc1nonc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856062
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COC(F)(F)F)C1 s275592__15865378__15842670__15856066
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CNC(=O)N2)C1 s275592__15865378__15842670__15856072
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cncs2)C1 s275592__15865378__15842670__15856078
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCN2CCCC2)C1 s275592__15865378__15842670__15856100
Cc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1N s275592__15865378__15842670__15856106
[N-]=[N+]=NCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856110
C#CCOCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856116
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2nnco2)C1 s275592__15865378__15842670__15856118
CN(CCO)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856124
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCS2)C1 s275592__15865378__15842670__15856128
COC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857874
CC(O)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857888
CCS(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857902
Nc1cncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15857944
N#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15842670__15857952
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2cccc2)C1 s275592__15865378__15842670__15857988
CC1=NOC(C)(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15859874
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccn(CO)n2)C1 s275592__15865378__15842670__15859886
C#CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859904
CC(=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)C s275592__15865378__15842670__15859962
COC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15861842
Cn1ncc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15861854
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CC2(F)F)C1 s275592__15865378__15842670__15861866
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(O)ncn2)C1 s275592__15865378__15842670__15861886
CC[C@H](C)[C@H](O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861908
CC1(C)CC1CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861942
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(O)c2c[nH]cn2)C1 s275592__15865378__15842670__15864266
CCC(C)(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864276
Nc1cncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15864294
CC=CC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864312
Cn1ncnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864328
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CC[C@@H](O)C2)C1 s275592__15865378__15842670__15864330
CS(=O)C=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864332
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CC=CCC2)C1 s275592__15865378__15842670__15864344
COCC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864348
[N-]=[N+]=N[C@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15864362
CC(=O)C(C)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864364
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3CC3C2)C1 s275592__15865378__15842670__15856140
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cncnc2)C1 s275592__15865378__15842670__15856158
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2C3CCC(=O)C32)C1 s275592__15865378__15842670__15856176
CS(=O)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856194
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(=O)C2CCCC2)C1 s275592__15865378__15842670__15856196
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cc1F s275592__15865378__15842670__15856210
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=C(Cl)Cl)C1 s275592__15865378__15842670__15856226
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnncc2O)C1 s275592__15865378__15842670__15856232
COc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n[nH]1 s275592__15865378__15842670__15856240
CC1CN(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15856250
CCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857998
CC1CCC(=CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15858032
C#CCC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858040
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15858064
C=CC(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858068
[N-]=[N+]=NCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858070
CC(O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858076
CC1(C)COC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858080
Cn1nncc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858092
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCCO1 s275592__15865378__15842670__15859990
CC1(CCCC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)N=N1 s275592__15865378__15842670__15860034
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C23CCC2C3)C1 s275592__15865378__15842670__15860044
CCCC(C)=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860050
C=C[C@H](C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860060
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=CC2CC2)C1 s275592__15865378__15842670__15860092
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C23CCC(CC2)O3)C1 s275592__15865378__15842670__15860096
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=CC2CCCO2)C1 s275592__15865378__15842670__15861948
Cc1oncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861960
CC(C)CC(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861966
CC1CC1(C#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861988
CCC(C#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861996
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2coc(CO)c2)C1 s275592__15865378__15842670__15862014
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CNC(=O)O2)C1 s275592__15865378__15842670__15862020
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C23CCC(CO2)C3)C1 s275592__15865378__15842670__15864376
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2C3CCC32)C1 s275592__15865378__15842670__15864378
C=C1CCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864388
C[C@@H]1C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[C@@H]1C s275592__15865378__15842670__15864392
Cc1nnn(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15864412
CCN(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864424
CC1(C)CC1(C#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864484
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3(C2)N=N3)C1 s275592__15865378__15842670__15856264
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)sn1 s275592__15865378__15842670__15856288
CC1(C)C(=O)CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856290
CC(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856300
CCCCCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856320
CC(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856322
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1 s275592__15865378__15842670__15856332
Nc1n[nH]cc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856354
CC(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856356
CCOC(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856372
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)ccn1 s275592__15865378__15842670__15856380
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)n1ccnc1 s275592__15865378__15842670__15858144
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccnc2O)C1 s275592__15865378__15842670__15858152
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15858154
Nc1cccnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858168
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CSC(F)F)C1 s275592__15865378__15842670__15858176
Cc1noc(N)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858188
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15858198
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccc[n+]2[O-])C1 s275592__15865378__15842670__15858200
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cs1 s275592__15865378__15842670__15858204
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=NNC(=O)C2)C1 s275592__15865378__15842670__15858220
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c[nH]1 s275592__15865378__15842670__15858222
COCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858228
CC1=C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15858230
N#CCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858238
N#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15858240
C=C1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15858242
CN(C)C(=O)C=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860112
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@]23C[C@@H](O)[C@@H]2C3)C1 s275592__15865378__15842670__15860130
N#C[C@]1(O)C[C@@H](C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15860176
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15860180
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCCCCF)C1 s275592__15865378__15842670__15860190
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3(C2)CC3F)C1 s275592__15865378__15842670__15860216
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C23CC(CO2)C3)C1 s275592__15865378__15842670__15860230
CC12COC(C(=O)N3CC(=C(F)CNC(=O)CSc4n[nH]c(=O)[nH]4)C3)(C1)C2 s275592__15865378__15842670__15862074
CC(=O)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862082
C#CC1(O)CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15862092
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]c1C s275592__15865378__15842670__15862108
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC3CCCC32)C1 s275592__15865378__15842670__15862146
CC1(C)CC(C)(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15862166
CC(C)(F)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864494
CC[C@H](CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)C s275592__15865378__15842670__15864540
CCC=CC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864546
CC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCO1 s275592__15865378__15842670__15864566
Cc1ncn(C)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864570
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2nncs2)C1 s275592__15865378__15842670__15864586
CC(=C(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__15864610
CN(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(N)=O s275592__15865378__15842670__15856410
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2nc(=O)[nH][nH]2)C1 s275592__15865378__15842670__15856424
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(F)CC2)C1 s275592__15865378__15842670__15856434
Nc1ncncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856466
CCN(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__15858258
CC(O)(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__15858266
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__15858272
Cc1scnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858282
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccc(F)n2)C1 s275592__15865378__15842670__15858288
COC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858294
CC(CC#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858308
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)n1cnnn1 s275592__15865378__15842670__15858340
O=NN1CCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858354
CCC1CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858366
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CCC(O)C2)C1 s275592__15865378__15842670__15860236
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)(C)O s275592__15865378__15842670__15860240
CN1CC2CC1(C(=O)N1CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C1)C2 s275592__15865378__15842670__15860250
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2COC(=O)O2)C1 s275592__15865378__15842670__15860258
Cn1nncc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860272
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C23COC(C2)C3)C1 s275592__15865378__15842670__15860284
CC(O)C1CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860286
C[C@@H]1C[C@@]2(C(=O)N3CC(=C(F)CNC(=O)CSc4n[nH]c(=O)[nH]4)C3)C[C@@H]12 s275592__15865378__15842670__15860334
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CO1 s275592__15865378__15842670__15860338
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2cncn2)C1 s275592__15865378__15842670__15860346
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccc(=O)o2)C1 s275592__15865378__15842670__15860352
CC(CN(C)C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862216
CNc1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__15862226
Cn1cc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nn1 s275592__15865378__15842670__15862236
C=CC(C)(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862244
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC2(O)CCC2)C1 s275592__15865378__15842670__15862246
CCC(C)(CO)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862252
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15862262
Cn1nc(O)cc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862272
CCc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15862276
CCCC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862286
CC=C(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862288
N#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCOC1 s275592__15865378__15842670__15862294
CCC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)C s275592__15865378__15842670__15862302
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cncc(F)n2)C1 s275592__15865378__15842670__15864618
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)co1 s275592__15865378__15842670__15864622
C[C@H](C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)N(C)C s275592__15865378__15842670__15864628
CC(C)C(CO)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864638
CCOC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864642
CCN1CCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864656
CSSCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856512
NC(=O)C(O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856518
CCC(C)=C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856520
COC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15856530
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=NNC(=O)CC2)C1 s275592__15865378__15842670__15856546
C=CCCC(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858382
CC(O)CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858388
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)on1 s275592__15865378__15842670__15858392
CC(=O)OCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858408
Nc1ccncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858424
Nc1cnccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858428
CC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858440
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2c[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858448
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cs1 s275592__15865378__15842670__15858468
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15858474
CN(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858478
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(F)(F)CO)C1 s275592__15865378__15842670__15858486
CC1(C#CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15860362
C=CC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15860378
CC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860380
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COC2CC2)C1 s275592__15865378__15842670__15860388
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ncc[nH]2)C1 s275592__15865378__15842670__15860394
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=CC2CCC2)C1 s275592__15865378__15842670__15860398
O=C1CC(C#CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15860408
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC(C3CC3)C2)C1 s275592__15865378__15842670__15860432
CSC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862328
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2nncs2)C1 s275592__15865378__15842670__15862356
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3CCCO[C@H]32)C1 s275592__15865378__15842670__15862374
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)no1 s275592__15865378__15842670__15862416
O=C1COC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15862436
CC(C)NC(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863680
C=C(Cl)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863686
CC1=C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCO1 s275592__15865378__15842670__15863704
C=Cn1nccc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863714
Cn1ccnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863724
CO[C@@H]1C[C@@]2(C(=O)N3CC(=C(F)CNC(=O)CSc4n[nH]c(=O)[nH]4)C3)C[C@@H]12 s275592__15865378__15842670__15864778
Cn1cnnc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864786
CCc1nonc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864792
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cnsn2)C1 s275592__15865378__15842670__15864798
C=CCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864800
CCC(C)CC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864832
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(F)n2cccn2)C1 s275592__15865378__15842670__15864846
CC(CO)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856640
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnoc2)C1 s275592__15865378__15842670__15856650
Nc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cs1 s275592__15865378__15842670__15856652
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCCCO)C1 s275592__15865378__15842670__15858500
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(=O)C2CC2)C1 s275592__15865378__15842670__15858504
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2COC(=O)N2)C1 s275592__15865378__15842670__15858518
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cncc(O)c2)C1 s275592__15865378__15842670__15858522
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2(O)CC2)C1 s275592__15865378__15842670__15858528
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC2F)C1 s275592__15865378__15842670__15858574
N#CCCCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858576
Cc1cnsc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860502
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(F)C2CCC2)C1 s275592__15865378__15842670__15860518
CC(OC(F)F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860520
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)O1 s275592__15865378__15842670__15860522
CC(C)(CCC#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860558
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__15860570
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2c[nH]cn2)C1 s275592__15865378__15842670__15862464
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2ncc[nH]2)C1 s275592__15865378__15842670__15862484
CCC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)COC1 s275592__15865378__15842670__15862492
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2cn[nH]c2)C1 s275592__15865378__15842670__15862500
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2CF)C1 s275592__15865378__15842670__15862520
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cnns2)C1 s275592__15865378__15842670__15862548
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(F)=C2CCC2)C1 s275592__15865378__15842670__15862554
CCC(CO)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862556
CC(C)(O)C(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862558
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC(O)C2CC2)C1 s275592__15865378__15842670__15863750
CC(C)CC(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863770
CC1(C#CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)COC1 s275592__15865378__15842670__15863772
CC(=CC1CC1)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863786
N#C[C@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863804
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2cocn2)C1 s275592__15865378__15842670__15863816
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2(CO)CCC2)C1 s275592__15865378__15842670__15863830
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cnco2)C1 s275592__15865378__15842670__15864872
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C[C@@H]2CC=CCC2)C1 s275592__15865378__15842670__15864876
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CN2CC3CC3C2)C1 s275592__15865378__15842670__15864884
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CC3CC3C2)C1 s275592__15865378__15842670__15864900
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=COCC2)C1 s275592__15865378__15842670__15856668
CC(C)(O)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856700
CCC(C#N)(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856756
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]1 s275592__15865378__15842670__15856770
CN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856776
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(O)CCCCC2)C1 s275592__15865378__15842670__15858626
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(O)CC2)C1 s275592__15865378__15842670__15858682
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCC2)C1 s275592__15865378__15842670__15858720
CC1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)=NO1 s275592__15865378__15842670__15860614
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CCCC[C@H]2O)C1 s275592__15865378__15842670__15860642
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C=CCCC1 s275592__15865378__15842670__15860644
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CC3(CC3)C2)C1 s275592__15865378__15842670__15860654
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1C s275592__15865378__15842670__15860672
CC(CF)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862566
CC(Cl)=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862574
CC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862586
CN1C(=O)NCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862588
CCC(F)(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862594
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1F s275592__15865378__15842670__15862600
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CCC(=O)O2)C1 s275592__15865378__15842670__15862656
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2C3CCOCC32)C1 s275592__15865378__15842670__15863872
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=CCF)C1 s275592__15865378__15842670__15863884
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(F)CC2CC2)C1 s275592__15865378__15842670__15863892
CCC(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__15863894
CC(C)CCC(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863902
CN1CCC(=CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15863906
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]c1C s275592__15865378__15842670__15863940
CCOC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15863948
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2COC(=O)N2)C1 s275592__15865378__15842670__15863964
N#CCCCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863976
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(CO)CC2)C1 s275592__15865378__15842670__15856792
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccno2)C1 s275592__15865378__15842670__15856830
[N-]=[N+]=NCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856874
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC(=O)N2)C1 s275592__15865378__15842670__15856878
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCSC2)C1 s275592__15865378__15842670__15856886
C[C@H](O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856892
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(F)o2)C1 s275592__15865378__15842670__15858752
CON=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858762
C#CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858766
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)N=[N+]=[N-] s275592__15865378__15842670__15858792
CC1(F)CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15858798
Cn1ncc(N)c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858800
CCC(C)(OC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858808
CC(C)[C@H](O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858830
CN(C)C(=O)C=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860752
C#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15860756
CCC1CN(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15860778
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2CCC(=O)O2)C1 s275592__15865378__15842670__15860782
Cc1cn(C)cc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860784
C=CC=CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860802
C#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15860826
CN1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860828
CCCC=CC(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15860832
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC=CCO2)C1 s275592__15865378__15842670__15860842
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2ncco2)C1 s275592__15865378__15842670__15862704
CC(CC1CCC1)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862718
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC3(C2)N=N3)C1 s275592__15865378__15842670__15862724
CC1(C)C=C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15862726
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2ccn[nH]2)C1 s275592__15865378__15842670__15862730
CC1(C)CC(O)(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15862772
CN(C)C(=O)C#CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862802
C#C[C@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863992
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nc1O s275592__15865378__15842670__15864000
[N-]=[N+]=NC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15864012
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2ncc[nH]2)C1 s275592__15865378__15842670__15864060
CCC(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)OC s275592__15865378__15842670__15864096
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nc1 s275592__15865378__15842670__15856920
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cscn2)C1 s275592__15865378__15842670__15856940
CC=C(CC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856970
Cc1[nH]nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1F s275592__15865378__15842670__15856978
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC23CC(C2)C3)C1 s275592__15865378__15842670__15856982
C#CCC(CC#C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15856994
CCC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)O s275592__15865378__15842670__15857002
COC(F)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858882
N#CC(=CC1CC1)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858896
CCc1cnoc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858900
NS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858910
Nc1ccnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15858948
N#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15858950
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=C2CCCC2)C1 s275592__15865378__15842670__15858972
CC(C)(C#N)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858978
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC(=O)NC2CC2)C1 s275592__15865378__15842670__15858984
COCC(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15858990
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCOC1 s275592__15865378__15842670__15860864
CN(C)[C@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15860888
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2(C3CC3)CC2)C1 s275592__15865378__15842670__15860906
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CC2(F)F)C1 s275592__15865378__15842670__15860916
N#C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862806
CCCC(CC)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862808
C=C(C)CCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862818
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nn1C s275592__15865378__15842670__15862852
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2C[C@@H](O)C2)C1 s275592__15865378__15842670__15862874
CC1(C)CC1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15862884
CC(=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)(C)C s275592__15865378__15842670__15862900
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=C(Cl)CC2)C1 s275592__15865378__15842670__15864120
Cc1nnnn1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864128
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@]23C[C@@H](F)[C@@H]2C3)C1 s275592__15865378__15842670__15864138
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2c[nH]c(=O)o2)C1 s275592__15865378__15842670__15864148
CC(C)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864156
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CC3CCCC23)C1 s275592__15865378__15842670__15864180
CCn1ncnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15864218
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(F)(F)C2CC2)C1 s275592__15865378__15842670__15857016
CC(=O)OC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15857018
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COCCO)C1 s275592__15865378__15842670__15857042
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)=NO1 s275592__15865378__15842670__15857048
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ncc(F)cn2)C1 s275592__15865378__15842670__15857050
CC(C)(CF)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857052
CC(C)[C@@H](O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857054
CC(C)(CO)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857066
C=CCC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857082
CC1CCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859060
CC1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15859064
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2C3CC4C(C3)C42)C1 s275592__15865378__15842670__15860980
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H](O)C2CCCC2)C1 s275592__15865378__15842670__15860990
CCn1cnnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861050
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(C3CCC3)CC2)C1 s275592__15865378__15842670__15861058
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CC[C@@H]3C[C@@H]32)C1 s275592__15865378__15842670__15861066
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC(F)C1 s275592__15865378__15842670__15862956
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]1 s275592__15865378__15842670__15862958
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C#CC2CCCO2)C1 s275592__15865378__15842670__15862984
C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863036
CC(C)(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857148
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CN2CCCCC2)C1 s275592__15865378__15842670__15857176
CN1CCCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15857180
Cn1cc[n+](CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15857214
Cc1nccnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857228
CSC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15857232
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=NOCC2)C1 s275592__15865378__15842670__15857252
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COc2ccon2)C1 s275592__15865378__15842670__15859122
Cc1coc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1C s275592__15865378__15842670__15859134
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cnccn2)C1 s275592__15865378__15842670__15859158
CC(C#N)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859162
Nc1ccnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15859176
CCC1OCCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859182
CN(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__15859226
Cn1cccc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859228
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCOC2CC2)C1 s275592__15865378__15842670__15861110
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCCCCO)C1 s275592__15865378__15842670__15861138
COC(=O)[C@@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861166
Cc1conc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861172
CCc1noc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15861194
Nc1cnn(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15863050
CC(CCO)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863056
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(F)=CC2CC2)C1 s275592__15865378__15842670__15863058
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CC(F)C2)C1 s275592__15865378__15842670__15863076
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H](O)CF)C1 s275592__15865378__15842670__15863130
CCC1(C)C=C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15863134
CCC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15863136
CCn1cnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15863154
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(CCO)CC2)C1 s275592__15865378__15842670__15857266
CC(C)C(C)(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857276
COC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15857302
COC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15842670__15857304
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__15857310
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2ccccn2)C1 s275592__15865378__15842670__15857374
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(O)CCC2)C1 s275592__15865378__15842670__15859240
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(O)C2CC2)C1 s275592__15865378__15842670__15859246
NC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15859256
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2cnnc2)C1 s275592__15865378__15842670__15859258
C=C(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859282
CC(C)(C#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859288
CC1=CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15859298
CCSCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859302
CC(=O)OCCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859304
CC(C)=C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859306
Cc1sncc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859338
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccncc2O)C1 s275592__15865378__15842670__15859340
CC1(CCC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)N=N1 s275592__15865378__15842670__15859356
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842670__15859360
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)COC2COC2)C1 s275592__15865378__15842670__15861226
C[C@@H]1C[C@]2(C(=O)N3CC(=C(F)CNC(=O)CSc4n[nH]c(=O)[nH]4)C3)C[C@H]12 s275592__15865378__15842670__15861228
CNC(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861240
CC(=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)F s275592__15865378__15842670__15861304
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC2(CC2)C1 s275592__15865378__15842670__15861316
CCOC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861322
Cn1cnnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863182
Nc1ncn(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15863202
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCOCC2)C1 s275592__15865378__15842670__15863212
C[C@@H]1OCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863214
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC(F)C2)C1 s275592__15865378__15842670__15863220
CCC(O)C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863232
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CC(=O)N2)C1 s275592__15865378__15842670__15863258
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(O)C2CCC2)C1 s275592__15865378__15842670__15863264
CN1CC(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15863276
Cc1nnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)s1 s275592__15865378__15842670__15863286
CC1(O)CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15863290
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15855626
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(O)cc2)C1 s275592__15865378__15842670__15855632
C=CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855634
CN(C)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855640
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15855648
N#CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855652
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cc1 s275592__15865378__15842670__15855660
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cccnc2F)C1 s275592__15865378__15842670__15857384
CCOC1C(C)C1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857420
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC2F)C1 s275592__15865378__15842670__15857454
CC1(OCC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15857466
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)N(C)C s275592__15865378__15842670__15857472
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cn1 s275592__15865378__15842670__15857478
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCF)C1 s275592__15865378__15842670__15857480
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(F)n[nH]2)C1 s275592__15865378__15842670__15857486
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2C=CCC2)C1 s275592__15865378__15842670__15857492
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC(=O)C1 s275592__15865378__15842670__15857496
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCC(O)C2)C1 s275592__15865378__15842670__15857500
N#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC(=O)C1 s275592__15865378__15842670__15857502
CCC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)COC1 s275592__15865378__15842670__15859370
C#CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859374
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=CC2CCOC2)C1 s275592__15865378__15842670__15859412
COC(C)C(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859432
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2CNC(=O)N2)C1 s275592__15865378__15842670__15859438
CCSC(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859462
CC1CN(C(C)C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15859468
CC1CCN1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859482
COC(C)(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC1 s275592__15865378__15842670__15859488
CN(C)CC=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861374
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC(C#N)C1 s275592__15865378__15842670__15861388
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCSC2)C1 s275592__15865378__15842670__15861398
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCCC(F)F)C1 s275592__15865378__15842670__15861400
CC1(C)CN(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15861410
CO[C@H](C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15863310
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C23CCC(C2)OC3)C1 s275592__15865378__15842670__15863334
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC23CC(O)C3)C1 s275592__15865378__15842670__15863340
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C=Cc2cc[nH]n2)C1 s275592__15865378__15842670__15863350
CC(CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)F s275592__15865378__15842670__15863380
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C[C@@H]2CCC[C@H]2O)C1 s275592__15865378__15842670__15863396
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2ccc(=O)oc2)C1 s275592__15865378__15842670__15855674
CC(=O)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855680
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2(O)CCCC2)C1 s275592__15865378__15842670__15855696
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCCC2O)C1 s275592__15865378__15842670__15855698
C[C@@H](O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855722
CCN(CC)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855728
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c1 s275592__15865378__15842670__15855744
CCOC=C(C#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855752
CC(C)(C#N)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855756
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nc1 s275592__15865378__15842670__15855764
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CN2CCC2)C1 s275592__15865378__15842670__15855766
CC(C)C(O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855768
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2COC(=O)C2)C1 s275592__15865378__15842670__15855790
CC1CC=C(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15857504
CC(O)C(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857506
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(O)CCOC2)C1 s275592__15865378__15842670__15857516
CCC(C)(C#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857522
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cc1O s275592__15865378__15842670__15857524
C=C1CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857536
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CC=CC2)C1 s275592__15865378__15842670__15857548
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2OCCO2)C1 s275592__15865378__15842670__15857568
COC(OC)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857572
N#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC=CC1 s275592__15865378__15842670__15857578
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCC[N+](=O)[O-])C1 s275592__15865378__15842670__15857582
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15857586
COC(=O)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857614
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCOC2)C1 s275592__15865378__15842670__15859502
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1(F)F s275592__15865378__15842670__15859514
Nc1nnn(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15859516
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)on1 s275592__15865378__15842670__15859520
CC(C)(C)C(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859522
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C(O)C2CCCC2)C1 s275592__15865378__15842670__15859546
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)COC1 s275592__15865378__15842670__15859548
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCCO2)C1 s275592__15865378__15842670__15859558
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCO1 s275592__15865378__15842670__15859562
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CC(=O)N2)C1 s275592__15865378__15842670__15859564
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(CO)on2)C1 s275592__15865378__15842670__15859574
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@@H]2CC(=O)N2)C1 s275592__15865378__15842670__15859582
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2=CCCCC2)C1 s275592__15865378__15842670__15859608
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c(N)n1 s275592__15865378__15842670__15859612
CCC[C@H](O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861464
C#CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCC1 s275592__15865378__15842670__15861488
CC(C)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)COC1 s275592__15865378__15842670__15861502
Nc1ccnn1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861512
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)c[nH]1 s275592__15865378__15842670__15861516
CCc1nnc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]1 s275592__15865378__15842670__15861528
CC1CC(C)(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15861556
Cn1ncnc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861562
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n(C)n1 s275592__15865378__15842670__15863462
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)N1CCC1 s275592__15865378__15842670__15863476
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)cc1 s275592__15865378__15842670__15863478
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2CC2(F)F)C1 s275592__15865378__15842670__15863508
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cn[nH]c2)C1 s275592__15865378__15842670__15863518
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)nc1 s275592__15865378__15842670__15855796
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2=NNC(=O)C2)C1 s275592__15865378__15842670__15855798
CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC(=O)C1 s275592__15865378__15842670__15855814
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cc[nH]c2)C1 s275592__15865378__15842670__15855816
CCCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855836
CCOC(C)(C)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855838
CC(O)(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCC1 s275592__15865378__15842670__15855864
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)O1 s275592__15865378__15842670__15855868
Cn1nccc1CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855880
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15855882
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2CSC2)C1 s275592__15865378__15842670__15855884
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(F)CCC2)C1 s275592__15865378__15842670__15855898
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnc[nH]2)C1 s275592__15865378__15842670__15857636
Cc1noc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15857642
CCOC(=O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857644
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15857654
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2ccnn2)C1 s275592__15865378__15842670__15857670
CN1CCCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857674
C=CC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15842670__15857684
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(O)COC2)C1 s275592__15865378__15842670__15857690
CCC(C)C(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857696
CC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)=C1CC1 s275592__15865378__15842670__15857712
CC1=CC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857746
CN(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15857748
CC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15859626
CCCC(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859672
CCCCC(O)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859676
COC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)O s275592__15865378__15842670__15859690
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CSC2CC2)C1 s275592__15865378__15842670__15859698
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCCC2CCC2)C1 s275592__15865378__15842670__15859702
CCC(O)CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859710
CN1C(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15859720
N#Cc1cn[nH]c1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861586
CNC(=O)CCC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861592
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCc2cnoc2)C1 s275592__15865378__15842670__15861604
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2cnsc2)C1 s275592__15865378__15842670__15861610
C=CCC(C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1)N(C)C s275592__15865378__15842670__15861626
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CCCCF)C1 s275592__15865378__15842670__15861646
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(O)ccn2)C1 s275592__15865378__15842670__15861668
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(O)cs2)C1 s275592__15865378__15842670__15861670
CC1CC(=O)NC1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861676
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cnsc2)C1 s275592__15865378__15842670__15861686
Cn1nc(N)cc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15861694
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15842670__15861700
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)[C@H]2CC(=O)N2)C1 s275592__15865378__15842670__15855518
Cn1cc(N)c(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15842670__15855526
CC(C)C=C(C#N)C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855536
Nc1csnc1C(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15855538
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cn2cncn2)C1 s275592__15865378__15842670__15855544
COC1(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842670__15855548
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CSC2)C1 s275592__15865378__15842670__15855552
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)CSc3n[nH]c(=O)[nH]3)C2)o1 s275592__15865378__15842670__15855558
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)CC2(CO)CC2)C1 s275592__15865378__15842670__15855560
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)Cc2nccs2)C1 s275592__15865378__15842670__15855582
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2CCC=CO2)C1 s275592__15865378__15842670__15855594
O=C(CSc1n[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)C2(O)CCCC2)C1 s275592__15865378__15842670__15855622
C=CC(=O)N1CC(=C(F)CNC(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842670__15909382
Cc1[nH]c(=O)nc(S)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842672__15859360
Cn1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cnc1S s275592__15865378__15842674__15862300
Cn1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cnc1S s275592__15865378__15842674__15859360
N=C(N)SCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842676__15862300
N=C(N)SCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842676__15859360
N=C(N)SCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842676__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)c1ccc(F)c(F)c1 s275592__15865378__15842678__15859360
O=C(CCC[N+](=O)[O-])NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842680__15862300
O=C(CCC[N+](=O)[O-])NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842680__15859360
O=C(CCC[N+](=O)[O-])NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842680__15857566
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C(F)(F)c2cccnc2)C1 s275592__15865378__15842682__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)c2cccnc2)C1 s275592__15865378__15842682__15859360
[N-]=[N+]=Nc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15842684__15862300
[N-]=[N+]=Nc1cncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15842684__15859360
Cn1ccc2cccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c21 s275592__15865378__15842686__15859360
CON1CCC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842688__15862300
CON1CCC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842688__15859360
CC(CF)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842692__15862300
CC(CF)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842692__15859360
CC(CF)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842692__15857566
O=C(C=Cc1cc2ccccc2o1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844430__15859360
Cn1ncc(Cl)c1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844432__15859360
Cc1cc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cccc2o1 s275592__15865378__15844434__15859360
O=C(C=Cc1cscn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844436__15862300
O=C(C=Cc1cscn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844436__15859360
O=C(C[C@@H]1COC[C@H]1O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844440__15862300
O=C(C[C@@H]1COC[C@H]1O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844440__15859360
O=C(CSc1cccc(F)c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844442__15859360
Cc1cc(F)sc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844444__15862300
Cc1cc(F)sc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844444__15859360
Cc1ccc([C@@H]2C[C@H]2C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15844448__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@H]1C[C@H]2[C@@H](C1)C2(F)F s275592__15865378__15844450__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@H]1C[C@H]2[C@@H](C1)C2(F)F s275592__15865378__15844450__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CC2(CCOCC2)C1 s275592__15865378__15844454__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CC2(CCOCC2)C1 s275592__15865378__15844454__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnc2occc2c1 s275592__15865378__15844458__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2occc2c1 s275592__15865378__15844458__15859360
O=C(CCCC1CCCC(=O)N1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844460__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCNS1(=O)=O s275592__15865378__15844462__15859360
CC(C)(C)c1nnn(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844466__15859360
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CC1(C)C=C(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15844494__15857566
O=C(CCC=CBr)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844496__15859360
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CC12CC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(C1)C1(CCC1)O2 s275592__15865378__15844502__15859360
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CC1CCC(F)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15844510__15862300
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O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC2(C1)CC2(F)F s275592__15865378__15844512__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)=Cc1c[nH]cn1 s275592__15865378__15844514__15862300
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CCN1CCOCC1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844522__15862300
CCN1CCOCC1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844522__15859360
O=C(Cc1nnc2n1CCOC2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844524__15859360
O=C(Cc1nnc2n1CCCC2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844526__15859360
CC1(C)CCOC1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844528__15862300
CC1(C)CCOC1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844528__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nc2ccccn2n1 s275592__15865378__15844530__15862300
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O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(Cc3cnn[nH]3)CCC2)C1 s275592__15865378__15844532__15859360
CC12CC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(C1)C1(COC1)O2 s275592__15865378__15844534__15859360
CC1(C)CC(O)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15844536__15862300
CC1(C)CC(O)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15844536__15859360
CC1(C)CC(O)(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15844536__15857566
CC(=Cc1c[nH]cn1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844540__15862300
CC(=Cc1c[nH]cn1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844540__15859360
O=C(Cn1nnnc1C1CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844542__15862300
O=C(Cn1nnnc1C1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844542__15859360
Cc1ccc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cnc2c1 s275592__15865378__15844544__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC(OC(F)F)C1 s275592__15865378__15846230__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CC4CC(CC(C4)O2)C3)C1 s275592__15865378__15846232__15859360
O=C(CC1(C2CC2)CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846234__15862300
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CC(C)[C@@H](NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846236__15862300
CC(C)[C@@H](NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846236__15859360
Cc1cccc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cnn12 s275592__15865378__15846238__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(C2CCC2)no1 s275592__15865378__15846240__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(C2CCC2)no1 s275592__15865378__15846240__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1CC1(F)F s275592__15865378__15846244__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CC1(F)F s275592__15865378__15846244__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)[C@@H]1CC1(F)F s275592__15865378__15846244__15857566
Cc1c[nH]c2ncc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15846246__15859360
CN(C)CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15846248__15859360
COC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)(CC1)C2 s275592__15865378__15846250__15862300
COC12CCC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)(CC1)C2 s275592__15865378__15846250__15859360
CC1CCCC(C)N1CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846252__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)C1CCOC1 s275592__15865378__15846254__15862300
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O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nn[nH]c1C1CC1 s275592__15865378__15846256__15862300
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CN(C)C1CCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15846258__15862300
CN(C)C1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15846258__15859360
CN(C)CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15846260__15862300
CN(C)CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15846260__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc(-n2cccn2)n1 s275592__15865378__15846262__15859360
C#Cc1ccc(OCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15846264__15859360
Cc1ccc(C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C2CC2)cc1 s275592__15865378__15846266__15859360
CN(C)[C@H]1CC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15846268__15862300
CN(C)[C@H]1CC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15846268__15859360
CN1CC=CCC1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846270__15862300
CN1CC=CCC1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846270__15859360
CCc1nc2ccccn2c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846274__15859360
O=C(CCC12CCC(CC1)C2)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846276__15862300
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Cc1cc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n(C)n1 s275592__15865378__15846278__15862300
Cc1cc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15846278__15859360
COc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc(F)c1F s275592__15865378__15846282__15859360
Cc1ccc2ncnc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15846284__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(O)CCn1cncn1 s275592__15865378__15846286__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)CCn1cncn1 s275592__15865378__15846286__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@H]2C[C@](F)(CO)C2)C1 s275592__15865378__15846288__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@H]2C[C@](F)(CO)C2)C1 s275592__15865378__15846288__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2CCCCCCC21 s275592__15865378__15846290__15859360
CC1CC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C(C)O1 s275592__15865378__15846292__15862300
CC1CC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C(C)O1 s275592__15865378__15846292__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnc2ncnn2c1 s275592__15865378__15846294__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2ncnn2c1 s275592__15865378__15846294__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1Cc2cscc2C1 s275592__15865378__15846296__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1Cc2cscc2C1 s275592__15865378__15846296__15859360
CCOc1sccc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846298__15862300
CCOc1sccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846298__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1C2CC3C(C2)C31 s275592__15865378__15846300__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1C2CC3C(C2)C31 s275592__15865378__15846300__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1C2CC3C(C2)C31 s275592__15865378__15846300__15857566
CC(C)(C)c1cccnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846302__15859360
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)noc1C1CC1 s275592__15865378__15846304__15862300
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)noc1C1CC1 s275592__15865378__15846304__15859360
Cn1c([N+](=O)[O-])cnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846306__15862300
Cn1c([N+](=O)[O-])cnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846306__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H](O)C1CCCC1 s275592__15865378__15846310__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H](O)C1CCCC1 s275592__15865378__15846310__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)[C@@H](O)C1CCCC1 s275592__15865378__15846310__15857566
CC1(C)CCCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15846312__15862300
CC1(C)CCCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15846312__15859360
Cc1nn2c(C)cccc2c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846314__15859360
COCC(C)(O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846316__15862300
COCC(C)(O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846316__15859360
CC1(C)CCCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15846318__15859360
C[C@]1(C(F)(F)F)C[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846320__15862300
C[C@]1(C(F)(F)F)C[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846320__15859360
CC(Cc1ccncc1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846322__15862300
CC(Cc1ccncc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846322__15859360
COC1CC(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15846326__15862300
COC1CC(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15846326__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2c(c1)CCOC2 s275592__15865378__15846328__15859360
CC(F)(F)[C@@H]1C[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846330__15862300
CC(F)(F)[C@@H]1C[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846330__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nnc2ccccn12 s275592__15865378__15846334__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nnc2ccccn12 s275592__15865378__15846334__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@]23C[C@@H]4C[C@@H]2C3[C@H]4O)C1 s275592__15865378__15846336__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@]23C[C@@H]4C[C@@H]2C3[C@H]4O)C1 s275592__15865378__15846336__15859360
C[C@@H](OCCN(C)C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846344__15862300
C[C@@H](OCCN(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846344__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2oc(=O)oc2c1 s275592__15865378__15846346__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(CCOCC2)CO1 s275592__15865378__15846350__15859360
CC(=O)NCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840832__15862300
CC(=O)NCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840832__15859360
CC(=O)NCCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840832__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCN1C(=O)C1CC1 s275592__15865378__15840834__15859360
O=C(CNC(=O)NC1CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840836__15862300
O=C(CNC(=O)NC1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840836__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1c[nH]c(=O)[nH]1 s275592__15865378__15840838__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c(=O)[nH]1 s275592__15865378__15840838__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1c[nH]c(=O)[nH]1 s275592__15865378__15840838__15857566
Cc1nc2ccccc2cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840842__15859360
O=C(C[C@H](O)c1ccccc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840850__15862300
O=C(C[C@H](O)c1ccccc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840850__15859360
CSc1ccccc1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840854__15859360
CNC(=O)N1CCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840858__15862300
CNC(=O)N1CCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840858__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(O)cc(O)n1 s275592__15865378__15840860__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(O)cc(O)n1 s275592__15865378__15840860__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2nsnc2c1 s275592__15865378__15840862__15859360
O=C(CC(O)c1ccccc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840864__15862300
O=C(CC(O)c1ccccc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840864__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(O)CCCCCC2)C1 s275592__15865378__15840868__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(O)CCCCCC2)C1 s275592__15865378__15840868__15859360
CNC(=O)N1CCC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840870__15862300
CNC(=O)N1CCC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840870__15859360
CC1CCCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840872__15862300
CC1CCCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840872__15859360
CC1CCCC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840872__15857566
CC1CCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15840874__15862300
CC1CCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15840874__15859360
CC1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15840876__15862300
CC1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15840876__15859360
CC1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15840876__15857566
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)sc2cncn12 s275592__15865378__15840878__15859360
CC1(C)CCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15840880__15862300
CC1(C)CCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15840880__15859360
C=C(C)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840886__15862300
C=C(C)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840886__15859360
C=C(C)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840886__15857566
Cc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(O)c1Cl s275592__15865378__15840888__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C(F)(F)c2ccccn2)C1 s275592__15865378__15840890__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)c2ccccn2)C1 s275592__15865378__15840890__15859360
CCc1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cnn1CC s275592__15865378__15840892__15862300
CCc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cnn1CC s275592__15865378__15840892__15859360
CCCn1nc(C)cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840896__15862300
CCCn1nc(C)cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840896__15859360
CC1=CCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15840898__15862300
CC1=CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15840898__15859360
CC1=CCC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15840898__15857566
CCSCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840900__15862300
CCSCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840900__15859360
CCSCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840900__15857566
CC(C)=C(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840902__15862300
CC(C)=C(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840902__15859360
CC(C)=C(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840902__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc(F)c1Cl s275592__15865378__15840910__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C(F)(F)C(F)F)C1 s275592__15865378__15840912__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)C(F)F)C1 s275592__15865378__15840912__15859360
CC(C)C(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)n1ccnc1 s275592__15865378__15840914__15862300
CC(C)C(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)n1ccnc1 s275592__15865378__15840914__15859360
COc1ccc(F)c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15840916__15862300
COc1ccc(F)c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15840916__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2nc(O)cn2c1 s275592__15865378__15840920__15859360
CN1C2CCC1CC(C(=O)NCC(F)=C1CN(C(=O)c3nsnc3O)C1)C2 s275592__15865378__15840922__15862300
CN1C2CCC1CC(C(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)C2 s275592__15865378__15840922__15859360
CCCC(O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840924__15862300
CCCC(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840924__15859360
CCCC(O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840924__15857566
CCCCC(O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840926__15862300
CCCCC(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840926__15859360
CCCCC(O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840926__15857566
O=C(Cc1ncncc1Cl)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840928__15862300
O=C(Cc1ncncc1Cl)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840928__15859360
O=C(CC(c1ccccc1)C1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840930__15859360
CC(C)(O)C1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15840932__15859360
O=C(CC1CC(=O)NC(=O)C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840934__15862300
O=C(CC1CC(=O)NC(=O)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840934__15859360
COC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)O s275592__15865378__15840936__15862300
COC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)O s275592__15865378__15840936__15859360
COC(C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)O s275592__15865378__15840936__15857566
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)ccn1C1CC1 s275592__15865378__15840938__15862300
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccn1C1CC1 s275592__15865378__15840938__15859360
O=C(CSC1CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840940__15862300
O=C(CSC1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840940__15859360
O=C(CSC1CC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840940__15857566
O=C(CCCC1CCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840944__15862300
O=C(CCCC1CCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840944__15859360
O=C(CCCC1CCC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840944__15857566
CC(C)(C)c1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)on1 s275592__15865378__15840946__15862300
CC(C)(C)c1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)on1 s275592__15865378__15840946__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cncc(C(F)F)c1 s275592__15865378__15840948__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc(C(F)F)c1 s275592__15865378__15840948__15859360
CCC(O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840950__15862300
CCC(O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840950__15859360
CCC(O)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840950__15857566
CC1(C)CCCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15842696__15862300
CC1(C)CCCC(O)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15842696__15859360
CC(=CC1CCC(C)CC1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842698__15859360
CC(Cl)=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842700__15862300
CC(Cl)=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842700__15859360
CC(Cl)=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842700__15857566
O=C(C=Cc1cccs1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842702__15862300
O=C(C=Cc1cccs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842702__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(N3CCOCC3)CC2)C1 s275592__15865378__15842704__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(N3CCOCC3)CC2)C1 s275592__15865378__15842704__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(Oc3ccccc3)CC2)C1 s275592__15865378__15842706__15859360
CC1(c2cc(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)no2)CC1 s275592__15865378__15842708__15862300
CC1(c2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)no2)CC1 s275592__15865378__15842708__15859360
CC=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842710__15862300
CC=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842710__15857566
CN1C(=O)NCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842712__15862300
CN1C(=O)NCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842712__15859360
CN1C(=O)NCC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842712__15857566
O=C(C=Cc1ccccc1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842714__15862300
O=C(C=Cc1ccccc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842714__15859360
CCC(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842716__15862300
CCC(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842716__15859360
CCC(F)(F)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842716__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCCC1F s275592__15865378__15842718__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCCC1F s275592__15865378__15842718__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1F s275592__15865378__15842720__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1F s275592__15865378__15842720__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1F s275592__15865378__15842720__15857566
CSCCCCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842722__15859360
CCC(F)(F)C(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842724__15862300
CCC(F)(F)C(C)(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842724__15859360
CC(=Cc1ccncc1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842734__15862300
CC(=Cc1ccncc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842734__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC2(CC1)CC2(F)F s275592__15865378__15842736__15859360
Cc1ccc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)ccc2c1 s275592__15865378__15842740__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CC[C@H](C(F)(F)F)O1 s275592__15865378__15842742__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(n3cnnn3)CC2)C1 s275592__15865378__15842744__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(n3cnnn3)CC2)C1 s275592__15865378__15842744__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCc2nnnn2C1 s275592__15865378__15842746__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCc2nnnn2C1 s275592__15865378__15842746__15859360
O=C(CSc1ccccn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842748__15862300
O=C(CSc1ccccn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842748__15859360
O=C(CC1CCC(F)(F)CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842750__15859360
O=C(Cc1ccc2[nH]nnc2c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842752__15859360
O=C1Cc2ccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc2N1 s275592__15865378__15842754__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2CC(O)CC(C2)C1 s275592__15865378__15842756__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@H]2C[C@@H](O)C2)C1 s275592__15865378__15842758__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@H]2C[C@@H](O)C2)C1 s275592__15865378__15842758__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)[C@H]2C[C@@H](O)C2)C1 s275592__15865378__15842758__15857566
CC(=Cc1ccco1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842760__15862300
CC(=Cc1ccco1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842760__15859360
O=C(CCC1CC1(Cl)Cl)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842762__15859360
CC1(C)CC1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842764__15862300
CC1(C)CC1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842764__15859360
CC1(C)CC1CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842764__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2ncccc12 s275592__15865378__15842768__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2ncccc12 s275592__15865378__15842768__15859360
O=C(CCc1cccnc1Cl)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842772__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(O)c1ccccc1 s275592__15865378__15842774__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)c1ccccc1 s275592__15865378__15842774__15859360
CCCCCCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842776__15862300
CCCCCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842776__15859360
CCCCCCCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842776__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc([N+](=O)[O-])cc1 s275592__15865378__15842780__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc([N+](=O)[O-])cc1 s275592__15865378__15842780__15859360
O=C(Cc1ccc([N+](=O)[O-])cc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842782__15859360
Cc1ccc(OCCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15842786__15859360
CC(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842788__15862300
CC(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842788__15859360
CC(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842788__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc([N+](=O)[O-])s1 s275592__15865378__15842790__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc([N+](=O)[O-])s1 s275592__15865378__15842790__15859360
O=C(C=CC(=O)N1CCOCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842794__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(O)CCOCC2)C1 s275592__15865378__15842798__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(O)CCOCC2)C1 s275592__15865378__15842798__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C(=O)NC3CC3)CCC2)C1 s275592__15865378__15842802__15859360
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)n1cccn1 s275592__15865378__15842806__15862300
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)n1cccn1 s275592__15865378__15842806__15859360
O=C(CSCC1CCCO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842808__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc([N+](=O)[O-])cn1 s275592__15865378__15842812__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc([N+](=O)[O-])cn1 s275592__15865378__15842812__15859360
CCC(=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15842814__15859360
CCSC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)C s275592__15865378__15842816__15862300
CCSC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15842816__15859360
C[C@@H](C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc(F)cc1 s275592__15865378__15844550__15862300
C[C@@H](C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15844550__15859360
COc1cc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)sn1 s275592__15865378__15844552__15859360
CN(C)C(=O)C#CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844554__15862300
CN(C)C(=O)C#CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844554__15859360
CN(C)C(=O)C#CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844554__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1C[C@H]1c1ccccn1 s275592__15865378__15844558__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1C[C@H]1c1ccccn1 s275592__15865378__15844558__15859360
C=C(C)CCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844564__15862300
C=C(C)CCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844564__15859360
C=C(C)CCCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844564__15857566
CC1(C)C(O)CC1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844566__15862300
CC1(C)C(O)CC1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844566__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1conc1C1CCC1 s275592__15865378__15844568__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1conc1C1CCC1 s275592__15865378__15844568__15859360
O=C(C=Cc1cnccn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844570__15862300
O=C(C=Cc1cnccn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844570__15859360
CCc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(C)n1 s275592__15865378__15844572__15862300
CCc1ncc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15844572__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc2c(n1)CCC2 s275592__15865378__15844574__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(n1)CCC2 s275592__15865378__15844574__15859360
CC(F)(F)C(C)(C)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844578__15862300
CC(F)(F)C(C)(C)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844578__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCC2(CCC2)C1 s275592__15865378__15844580__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCC2(CCC2)C1 s275592__15865378__15844580__15859360
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nn1C s275592__15865378__15844582__15862300
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15844582__15859360
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)nn1C s275592__15865378__15844582__15857566
CC(C)c1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)co1 s275592__15865378__15844584__15862300
CC(C)c1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)co1 s275592__15865378__15844584__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1conc1C1CCCO1 s275592__15865378__15844586__15859360
O=C(Cc1csc(Cl)c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844588__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC(F)C1 s275592__15865378__15844590__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC(F)C1 s275592__15865378__15844590__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC(F)C1 s275592__15865378__15844590__15857566
CCc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15844592__15862300
CCc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15844592__15859360
CCc1ccc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)[nH]1 s275592__15865378__15844592__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1nc(=O)[nH]c(=O)[nH]1 s275592__15865378__15844596__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nc(=O)[nH]c(=O)[nH]1 s275592__15865378__15844596__15859360
CCc1ccnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15844602__15862300
CCc1ccnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844602__15859360
Cc1cccc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)nccc12 s275592__15865378__15844604__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)C1CCCCC1 s275592__15865378__15844608__15859360
CC(C)C1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C(=O)N1 s275592__15865378__15844612__15859360
O=C(C#CC1CCCO1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844614__15862300
O=C(C#CC1CCCO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844614__15859360
O=C(C#CC1CCCO1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844614__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CC[C@H]2[C@@H](C1)C2(F)F s275592__15865378__15844616__15859360
C=CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC=CC1 s275592__15865378__15844618__15862300
C=CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC=CC1 s275592__15865378__15844618__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23CCCC(C2)OC3)C1 s275592__15865378__15844620__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CCCC(C2)OC3)C1 s275592__15865378__15844620__15859360
CC1OCCC1(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844622__15862300
CC1OCCC1(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844622__15859360
CC1(C)OCc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)n[nH]c21 s275592__15865378__15844624__15859360
Cc1ncc(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)s1 s275592__15865378__15844632__15862300
Cc1ncc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15844632__15859360
CCc1scnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844634__15862300
CCc1scnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844634__15859360
Cn1ncc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)sc21 s275592__15865378__15844636__15859360
Cc1cccc(SCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844640__15859360
Cc1cccc(C(O)C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15844642__15862300
Cc1cccc(C(O)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844642__15859360
O=C(Cn1cc2ncccc2n1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844644__15859360
O=C(COCCc1cccs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844648__15859360
O=C1CC2CCC(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)CC2N1 s275592__15865378__15844652__15859360
C[C@@H]1C[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844656__15862300
C[C@@H]1C[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844656__15859360
C[C@@H]1C[C@H]1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844656__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)c2cncs2)C1 s275592__15865378__15844658__15859360
CC1(C)C2CCC1(CC(=O)NCC(F)=C1CN(C(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15844664__15859360
CC(F)(F)c1cccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844666__15859360
O=C(CN1Cc2ccccc2C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844670__15859360
CNC(=O)NC(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846352__15862300
CNC(=O)NC(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846352__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23COC(CCO2)C3)C1 s275592__15865378__15846360__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23COC(CCO2)C3)C1 s275592__15865378__15846360__15859360
CCn1cnnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846362__15862300
CCn1cnnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846362__15859360
CCn1cnnc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15846362__15857566
CCC(=Cc1ccccc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846366__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(C3CCC3)CC2)C1 s275592__15865378__15846368__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C3CCC3)CC2)C1 s275592__15865378__15846368__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(C3CCC3)CC2)C1 s275592__15865378__15846368__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(=O)[nH]ncc2c1 s275592__15865378__15846372__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@@H]1CC[C@@H]2C[C@@H]21 s275592__15865378__15846376__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1CC[C@@H]2C[C@@H]21 s275592__15865378__15846376__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)[C@@H]1CC[C@@H]2C[C@@H]21 s275592__15865378__15846376__15857566
CC1(C)C(C)(C)C1(F)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846378__15862300
CC1(C)C(C)(C)C1(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846378__15859360
C[C@@H]1C(=O)N(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C(=O)[C@@H]1C s275592__15865378__15846380__15859360
CC(C)[C@@H]1CCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846382__15862300
CC(C)[C@@H]1CCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846382__15859360
CC(C)Cc1nccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15846384__15859360
O=C(CC1CC2(CCCC2)CO1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846388__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC2(CCOCC2)O1 s275592__15865378__15846390__15859360
O=C(COC1COC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846396__15862300
O=C(COC1COC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846396__15859360
O=C(COC1COC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15846396__15857566
C[C@@H]1C[C@]2(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)C[C@H]12 s275592__15865378__15846398__15862300
C[C@@H]1C[C@]2(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)C[C@H]12 s275592__15865378__15846398__15859360
C[C@@H]1C[C@]2(C(=O)NCC(F)=C3CN(C(=O)CSc4n[nH]c(=O)[nH]4)C3)C[C@H]12 s275592__15865378__15846398__15857566
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nn1CCO s275592__15865378__15846400__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1CCO s275592__15865378__15846400__15859360
Cc1ccnc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15846404__15862300
Cc1ccnc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15846404__15859360
O=C1N[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[C@@H]2CC[C@H]12 s275592__15865378__15846406__15862300
O=C1N[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[C@@H]2CC[C@H]12 s275592__15865378__15846406__15859360
CNC(=O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846408__15862300
CNC(=O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846408__15859360
CNC(=O)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15846408__15857566
CC(OC1COC1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15846416__15862300
CC(OC1COC1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15846416__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2c(c1)COCC2 s275592__15865378__15846418__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCCC1(F)F s275592__15865378__15846420__15859360
C#Cc1cccc(OCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15846422__15859360
Cn1cc([N+](=O)[O-])c(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15846424__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCOC1 s275592__15865378__15846428__15862300
COC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCOC1 s275592__15865378__15846428__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@]23C[C@H]2[C@H](c2ccccc2)C3)C1 s275592__15865378__15846432__15859360
CCCCC[C@@H](O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840954__15862300
CCCCC[C@@H](O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840954__15859360
CN1C(=O)CCC1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840956__15862300
CN1C(=O)CCC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840956__15859360
CN1C(=O)CCC1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840956__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn2ccsc12 s275592__15865378__15840958__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn2ccsc12 s275592__15865378__15840958__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(c3ccc(F)cn3)CC2)C1 s275592__15865378__15840960__15859360
O=C(C[C@@H]1CCCC[C@H]1O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840962__15862300
O=C(C[C@@H]1CCCC[C@H]1O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840962__15859360
CCn1nnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1C s275592__15865378__15840964__15862300
CCn1nnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1C s275592__15865378__15840964__15859360
CC(=NO)C1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15840966__15859360
Cc1cnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc1Cl s275592__15865378__15840970__15862300
Cc1cnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15840970__15859360
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc1CO s275592__15865378__15840972__15862300
Cc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1CO s275592__15865378__15840972__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(c1)B(O)OC2 s275592__15865378__15840978__15859360
COc1sccc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840980__15862300
COc1sccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840980__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(O)CC1CCCCC1 s275592__15865378__15840982__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)CC1CCCCC1 s275592__15865378__15840982__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1c[nH]nc1C(F)F s275592__15865378__15840984__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]nc1C(F)F s275592__15865378__15840984__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)N1CCSCC1 s275592__15865378__15840988__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2CCCC(C2)C1 s275592__15865378__15840992__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2CCCC(C2)C1 s275592__15865378__15840992__15859360
CCC1CN(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15840994__15862300
CCC1CN(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15840994__15859360
CCC1CN(CC(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15840994__15857566
Cc1cn(C)cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15840996__15862300
Cc1cn(C)cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15840996__15859360
Cc1cn(C)cc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15840996__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CN(C2CCOCC2)C1 s275592__15865378__15840998__15859360
O=C(C=Cc1ccc(Cl)cc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841000__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(N3CCCC3)CCC2)C1 s275592__15865378__15841002__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(N3CCCC3)CCC2)C1 s275592__15865378__15841002__15859360
C=CC=CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841006__15862300
C=CC=CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841006__15859360
C=CC=CCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841006__15857566
C=CCC(CC(C)C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841008__15862300
C=CCC(CC(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841008__15859360
O=C(COCc1ccccn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841010__15862300
O=C(COCc1ccccn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841010__15859360
O=C(COc1nc(=O)[nH]c(=O)[nH]1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841012__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2CCC(C1)S2 s275592__15865378__15841014__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2CCC(C1)S2 s275592__15865378__15841014__15859360
O=C(C=CCl)NCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841016__15859360
Cn1ncc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)ncnc21 s275592__15865378__15841018__15859360
CCc1ccc(C(C)=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841020__15859360
O=C(C=Cc1cncc(F)c1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841022__15862300
O=C(C=Cc1cncc(F)c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841022__15859360
C#CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15841024__15862300
C#CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841024__15859360
C#CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC1 s275592__15865378__15841024__15857566
CN1CCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841026__15862300
CN1CCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841026__15859360
CN1CCC[C@H]1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841026__15857566
CCCC=CC(O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841030__15862300
CCCC=CC(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841030__15859360
CCCC=CC(O)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841030__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCOC2(CCCC2)C1 s275592__15865378__15841032__15859360
O=C(Cc1nc(C2CC2)cs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841034__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC=CCO1 s275592__15865378__15841036__15862300
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O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC=CCO1 s275592__15865378__15841036__15857566
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23CCOC2CCOC3)C1 s275592__15865378__15841038__15862300
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CC(C)(CCCO)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841040__15862300
CC(C)(CCCO)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841040__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccn(CCF)n1 s275592__15865378__15841042__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn(CCF)n1 s275592__15865378__15841042__15859360
O=C(COc1ccsn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841044__15862300
O=C(COc1ccsn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841044__15859360
O=C(CCN1CCC(F)C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841046__15862300
O=C(CCN1CCC(F)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841046__15859360
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)cc(=O)[nH]1 s275592__15865378__15841048__15862300
Cc1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc(=O)[nH]1 s275592__15865378__15841048__15859360
CN1CCCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1=O s275592__15865378__15841052__15862300
CN1CCCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841052__15859360
O=C(CCOC1CC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841054__15862300
O=C(CCOC1CC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841054__15859360
O=C(CCOC1CC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841054__15857566
Cn1cncc1C=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841056__15862300
Cn1cncc1C=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841056__15859360
Cc1cccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15841058__15862300
Cc1cccc(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841058__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnccn1 s275592__15865378__15841060__15862300
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnccn1 s275592__15865378__15841060__15859360
CCCCC(O)CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841064__15862300
CCCCC(O)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841064__15859360
CC1(C)Cc2ccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc2C1 s275592__15865378__15841066__15859360
COC1CN(C)C(C)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15841068__15862300
COC1CN(C)C(C)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841068__15859360
O=C(CCCCCO)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841070__15862300
O=C(CCCCCO)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841070__15859360
O=C(CCCCCO)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841070__15857566
Cc1n[nH]c2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cccc12 s275592__15865378__15841072__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CS(=O)CCC1 s275592__15865378__15841074__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CS(=O)CCC1 s275592__15865378__15841074__15859360
NS(=O)(=O)NCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841076__15862300
NS(=O)(=O)NCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841076__15859360
CCSc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15842818__15859360
CCCC(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842822__15862300
CCCC(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842822__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cscn1 s275592__15865378__15842824__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cscn1 s275592__15865378__15842824__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cscn1 s275592__15865378__15842824__15857566
CCCCc1csc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15842826__15859360
CC(c1ccccc1)C(O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842828__15859360
CNC(=O)NC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15842834__15859360
Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842836__15859360
CSc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)ccn1 s275592__15865378__15842838__15862300
CSc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15842838__15859360
O=C(CCN1CCCCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842840__15862300
O=C(CCN1CCCCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842840__15859360
Cc1nc(C)n(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15842844__15862300
Cc1nc(C)n(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15842844__15859360
O=C(CN1CCCCC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842848__15862300
O=C(CN1CCCCC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842848__15859360
O=C(CN1CCCCC1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842848__15857566
O=C(Cn1ccc([N+](=O)[O-])n1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842850__15862300
O=C(Cn1ccc([N+](=O)[O-])n1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842850__15859360
Cc1n[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1Cl s275592__15865378__15842854__15862300
Cc1n[nH]c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15842854__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(CO)CCC2)C1 s275592__15865378__15842856__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(CO)CCC2)C1 s275592__15865378__15842856__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(CO)CCC2)C1 s275592__15865378__15842856__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCCC1O s275592__15865378__15842858__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCCC1O s275592__15865378__15842858__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CCCCC1O s275592__15865378__15842858__15857566
Cn1ccnc1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842860__15862300
Cn1ccnc1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842860__15859360
Cn1ccnc1CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842860__15857566
CC(C)(CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[N+](=O)[O-] s275592__15865378__15842862__15862300
CC(C)(CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[N+](=O)[O-] s275592__15865378__15842862__15859360
CN1C(=O)CSC1=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842864__15862300
CN1C(=O)CSC1=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842864__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(C1)CC(F)(F)C2 s275592__15865378__15842866__15859360
COC1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842868__15862300
COC1CCC(C)(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842868__15859360
CC1C(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCN1C s275592__15865378__15842870__15862300
CC1C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCN1C s275592__15865378__15842870__15859360
CC1C(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCN1C s275592__15865378__15842870__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cncc(O)n1 s275592__15865378__15842872__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc(O)n1 s275592__15865378__15842872__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cncc(O)n1 s275592__15865378__15842872__15857566
CN1CCCCC1CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842876__15862300
CN1CCCCC1CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842876__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1c[nH]c(=O)s1 s275592__15865378__15842878__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c[nH]c(=O)s1 s275592__15865378__15842878__15859360
NC(=O)CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842880__15862300
NC(=O)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842880__15859360
NC(=O)CCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842880__15857566
C=CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15842882__15862300
C=CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842882__15859360
C=CCC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__15842882__15857566
O=C(COC(F)F)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842884__15862300
O=C(COC(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842884__15859360
O=C(COC(F)F)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842884__15857566
O=C(CC1COc2ccccc21)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842888__15859360
COC(=Cc1ccccc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842890__15859360
Cc1nc(=O)[nH]c(C)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842892__15862300
Cc1nc(=O)[nH]c(C)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842892__15859360
Cc1nc2cccnn2c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842894__15859360
[N-]=[N+]=NCc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15842900__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC(=O)N1 s275592__15865378__15842904__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC(=O)N1 s275592__15865378__15842904__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCC(=O)N1 s275592__15865378__15842904__15857566
COC(C)(C)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842906__15862300
COC(C)(C)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842906__15859360
COC(C)(C)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842906__15857566
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)c2nccs2)C1 s275592__15865378__15842910__15859360
O=C(Cc1ccc2ncccc2c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842912__15859360
O=C(CC1CCCC(O)C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842914__15862300
O=C(CC1CCCC(O)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842914__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)C2CCOCC2)C1 s275592__15865378__15842916__15859360
CC(O)CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842918__15862300
CC(O)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842918__15859360
CC(O)CCC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842918__15857566
CC1(C)CC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCO1 s275592__15865378__15842924__15862300
CC1(C)CC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15842924__15859360
CCS(=O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842928__15862300
CCS(=O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842928__15859360
CCS(=O)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842928__15857566
CN(C)C(=O)CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842930__15862300
CN(C)C(=O)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842930__15859360
C#CCC(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842932__15862300
C#CCC(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842932__15859360
C#CCC(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842932__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cncc(Cl)c1O s275592__15865378__15842934__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc(Cl)c1O s275592__15865378__15842934__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(OC2CC2)cc1 s275592__15865378__15842938__15859360
O=C(Cn1ncc2ncccc21)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842940__15859360
CC(CCO)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844674__15862300
CC(CCO)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844674__15859360
CC(CCO)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844674__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)=CC1CC1 s275592__15865378__15844676__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)=CC1CC1 s275592__15865378__15844676__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)=CC1CC1 s275592__15865378__15844676__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@@H]1COC[C@H]1C(F)(F)F s275592__15865378__15844678__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nc2c(s1)COCC2 s275592__15865378__15844680__15859360
CC(C)N1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1=O s275592__15865378__15844682__15859360
CC(C)(C)c1ccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]1 s275592__15865378__15844688__15862300
CC(C)(C)c1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15844688__15859360
O=C(CC1CC(F)C1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844690__15862300
O=C(CC1CC(F)C1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844690__15859360
O=C(CC1CC(F)C1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844690__15857566
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nc(C)n1 s275592__15865378__15844692__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc(C)n1 s275592__15865378__15844692__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)CC1CCC1 s275592__15865378__15844694__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)CC1CCC1 s275592__15865378__15844694__15859360
COc1nc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)ncc1F s275592__15865378__15844696__15862300
COc1nc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)ncc1F s275592__15865378__15844696__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCN2CCOCC12 s275592__15865378__15844700__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCN2CCOCC12 s275592__15865378__15844700__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)CC1CCCC1 s275592__15865378__15844702__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)CC1CCCC1 s275592__15865378__15844702__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC2C(CC1)C2(F)F s275592__15865378__15844704__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2(C1)CC2(F)F s275592__15865378__15844706__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(C1)CC2(F)F s275592__15865378__15844706__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ncccc1CO s275592__15865378__15844708__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ncccc1CO s275592__15865378__15844708__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)=Cc1cnc[nH]1 s275592__15865378__15844710__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)=Cc1cnc[nH]1 s275592__15865378__15844710__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2ccncc2c(O)n1 s275592__15865378__15844712__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)CCn2cccn2)C1 s275592__15865378__15844714__15859360
Cc1ncc2ccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cn12 s275592__15865378__15844718__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc2ccsc12 s275592__15865378__15844720__15859360
CCC(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)n1cccn1 s275592__15865378__15844722__15862300
CCC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)n1cccn1 s275592__15865378__15844722__15859360
O=C(CCC1CCC(=O)NC1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844728__15862300
O=C(CCC1CCC(=O)NC1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844728__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2c(n1)CCCC2 s275592__15865378__15844730__15859360
O=C(C[C@@H]1CCC[C@H](C2CC2)O1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844734__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)[C@H](O)CF s275592__15865378__15844736__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@H](O)CF s275592__15865378__15844736__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)[C@H](O)CF s275592__15865378__15844736__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CC2(CCOC2)C1 s275592__15865378__15844738__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CC2(CCOC2)C1 s275592__15865378__15844738__15859360
CCC1(C)C=C(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15844740__15862300
CCC1(C)C=C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15844740__15859360
CCC1(C)C=C(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15844740__15857566
CCC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15844742__15862300
CCC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15844742__15859360
CCC1(C)CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)C1 s275592__15865378__15844742__15857566
Cc1nnc(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1C s275592__15865378__15844744__15862300
Cc1nnc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1C s275592__15865378__15844744__15859360
O=C(Cn1nc2c(n1)CCCC2)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844746__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2ccoc2cc1F s275592__15865378__15844748__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1coc2c1COC2 s275592__15865378__15844750__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1coc2c1COC2 s275592__15865378__15844750__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)[C@H]2C[C@H](n3cnnc3)C2)C1 s275592__15865378__15844752__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)[C@H]2C[C@H](n3cnnc3)C2)C1 s275592__15865378__15844752__15859360
CC(C(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15844754__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc2n(n1)CC(F)C2 s275592__15865378__15844756__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc2n(n1)CC(F)C2 s275592__15865378__15844756__15859360
CCn1cnc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844758__15862300
CCn1cnc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844758__15859360
CCn1cnc(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)n1 s275592__15865378__15844758__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2(C1)CC1(CCC1)C2 s275592__15865378__15844760__15859360
CN1CCOCC1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844764__15862300
CN1CCOCC1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844764__15859360
C=CCCCc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15844766__15859360
CCCC(C)(O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844768__15862300
CCCC(C)(O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844768__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCCSS1 s275592__15865378__15844776__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCCSS1 s275592__15865378__15844776__15859360
Cc1ccc(C(C)CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15844778__15859360
Cn1cnnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844782__15862300
Cn1cnnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844782__15859360
Cn1cnnc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844782__15857566
O=C(CC1C[C@@H]2COC[C@H]12)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844784__15862300
O=C(CC1C[C@@H]2COC[C@H]12)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844784__15859360
CCCC(CC)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844786__15862300
CCCC(CC)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844786__15859360
CCCC(CC)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844786__15857566
Cc1cc(F)cc(C(C)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15844790__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccc2c(c1)CC2 s275592__15865378__15844792__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2c(c1)CC2 s275592__15865378__15844792__15859360
Cc1nc(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)[nH]c1C s275592__15865378__15844794__15862300
Cc1nc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)[nH]c1C s275592__15865378__15844794__15859360
COC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCSC1 s275592__15865378__15841078__15862300
COC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCSC1 s275592__15865378__15841078__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1csnc1Cl s275592__15865378__15841080__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1csnc1Cl s275592__15865378__15841080__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C(F)F)CCOCC2)C1 s275592__15865378__15841084__15859360
CCn1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nc2ccccc21 s275592__15865378__15841086__15859360
Cc1ncc([N+](=O)[O-])n1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841090__15859360
Cc1conc1CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841094__15862300
Cc1conc1CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841094__15859360
Cc1conc1CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841094__15857566
CCOCC(N=[N+]=[N-])C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841096__15862300
CCOCC(N=[N+]=[N-])C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841096__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCC(F)(F)CO1 s275592__15865378__15841098__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC(F)(F)CO1 s275592__15865378__15841098__15859360
C#Cc1cccc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c1 s275592__15865378__15841100__15862300
C#Cc1cccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841100__15859360
CSCc1ccc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841108__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(O)CCCCC2)C1 s275592__15865378__15841110__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(O)CCCCC2)C1 s275592__15865378__15841110__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(O)CCCCC2)C1 s275592__15865378__15841110__15857566
O=C(CSCc1cccnc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841114__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnccc1Cl s275592__15865378__15841116__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnccc1Cl s275592__15865378__15841116__15859360
O=C(Cn1cc([N+](=O)[O-])cn1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841118__15862300
O=C(Cn1cc([N+](=O)[O-])cn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841118__15859360
CC(C)CN1CCCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841120__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1c(F)cccc1[N+](=O)[O-] s275592__15865378__15841122__15859360
CS(=O)(=O)NCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841126__15862300
CS(=O)(=O)NCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841126__15859360
CC(C)CC(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841130__15859360
O=C(CC1CC(F)(F)C1(F)F)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841132__15859360
O=C(Cn1[nH]c(=O)ccc1=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841136__15862300
O=C(Cn1[nH]c(=O)ccc1=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841136__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(O)CC2)C1 s275592__15865378__15841140__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(O)CC2)C1 s275592__15865378__15841140__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C2(O)CC2)C1 s275592__15865378__15841140__15857566
C=CCn1ccnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841142__15862300
C=CCn1ccnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841142__15859360
CC(Sc1nncn1C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841144__15859360
O=C(CSc1nncs1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841146__15859360
CN(CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ncccn1 s275592__15865378__15841150__15862300
CN(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ncccn1 s275592__15865378__15841150__15859360
NS(=O)(=O)CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841154__15862300
NS(=O)(=O)CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841154__15859360
NS(=O)(=O)CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841154__15857566
NS(=O)(=O)CCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841156__15862300
NS(=O)(=O)CCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841156__15859360
Cc1nn2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)nc2s1 s275592__15865378__15841158__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc2cnsc2c1 s275592__15865378__15841160__15859360
Cc1sncc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15841162__15862300
Cc1sncc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841162__15859360
Cc1sncc1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15841162__15857566
O=C(CCSc1ccccn1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841164__15859360
CC(C)c1nnc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841166__15859360
Cc1ccccc1C(F)(F)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15841168__15859360
O=C(NCC(F)=C1CN(C(=O)CC2CCC3(CCC3)CO2)C1)c1cc(O)no1 s275592__15865378__15841170__14128900
O=C(NCC(F)=C1CN(C(=O)CC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186218
CC(C)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186220
CC(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186222
O=C(NCC(F)=C1CN(C(=O)c2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186226
O=C(NCC(F)=C1CN(C(=O)c2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186228
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186230
O=C(NCC(F)=C1CN(C(=O)c2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186234
O=C(NCC(F)=C1CN(C(=O)Cc2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__13186236
O=C(NCC(F)=C1CN(C(=O)c2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__13186238
CC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186240
Cc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186242
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__13186244
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__13186246
O=C(NCC(F)=C1CN(C(=O)c2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__13186248
O=C(NCC(F)=C1CN(C(=O)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186250
CC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186252
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186254
O=C(NCC(F)=C1CN(C(=O)c2cnccn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186256
Cc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186258
O=C(NCC(F)=C1CN(C(=O)CC2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186260
O=C(NCC(F)=C1CN(C(=O)CCC2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186262
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Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__13186268
O=C(NCC(F)=C1CN(C(=O)Cc2ccsc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186270
CC1CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186272
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__13186274
CCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186276
CC(C)=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186278
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O=C(NCC(F)=C1CN(C(=O)c2cc[n+]([O-])cc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186282
O=C(NCC(F)=C1CN(C(=O)C2CC3C=CC2C3)C1)c1cc(O)no1 s275592__15865378__15841170__13186284
CC(=O)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186286
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__13186288
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__13186290
O=C(NCC(F)=C1CN(C(=O)CC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186292
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CSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186296
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__13186298
CSCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186300
CC(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186302
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Cc1occc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186308
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O=C(NCC(F)=C1CN(C(=O)Cn2cnnn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186312
O=C(NCC(F)=C1CN(C(=O)CN2CCCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__13186314
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__13186316
Cc1noc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186318
Cc1nnsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186320
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__13186322
O=C(NCC(F)=C1CN(C(=O)C2CC=CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186324
O=C(NCC(F)=C1CN(C(=O)CCc2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__13186326
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__13186328
O=C(NCC(F)=C1CN(C(=O)c2ccc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__13186330
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)c[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__13186332
CC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186334
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1C s275592__15865378__15841170__13186336
O=C(NCC(F)=C1CN(C(=O)c2ccoc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186338
O=C(NCC(F)=C1CN(C(=O)Cn2cccn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186340
Cc1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186342
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC2C3)C1)c1cc(O)no1 s275592__15865378__15841170__13186344
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)o2)C1)c1cc(O)no1 s275592__15865378__15841170__13186346
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__13186348
CCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186350
CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186352
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__13186354
Cn1cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186356
O=C(NCC(F)=C1CN(C(=O)CCn2cncn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186358
CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186362
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__13186364
O=C(NCC(F)=C1CN(C(=O)CCn2cccn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186368
O=C(NCC(F)=C1CN(C(=O)c2ccccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__13186370
CCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186372
CC(C)SCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186374
N#CCSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186376
CC(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186378
CCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186380
CC(C)OCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186382
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__13186384
O=C(NCC(F)=C1CN(C(=O)CCC2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__13186386
O=C(NCC(F)=C1CN(C(=O)C2COCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__13186388
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__13186390
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cccn1 s275592__15865378__15841170__13186392
CCCCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186394
CSC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186396
CCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186398
CC(C)COCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186400
CCOCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186402
O=C(NCC(F)=C1CN(C(=O)COCC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186404
O=C(NCC(F)=C1CN(C(=O)CC2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__13186406
Cc1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186408
O=C(NCC(F)=C1CN(C(=O)c2cn[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__13186410
O=C(NCC(F)=C1CN(C(=O)CNC(=O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186412
COCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186414
O=C(NCC(F)=C1CN(C(=O)COC2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186416
Cc1ncncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186418
CCSCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186420
CCOC1CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186422
O=C(NCC(F)=C1CN(C(=O)c2cnsn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186424
O=C(NCC(F)=C1CN(C(=O)c2cnns2)C1)c1cc(O)no1 s275592__15865378__15841170__13186426
COC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186428
O=C(NCC(F)=C1CN(C(=O)c2ccon2)C1)c1cc(O)no1 s275592__15865378__15841170__13186430
CCCSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186432
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__13186434
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__13186436
O=C(NCC(F)=C1CN(C(=O)c2cncs2)C1)c1cc(O)no1 s275592__15865378__15841170__13186438
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__13186440
Cc1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__13186446
CC(C)COC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186448
CCCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186450
CCC=C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186452
CS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186454
O=C(NCC(F)=C1CN(C(=O)C=C2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186456
Cc1ocnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186458
CCOC(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186460
O=C(NCC(F)=C1CN(C(=O)CC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__13186462
COC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186464
CC(C)OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186466
CC(OCC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186468
CCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186470
CCCCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186472
C=CCCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186474
O=C(NCC(F)=C1CN(C(=O)C2CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186476
O=C(NCC(F)=C1CN(C(=O)c2ccnc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__13186478
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__13186480
Cn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186482
CCC(OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186484
COCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186486
CCCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186488
COC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186490
Cn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__13186492
O=C(NCC(F)=C1CN(C(=O)C2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186494
C=CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186496
O=C(NCC(F)=C1CN(C(=O)C2=COCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186498
COC(=O)C1CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186500
O=C(NCC(F)=C1CN(C(=O)C2CCCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186504
CCOCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186506
CCNC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186508
O=C(NCC(F)=C1CN(C(=O)c2cscn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186510
COCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186512
CC(C)(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186514
C=CCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186516
O=C(NCC(F)=C1CN(C(=O)c2cocn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186518
O=C1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__13186520
O=C(NCC(F)=C1CN(C(=O)CC2=CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186522
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__13186524
CSCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186526
CN1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186528
CCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186530
CC(C)(C)/C=C/C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186532
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186534
CC(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186536
COCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186538
CCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186540
Cc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186542
CC(C)(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186544
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC2O3)C1)c1cc(O)no1 s275592__15865378__15841170__13186546
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__13186548
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__13186550
Nc1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186552
O=C(NCC(F)=C1CN(C(=O)CCC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186554
Cc1[nH]nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__13186556
O=C(NCC(F)=C1CN(C(=O)CC2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186558
CCCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186560
O=C(NCC(F)=C1CN(C(=O)Cc2ccon2)C1)c1cc(O)no1 s275592__15865378__15841170__13186562
CCc1ocnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186566
O=C(NCC(F)=C1CN(C(=O)CC2CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186568
O=C(NCC(F)=C1CN(C(=O)C2CC=CC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186570
O=C(NCC(F)=C1CN(C(=O)Cc2ccn[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__13186572
O=C(NCC(F)=C1CN(C(=O)c2ccncc2F)C1)c1cc(O)no1 s275592__15865378__15841170__13186574
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nnn1C s275592__15865378__15841170__13186576
Cc1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186578
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__13186580
CN1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__13186582
Cc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__13186584
O=C(NCC(F)=C1CN(C(=O)CCC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__13186586
C=CCOCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186588
O=C(NCC(F)=C1CN(C(=O)CC2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186592
O=C(NCC(F)=C1CN(C(=O)c2cccc(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__13186596
CC1(C)C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__13186598
Cc1ncoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186600
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__13186602
O=C(NCC(F)=C1CN(C(=O)C2C3CCCC32)C1)c1cc(O)no1 s275592__15865378__15841170__13186604
N#Cc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__13186606
Cc1cscc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186608
O=C(NCC(F)=C1CN(C(=O)CCC2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186610
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__13186612
O=C(NCC(F)=C1CN(C(=O)CCc2nnc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__13186614
Cc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186616
Cc1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186618
CC=C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186620
O=C(NCC(F)=C1CN(C(=O)CCC2CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186622
O=C(NCC(F)=C1CN(C(=O)CCc2ccoc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186624
O=C(NCC(F)=C1CN(C(=O)C2CC(F)(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__13186626
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__13186628
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)=C1CCCC1 s275592__15865378__15841170__13186630
O=C(NCC(F)=C1CN(C(=O)CC2CCCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__13186632
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__13186634
O=C(NCC(F)=C1CN(C(=O)C=C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186636
O=C(NCC(F)=C1CN(C(=O)c2cncc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__13186638
CCC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CC s275592__15865378__15841170__13186640
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c(=O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__13186642
CC(C)=C(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186644
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCN1 s275592__15865378__15841170__13186646
O=C(NCC(F)=C1CN(C(=O)C2=CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186648
O=C(NCC(F)=C1CN(C(=O)C(F)=C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186650
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__13186652
Cn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__13186654
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__13186656
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc1C s275592__15865378__15841170__13186658
O=C(NCC(F)=C1CN(C(=O)Cc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186660
O=C(NCC(F)=C1CN(C(=O)C2CCCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__13186662
Cc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__13186664
CCC(SC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186666
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cccc1 s275592__15865378__15841170__13186668
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncn1 s275592__15865378__15841170__13186670
CC1(C)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186672
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__13186674
CCC(C)OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186676
CC1(C)C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186678
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__13186680
CC(O)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__13186682
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15841170__13186684
CSC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186686
O=C(NCC(F)=C1CN(C(=O)CN2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186688
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__13186690
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cncn1 s275592__15865378__15841170__13186692
NC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__13186694
CN1CCOCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186696
Cc1nscc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186698
C#CCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186700
CC(C)(C)OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186702
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__13186704
C#CCNC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186706
CCNC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186708
CNC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186710
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__13186714
COC(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186716
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__13186718
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186720
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__13186722
O=C(NCC(F)=C1CN(C(=O)c2cncnc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186724
O=C(NCC(F)=C1CN(C(=O)c2ncccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__13186726
O=C(NCC(F)=C1CN(C(=O)C2=CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186730
O=C(NCC(F)=C1CN(C(=O)Cc2ccoc2)C1)c1cc(O)no1 s275592__15865378__15841170__13186732
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__13186736
O=C(NCC(F)=C1CN(C(=O)C2=CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186740
C[C@H](NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186742
O=C(NCC(F)=C1CN(C(=O)CC2OCCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__13186744
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__13186746
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__13186748
Cc1ccn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186750
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1 s275592__15865378__15841170__13186752
O=C(NCC(F)=C1CN(C(=O)CCn2ccnn2)C1)c1cc(O)no1 s275592__15865378__15841170__13186754
CC(=O)N1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__13186756
Cn1oc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15841170__13186758
CCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186760
COC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__13186762
CC1OCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186764
C#CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186766
O=C(NCC(F)=C1CN(C(=O)c2ccoc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__13186768
C=CC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186770
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ns1 s275592__15865378__15841170__13186772
CCn1ccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186778
O=C(NCC(F)=C1CN(C(=O)C2CCCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186780
O=C(NCC(F)=C1CN(C(=O)CCc2ncc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__13186782
O=C(NCC(F)=C1CN(C(=O)C2CCC(O)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186784
CC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186786
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__13186788
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__13186790
CCc1occc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186792
Cc1cc[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186794
Cn1nncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186796
O=C1NC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__13186798
CCCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186800
CC1CC(C)C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__13186802
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@@H]2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__13186804
Cc1coc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186806
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__13186810
CCc1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186812
CC(C)[C@@H](O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186814
CCOC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__13186816
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__13186818
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__13186820
Cc1nnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__13186822
Cn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__13186824
CNC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186826
O=C(NCC(F)=C1CN(C(=O)c2sccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__13186828
CCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__13186830
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__13186832
CCn1nncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186834
Cc1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__13186836
O=C(NCC(F)=C1CN(C(=O)C2CC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__13186838
CCC(C)=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186840
Cc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186842
CC(C)C#CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186846
Cc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186848
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186850
Cc1c[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186852
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)=C1CCC1 s275592__15865378__15841170__13186854
O=C(NCC(F)=C1CN(C(=O)C#CC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186856
CC(C)(C)C#CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186858
Cc1n[nH]c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__13186860
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__13186862
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__13186864
Cc1cn(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186866
O=C(NCC(F)=C1CN(C(=O)C2CCCC(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__13186868
Cn1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__13186870
COCC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__13186872
COCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__13186204
O=C(NCC(F)=C1CN(C(=O)C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186212
O=C(NCC(F)=C1CN(C(=O)C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186214
O=C(NCC(F)=C1CN(C(=O)C2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__13186216
CCCCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__14130356
C=CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14130358
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)C=CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130360
O=C(NCC(F)=C1CN(C(=O)CCNC(=O)C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130362
CC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14130366
Cc1cn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc12 s275592__15865378__15841170__14130368
CS(=O)(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130370
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)COC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130372
Cc1ccc2c(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c[nH]c2c1 s275592__15865378__15841170__14130374
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCCC1 s275592__15865378__15841170__14130376
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__14130378
CCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130382
O=C(NCC(F)=C1CN(C(=O)c2ccc3n[nH]c(=O)n3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130388
Cc1nnc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cn12 s275592__15865378__15841170__14130390
O=C(NCC(F)=C1CN(C(=O)c2ccc3nncn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130392
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3ccnc3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14130394
O=C(NCC(F)=C1CN(C(=O)c2cccn3ccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14130396
CNC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130398
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3cn[nH]c3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130400
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130402
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(=O)N1 s275592__15865378__15841170__14130406
Cc1noc(Cl)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130408
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14130412
O=C(CC1CCCC1)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130414
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3cnnc3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130418
O=C(NCC(F)=C1CN(C(=O)c2cncc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130420
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)(F)F)n[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14130426
Cc1cccn2cc(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nc12 s275592__15865378__15841170__14130428
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2[nH]ncc2c1 s275592__15865378__15841170__14130430
Cc1nccn1CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130432
Cc1noc(C)c1C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130434
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14130436
CC(C)(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14130438
O=C(NCC(F)=C1CN(C(=O)CCCCN2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130440
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14130442
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1F s275592__15865378__15841170__14130444
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1c(C)noc1C s275592__15865378__15841170__14130446
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3cccn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130448
CC1Cc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2O1 s275592__15865378__15841170__14130450
CN(C)Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14130452
O=C(NCC(F)=C1CN(C(=O)CCN2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130454
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCOCC1 s275592__15865378__15841170__14130458
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCc2ccccc21 s275592__15865378__15841170__14130460
O=C(NCC(F)=C1CN(C(=O)COc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130462
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__14130464
Cc1cc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__14130466
CCc1ccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14130468
CC(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14130470
CCN(CC)C(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130474
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130478
CC(=O)NC(CCC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130480
O=C(NCC(F)=C1CN(C(=O)C2CCOc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14130482
O=C(NCC(F)=C1CN(C(=O)CCn2cc[nH]c(=O)c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14130484
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1F s275592__15865378__15841170__14130486
Cn1ccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15841170__14130488
CC(=O)NCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14130490
CC(C)CCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130492
CC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(C)(C)C1 s275592__15865378__15841170__14130496
CCn1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14130498
CC(C)CC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130504
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C(F)F s275592__15865378__15841170__14130508
CCCCCCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130510
O=C(NCC(F)=C1CN(C(=O)c2ccc3nccn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130514
CCCN(CCC)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130516
CC(=O)Nc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14135178
O=C(NCC(F)=C1CN(C(=O)CN2CCCCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14135180
Cc1nc[nH]c(=O)c1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135182
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1=O s275592__15865378__15841170__14135184
COCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135188
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__14135190
CCCc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__14135192
CCn1nc(C(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135196
Cc1ccc2[nH]nc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__14135198
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2-c2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__14135200
O=C(NCC(F)=C1CN(C(=O)CN2CCCNC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14135202
O=C(NCC(F)=C1CN(C(=O)c2ccn(-c3ccccc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14135204
O=C(Nc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135206
CC(C)NC(=O)CN(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135208
O=C(NCC(F)=C1CN(C(=O)c2cn3cccnc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14135214
O=C(NCC(F)=C1CN(C(=O)C23CCCN2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135218
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(n2)OCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14135224
O=C(NCC(F)=C1CN(C(=O)c2coc(-c3ccccn3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14135226
CCc1ccc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135228
O=C(NCC(F)=C1CN(C(=O)c2cccn3nccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14135230
O=C1Cc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccnc2N1 s275592__15865378__15841170__14135232
O=C(NCC(F)=C1CN(C(=O)c2[nH]nc(C3CC3)c2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14135236
O=C(NCC(F)=C1CN(C(=O)c2cccnc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135238
Cc1cccc(Cl)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135240
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2OCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135244
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(OC)n1 s275592__15865378__15841170__14135246
CCOc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__14135248
O=C(NCC(F)=C1CN(C(=O)c2coc(C(F)(F)F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14135250
O=C(NCC(F)=C1CN(C(=O)c2ncnc3[nH]ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14135252
COc1cc(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14135254
O=C(NCC(F)=C1CN(C(=O)c2coc(-c3cccnc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14135256
Cc1nn(C)c(Cl)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135258
O=C(NCC(F)=C1CN(C(=O)c2cc3cnccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__14135260
O=C(NCC(F)=C1CN(C(=O)c2ccn3cncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14135262
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c(=O)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14135264
Cc1nnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135266
O=C(NCC(F)=C1CN(C(=O)c2ccnc(C3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14135268
COCc1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14135272
CC(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14135274
Cc1nnc(COCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14135278
Cn1cc(C(N)=O)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135280
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCOCC1 s275592__15865378__15841170__14135288
O=C(NCC(F)=C1CN(C(=O)c2cc3c(cn2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135290
O=C1CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__14135292
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14135296
COc1cncc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14135298
Cc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1C s275592__15865378__15841170__14135300
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__14135302
Cc1ccc2nc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2c1 s275592__15865378__15841170__14135304
Cc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__14135306
CCCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135308
COc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14135310
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__14135312
O=C(NCC(F)=C1CN(C(=O)c2cccnc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14135316
Cc1cncc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14135318
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14135320
Cc1occc(=O)c1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135322
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14135324
O=C(NCC(F)=C1CN(C(=O)c2nc3cnccc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14135326
O=C(NCC(F)=C1CN(C(=O)C2CCCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135328
O=C(NCC(F)=C1CN(C(=O)C2CCCC2c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14135330
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3ccco3)o2)C1)c1cc(O)no1 s275592__15865378__15841170__14135334
COCCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14135336
Cn1ccc(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14135338
Cc1cnc(COCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14135340
O=C(NCC(F)=C1CN(C(=O)c2ccnc3nn[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14135342
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130524
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__14130526
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(F)(F)C1 s275592__15865378__15841170__14130528
O=C(NCC(F)=C1CN(C(=O)c2cc3c([nH]2)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130530
CC(C)Oc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__14130532
CC(C)c1scnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130534
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15841170__14130536
COCc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14130540
O=C(NCC(F)=C1CN(C(=O)c2[nH]ccc2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130542
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3ccnn3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130546
COCc1nocc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130550
CC(C)n1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14130552
Cc1nn(C(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130554
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3ccnc3)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14130558
CCc1oc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14130562
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCC1=O s275592__15865378__15841170__14130564
Cn1nc2c(c1C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CCC2 s275592__15865378__15841170__14130568
CN1CCCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__14130570
Cc1cccn2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__14130572
Cc1nc2nccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)n2n1 s275592__15865378__15841170__14130574
O=C(NCC(F)=C1CN(C(=O)c2cccn3c(=O)[nH]nc23)C1)c1cc(O)no1 s275592__15865378__15841170__14130576
CN1C(=O)CN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__14130578
O=C(NCC(F)=C1CN(C(=O)C2CCc3[nH]ncc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14130580
COc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c(=O)[nH]c1=O s275592__15865378__15841170__14130584
O=C(NCC(F)=C1CN(C(=O)c2ccc3oc(=O)[nH]c3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14130586
CCCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__14130588
O=C(NCC(F)=C1CN(C(=O)c2cc(=O)n3ncnc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14130590
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCOCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14130592
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)s2)C1)c1cc(O)no1 s275592__15865378__15841170__14130594
COCc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130596
CCCc1occc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130598
Cc1ccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130600
CCOCCOCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130602
CC(C)(C)S(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130604
CC(C)(C)C(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130606
CC(CCC(C)(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130608
CCCCCCC(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130610
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)c1C s275592__15865378__15841170__14130614
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCCC1 s275592__15865378__15841170__14130620
CN(C)C1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14130622
O=C(NCC(F)=C1CN(C(=O)c2cccc(C3CCC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130624
O=C(NCC(F)=C1CN(C(=O)c2cccc(C3CCCC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130626
CC1(C)CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14130628
CN1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14130638
Cn1cncc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130640
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3cccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14130644
O=C(NCC(F)=C1CN(C(=O)COc2ccsc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130646
CCCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14130648
O=C(NCC(F)=C1CN(C(=O)C(F)CC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130650
CCc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14130652
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc1CC s275592__15865378__15841170__14130658
Cc1cccc2c1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)O2 s275592__15865378__15841170__14130660
Cc1cc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)oc2cc1C s275592__15865378__15841170__14130662
COc1cc[nH]c(=O)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130664
CC(C)Cc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14130666
CCn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14130668
CN(C)c1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130670
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCC=C3)C1)c1cc(O)no1 s275592__15865378__15841170__14130672
CCC(CC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130674
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(=O)ccoc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130676
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccco1 s275592__15865378__15841170__14130678
CC(Oc1ccccn1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130680
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__14130682
Cc1sc(Cl)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135344
O=C(NCC(F)=C1CN(C(=O)c2ccn3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14135346
O=C(NCC(F)=C1CN(C(=O)c2nncc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14135348
Cc1n[nH]c2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__14135350
C[C@H](OCc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135352
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14135354
COc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14135356
COc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14135358
O=C(NCC(F)=C1CN(C(=O)c2ccn(-c3ccncc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14135360
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14135364
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135366
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135368
CC(C)(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14135370
O=C(NCC(F)=C1CN(C(=O)C2CC3CC2C2CC32)C1)c1cc(O)no1 s275592__15865378__15841170__14135372
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(C)O1 s275592__15865378__15841170__14135374
O=C(NCC(F)=C1CN(C(=O)c2scnc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14135376
O=C(NCC(F)=C1CN(C(=O)C23CCCCC2OCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135378
CC(C)(C)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135380
O=C(NCC(F)=C1CN(C(=O)[C@]23CCC[C@H]2OCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135382
CC1CC1C1CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135384
COc1ccnc(OC)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135386
CC1(C)COC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14135388
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCCO3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135392
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135394
CCOC1COCCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135398
NC(=O)[C@@H]1CC[C@H](CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__14135400
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CC(F)F s275592__15865378__15841170__14135402
O=C(NCC(F)=C1CN(C(=O)Cn2ncc3cccnc32)C1)c1cc(O)no1 s275592__15865378__15841170__14135404
O=C(NCC(F)=C1CN(C(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__14135406
CC1(C)CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)OC1 s275592__15865378__15841170__14135408
O=C(NCC(F)=C1CN(C(=O)C2CCc3nncn3CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135410
Cc1cc2ccccc2nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135412
CC1CCc2n[nH]cc2C1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135416
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3O[C@H]2[C@H]2C[C@@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__14135418
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2C[C@H]2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135422
CC1COC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14135424
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc1=O s275592__15865378__15841170__14135430
Cc1nc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14135432
O=C(NCC(F)=C1CN(C(=O)[C@@]23CCC[C@@H]2C3)C1)c1cc(O)no1 s275592__15865378__15841170__14135434
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__14135436
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCO[C@H]2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135438
CC(C)n1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14135442
CCOc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14135446
CC[C@@H]1OCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135448
O=C(NCC(F)=C1CN(C(=O)CC2CCC(C3CC3)O2)C1)c1cc(O)no1 s275592__15865378__15841170__14135452
Cc1nc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccnc2[nH]1 s275592__15865378__15841170__14135456
CCc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__14135458
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__14135460
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14135462
O=C(NCC(F)=C1CN(C(=O)c2nccc3occc23)C1)c1cc(O)no1 s275592__15865378__15841170__14135466
O=C(NCC(F)=C1CN(C(=O)C2CC[C@H]3C[C@H]3CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135470
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2C[C@H]2Cc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14135474
CCn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14135476
Cn1nccc1[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135478
CC1CC2CC2CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135480
CC1CC2CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CN2C1 s275592__15865378__15841170__14135484
O=C(NCC(F)=C1CN(C(=O)[C@@H]2OC[C@@H]3COCC[C@@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__14135486
Cn1ccnc1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135492
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3CCCC[C@@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__14135494
C[C@H](CC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135498
O=C(NCC(F)=C1CN(C(=O)[C@@H]2Cc3cncn3C(=O)N2)C1)c1cc(O)no1 s275592__15865378__15841170__14135500
C[C@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130686
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14130688
O=C(NCC(F)=C1CN(C(=O)c2coc(-c3ccccc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14130690
Cc1ccn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2n1 s275592__15865378__15841170__14130692
CNC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14130696
Cc1cccc2[nH]cc(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c12 s275592__15865378__15841170__14130702
COC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130704
CN(C)C(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130706
CCNC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130708
CCCNC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130710
CCn1nc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14130712
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccnc1 s275592__15865378__15841170__14130714
CCCNC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130716
CC(C)NC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130718
O=C(NCC(F)=C1CN(C(=O)Cn2cc3ccccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14130722
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3ncon3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130726
O=C(NCC(F)=C1CN(C(=O)c2cc3c(s2)CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130728
Cc1ccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14130730
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__14130732
Cn1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15841170__14130734
C#CCOc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130736
Cc1ccc(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14130740
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14130744
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14130746
CN(C)CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130748
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14130750
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14130752
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cccc1 s275592__15865378__15841170__14130754
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130762
CO[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130764
O=C1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__14130766
CC(=O)N1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130768
COc1cc(C)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130770
CC(=O)N[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14130772
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc21 s275592__15865378__15841170__14130774
CC(=O)N[C@@H](CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130776
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130778
CC(=O)N[C@H](CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130780
C[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130782
CC[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130784
O=C(NCC(F)=C1CN(C(=O)c2ncccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14130786
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14130788
Cc1cc(F)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130790
COc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__14130792
Cc1ccc(F)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14130794
Cc1ccc2oc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2n1 s275592__15865378__15841170__14130800
Cc1ccc(=O)n(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14130802
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__14130804
O=C(NCC(F)=C1CN(C(=O)c2cccc(C(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130806
CCCN(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130808
CC(C)Oc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130812
O=C(NCC(F)=C1CN(C(=O)CCCc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14130814
O=C(NCC(F)=C1CN(C(=O)c2cnc(C3CC3)s2)C1)c1cc(O)no1 s275592__15865378__15841170__14130816
CNC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14130818
COc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130822
CCCN(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130824
O=C(NCC(F)=C1CN(C(=O)CC2CCCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14130826
O=C(NCC(F)=C1CN(C(=O)c2ncoc2-c2ccon2)C1)c1cc(O)no1 s275592__15865378__15841170__14130828
O=C(NCC(F)=C1CN(C(=O)CC2CCc3ccccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14130830
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__14130832
COc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130834
CCCCCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130836
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3c(c2)COC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130838
O=C(NCC(F)=C1CN(C(=O)c2cnn3cc[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14130840
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCO1 s275592__15865378__15841170__14130842
O=C(NCC(F)=C1CN(C(=O)c2occ3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130844
CC1(C)COC(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14130846
COCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14130850
COCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__14130852
CCC[C@@H](NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130854
O=C1CCCCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__14130858
C#Cc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130860
Cc1[nH]cnc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130862
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCCC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130864
O=C(NCC(F)=C1CN(C(=O)c2cc3[nH]ccc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14130866
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CC(F)(F)F s275592__15865378__15841170__14130868
O=C(NCC(F)=C1CN(C(=O)Cn2c(=O)[nH][nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14130872
Cc1csc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130874
O=C(NCC(F)=C1CN(C(=O)COCc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130878
O=C(NCC(F)=C1CN(C(=O)C2Cc3cccnc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14130880
COc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__14130882
CC(F)(F)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130884
Cn1nnc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc21 s275592__15865378__15841170__14130886
Cc1ccsc1CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130888
O=C(NCC(F)=C1CN(C(=O)C23CCCN(CC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__14130890
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)cc1F s275592__15865378__15841170__14130892
Cc1ccccc1C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14130894
CC(=O)N(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130896
O=C(NCC(F)=C1CN(C(=O)c2coc3ccc(F)cc23)C1)c1cc(O)no1 s275592__15865378__15841170__14130898
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCC1 s275592__15865378__15841170__14130900
CC(OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1nccn1C s275592__15865378__15841170__14130902
COCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130904
O=C(NCC(F)=C1CN(C(=O)c2cc3c(cn2)OCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130906
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)nn1C s275592__15865378__15841170__14130908
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__14130910
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1CC(C)C s275592__15865378__15841170__14130916
COCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14130918
CC1CCn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2C1 s275592__15865378__15841170__14130920
O=C(NCC(F)=C1CN(C(=O)c2ccccc2C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130922
O=C(NCC(F)=C1CN(C(=O)CC2OCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14130924
Cc1nn(C)c(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130926
C[C@H](CC1CCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130928
O=C(NCC(F)=C1CN(C(=O)c2ccsc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14130930
O=C(NCC(F)=C1CN(C(=O)c2sccc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14130932
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)o2)C1)c1cc(O)no1 s275592__15865378__15841170__14130934
Cc1cc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130940
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15841170__14130942
CCc1nc[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130946
CN(C)S(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130948
CNC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14130952
CN1C(=O)CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130954
CC(C)Oc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130956
O=C(NCC(F)=C1CN(C(=O)C2CCC(C(F)F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130960
O=C(NCC(F)=C1CN(C(=O)C2CCC(C3CC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130962
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccc(Cl)cc32)C1)c1cc(O)no1 s275592__15865378__15841170__14130964
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3cn[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130966
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14130968
O=C(NCC(F)=C1CN(C(=O)c2cncnc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130970
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C2CC2)n1 s275592__15865378__15841170__14130972
O=C(NCC(F)=C1CN(C(=O)[C@@H]2Cc3ccccc3CO2)C1)c1cc(O)no1 s275592__15865378__15841170__14130974
CC(=O)N1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14130976
CN1CCc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc21 s275592__15865378__15841170__14130978
Cn1cncc1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130982
Cc1nn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)n1C s275592__15865378__15841170__14130984
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14130992
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C(C)(C)C)n1 s275592__15865378__15841170__14130996
Cc1n[nH]c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131000
Cc1n[nH]c(C)c1C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131002
CCCCCCN(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131004
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2-c2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14131006
O=C(NCC(F)=C1CN(C(=O)Cn2ncc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14131008
CN(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14131012
O=C(NCC(F)=C1CN(C(=O)c2cnn3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131014
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)c1 s275592__15865378__15841170__14131018
O=C(NCC(F)=C1CN(C(=O)c2nccn3ccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131024
O=C(NCC(F)=C1CN(C(=O)CNC(=O)C2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131028
CCN(CC)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14131032
CCn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1=O s275592__15865378__15841170__14131038
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__14131042
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1F s275592__15865378__15841170__14131048
Cc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131050
O=C(NCC(F)=C1CN(C(=O)c2ccc3cccnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131052
Cc1ccc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131054
CC(C)CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131056
O=C(NCC(F)=C1CN(C(=O)C2CCc3ccccc3O2)C1)c1cc(O)no1 s275592__15865378__15841170__14131058
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3cccc3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__14131062
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__14131066
CC(C)(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131068
O=C(NCC(F)=C1CN(C(=O)c2ccncn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131070
O=C(NCC(F)=C1CN(C(=O)CC2CCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14131072
O=C(NCC(F)=C1CN(C(=O)c2nc3ncccn3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131074
CCCCCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131076
CC(=O)Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__14131080
O=C(NCC(F)=C1CN(C(=O)CCc2ncccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131082
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__14131084
O=C(NCC(F)=C1CN(C(=O)c2cc3ncccn3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131088
O=C(NCC(F)=C1CN(C(=O)Cc2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__14131092
Cc1ccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2n1 s275592__15865378__15841170__14131094
COc1ccc(F)cc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131096
O=C(NCC(F)=C1CN(C(=O)c2ncccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131098
CCC(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131100
CC(C)(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14131102
COc1cc(Cl)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14131104
CC(C)c1nnsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131108
O=C(NCC(F)=C1CN(C(=O)c2cccc3[nH]cnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131110
O=C(NCC(F)=C1CN(C(=O)c2cccnn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131112
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__14131114
CC1(C)CC1(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14131116
CCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14131120
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14131126
Cc1[nH]c(=O)[nH]c(=O)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131128
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__14131130
O=C(NCC(F)=C1CN(C(=O)c2cccc3nccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131132
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__14131134
O=C(NCC(F)=C1CN(C(=O)CCn2cnnn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131136
CC1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14131138
O=C(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)NC1CCCC1 s275592__15865378__15841170__14131142
CCCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14131144
CCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__14131146
O=C(NCC(F)=C1CN(C(=O)c2ncccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14131150
O=C(NCC(F)=C1CN(C(=O)Cc2coc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131154
CC(C)[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14131156
O=C(NCC(F)=C1CN(C(=O)COCc2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__14131162
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccnc1 s275592__15865378__15841170__14131164
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14131166
CCOCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14131170
Cn1ncc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc21 s275592__15865378__15841170__14131172
CC1OCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131176
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOC1 s275592__15865378__15841170__14131178
O=C(NCC(F)=C1CN(C(=O)c2cnn(C(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131180
CC(C)Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14131182
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccccn3)no2)C1)c1cc(O)no1 s275592__15865378__15841170__14131186
CCOc1c(F)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131188
NC(=O)c1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14131190
CCC(CC)(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131192
Cc1cc(C)n(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)n1 s275592__15865378__15841170__14131194
CCCC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__14131196
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__14131198
CCCC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131200
CCC(CC)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131202
CCC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131204
CCCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131208
Cc1nc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2[nH]1 s275592__15865378__15841170__14131210
O=C(NCC(F)=C1CN(C(=O)c2cnn(-c3ccncc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131212
CCOCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14131214
O=C(NCC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131216
O=C(NCC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131218
CC1CCCC(C)N1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131220
O=C(NCC(F)=C1CN(C(=O)c2cccn2C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131222
O=C(NCC(F)=C1CN(C(=O)CCCc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14131224
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__14131228
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCOC1 s275592__15865378__15841170__14131230
CN1CCC(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14131232
O=C(NCC(F)=C1CN(C(=O)c2cn(CC3CC3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131234
CCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14131236
CC(C)n1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14131238
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nnn1C(C)C s275592__15865378__15841170__14131240
CC(C)N(C)C(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14131242
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14131246
CC(Cc1cnn(C)c1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131252
O=C(NCC(F)=C1CN(C(=O)CCC2CCCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131254
O=C(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)NCC(F)(F)F s275592__15865378__15841170__14131256
O=C(NCC(F)=C1CN(C(=O)CCn2cnccc2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14131258
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3cncn3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131260
CC(C)Oc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131262
O=C(NCC(F)=C1CN(C(=O)c2coc(C3CCCC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131264
COCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__14131266
O=C(NCC(F)=C1CN(C(=O)c2coc(CC3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131268
Cc1oc(C2CC2)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131270
Cc1nc2ccnn2cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131272
O=C(NCC(F)=C1CN(C(=O)C2CC2C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131274
O=C(NCC(F)=C1CN(C(=O)c2c[nH]cc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131278
CCC1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131282
CCC1(C(C)C)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131284
CCC1(C)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131286
O=C(NCC(F)=C1CN(C(=O)C2CC23CCc2ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131288
CC(C)C1(C)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131290
O=C(NCC(F)=C1CN(C(=O)C2(N3CCOCC3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131292
Cn1cc(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14131294
CS(=O)(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14131296
COCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131300
CCS(=O)(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131302
CCc1c[nH]c(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14131304
CCOc1nc(C)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131310
COCCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131314
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14131318
Cc1nonc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131322
CC1CCc2n[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2C1 s275592__15865378__15841170__14131324
O=C(NCC(F)=C1CN(C(=O)c2cccc3nsnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131326
Cc1ccc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c(C)c2c1 s275592__15865378__15841170__14131328
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14131330
Cc1ncsc1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131332
O=C(NCC(F)=C1CN(C(=O)c2cnoc2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14131334
O=C(NCC(F)=C1CN(C(=O)c2ccc3sccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131338
CC1CCc2onc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2C1 s275592__15865378__15841170__14131342
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14131344
Cc1oc(C(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131346
O=C(NCC(F)=C1CN(C(=O)c2cccc3ccncc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131348
COc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__14131350
CCCCCCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131850
C=CCCOCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131852
Cc1nc(C2CC2)sc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131854
O=C(NCC(F)=C1CN(C(=O)COC2CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131856
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)NC(N)=O s275592__15865378__15841170__14131860
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCCC1=O s275592__15865378__15841170__14131862
CC(C)(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__14131864
Cc1oc(C(C)C)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131866
Cc1cccn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15841170__14131868
CCC(OC1CCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131872
Cc1ccsc1[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131874
O=C(NCC(F)=C1CN(C(=O)c2cccc3scnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131878
COCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__14131880
COCCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14131882
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131884
O=C(NCC(F)=C1CN(C(=O)C2CCCC3(CC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14131886
O=C(NCC(F)=C1CN(C(=O)C2(c3ccccn3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131888
O=C(NCC(F)=C1CN(C(=O)c2cnn(C3CCC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131890
CCOC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1=CCCC1 s275592__15865378__15841170__14131892
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCCN3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14131894
CC(C)Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__14131902
CN(C)c1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14131906
CC(C)Oc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14131908
Cc1cnc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccn12 s275592__15865378__15841170__14131910
Cn1nnc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccnc21 s275592__15865378__15841170__14133582
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14133584
NC(=O)Cc1occc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133586
Cn1cc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14133590
O=C(NCC(F)=C1CN(C(=O)C(C2CCC2)C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133592
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(C)n1 s275592__15865378__15841170__14133594
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133596
CCc1ccccc1[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133604
CN(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133608
Cc1ncc2n1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__14133610
O=C(NCC(F)=C1CN(C(=O)C2CCCc3[nH]nnc32)C1)c1cc(O)no1 s275592__15865378__15841170__14133612
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]ncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133614
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14133618
O=C(NCC(F)=C1CN(C(=O)c2nccc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133620
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc2ccccc21 s275592__15865378__15841170__14133622
COc1cc(Cl)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133624
CCCC(CCC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133626
CCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133628
O=C(NCC(F)=C1CN(C(=O)Cc2cc(F)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14133630
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133632
O=C(NCC(F)=C1CN(C(=O)c2cccc(F)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14133634
CC(C)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14131352
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131354
O=C(NCC(F)=C1CN(C(=O)c2cccc(-c3cnco3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131356
O=C(NCC(F)=C1CN(C(=O)c2ccc3scnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131358
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__14131360
O=C(NCC(F)=C1CN(C(=O)C2(c3ccccc3F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131362
O=C(NCC(F)=C1CN(C(=O)c2cnoc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131364
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131366
CC(C)c1oncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131368
Cn1cnc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc21 s275592__15865378__15841170__14131370
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3ccnc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131372
CC1(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14131376
Cc1cnoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131378
O=C(NCC(F)=C1CN(C(=O)c2scc3c2OCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14131380
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3c[nH]cn3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14131382
O=C(NCC(F)=C1CN(C(=O)c2cc(-n3ccnc3)ccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131384
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cnc2ccccc21 s275592__15865378__15841170__14131386
COc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14131388
Cc1cc(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__14131390
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3ncn[nH]3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14131394
O=C(NCC(F)=C1CN(C(=O)c2cc3cccnc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14131398
O=C(NCC(F)=C1CN(C(=O)c2cc3sccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14131406
Cn1nc2ccccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131410
CC(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14131412
O=C(NCC(F)=C1CN(C(=O)c2nc3ccccn3c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14131414
O=C(NCC(F)=C1CN(C(=O)C2(F)CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131416
Cn1ccc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc21 s275592__15865378__15841170__14131418
O=C(NCC(F)=C1CN(C(=O)c2cccc3ccsc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131420
CC1(C)C(=O)NC(=O)N1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131422
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14131426
O=C(NCC(F)=C1CN(C(=O)c2ncoc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131428
CCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14131430
Cc1nc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc2[nH]1 s275592__15865378__15841170__14131432
CCN(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131434
O=C(NCC(F)=C1CN(C(=O)C2CC23CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14131436
O=C(NCC(F)=C1CN(C(=O)CCc2cnccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131440
Cc1cc(C)cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14131444
CC(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__14131446
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14131448
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131452
O=C(NCC(F)=C1CN(C(=O)CCCn2cncn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131454
O=C(NCC(F)=C1CN(C(=O)c2ccc3cnccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131456
O=C(NCC(F)=C1CN(C(=O)c2csc(Cl)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131458
CC(C)(CC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131460
CN1CCc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc21 s275592__15865378__15841170__14131462
Cc1conc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131468
CC(C)c1ocnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131470
CC(C)(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131472
O=C1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(=O)N1 s275592__15865378__15841170__14131474
O=C(NCC(F)=C1CN(C(=O)c2cc3c([nH]2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14131478
CCC(=O)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14131484
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cscn1 s275592__15865378__15841170__14131486
COC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15841170__14131490
O=C(NCC(F)=C1CN(C(=O)c2cnn(CC3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131496
O=C(NCC(F)=C1CN(C(=O)c2cccc(-c3ccoc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131500
CC(C)C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__14131502
CCC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__14131504
CCC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__14131506
O=C(NCC(F)=C1CN(C(=O)C2CCc3[nH]cnc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14131508
CC(=O)N1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14131510
Cc1cn2ccnc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2n1 s275592__15865378__15841170__14131512
CCc1nn(C)c(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131516
O=C(NCC(F)=C1CN(C(=O)c2ccnn2CC(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14131918
Cc1ccc(F)c(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14131920
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCCC1 s275592__15865378__15841170__14131922
O=C(NCC(F)=C1CN(C(=O)Cc2n[nH]c3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14131924
O=C(NCC(F)=C1CN(C(=O)C2CCCc3[nH]ncc32)C1)c1cc(O)no1 s275592__15865378__15841170__14131926
COC(C)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14131932
COC(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14131934
Cc1nc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14131936
Cc1nn(C)c(C)c1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131938
CCOCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14131944
CC1(C)CC(=O)N(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__14131946
O=C(NCC(F)=C1CN(C(=O)c2ccnn2CC2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131950
CCc1ccc2occ(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__14131954
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__14131956
Cc1nc(CC2CC2)oc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131958
Cn1nc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc21 s275592__15865378__15841170__14131960
O=C(NCC(F)=C1CN(C(=O)CCOCC(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14131962
O=C(NCC(F)=C1CN(C(=O)Cn2ncnn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131964
Cn1ncc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131966
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncn1 s275592__15865378__15841170__14131968
O=C(NCC(F)=C1CN(C(=O)C2CN3CCC2CC3)C1)c1cc(O)no1 s275592__15865378__15841170__14131970
CCCC[C@@H](C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131972
CCc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14131974
O=C(NCC(F)=C1CN(C(=O)CC2Cc3ccccc3O2)C1)c1cc(O)no1 s275592__15865378__15841170__14131976
O=C(NCC(F)=C1CN(C(=O)c2cccc3nn[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14131978
CC1=C(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14131980
CC(C)(C)CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131982
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14131986
CC(C)(C)n1nnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131988
Cc1oc2ccccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131990
Cc1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__14131992
O=C(NCC(F)=C1CN(C(=O)c2nsc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131994
C=CCC(CC=C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131996
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC=CCC1 s275592__15865378__15841170__14132000
Cn1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14132002
O=C(NCC(F)=C1CN(C(=O)C2CS(=O)(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132004
Cc1scc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14132006
CCn1ncc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132008
CCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132012
CCCC(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132014
CCC(C)CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132016
CC(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132018
COc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__14132020
Cc1ccnc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__14132024
Cc1ccn(CC(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14132026
Cc1cc(C(F)F)n(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14132030
O=C(NCC(F)=C1CN(C(=O)c2cccn3nnnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132032
C=C(Cl)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132034
CC(C)n1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132036
O=C(NCC(F)=C1CN(C(=O)c2ccn(C(F)F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132040
O=C(NCC(F)=C1CN(C(=O)c2ccnn2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14132042
C=CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132044
O=C(NCC(F)=C1CN(C(=O)c2ccoc2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14132048
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(C)n1 s275592__15865378__15841170__14132050
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3c(=O)o2)C1)c1cc(O)no1 s275592__15865378__15841170__14132054
O=C(NCC(F)=C1CN(C(=O)Cn2nccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132056
Cc1nc(Cl)sc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132058
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14132060
Cn1nc2c(c1C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CCCC2 s275592__15865378__15841170__14132064
CCCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132068
CCCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14132070
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C2CC2)n1 s275592__15865378__15841170__14132072
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C2CC2)n1 s275592__15865378__15841170__14132074
Cc1c(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__14132076
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ccncc3c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14132080
COc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__14132082
O=C(NCC(F)=C1CN(C(=O)Cc2c(F)cccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14133638
CC1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133642
CC1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133644
O=C(NCC(F)=C1CN(C(=O)c2cc(F)c(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14133646
COC1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133648
COC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133650
CCCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14133652
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(F)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14133654
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccncc3)on2)C1)c1cc(O)no1 s275592__15865378__15841170__14133656
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133658
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccc(F)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14133660
Cc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133662
Cn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc21 s275592__15865378__15841170__14133664
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14133672
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]ccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133676
Cc1[nH]c2ccccc2c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133678
O=C(NCC(F)=C1CN(C(=O)c2c(F)cc(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14133680
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3cccnc3)on2)C1)c1cc(O)no1 s275592__15865378__15841170__14133682
C=CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133684
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15841170__14133686
NS(=O)(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133688
CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133690
CCCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133692
Cc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133694
NC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133696
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__14133698
O=C(NCC(F)=C1CN(C(=O)CCCCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133700
O=C(NCC(F)=C1CN(C(=O)c2ccc3nonc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133706
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133708
O=C(NCC(F)=C1CN(C(=O)CCOc2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133710
O=C(NCC(F)=C1CN(C(=O)c2cccc(Cl)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14133714
O=C(NCC(F)=C1CN(C(=O)CCCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133716
Cc1nocc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133720
Cc1cc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__14133722
Cc1cc(C)cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133724
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(Cl)cc1 s275592__15865378__15841170__14133726
O=C(NCC(F)=C1CN(C(=O)c2ccccc2-n2cccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133728
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1Cl s275592__15865378__15841170__14133730
Cc1cc(Cl)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133732
Cc1ccc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14133736
O=C(NCC(F)=C1CN(C(=O)c2ccc3ncccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133738
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__14133740
CC(CC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133742
COc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133744
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14133746
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133750
CCCOc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133752
Cc1ccc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133756
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14133760
Cn1nc(C(C)(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133762
Cc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__14133764
Cc1cccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133766
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC=CC1 s275592__15865378__15841170__14133772
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c1=O s275592__15865378__15841170__14133774
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14133776
CC1CC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133778
CCCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133780
C=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133782
C=CCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133784
C=CC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133786
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133788
O=C(NCC(F)=C1CN(C(=O)C[C@H]2CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133790
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14133792
O=C(NCC(F)=C1CN(C(=O)CC2=CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133794
CCc1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133796
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133798
CC(C)[C@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__14133800
CCC1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133804
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)no2)C1)c1cc(O)no1 s275592__15865378__15841170__14128902
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c(=O)c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14128906
CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14128908
O=C(NCC(F)=C1CN(C(=O)c2ccccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14128910
O=C(NCC(F)=C1CN(C(=O)Cc2cccc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14128912
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14128914
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14128916
CCCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14128918
COc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14128920
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14128922
CC(C)(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14128924
O=C(NCC(F)=C1CN(C(=O)c2c(F)cccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14128926
CCCCCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14128928
O=C(NCC(F)=C1CN(C(=O)c2ccccc2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14128930
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)(F)F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14128932
O=C(NCC(F)=C1CN(C(=O)c2cccc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14128934
O=C(NCC(F)=C1CN(C(=O)c2cccc(C(F)(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14128936
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14128938
O=C(NCC(F)=C1CN(C(=O)C23CC4CC(CC(C4)C2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__14128944
CC(=O)Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14128946
CCCCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14128948
O=C(NCC(F)=C1CN(C(=O)CCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14128950
O=C(NCC(F)=C1CN(C(=O)Cc2c[nH]c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14128952
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14128954
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14128958
O=C(NCC(F)=C1CN(C(=O)COc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14128960
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14128962
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14128964
COc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14128966
O=C(NCC(F)=C1CN(C(=O)Cc2c(F)cccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14128970
O=C(NCC(F)=C1CN(C(=O)c2c(F)cccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14128982
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1OC s275592__15865378__15841170__14128984
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(OC)c1 s275592__15865378__15841170__14128986
COc1cccc(OC)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14128988
COc1cc(OC)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14128990
CN(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14128992
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14128994
Cc1ccc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14128996
Cc1cc(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14128998
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(Cl)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129002
O=C(NCC(F)=C1CN(C(=O)COc2ccc(Cl)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129004
CCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129006
CCOc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129008
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129010
CCOc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129012
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14129014
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14129016
O=C(NCC(F)=C1CN(C(=O)c2cc(=O)c3ccccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__14129018
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1OC s275592__15865378__15841170__14129022
O=C(NCC(F)=C1CN(C(=O)C2CC23CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__14131518
O=C(NCC(F)=C1CN(C(=O)c2cn(C3CCOC3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131520
O=C(NCC(F)=C1CN(C(=O)c2cc(-n3cccc3)ccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14131522
CCC1CCCN1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131524
COCCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131526
CCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131528
CCCCCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14131530
COCCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14131534
COCCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131536
COCCCOCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131538
CC(C)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131540
O=C(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)NCC1CC1 s275592__15865378__15841170__14131542
CCCn1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14131544
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cccn1 s275592__15865378__15841170__14131546
O=C(NCC(F)=C1CN(C(=O)c2coc(C3CCC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131548
Cc1n[nH]c(C(C)C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131556
NC(=O)CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131560
COCc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14131564
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(Cl)s1 s275592__15865378__15841170__14131566
CC1CCN(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14131570
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cc2ccccc2o1 s275592__15865378__15841170__14131572
O=C(NCC(F)=C1CN(C(=O)C(C2CC2)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131574
CCCCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14131582
CCCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__14131586
CCC(C)n1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14131588
O=C(NCC(F)=C1CN(C(=O)CCOC2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131592
O=C(NCC(F)=C1CN(C(=O)CCCOC2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131594
CCn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C1CC1 s275592__15865378__15841170__14131596
CCc1noc(COCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131598
Cc1nc(C)n(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131600
O=C(NCC(F)=C1CN(C(=O)Cc2nc[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131602
C=CCOc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131604
COCCCNC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131606
CN(C)C(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14131610
O=C(NCC(F)=C1CN(C(=O)C2CCN(CC3CC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131612
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C(C)C s275592__15865378__15841170__14131614
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCC1 s275592__15865378__15841170__14131618
NC(=O)N1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131622
CC(C)(C)c1n[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131624
CC(NC(=O)CC(C)(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131634
CCn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14131638
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cnn(C)c1 s275592__15865378__15841170__14131640
CCCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14131642
O=C(NCC(F)=C1CN(C(=O)CCC2CCCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__14131644
O=C(NCC(F)=C1CN(C(=O)c2cc3cc(F)ccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__14131646
O=C(NCC(F)=C1CN(C(=O)C2Cc3cc(F)ccc3O2)C1)c1cc(O)no1 s275592__15865378__15841170__14131648
CCC(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131650
CCC(OC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131652
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3ccccc3c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14131654
COc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)nn1C s275592__15865378__15841170__14131656
CC(C)n1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131658
CN(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__14131660
CS(=O)(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14131662
CCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14131664
NC(=O)C1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14131666
CC1CCCC(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14131672
O=C(NCC(F)=C1CN(C(=O)c2ccnc(C3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131674
O=C(NCC(F)=C1CN(C(=O)c2cnn(-c3ccccn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131676
O=C(NCC(F)=C1CN(C(=O)c2csc3cncn23)C1)c1cc(O)no1 s275592__15865378__15841170__14131678
CC1CCCCC1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131680
O=C(NCC(F)=C1CN(C(=O)COC2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131682
O=C(NCC(F)=C1CN(C(=O)c2ccnc3[nH]cnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132086
Cc1cccc(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132088
O=C(NCC(F)=C1CN(C(=O)C2C=CC=CC=C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132090
C=C(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132092
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]cnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132094
Cc1ccc2occ(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__14132096
O=C(NCC(F)=C1CN(C(=O)CCc2ccncn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132098
CC(C)Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14132100
O=C(NCC(F)=C1CN(C(=O)c2ccn(C3CCCC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132102
CCC(C)n1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132104
CC(C)Cn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132106
O=C(NCC(F)=C1CN(C(=O)c2ccnn2C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132108
Cn1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14132110
Cn1nccc1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132112
Cn1nc(C2CC2)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132114
O=C(NCC(F)=C1CN(C(=O)c2cc3occc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14132116
O=C(NCC(F)=C1CN(C(=O)c2ccns2)C1)c1cc(O)no1 s275592__15865378__15841170__14132118
C=C(C)C(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)OCC s275592__15865378__15841170__14132122
CCN(CC)CC(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132124
CN(C)Cc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132126
CCC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__14132128
Cc1nc2ccccc2cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132132
O=C(NCC(F)=C1CN(C(=O)c2cn3c(n2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132136
Cc1n[nH]c(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132142
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2-c2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132146
O=C(NCC(F)=C1CN(C(=O)c2ocnc2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132150
O=C(NCC(F)=C1CN(C(=O)Cn2ccc(C(F)F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132152
COCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14132154
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14132156
Cc1c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__14132160
O=C(NCC(F)=C1CN(C(=O)c2[nH]ccc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132164
CCn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C1CC1 s275592__15865378__15841170__14132168
Cc1cnc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14132172
Cc1nc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc2[nH]1 s275592__15865378__15841170__14132174
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__14132176
COC1CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14132180
COCC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132182
CCC(CC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132184
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC(C)CC1 s275592__15865378__15841170__14132186
CC(C)(CC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132188
Cn1ncc(C2CC2)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132192
O=C(NCC(F)=C1CN(C(=O)c2[nH]ncc2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14132194
O=C(NCC(F)=C1CN(C(=O)c2cc3c(o2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132196
O=C(NCC(F)=C1CN(C(=O)c2c(C3CC3)n[nH]c2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14132200
O=C(NCC(F)=C1CN(C(=O)c2conc2C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132202
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)[nH]c(=O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132204
O=C(NCC(F)=C1CN(C(=O)C2CCc3ncncc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132206
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2COCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132208
CCc1n[nH]c(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132210
COC1COCCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132212
O=C(NCC(F)=C1CN(C(=O)CC2(C(F)(F)F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132214
O=C(NCC(F)=C1CN(C(=O)c2cc3c([nH]2)CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132216
O=C(NCC(F)=C1CN(C(=O)Cc2cc(C3CC3)no2)C1)c1cc(O)no1 s275592__15865378__15841170__14132218
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ccnn23)C1)c1cc(O)no1 s275592__15865378__15841170__14132220
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15841170__14132222
O=C(NCC(F)=C1CN(C(=O)CC2CC3CCC2O3)C1)c1cc(O)no1 s275592__15865378__15841170__14132224
CCn1nnc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132226
CC(C)c1nocc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132228
O=C(NCC(F)=C1CN(C(=O)CC2CCNC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14132230
Cc1ncc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14132232
O=C(NCC(F)=C1CN(C(=O)c2cnn(-c3cccnc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132234
CC(C)CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14132236
CCOC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14132238
O=C(NCC(F)=C1CN(C(=O)C2CCCCS2(=O)=O)C1)c1cc(O)no1 s275592__15865378__15841170__14132240
O=C(NCC(F)=C1CN(C(=O)Cn2cc(C3CC3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132242
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14132244
CC1CCCC1(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133806
CC(F)(F)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133808
COC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133810
CCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133812
C[C@@]1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(=O)N1 s275592__15865378__15841170__14133814
CCc1nocc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133818
CC1COCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133820
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1C s275592__15865378__15841170__14133822
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14133824
COCC(OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133826
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133828
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCO1 s275592__15865378__15841170__14133830
CCC[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133832
O=C(NCC(F)=C1CN(C(=O)C23CCCCC2C3)C1)c1cc(O)no1 s275592__15865378__15841170__14133834
CC(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133836
C=C1CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133838
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)F s275592__15865378__15841170__14133840
Cc1ccoc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133842
CCc1ncoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133844
C#Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133846
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3cncn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133848
CCOc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__14133852
CC(OC1CCCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133854
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(F)c1 s275592__15865378__15841170__14133860
CC(Oc1cccnc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133864
COCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15841170__14133866
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cccc1=O s275592__15865378__15841170__14133870
O=C(NCC(F)=C1CN(C(=O)C2(CF)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133872
O=C(NCC(F)=C1CN(C(=O)C2CC3(CC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14133874
Cc1cc(=O)[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133876
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)F)[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__14133880
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14133882
O=C(NCC(F)=C1CN(C(=O)c2conc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133884
Cn1cnc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccnc21 s275592__15865378__15841170__14133886
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(CC)CC s275592__15865378__15841170__14133888
O=C(NCC(F)=C1CN(C(=O)c2ccnc(-n3cccn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133890
O=C(NCC(F)=C1CN(C(=O)c2cc(-n3cccn3)ccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14133894
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3cccn3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14133896
NC(=O)c1coc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133902
O=C(NCC(F)=C1CN(C(=O)C2CCCC(F)(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14133904
CC1(c2ccccc2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14133906
O=C(NCC(F)=C1CN(C(=O)c2ccc(N3CC=CC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133908
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccsc1 s275592__15865378__15841170__14133912
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccs1 s275592__15865378__15841170__14133914
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccco1 s275592__15865378__15841170__14133916
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(F)c1 s275592__15865378__15841170__14133918
CC(C)CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14133920
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nnn1CC s275592__15865378__15841170__14133922
CC(Cc1ccccc1F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133928
O=C(NCC(F)=C1CN(C(=O)c2cc3occc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14133932
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCNC1=O s275592__15865378__15841170__14133934
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133936
NC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__14133942
O=C(NCC(F)=C1CN(C(=O)c2ncsc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133944
CCOC1CC2(C1)CC2C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133946
Cn1cnc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nc21 s275592__15865378__15841170__14133948
Cc1ncccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133950
O=C(NCC(F)=C1CN(C(=O)c2ocnc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133952
Cn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15841170__14133954
CC(C)(C)n1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14133958
Cc1cn2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2n1 s275592__15865378__15841170__14133960
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c2C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133962
CC1CCCN1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133964
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14133966
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1C s275592__15865378__15841170__14133970
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129024
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129026
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__14129028
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14129030
Cc1ccccc1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129032
O=C(NCC(F)=C1CN(C(=O)c2cccc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129034
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3oc2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14129036
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14129038
CC(C)(C)C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14129040
O=C(NCC(F)=C1CN(C(=O)CC2CC3CCC2C3)C1)c1cc(O)no1 s275592__15865378__15841170__14129044
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14129046
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129048
CC(Oc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129050
COc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129052
O=C(NCC(F)=C1CN(C(=O)CCC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129054
CCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129058
CCc1ccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129062
O=C(NCC(F)=C1CN(C(=O)CCOc2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14129064
CCc1ccccc1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129066
O=C(NCC(F)=C1CN(C(=O)C2COc3ccccc3O2)C1)c1cc(O)no1 s275592__15865378__15841170__14129074
Cc1ccnc2nc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nn12 s275592__15865378__15841170__14129078
O=C(NCC(F)=C1CN(C(=O)CNC(=O)C2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129080
O=C(NCC(F)=C1CN(C(=O)CNC(=O)c2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__14129082
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccco1 s275592__15865378__15841170__14129088
O=C(NCC(F)=C1CN(C(=O)c2cn3ccccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14129090
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc2n1 s275592__15865378__15841170__14129092
O=C(NCC(F)=C1CN(C(=O)CCc2c[nH]c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129096
O=C(NCC(F)=C1CN(C(=O)CCCOc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129100
O=C(NCC(F)=C1CN(C(=O)c2ccc3ncsc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129102
CC1(C)NC(=O)N(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__14129104
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)s2)C1)c1cc(O)no1 s275592__15865378__15841170__14129106
CC(C)Oc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129112
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__14129114
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129118
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129120
O=C(NCC(F)=C1CN(C(=O)CCCC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129124
COc1ccc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129128
O=C(NCC(F)=C1CN(C(=O)c2cc3c(s2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129130
O=C(NCC(F)=C1CN(C(=O)c2cc3c(s2)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129132
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc2ccccc12 s275592__15865378__15841170__14129134
CCOc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129136
O=C(NCC(F)=C1CN(C(=O)c2sccc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129140
CCCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129144
O=C(NCC(F)=C1CN(C(=O)CCC(=O)N2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129146
NC(=O)Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129148
CC(=O)NCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129154
O=C(NCC(F)=C1CN(C(=O)C2(c3ccccc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129156
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129160
O=C(NCC(F)=C1CN(C(=O)C2(c3ccccc3)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129162
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14129164
CCc1cccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129166
Cc1ccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129172
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1=O s275592__15865378__15841170__14129174
CCCCC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14129176
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129178
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__14129180
COc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129182
COc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129186
Cc1ccc(OC(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129188
Cc1cccc(OC(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129190
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3cnnn3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129192
O=C(NCC(F)=C1CN(C(=O)COCC2CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131684
O=C(NCC(F)=C1CN(C(=O)C2CCCS(=O)(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14131686
O=C(NCC(F)=C1CN(C(=O)C2CCS(=O)(=O)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131688
CC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131690
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)n(C)c1=O s275592__15865378__15841170__14131694
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)S(C)(=O)=O s275592__15865378__15841170__14131696
CC(CC1CCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131700
CCC(CC1CCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131702
CC(CC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131708
CCC(CC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131710
CCCC(CC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131712
CC(C)C(CC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131714
CCOc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1C s275592__15865378__15841170__14131716
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131718
CN1C(=O)C(=O)N(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__14131720
CCNC(=O)NC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131722
Cc1nc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14131726
Cc1nn(C)cc1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131728
O=C(NCC(F)=C1CN(C(=O)C2(c3cccc(F)c3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131730
Cc1ccccc1C(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131732
CC(C)c1nccn1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131734
O=C(NCC(F)=C1CN(C(=O)CCC2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131736
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccnc1 s275592__15865378__15841170__14131738
NC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14131740
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14131742
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C(C)C)n1 s275592__15865378__15841170__14131746
COc1cc(C)sc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131748
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCCCC1 s275592__15865378__15841170__14131750
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__14131752
CC(C)N1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131756
CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131758
CCC(CC)n1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131760
C[C@H]1CC[C@@](C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__14131764
Cc1cccc2c(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c[nH]c12 s275592__15865378__15841170__14131766
CC(C)CCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131768
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)cs2)C1)c1cc(O)no1 s275592__15865378__15841170__14131772
O=C(NCC(F)=C1CN(C(=O)c2csc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14131774
CC(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14131776
O=C(NCC(F)=C1CN(C(=O)c2ccsc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14131780
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14131782
C=C(C)CC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131784
CCCCCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131788
Cc1ncc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131790
COc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14131794
CC(=O)N[C@@H](CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(N)=O s275592__15865378__15841170__14131796
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1Cl s275592__15865378__15841170__14131798
Cc1sccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131800
O=C(NCC(F)=C1CN(C(=O)Cc2csc(C3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14131804
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__14131808
Cc1nc2ccccc2n1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131810
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14131812
C#CCCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14131814
CCC1CCCCC1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131816
CC(C)CC(C)OCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131818
O=C(NCC(F)=C1CN(C(=O)CNC(=O)N2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131822
C#CCOCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131824
COCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14131826
C#CCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131828
Cc1nn(C(C)(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131830
CC(C)N1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131832
O=C(NCC(F)=C1CN(C(=O)CCOCC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14131836
CNS(=O)(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131840
CC1CC1c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14131844
CCCc1onc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14131846
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3ccncc3)o2)C1)c1cc(O)no1 s275592__15865378__15841170__14132252
CN(C)C(Cn1cccn1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132256
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__14132258
CCC(CC)n1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132260
Cc1cn2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)sc2n1 s275592__15865378__15841170__14132266
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14132268
CC(C)N1CCCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132270
O=C(NCC(F)=C1CN(C(=O)C2CCCN2C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132272
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3c(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14132278
O=C(NCC(F)=C1CN(C(=O)c2cncn2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132288
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3cccn3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132290
O=C(NCC(F)=C1CN(C(=O)CCc2ccsc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132292
O=C(NCC(F)=C1CN(C(=O)c2cnc3ccccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132296
Cc1csc(=O)n1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132298
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132300
O=C(NCC(F)=C1CN(C(=O)c2cc(F)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14132302
O=C(NCC(F)=C1CN(C(=O)C2C3CC4CC(C3)CC2C4)C1)c1cc(O)no1 s275592__15865378__15841170__14132304
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3cncn3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132310
Cc1cc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14132312
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__14132314
Cc1noc(C(C)C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132318
Cc1ccn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__14132322
O=C(NCC(F)=C1CN(C(=O)c2snnc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132324
CC(C)(C)c1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14132326
Cc1c(Cl)cncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132328
CC(C)(C(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132330
Cc1nc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2o1 s275592__15865378__15841170__14132332
O=C(NCC(F)=C1CN(C(=O)c2ccc3oc(=O)[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132336
CC(C)[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__14132338
Cc1ncn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132342
Cc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__14132344
O=C(NCC(F)=C1CN(C(=O)CCCc2ccsc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132346
O=C(NCC(F)=C1CN(C(=O)c2ccc3cc[nH]c3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132348
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]ccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132350
O=C(NCC(F)=C1CN(C(=O)Cc2cncs2)C1)c1cc(O)no1 s275592__15865378__15841170__14132352
Cc1cc(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1C s275592__15865378__15841170__14132354
O=C(NCC(F)=C1CN(C(=O)c2cnc(-c3ccccc3)o2)C1)c1cc(O)no1 s275592__15865378__15841170__14132358
O=C(NCC(F)=C1CN(C(=O)c2ccnc(-n3cccc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132360
O=C(NCC(F)=C1CN(C(=O)c2cn[nH]c(=O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132362
Cc1[nH]c(=O)[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132366
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CCCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132368
CC(C)CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1ccnc1 s275592__15865378__15841170__14132374
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)(F)F)no2)C1)c1cc(O)no1 s275592__15865378__15841170__14132376
O=C(NCC(F)=C1CN(C(=O)c2cscc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14132378
O=C(NCC(F)=C1CN(C(=O)c2ccn(CC(F)F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132380
Cc1nn(CC(F)F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132382
CCc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132384
O=C(NCC(F)=C1CN(C(=O)C2(C3CC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132386
O=C(NCC(F)=C1CN(C(=O)c2cc(=O)[nH]c(C3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132388
COC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14132390
O=C1CCC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__14132392
Cn1ccnc1COCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132394
CN1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__14132396
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132400
CC(C)(C)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132402
O=C(NCC(F)=C1CN(C(=O)c2ncn(-c3ccccc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132404
O=C(NCC(F)=C1CN(C(=O)c2ccnc(-c3ccco3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132414
CC1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133972
CC(C)(C)N1CCC(F)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133974
O=C(NCC(F)=C1CN(C(=O)C2(CF)CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133976
Cc1ncc2n1CCC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__14133978
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccncc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14133986
O=C(NCC(F)=C1CN(C(=O)CC(F)(F)C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14133994
CC1(C)CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133996
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CC(C)(C)C s275592__15865378__15841170__14133998
O=C(NCC(F)=C1CN(C(=O)CCc2cncs2)C1)c1cc(O)no1 s275592__15865378__15841170__14134002
NC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14134006
NC(=O)[C@@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134008
O=C(NCC(F)=C1CN(C(=O)CC(C2CCC2)C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134010
O=C(NCC(F)=C1CN(C(=O)c2ocnc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14134012
Cn1ncc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14134014
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__14134016
CC(F)(F)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14134018
O=C(NCC(F)=C1CN(C(=O)Cn2nnc3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134020
Cc1nc(C(C)C)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134022
CC[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__14134026
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(F)F s275592__15865378__15841170__14134028
CCc1ncnc(CC)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134032
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)[nH]1 s275592__15865378__15841170__14134034
O=C(NCC(F)=C1CN(C(=O)c2nccn3ccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134036
Cc1nc(C2CC2)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134038
Cc1ccn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14134040
O=C(NCC(F)=C1CN(C(=O)c2nccc3[nH]ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134042
CC(COCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCC1 s275592__15865378__15841170__14134044
COc1cc(=O)[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134046
CC(OCc1ccncc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134048
Cn1cncc1[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134052
O=C(NCC(F)=C1CN(C(=O)CCc2c[nH]nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134054
O=C(NCC(F)=C1CN(C(=O)C2(CF)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134056
C=C[C@@H]1OCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134058
CC(C)C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134062
CC[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134064
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc1C(N)=O s275592__15865378__15841170__14134068
O=C(NCC(F)=C1CN(C(=O)C2CCc3nnnn3CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134074
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]3CC[C@@H]2O3)C1)c1cc(O)no1 s275592__15865378__15841170__14134076
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2c1CCCC2 s275592__15865378__15841170__14134080
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC(=O)N1 s275592__15865378__15841170__14134082
Cc1c[nH]c(CC(N)=O)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134084
Cn1cc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14134086
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__14134088
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134090
COc1cccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134092
O=C(NCC(F)=C1CN(C(=O)c2cccc3cc[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14134096
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccnc1 s275592__15865378__15841170__14134098
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__14134100
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134102
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)c1 s275592__15865378__15841170__14134104
COc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__14134106
CCC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134108
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3ccccc3)o2)C1)c1cc(O)no1 s275592__15865378__15841170__14134110
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15841170__14134112
O=C(NCC(F)=C1CN(C(=O)c2cccc3[nH]ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134114
CC(C)=CCCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134116
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1F s275592__15865378__15841170__14134118
C=Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14134120
CC(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134122
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2OCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134124
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14134126
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccco3)[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__14134128
O=C(NCC(F)=C1CN(C(=O)C2(C(F)(F)F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134130
COc1ccccc1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129194
Cc1ccc2c(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)coc2c1 s275592__15865378__15841170__14129196
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14129202
Cc1cccc(C)c1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129204
O=C(NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccco1 s275592__15865378__15841170__14129208
O=C(NCC(F)=C1CN(C(=O)Cn2cncn2)C1)c1cc(O)no1 s275592__15865378__15841170__14129210
O=C(NCC(F)=C1CN(C(=O)CCc2ccccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14129212
Cc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14129214
O=C(NCC(F)=C1CN(C(=O)c2csc3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129216
O=C(NCC(F)=C1CN(C(=O)CCCc2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__14129218
CCc1sc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14129222
O=C(NCC(F)=C1CN(C(=O)c2ccc3nccnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129224
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sc1C s275592__15865378__15841170__14129226
O=C(NCC(F)=C1CN(C(=O)CN2C(=O)CNC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14129228
CN1CC(=O)N(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__14129230
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14129232
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sc1C s275592__15865378__15841170__14129234
O=C(NCC(F)=C1CN(C(=O)CN2CCCCCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14129238
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sc1C s275592__15865378__15841170__14129240
Cc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14129242
O=C(NCC(F)=C1CN(C(=O)COc2cccc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129244
O=C1NC(=O)C(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__14129246
NC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129250
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129252
NC(=O)c1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129254
O=C(NCC(F)=C1CN(C(=O)CCn2ccc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14129256
CC(Oc1ccc(F)cc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129258
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3ccccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129260
O=C(NCC(F)=C1CN(C(=O)CN2C(=O)CCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14129268
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1C s275592__15865378__15841170__14129270
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1C(C)C s275592__15865378__15841170__14129272
NC(=O)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14129274
CC(=O)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14129276
O=C(NCC(F)=C1CN(C(=O)CCCN2C(=O)CNC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14129278
Cc1cccc2nc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cn12 s275592__15865378__15841170__14129280
Cc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129282
O=C(NCC(F)=C1CN(C(=O)c2cnn(-c3ccccc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14129284
NC(=O)Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129286
COc1ccc(OC)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129290
O=C(NCC(F)=C1CN(C(=O)CCc2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__14129292
CC(C)Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129294
O=C(NCC(F)=C1CN(C(=O)Cn2ccccc2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14129296
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3c(c2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129298
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129300
Cc1noc(C)c1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129302
COCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129304
Cc1[nH]c2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2c1C s275592__15865378__15841170__14129312
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3cnnn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129314
CCc1onc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129316
O=C(NCC(F)=C1CN(C(=O)c2ccccc2-n2cnnn2)C1)c1cc(O)no1 s275592__15865378__15841170__14129320
CCCn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1=O s275592__15865378__15841170__14129324
O=C(NCC(F)=C1CN(C(=O)COc2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129326
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]nnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129330
Cc1ccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__14129338
Cc1n[nH]c(C)c1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129340
O=C(NCC(F)=C1CN(C(=O)COCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129344
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129348
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3c(c2)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129350
Cc1ccc(NC(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129352
O=C(NCC(F)=C1CN(C(=O)CCc2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14129354
Cc1csc(=O)n1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129356
CCn1nc(C2CC2)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132416
COCCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132420
Cc1cnc2nc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nn2c1 s275592__15865378__15841170__14132424
Cc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132428
Cc1ccc2cccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2n1 s275592__15865378__15841170__14132430
Cc1nc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2o1 s275592__15865378__15841170__14132432
O=C(NCC(F)=C1CN(C(=O)c2cnc3cc[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132434
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]ncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132436
O=C(NCC(F)=C1CN(C(=O)C2CCC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14132438
O=C(NCC(F)=C1CN(C(=O)c2ccsn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132440
CCOc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__14132442
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)cc1F s275592__15865378__15841170__14132444
Cc1noc(C(F)F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132446
Cc1cc(COCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14132448
Cc1cc(COCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__14132450
Cn1nccc1COCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132452
O=C(NCC(F)=C1CN(C(=O)c2ccc3nc[nH]c3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132454
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]c1C s275592__15865378__15841170__14132456
O=C(NCC(F)=C1CN(C(=O)c2cc3cccn3cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132460
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3cccnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132462
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)s1 s275592__15865378__15841170__14132464
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC1 s275592__15865378__15841170__14132466
CCc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132468
O=C(NCC(F)=C1CN(C(=O)CC2C=CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132470
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__14132472
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132474
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)c1 s275592__15865378__15841170__14132476
CCc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14132478
O=C(NCC(F)=C1CN(C(=O)C2CCn3cncc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132480
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(F)(F)CC1 s275592__15865378__15841170__14132482
CCOCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14132486
O=C(NCC(F)=C1CN(C(=O)c2cnoc2-c2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__14132490
Cc1noc(C)c1C(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132494
O=C(NCC(F)=C1CN(C(=O)CC2CC(F)(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132496
O=C(NCC(F)=C1CN(C(=O)C2CCc3n[nH]c(=O)n3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132502
COCc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132504
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C2CCC2)n1 s275592__15865378__15841170__14132506
CCc1nnc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132508
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3cn[nH]c3)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132510
Cn1cnc2cccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c21 s275592__15865378__15841170__14132512
Cc1n[nH]c(C)c1C(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132516
O=C(NCC(F)=C1CN(C(=O)C2CC3C=CC2O3)C1)c1cc(O)no1 s275592__15865378__15841170__14132520
CCCCC(C)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132522
O=C(NCC(F)=C1CN(C(=O)C2CCc3nccn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132524
O=C(NCC(F)=C1CN(C(=O)C2CCn3ccnc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132526
O=C(NCC(F)=C1CN(C(=O)C2CCc3cncn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132528
Cn1cnc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc21 s275592__15865378__15841170__14132534
COC1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132536
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__14132538
O=C(NCC(F)=C1CN(C(=O)C2CCCC3CC32)C1)c1cc(O)no1 s275592__15865378__15841170__14132540
O=C(NCC(F)=C1CN(C(=O)CC2CCC3CC23)C1)c1cc(O)no1 s275592__15865378__15841170__14132542
O=C(NCC(F)=C1CN(C(=O)C2CCC3CC3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132544
CCC(C)C(OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132546
COC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14132548
CN1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__14132550
CN(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccncc1 s275592__15865378__15841170__14132552
O=C(NCC(F)=C1CN(C(=O)CCCn2c(=O)[nH][nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14132554
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(=O)[nH]ccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132556
Cc1c(F)ccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132558
O=C(NCC(F)=C1CN(C(=O)Cn2cc(C3CC3)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14132560
O=C(NCC(F)=C1CN(C(=O)CC2CC(c3ccccc3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132562
CCCC1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132564
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C2Cc3ccccc3C21 s275592__15865378__15841170__14132566
O=C(NCC(F)=C1CN(C(=O)C23CC4CC(C(=O)N2)C3C4)C1)c1cc(O)no1 s275592__15865378__15841170__14132568
CCC(CC)C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132570
O=C(NCC(F)=C1CN(C(=O)CC2CS(=O)(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132572
O=C(NCC(F)=C1CN(C(=O)c2ncoc2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14132574
Cn1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15841170__14132578
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__14134134
O=C(NCC(F)=C1CN(C(=O)CCCC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14134136
O=C(NCC(F)=C1CN(C(=O)c2cc(F)c(F)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134138
O=C(NCC(F)=C1CN(C(=O)CCCc2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134140
Cc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134142
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CC(C)(C)C s275592__15865378__15841170__14134146
CCn1nc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134148
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14134150
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134152
O=C(NCC(F)=C1CN(C(=O)c2noc3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134154
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134156
O=C(NCC(F)=C1CN(C(=O)c2cc(F)ccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14134158
O=C(NCC(F)=C1CN(C(=O)c2ccncc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14134160
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)c(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134164
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__14134166
Cc1ccccc1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134168
O=C(NCC(F)=C1CN(C(=O)C2C3CCCCCCC32)C1)c1cc(O)no1 s275592__15865378__15841170__14134172
O=C(NCC(F)=C1CN(C(=O)C2CC23CC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134174
O=C(NCC(F)=C1CN(C(=O)c2ccc3cnccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14134176
O=C(NCC(F)=C1CN(C(=O)c2cccc(F)c2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14134178
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(Cl)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134180
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)(F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134184
O=C(NCC(F)=C1CN(C(=O)Cc2cc(F)c(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134188
O=C(NCC(F)=C1CN(C(=O)c2ccccc2-n2cccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134190
O=C(NCC(F)=C1CN(C(=O)c2cnnc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134194
O=C(NCC(F)=C1CN(C(=O)C2CCc3ccccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14134196
Cc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134198
CC(NS(C)(=O)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134200
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__14134206
O=C(NCC(F)=C1CN(C(=O)c2cnc3ccccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134208
O=C(NCC(F)=C1CN(C(=O)c2ccc3cc[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134212
CCOc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134214
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14134216
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc12 s275592__15865378__15841170__14134220
O=C(NCC(F)=C1CN(C(=O)Cc2cnc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14134222
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(F)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134224
O=C(NCC(F)=C1CN(C(=O)CC2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134228
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14134230
C[C@@H](OCc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134234
C=CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134236
Cc1oc(C(C)(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134238
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)[nH]1 s275592__15865378__15841170__14134240
O=C(NCC(F)=C1CN(C(=O)C(F)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134242
O=C(NCC(F)=C1CN(C(=O)C2CC23CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134246
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]c(=O)[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134250
O=C1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)NC(=O)N1 s275592__15865378__15841170__14134252
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(-c3ccccc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14134254
O=C(NCC(F)=C1CN(C(=O)c2cccc(N3CC=CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134256
O=C(NCC(F)=C1CN(C(=O)CCc2cc(Cl)cs2)C1)c1cc(O)no1 s275592__15865378__15841170__14134260
Cc1cccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134262
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C(C)C)n1 s275592__15865378__15841170__14134268
O=C(NCC(F)=C1CN(C(=O)Cn2cc(Cl)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134270
Cc1cccc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134132
O=C(NCC(F)=C1CN(C(=O)c2cnnn2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134272
CN(C)S(=O)(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134276
CCc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14134278
CCCN1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__14134280
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1ccnc1 s275592__15865378__15841170__14134282
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__14134284
Cc1c(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__14134286
Cc1ccnn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134288
O=C(NCC(F)=C1CN(C(=O)c2noc3c2CCCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134292
CCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14134294
Cc1cnc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnn2c1 s275592__15865378__15841170__14134296
Cc1ccn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)c1 s275592__15865378__15841170__14134298
Cc1noc(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129364
Cc1n[nH]c(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129366
CCc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129368
CC(C)(C)C(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129370
CCc1noc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129372
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)OCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14129374
COc1ccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129380
O=C(NCC(F)=C1CN(C(=O)COc2ccccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14129382
Cc1cccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129384
Cc1cc(C)cc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129386
COc1ccccc1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129388
O=C(NCC(F)=C1CN(C(=O)COc2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129390
Cc1ccc(C)c(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129392
Cc1ccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14129394
Cc1cccc(OCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129396
O=C(NCC(F)=C1CN(C(=O)CCOc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129398
Cc1ccccc1OCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129402
O=C(NCC(F)=C1CN(C(=O)COc2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14129404
Cc1noc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14129410
CCc1noc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14129414
Cc1cc(NC(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14129416
Cc1nc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__14129418
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]c1=O s275592__15865378__15841170__14129420
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(Cl)s2)C1)c1cc(O)no1 s275592__15865378__15841170__14129422
CC(C)c1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129426
Cc1nc(C(C)C)sc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129432
CCCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14129434
CN(C)c1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129436
Cc1c[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129438
O=C(NCC(F)=C1CN(C(=O)Cc2nc3ncccn3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14129440
O=C(NCC(F)=C1CN(C(=O)c2c[nH]cc2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129444
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14129446
O=C(NCC(F)=C1CN(C(=O)c2cccc3cnccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129448
Cc1[nH]nc2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__14129450
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccoc3)n[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14129454
Cc1cc(C)n(C(C)CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14129458
O=C(NCC(F)=C1CN(C(=O)c2cc3c([nH]c2=O)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129460
Cc1nccn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129462
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2CCCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129464
CC(CN1CCOCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129466
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14129468
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(=O)[nH]cnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129470
O=C(NCC(F)=C1CN(C(=O)Cc2csc3nccn23)C1)c1cc(O)no1 s275592__15865378__15841170__14129472
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__14129474
CC(COc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129476
CCn1cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129478
CC(C)n1cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129480
Cc1cc(C)cc(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2)c1 s275592__15865378__15841170__14129482
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C(C)(C)C s275592__15865378__15841170__14129486
O=C(NCC(F)=C1CN(C(=O)c2scnc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14129488
CCn1cc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129492
CCc1ncncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129494
CC(C)c1ncncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129496
Cc1nn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1Cl s275592__15865378__15841170__14129498
O=C(NCC(F)=C1CN(C(=O)CC2CCCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129500
O=C(NCC(F)=C1CN(C(=O)C2CCC=CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129502
NC(=O)c1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129504
O=C(NCC(F)=C1CN(C(=O)C2CCS(=O)(=O)N2)C1)c1cc(O)no1 s275592__15865378__15841170__14129506
Cc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14129508
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(C)c1F s275592__15865378__15841170__14129510
Cc1nn2cccnc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129512
O=C(NCC(F)=C1CN(C(=O)CCCN2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129514
CCC(C)C(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129516
O=C(NCC(F)=C1CN(C(=O)CCN2CCCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14129518
O=C(NCC(F)=C1CN(C(=O)c2ccnc(-n3ccnc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129520
CNS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129522
CCCS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129526
CC(C)S(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129528
O=C(NCC(F)=C1CN(C(=O)c2cnc3ccccn23)C1)c1cc(O)no1 s275592__15865378__15841170__14132582
Cc1ccn2cnc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__14132586
Cc1ccc2[nH]ncc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132588
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc3ccoc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132592
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]c(=O)[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132594
CC(=O)Nc1c[nH]c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132596
CCc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132598
CCN1CCOCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132600
O=C(NCC(F)=C1CN(C(=O)C2(F)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132604
CCc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132606
O=C(NCC(F)=C1CN(C(=O)c2coc3cc(F)ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132608
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccnc1 s275592__15865378__15841170__14132610
Cc1nnc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cn12 s275592__15865378__15841170__14132612
CCC(C)n1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14132616
CN(C)Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14132620
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3ccnc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132622
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc2cncn12 s275592__15865378__15841170__14132624
O=C(NCC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132628
O=C(NCC(F)=C1CN(C(=O)C2CCc3ccccc3CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132630
O=C(NCC(F)=C1CN(C(=O)c2cnn(CCF)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132634
Cc1cc(C)nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14132636
O=C(NCC(F)=C1CN(C(=O)c2cccc3ncnn23)C1)c1cc(O)no1 s275592__15865378__15841170__14132642
Cn1cncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132644
O=C(NCC(F)=C1CN(C(=O)c2cccc3cccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132646
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132650
O=C(NCC(F)=C1CN(C(=O)CCc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132654
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__14132656
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14132658
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132666
Cc1ccn2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nc2c1 s275592__15865378__15841170__14132672
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3cccc3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132674
O=C(NCC(F)=C1CN(C(=O)CCc2nc3ccccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14132676
O=C(NCC(F)=C1CN(C(=O)Cn2ccc(=O)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14132678
COCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14132680
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc21 s275592__15865378__15841170__14132686
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)s1 s275592__15865378__15841170__14132688
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3cccc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132692
NC(=O)NCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132694
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14132698
COc1ccc(C)cc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132700
CCn1c(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14132702
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14132704
CCc1nnsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132706
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132708
COc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__14132710
COc1ccc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132712
O=C(NCC(F)=C1CN(C(=O)c2cc(=O)c3ccccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14132716
O=C(NCC(F)=C1CN(C(=O)CC2CCS(=O)(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132718
O=C(NCC(F)=C1CN(C(=O)c2cc(Br)c[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14132720
O=C(NCC(F)=C1CN(C(=O)Cc2noc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132726
O=C(NCC(F)=C1CN(C(=O)c2cnn(-c3ccccc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132732
O=C(NCC(F)=C1CN(C(=O)CCN2C(=O)CCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14132734
O=C(NCC(F)=C1CN(C(=O)C2CCS(=O)(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132736
Cc1cc2ccccc2n1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132738
CC(=O)N1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14132740
O=C(NCC(F)=C1CN(C(=O)CCn2cnc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14132742
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3O2)C1)c1cc(O)no1 s275592__15865378__15841170__14132744
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14132746
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)no2)C1)c1cc(O)no1 s275592__15865378__15841170__14134302
CCc1oncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134304
CC(Cc1cccs1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134306
CC(C)c1nccn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134308
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__14134312
O=C(NCC(F)=C1CN(C(=O)c2cnc(C3CC3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134314
Cc1nc(C(C)C)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134316
O=C(NCC(F)=C1CN(C(=O)Cc2cscn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134318
Cc1nc(N(C)C)sc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134320
CC1CCN(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14134322
CC1CCCN(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14134324
COc1nc(C)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134326
O=C(NCC(F)=C1CN(C(=O)c2coc(C3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14134328
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@@H]2c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134330
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCCN2C(=O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134332
O=C(NCC(F)=C1CN(C(=O)c2cnc(C3CC3)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14134334
O=C(NCC(F)=C1CN(C(=O)C2C3Cc4ccccc4C32)C1)c1cc(O)no1 s275592__15865378__15841170__14134336
COCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14134338
COCC(=O)N[C@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14134340
O=C(NCC(F)=C1CN(C(=O)CCc2nc(C3CC3)no2)C1)c1cc(O)no1 s275592__15865378__15841170__14134346
Cc1noc(C)c1CC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134348
O=C(NCC(F)=C1CN(C(=O)c2ccc3cccnn23)C1)c1cc(O)no1 s275592__15865378__15841170__14134352
O=C(NCC(F)=C1CN(C(=O)c2cnn3c(=O)cc[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14134354
O=C(NCC(F)=C1CN(C(=O)c2cnc3cccnn23)C1)c1cc(O)no1 s275592__15865378__15841170__14134356
CN(C)C(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134358
C#CCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14134362
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(Cl)s2)C1)c1cc(O)no1 s275592__15865378__15841170__14134364
Cc1ccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14134366
CC(C)(NS(C)(=O)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134368
CCC(CC)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__14134370
CCC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__14134372
CC1(C)C2CCC1(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__14134380
Cc1cc(C)n(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14134300
C=CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14134384
CC(C)c1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134388
CC(C)(C)c1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134390
O=C(NCC(F)=C1CN(C(=O)c2scnc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134392
COCc1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134394
CC(C)c1nnnn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134396
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCCC1 s275592__15865378__15841170__14134398
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(=O)[nH]1 s275592__15865378__15841170__14134400
Cc1nc(C2CC2)oc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134406
Cc1nc(C(C)C)oc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134408
Cc1nc(CC(C)C)oc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134410
Cc1ccccc1COCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134412
Cc1ccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14134414
Cc1ccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14134422
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134424
O=C(NCC(F)=C1CN(C(=O)CCc2cn[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134428
CC(Cc1cnc[nH]1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134436
C=CCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14134438
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134440
C[C@]1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C[C@@H]1c1ccccc1 s275592__15865378__15841170__14134442
O=C(NCC(F)=C1CN(C(=O)C2CCCC3CCCN32)C1)c1cc(O)no1 s275592__15865378__15841170__14134444
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134448
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129530
O=C(NCC(F)=C1CN(C(=O)CN2CCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14129536
O=C(NCC(F)=C1CN(C(=O)CCOCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129538
O=C(NCC(F)=C1CN(C(=O)CCCn2cccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14129540
CC(C)C(=O)N1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129548
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccsc1 s275592__15865378__15841170__14129550
CC(C)(C)CC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129552
O=C(NCC(F)=C1CN(C(=O)Cn2ccc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14129554
O=C(NCC(F)=C1CN(C(=O)CCc2nccs2)C1)c1cc(O)no1 s275592__15865378__15841170__14129558
COCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129568
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCC1=O s275592__15865378__15841170__14129572
CCn1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__14129574
CC1OC(C)C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1C s275592__15865378__15841170__14129578
Cc1n[nH]c(C)c1CC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129580
O=C(NCC(F)=C1CN(C(=O)c2cn[nH]c2-c2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__14129586
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c3occc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129590
COC(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129592
CCC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129596
CNC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129598
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1F s275592__15865378__15841170__14129600
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)c(F)c1 s275592__15865378__15841170__14129602
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(Cl)c1 s275592__15865378__15841170__14129604
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(F)c1 s275592__15865378__15841170__14129606
C[C@H](NC(=O)c1ccco1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129608
O=C(NCC(F)=C1CN(C(=O)C2Cc3cccc(F)c3O2)C1)c1cc(O)no1 s275592__15865378__15841170__14129612
O=C(NCC(F)=C1CN(C(=O)c2cc3cccc(F)c3o2)C1)c1cc(O)no1 s275592__15865378__15841170__14129614
CCCCCCC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129616
O=C(NCC(F)=C1CN(C(=O)C2CCCS2(=O)=O)C1)c1cc(O)no1 s275592__15865378__15841170__14129618
O=C(NCC(F)=C1CN(C(=O)c2noc3c2COCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129620
O=C(NCC(F)=C1CN(C(=O)C2CCc3cn[nH]c3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14129624
Cn1nc(C2CC2)nc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129628
CCN1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14129634
O=C(NCC(F)=C1CN(C(=O)CCCOc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129636
CC1CCC(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__14129640
Cc1cc(=O)[nH]c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129644
C[C@@H](Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129646
C[C@H](Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129648
C=CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129650
O=C(NCC(F)=C1CN(C(=O)C23CCC(CC2)CC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129652
CCCCCCCCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129654
CCCCCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129660
CC[C@H](C)[C@H](NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129666
CCCCCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129668
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129672
C=CCC(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129674
CC1=CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14129676
CC(C)(C)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129682
CC(C)(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14129686
C=CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129688
NC(=O)N1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14132748
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__14132750
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccccc3)[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132752
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1C s275592__15865378__15841170__14132754
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14132756
CCCCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14132758
O=C(NCC(F)=C1CN(C(=O)C2(c3ccccc3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132762
O=C(NCC(F)=C1CN(C(=O)C2COc3ccccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14132766
Cc1[nH]c2ccccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132768
O=C(NCC(F)=C1CN(C(=O)c2occc2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132770
CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc21 s275592__15865378__15841170__14132772
Cc1oc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14132776
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14132778
O=C(NCC(F)=C1CN(C(=O)CCc2cc3ccccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__14132782
Cc1cc(C)n(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14132786
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccccc3)on2)C1)c1cc(O)no1 s275592__15865378__15841170__14132788
COCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14132792
Cc1cc(=O)oc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132794
Cn1cc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132796
CC(C)=CC1C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__14132798
CC(=O)NC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCC1 s275592__15865378__15841170__14132800
COc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1C s275592__15865378__15841170__14132802
Cc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14132806
COc1cccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14132812
O=C(NCC(F)=C1CN(C(=O)Cc2cccc3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14132814
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3cnccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132816
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3[nH]ncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132818
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(C(F)F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132820
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(C(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132822
Cc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__14132824
O=C(NCC(F)=C1CN(C(=O)c2ccn3ccnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132830
O=C(NCC(F)=C1CN(C(=O)c2cccc3nccn23)C1)c1cc(O)no1 s275592__15865378__15841170__14132832
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]ccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132834
O=C(NCC(F)=C1CN(C(=O)c2ccc3nnnn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132836
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__14132840
Cc1ccc2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)n2c1 s275592__15865378__15841170__14132844
O=C(NCC(F)=C1CN(C(=O)c2ncc(Cl)s2)C1)c1cc(O)no1 s275592__15865378__15841170__14132846
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccn12 s275592__15865378__15841170__14132850
O=C(NCC(F)=C1CN(C(=O)c2ncc3ccccn23)C1)c1cc(O)no1 s275592__15865378__15841170__14132852
O=C(NCC(F)=C1CN(C(=O)c2onc3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132856
O=C(NCC(F)=C1CN(C(=O)C(c2ccccc2)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132858
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14132860
COCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132862
O=C(NCC(F)=C1CN(C(=O)c2cnc3nccn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132876
O=C(NCC(F)=C1CN(C(=O)CCc2ccon2)C1)c1cc(O)no1 s275592__15865378__15841170__14132878
O=C(NCC(F)=C1CN(C(=O)CCc2cncnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132880
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C(F)F s275592__15865378__15841170__14132884
COc1coc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15841170__14132886
COc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15841170__14132888
Cc1cc(Cl)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14132890
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1c(F)cccc1F s275592__15865378__15841170__14132892
O=C(NCC(F)=C1CN(C(=O)c2ccc3cncn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132894
CCc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14132896
Cc1csc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14132898
O=C(NCC(F)=C1CN(C(=O)c2cnc3cnccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132900
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1C s275592__15865378__15841170__14132902
Cc1cncn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132904
O=C(NCC(F)=C1CN(C(=O)c2conc2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14132908
O=C(NCC(F)=C1CN(C(=O)CCc2ccc3[nH]ccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132910
O=C(NCC(F)=C1CN(C(=O)c2nnc3ccccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132912
CN(C)CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14134454
Cc1cccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134458
Cc1ccccc1[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134460
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)S1(=O)=O s275592__15865378__15841170__14134464
C=C(C)[C@@H]1OCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134470
CC1(C)[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[C@H]1c1ccccc1 s275592__15865378__15841170__14134472
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2C[C@H]2c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134474
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)F)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134476
O=C(NCC(F)=C1CN(C(=O)c2cn(C3CCC3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134480
O=C(NCC(F)=C1CN(C(=O)c2cscc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14134482
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(C(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134484
O=C(NCC(F)=C1CN(C(=O)c2cccc(C(F)F)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134486
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCCO1 s275592__15865378__15841170__14134488
O=C(NCC(F)=C1CN(C(=O)c2ccnn2C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134490
CN(C)CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14134502
CC(C)(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14134506
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccnn1C s275592__15865378__15841170__14134508
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sn1 s275592__15865378__15841170__14134518
O=C(NCC(F)=C1CN(C(=O)c2cn3c(n2)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134522
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134524
C[C@@H]1[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCN1C s275592__15865378__15841170__14134526
CC(C)(C)c1nc[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134528
CC(C)(C)C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134532
CCc1nccn1C(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134534
O=C(NCC(F)=C1CN(C(=O)c2ncnc3sccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134536
NC(=O)c1ncn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14134538
CC[C@@H]1[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCN1C s275592__15865378__15841170__14134540
CS(=O)(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__14134542
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3C=C[C@H]2CC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134544
CCN(CC)C(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129696
C=CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129700
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14129704
Cc1ccccc1C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129710
O=C(NCC(F)=C1CN(C(=O)CCC2CCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14129714
O=C(NCC(F)=C1CN(C(=O)C(F)Cc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129716
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14129720
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15841170__14129726
COc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__14129728
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__14129730
Cc1nnc2n1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__14129732
CN(C)S(=O)(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129734
CCCC(=O)N1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129738
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__14129744
CCN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129746
CC(C)c1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129748
CCc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129752
CC1CCC(C)N1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129754
O=C(NCC(F)=C1CN(C(=O)C2CCc3nncn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14129756
CCn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc2ccccc21 s275592__15865378__15841170__14129762
O=C(NCC(F)=C1CN(C(=O)CCn2cc(Cl)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14129768
CCOCCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129772
O=C(NCC(F)=C1CN(C(=O)c2cncc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129774
Cn1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14129776
O=C(NCC(F)=C1CN(C(=O)CCCN2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129778
CN(C)Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129780
O=C(Cn1cncn1)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129788
O=C(NCC(F)=C1CN(C(=O)Cc2n[nH]c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129790
Cc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14129792
CNC(=O)NC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129794
CCCNC(=O)NC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129796
CCc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14129798
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14129802
C#CCN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14129804
O=C(NCC(F)=C1CN(C(=O)CCN2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129808
Cc1ccc(C)n1C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129810
COc1cccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129812
Cc1cnn(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129814
Cc1ccc2oc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2c1 s275592__15865378__15841170__14129816
CN(C)Cc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129818
CCS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129820
Cc1sc(=O)n(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14129824
C=CCNC(=O)NC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129826
O=C(NCC(F)=C1CN(C(=O)CCc2cc(F)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14129830
NC(=O)Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14129832
CCc1cccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c[nH]c12 s275592__15865378__15841170__14129836
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc2c(C)cccc12 s275592__15865378__15841170__14129838
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129840
CCN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129844
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCCC1 s275592__15865378__15841170__14129846
O=C(NCC(F)=C1CN(C(=O)[C@H]2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__14129852
Cc1cccc(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2)c1 s275592__15865378__15841170__14129854
CN(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14129856
O=C(NCC(F)=C1CN(C(=O)CCC(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14132916
O=C(NCC(F)=C1CN(C(=O)c2cccc3oc(=O)[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14132918
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CCCC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132920
O=C(NCC(F)=C1CN(C(=O)C2CCc3cc(F)ccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14132926
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(=O)[nH]1 s275592__15865378__15841170__14132928
O=C(NCC(F)=C1CN(C(=O)Cn2cnc3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132932
CCOc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__14132934
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CC2)CC3)C1)c1cc(O)no1 s275592__15865378__15841170__14132936
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14132938
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccncc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14132940
O=C(NCC(F)=C1CN(C(=O)CCC2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132942
Cc1onc(C2CC2)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132946
Cc1noc(C2CC2)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132948
O=C(NCC(F)=C1CN(C(=O)c2cc3ncccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__14132950
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(=O)[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132952
CC(CC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132954
Cn1nnc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc21 s275592__15865378__15841170__14132956
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc2ccccc12 s275592__15865378__15841170__14132958
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ncccc12 s275592__15865378__15841170__14132960
CC1Cc2cccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2O1 s275592__15865378__15841170__14132962
O=C(NCC(F)=C1CN(C(=O)c2cc(F)c[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14132964
O=C(NCC(F)=C1CN(C(=O)c2cc3cscc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14132966
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14132968
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(Br)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132970
CCCCC(CC)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14132972
CCC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(=O)N1 s275592__15865378__15841170__14132974
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CNC(=O)C1 s275592__15865378__15841170__14132976
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1Cl s275592__15865378__15841170__14132982
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(C3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14132984
Cc1cc(F)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__14132986
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2-c2ccoc2)C1)c1cc(O)no1 s275592__15865378__15841170__14132988
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2CC2C1 s275592__15865378__15841170__14132994
O=C(NCC(F)=C1CN(C(=O)c2cnc(CC3CC3)s2)C1)c1cc(O)no1 s275592__15865378__15841170__14132996
O=C(NCC(F)=C1CN(C(=O)C2(CCF)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14132998
COCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133000
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cnn(C)c1 s275592__15865378__15841170__14133004
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133006
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2nccn2c1 s275592__15865378__15841170__14133008
Cc1ccc(C2CC2)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133010
CC(C)Oc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133012
CCOc1nccc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133016
Cc1nccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14133020
Cn1cnn(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15841170__14133022
O=C(NCC(F)=C1CN(C(=O)COCC(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14133024
CC(C)(COCC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133026
CCCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)S(N)(=O)=O s275592__15865378__15841170__14133028
O=C(NCC(F)=C1CN(C(=O)CCCCc2c[nH]nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14133030
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__14133032
CN(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14133036
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)nn1 s275592__15865378__15841170__14133040
O=C(NCC(F)=C1CN(C(=O)c2ocnc2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14133044
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14133046
O=C(NCC(F)=C1CN(C(=O)C2(C3CC3)CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133048
CC(C)n1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133050
CN(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCCC1 s275592__15865378__15841170__14133052
Cc1cc2occ(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2cc1C s275592__15865378__15841170__14133060
CN(C)C1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14133066
CNS(=O)(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133068
O=C(NCC(F)=C1CN(C(=O)c2cncc(-n3ccnn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133070
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCN1 s275592__15865378__15841170__14133072
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ccncc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133074
O=C(NCC(F)=C1CN(C(=O)c2occ3c2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14133076
O=C(NCC(F)=C1CN(C(=O)c2occ3c2CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__14133078
Cc1cncc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133080
CCn1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14134546
Cn1ncc(C2CCC2)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134548
O=C(NCC(F)=C1CN(C(=O)[C@@]23COC[C@@H]2C3)C1)c1cc(O)no1 s275592__15865378__15841170__14134550
O=C(NCC(F)=C1CN(C(=O)c2cncc3nc[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14134554
CC1CCCc2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)n21 s275592__15865378__15841170__14134556
O=C(NCC(F)=C1CN(C(=O)c2cn(-c3ccccc3)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134558
O=C(NCC(F)=C1CN(C(=O)Cc2cn3c(n2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134560
CC(C)(C)n1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14134564
O=C(NCC(F)=C1CN(C(=O)C(F)C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14134568
O=C(NCC(F)=C1CN(C(=O)c2ccc3cccnc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14134570
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134572
Cc1c(F)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134574
COc1c(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14134576
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14134582
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__14134584
CCS(=O)(=O)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134586
Cc1c(Cl)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134588
O=C(NCC(F)=C1CN(C(=O)c2sccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__14134590
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccncc1 s275592__15865378__15841170__14134594
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134596
CC1CCCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134598
COc1cccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134600
O=C(NCC(F)=C1CN(C(=O)CNC(=O)C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134602
Cc1occc1C(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134604
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccoc1 s275592__15865378__15841170__14134606
CC(Oc1ccccc1F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134610
CC(Oc1cccc(F)c1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134612
CCC(=O)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134614
CC(NC(=O)C1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134616
CC(NC(=O)c1ccoc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134618
CCC(=O)N1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14134626
CCC(=O)N1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134632
CC(C)C(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134634
CCS(=O)(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134636
CS(=O)(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134638
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)S(C)(=O)=O s275592__15865378__15841170__14134640
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(=O)C1CC1 s275592__15865378__15841170__14134642
COCC(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134646
COCCN1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__14134654
CC(C)(C)N1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__14134656
CN1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__14134658
CCN1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__14134660
CC(C)CN1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__14134662
COCC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134666
O=C(NCC(F)=C1CN(C(=O)CCCNC(=O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134668
CCCOc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134670
O=C(NCC(F)=C1CN(C(=O)COc2ccc(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134676
O=C(NCC(F)=C1CN(C(=O)CCn2ccccc2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14134678
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1C(=O)CCC1=O s275592__15865378__15841170__14134680
O=C(NCC(F)=C1CN(C(=O)CCOc2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134690
CCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14134694
O=C(NCC(F)=C1CN(C(=O)CCCN2C(=O)CCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14134696
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2OCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14134700
Cn1c(=O)ccn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15841170__14134702
O=C(NCC(F)=C1CN(C(=O)c2ncoc2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134704
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__14129862
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]c(=O)oc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129864
CN1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1=O s275592__15865378__15841170__14129868
COc1cccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129870
CC(C)(C)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14129872
CCOCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129876
O=C(NCC(F)=C1CN(C(=O)CC(C2CC2)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129878
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__14129880
Cc1cccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)oc12 s275592__15865378__15841170__14129882
NC(=O)c1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129884
O=C(NCC(F)=C1CN(C(=O)C2CCC3CCCCC3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14129886
CN(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccnc1 s275592__15865378__15841170__14129888
CCCCS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129890
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC2CC3)C1)c1cc(O)no1 s275592__15865378__15841170__14129892
CCOc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14129894
CC(CS(C)(=O)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129898
CCc1oc2ccccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129900
O=C(NCC(F)=C1CN(C(=O)c2nn[nH]c2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129902
CCCCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14129904
CC(C)CC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129906
CCC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129908
O=C(NCC(F)=C1CN(C(=O)CCCC2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14129910
Cc1ccc(CC(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14129912
Cc1ccc2[nH]cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__14129918
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)c1=O s275592__15865378__15841170__14129920
Cc1nsc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129922
O=C(NCC(F)=C1CN(C(=O)c2cccc(C3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129924
O=C(NCC(F)=C1CN(C(=O)C23CC(c4ccccc4)(C2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__14129926
O=C(NCC(F)=C1CN(C(=O)Cc2c[nH]c3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14129930
CCCCCC(C)(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129932
O=C(NCC(F)=C1CN(C(=O)C2CCCCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14129936
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2c1CCC2 s275592__15865378__15841170__14129938
CC1CC(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14129942
O=C(NCC(F)=C1CN(C(=O)COc2cc(F)cc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14129946
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__14129948
CC(=O)N1CCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129950
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14129952
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14129956
CC1(C)CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14129958
Cc1ccccc1CC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129960
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14129962
NC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14129964
O=C(NCC(F)=C1CN(C(=O)c2ccc(CF)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14129966
Cc1nc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc2o1 s275592__15865378__15841170__14129968
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)s1 s275592__15865378__15841170__14129970
Cc1cccc2oc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__14129972
Cn1c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc2ccccc21 s275592__15865378__15841170__14129974
CCCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129976
CC(=O)NC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__14129978
O=C(NCC(F)=C1CN(C(=O)C2CCCC3CCCCC32)C1)c1cc(O)no1 s275592__15865378__15841170__14129980
CC1(C)CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129984
CC1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14129986
Cc1ccc(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CCC2)cc1 s275592__15865378__15841170__14129990
CC(C)Cc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14129992
NC(=O)c1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14130000
CC(C)(C)C12CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(C1)C2 s275592__15865378__15841170__14130002
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc2ccccc12 s275592__15865378__15841170__14130004
O=C(NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3[C@@H]4CC[C@@H](C4)[C@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__14130006
O=C(NCC(F)=C1CN(C(=O)C2Cc3c(Cl)cccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14130008
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130010
COCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14130012
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14130014
CC(CC1CCCO1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130016
CC(C)c1occc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130018
C=CC(C)(CCOC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133082
O=C(NCC(F)=C1CN(C(=O)CC2CCCS2(=O)=O)C1)c1cc(O)no1 s275592__15865378__15841170__14133084
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cnn(C)c1 s275592__15865378__15841170__14133086
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCOC1 s275592__15865378__15841170__14133090
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCOCC1 s275592__15865378__15841170__14133092
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCC1 s275592__15865378__15841170__14133094
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCOC1 s275592__15865378__15841170__14133096
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(C)(C)C1 s275592__15865378__15841170__14133098
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOC1 s275592__15865378__15841170__14133100
O=C(NCC(F)=C1CN(C(=O)C2(C3CC3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133108
CC(C)n1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__14133110
COc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__14133112
CCOc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14133114
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC1 s275592__15865378__15841170__14133122
O=C(NCC(F)=C1CN(C(=O)C2(C3CCC3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133124
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(C3CCC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133126
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C(C)C)n1 s275592__15865378__15841170__14133128
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C2CC2)n1 s275592__15865378__15841170__14133130
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC1 s275592__15865378__15841170__14133132
Cc1cccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133136
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3ccnc3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133138
O=C(NCC(F)=C1CN(C(=O)c2csnn2)C1)c1cc(O)no1 s275592__15865378__15841170__14133140
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(Cl)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133142
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__14133144
O=C(NCC(F)=C1CN(C(=O)CCc2cccc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133148
Cc1cc(C)c2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)[nH]c2c1 s275592__15865378__15841170__14133150
Cc1ccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)[nH]c2c1 s275592__15865378__15841170__14133152
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133154
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)on2)C1)c1cc(O)no1 s275592__15865378__15841170__14133156
O=C(NCC(F)=C1CN(C(=O)c2csc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133158
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14133160
Cc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__14133166
Cc1ccc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133168
Cc1nn(C)c(C)c1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133170
Cc1nn(C)c(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133172
O=C(NCC(F)=C1CN(C(=O)c2cnco2)C1)c1cc(O)no1 s275592__15865378__15841170__14133174
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccco3)on2)C1)c1cc(O)no1 s275592__15865378__15841170__14133176
O=C(NCC(F)=C1CN(C(=O)c2cccc3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133178
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__14133180
Cc1nn(C)c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133182
Cc1nn(C)c(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133190
Cc1cc(C)n(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14133194
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3c(c2)CCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14133196
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)c(Cl)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14133198
O=C(NCC(F)=C1CN(C(=O)CCn2ccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133200
O=C(NCC(F)=C1CN(C(=O)Cc2cccc3cccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133206
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14133208
COc1ccc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133216
O=C(NCC(F)=C1CN(C(=O)c2cc3ccsc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14133218
O=C(NCC(F)=C1CN(C(=O)Cc2cc3ccccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__14133222
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3cccn3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133226
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3cncn3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133228
Cc1noc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14133230
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3ccnc3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133232
CC(C)(C)C(=O)NCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133234
CC(NC(=O)C(C)(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133240
CC(C)(C)C(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133242
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C(C)(C)C s275592__15865378__15841170__14134712
CNC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134714
CC(C)Oc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14134722
O=C(NCC(F)=C1CN(C(=O)CN2CCCCCCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14134724
O=C(NCC(F)=C1CN(C(=O)CN2CCCS2(=O)=O)C1)c1cc(O)no1 s275592__15865378__15841170__14134728
O=C(NCC(F)=C1CN(C(=O)C2(c3ccc(F)cc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134730
Cc1ccc(COCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14134732
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14134736
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14134738
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__14134740
O=C(NCC(F)=C1CN(C(=O)CCCC2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134742
CC1CC2(CCO1)CC2C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134744
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CCC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134746
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C1CC1 s275592__15865378__15841170__14134748
CC(C)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134750
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]nnc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14134754
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn2c1OCCC2 s275592__15865378__15841170__14134756
O=C(NCC(F)=C1CN(C(=O)c2cc(F)c3ccccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134758
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134762
CCc1ncsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134764
O=C(NCC(F)=C1CN(C(=O)c2cn(-c3cccnc3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134766
COc1nc(C)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134768
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134772
CC(=O)Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14134774
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14134776
COc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__14134778
O=C(NCC(F)=C1CN(C(=O)c2ncnc3ccsc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134780
CC(C)(C)n1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14134782
CC(=O)Nc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134784
Cc1cc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cn2c1 s275592__15865378__15841170__14134786
O=C(NCC(F)=C1CN(C(=O)c2ccccc2-c2cn[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134788
O=C(NCC(F)=C1CN(C(=O)C2(F)CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134790
O=C(NCC(F)=C1CN(C(=O)CCc2c[nH]cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134792
O=C(NCC(F)=C1CN(C(=O)CC2CCC(F)(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14134794
O=C(NCC(F)=C1CN(C(=O)CC2(c3ccccc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134796
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134800
C=CCn1cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134804
CCCCCCCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134806
O=C(NCC(F)=C1CN(C(=O)c2cc3ccncc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14134808
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC1 s275592__15865378__15841170__14134810
O=C(NCC(F)=C1CN(C(=O)c2nc[nH]c2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14134812
Cc1cccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)coc12 s275592__15865378__15841170__14134814
O=C(NCC(F)=C1CN(C(=O)c2nc3cccnc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14134816
O=C(NCC(F)=C1CN(C(=O)c2cnn3ccncc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134820
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14134822
O=C(NCC(F)=C1CN(C(=O)CN2CCOCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14134824
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]nnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134826
CCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14134828
O=C(NCC(F)=C1CN(C(=O)c2cnn3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134830
Cc1nn(C)cc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134832
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C(F)F)n1 s275592__15865378__15841170__14134838
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCC1 s275592__15865378__15841170__14134842
CC(C)Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14134844
O=C(NCC(F)=C1CN(C(=O)c2cnc3nccnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134846
O=C(NCC(F)=C1CN(C(=O)C2(Cc3ccccc3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134848
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCCC1 s275592__15865378__15841170__14134852
CCc1noc(CC)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134856
COc1cc(C)cnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134858
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sc2nccn12 s275592__15865378__15841170__14134860
O=C(NCC(F)=C1CN(C(=O)c2cc3c(cn2)OCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__14134864
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134866
O=C(NCC(F)=C1CN(C(=O)C2(Cc3ccccc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134868
CCOCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130024
CNC(=O)CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130026
CC(C)(CS(C)(=O)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130028
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCc2ccccc21 s275592__15865378__15841170__14130030
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__14130032
CC(C)(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14130034
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1C s275592__15865378__15841170__14130036
COC1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130038
CC1CCC(C)N1C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130046
C=CCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130048
C=CCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130050
CC(C)CCOC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130052
CC(OCC1CCCCO1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130054
CC(OCC1CCCO1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130056
Cc1noc(Cl)c1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130062
CCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130066
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130070
COCCOCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130072
CC(Cc1cccc(F)c1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130074
CC1CCCCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130076
CCOC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130078
O=C(NCC(F)=C1CN(C(=O)CCc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14130082
CC(Cc1ccc(F)cc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130084
O=C(NCC(F)=C1CN(C(=O)CCc2cscn2)C1)c1cc(O)no1 s275592__15865378__15841170__14130086
Cc1cc(C)n(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14130088
O=C(NCC(F)=C1CN(C(=O)CCCCN2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130090
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130092
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)Cc1ccccc1 s275592__15865378__15841170__14130096
CCCCC(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130098
CN(C)c1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14130100
O=C(NCC(F)=C1CN(C(=O)CCCn2ccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130102
COCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14130108
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14130110
CC1CCC(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130116
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCC1=O s275592__15865378__15841170__14130118
O=C(NCC(F)=C1CN(C(=O)c2csc(C3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__14130120
CCN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14130124
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3ccccc3)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14130126
CC(C)Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__14130128
CC(C)Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130130
CC(C)OCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130132
NC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130134
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130138
O=C(NCC(F)=C1CN(C(=O)c2ccnc(-n3cncn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130142
NC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14130144
O=C(NCC(F)=C1CN(C(=O)C2COc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14130146
O=C(NCC(F)=C1CN(C(=O)c2coc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14130148
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C1CC1 s275592__15865378__15841170__14130150
O=C(NCC(F)=C1CN(C(=O)COCCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130152
Cc1ccccc1C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130158
NC(=O)N1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130162
COc1ncnc(OC)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130166
O=C(NCC(F)=C1CN(C(=O)CCNC(=O)C2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__14130168
CC(C)CC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130170
O=C(NCC(F)=C1CN(C(=O)C2(C(F)(F)F)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130174
Cc1cccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130176
O=C(NCC(F)=C1CN(C(=O)COc2ccc(F)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130178
CC(=O)NC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130184
Cc1ccccc1C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130188
CC(C)c1noc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14133248
Cc1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133250
Cc1noc2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__14133252
Cc1cccc(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CCC2)c1 s275592__15865378__15841170__14133264
O=C(NCC(F)=C1CN(C(=O)c2cc3cc(F)ccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14133266
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__14133268
O=C(NCC(F)=C1CN(C(=O)c2cccc3[nH]ncc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133272
O=C(NCC(F)=C1CN(C(=O)c2cccnc2-n2cccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14133274
Cc1nn(C)c(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14133276
O=C(NCC(F)=C1CN(C(=O)c2cccc3cn[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14133282
Cc1ccc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2c1 s275592__15865378__15841170__14133284
Cc1n[nH]c(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14133286
O=C(NCC(F)=C1CN(C(=O)C2OCCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14133288
O=C(NCC(F)=C1CN(C(=O)c2cnn3cccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133294
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14133296
O=C(NCC(F)=C1CN(C(=O)c2coc(=O)c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133298
Cc1n[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133302
COc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133304
Cc1cc(F)cc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133306
O=C(NCC(F)=C1CN(C(=O)c2cccc(-c3ncn[nH]3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133310
COc1c(F)ccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133312
COc1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133314
CN1C(=O)CCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133316
O=C(NCC(F)=C1CN(C(=O)CCc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__14133320
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)cc1Cl s275592__15865378__15841170__14133322
Cn1cnc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc21 s275592__15865378__15841170__14133324
O=C(NCC(F)=C1CN(C(=O)c2ccn3nnnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133326
COc1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133328
O=C(NCC(F)=C1CN(C(=O)c2cc3ncccc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14133332
CCCC(OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133336
Cc1nc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2n1C s275592__15865378__15841170__14133338
C=C(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133340
Cc1ccn(C(C)CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14133344
O=C1CN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCN1 s275592__15865378__15841170__14133348
Cc1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__14133350
O=C(NCC(F)=C1CN(C(=O)c2cnc3ccsc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133356
CCCCCCC(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133358
CC(C)Oc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133362
O=C(NCC(F)=C1CN(C(=O)c2ncoc2C2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__14133364
CC(CC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133366
NC(=O)C1CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133368
Cc1ccc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2c1C s275592__15865378__15841170__14133370
O=C(NCC(F)=C1CN(C(=O)CCCn2ccccc2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14133372
O=C(NCC(F)=C1CN(C(=O)C2CCNC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14133374
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]c1=O s275592__15865378__15841170__14133376
CN1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)NC1=O s275592__15865378__15841170__14133378
C=CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133380
C#CCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133382
CN1CCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133386
C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133388
O=C(NCC(F)=C1CN(C(=O)CC2CC=CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133390
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14133392
CCC(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133394
O=C(NCC(F)=C1CN(C(=O)CCCF)C1)c1cc(O)no1 s275592__15865378__15841170__14133398
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15841170__14133400
Cc1cocc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133402
C[C@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133404
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C=CCC1 s275592__15865378__15841170__14133406
CN1C(=O)CC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133410
Cn1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14133412
CC1(C)CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133414
O=C(NCC(F)=C1CN(C(=O)c2cccc3[nH]c(=O)[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__14134872
O=C(NCC(F)=C1CN(C(=O)c2ccn3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134876
O=C(NCC(F)=C1CN(C(=O)COCC2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134878
CCc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__14134880
O=C(NCC(F)=C1CN(C(=O)c2nccc3cccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134882
O=C(NCC(F)=C1CN(C(=O)Cc2cnn3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134886
O=C(NCC(F)=C1CN(C(=O)CC=Cc2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14134888
O=C(NCC(F)=C1CN(C(=O)c2cnc(C3CC3)o2)C1)c1cc(O)no1 s275592__15865378__15841170__14134890
O=C1NC(=O)[C@H](CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__14134892
COCc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134898
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134900
C#CCN1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134902
Cc1ccncc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134906
C[C@@H]1OCCO[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134914
Cn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15841170__14134916
CCc1cnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__14134918
O=C(NCC(F)=C1CN(C(=O)[C@H]2CC[C@H](C3CCC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134924
O=C(NCC(F)=C1CN(C(=O)Cc2cncc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134926
Cc1ccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnn2c1C s275592__15865378__15841170__14134928
Cn1cnc2cncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c21 s275592__15865378__15841170__14134930
CN1CCCC1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134932
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCNC1=O s275592__15865378__15841170__14134940
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCNC1=O s275592__15865378__15841170__14134944
CC[C@@H]1CCO[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134946
O=C(NCC(F)=C1CN(C(=O)CC=CCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134948
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2c[nH]cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14134954
O=C(NCC(F)=C1CN(C(=O)c2nccc3ccsc23)C1)c1cc(O)no1 s275592__15865378__15841170__14134956
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134958
O=C(NCC(F)=C1CN(C(=O)Cc2cnn3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134960
Cc1cc(C(F)F)oc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134962
O=C(NCC(F)=C1CN(C(=O)C2CCC=CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14134964
Cc1cn(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14134968
O=C(NCC(F)=C1CN(C(=O)C23CCCN(CCC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__14134972
O=C(NCC(F)=C1CN(C(=O)CC=Cc2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14134974
O=C(NCC(F)=C1CN(C(=O)CC=Cc2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14134976
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14134978
COc1ccncc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14134980
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@@H](c3ccccc3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14134982
CC1C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1C1CC1 s275592__15865378__15841170__14134986
Cc1ccnc(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14134988
O=C(NCC(F)=C1CN(C(=O)C2CCC3CCCCN32)C1)c1cc(O)no1 s275592__15865378__15841170__14134990
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc1Cl s275592__15865378__15841170__14134992
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccncc1 s275592__15865378__15841170__14134994
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCNC(=O)C1 s275592__15865378__15841170__14134998
O=C(NCC(F)=C1CN(C(=O)C2CCCC23CC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135000
O=C(NCC(F)=C1CN(C(=O)COCc2cc[nH]c(=O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14135006
Cc1ccc2nc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cn2c1 s275592__15865378__15841170__14135008
O=C(NCC(F)=C1CN(C(=O)CCc2cccc(F)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__14130192
Cc1nn(C)c(C)c1C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130194
O=C(NCC(F)=C1CN(C(=O)COCC2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__14130200
CC(NC(=O)C1CCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130204
C#CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130208
CC(C)(C)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14130210
CC(=O)N[C@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__14130212
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3ccnn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130214
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__14130216
O=C(NCC(F)=C1CN(C(=O)c2ccccc2-n2ccnn2)C1)c1cc(O)no1 s275592__15865378__15841170__14130218
CCOc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14130220
CCn1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14130222
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ccc(F)cc23)C1)c1cc(O)no1 s275592__15865378__15841170__14130224
O=C(NCC(F)=C1CN(C(=O)CCc2cncc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14130226
Cn1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__14130228
COCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130230
Cc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130232
CC(C)CC(C(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130234
O=C(NCC(F)=C1CN(C(=O)CC(F)(F)C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14130236
COC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130240
CC1(C)C(C)(C)C1(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130242
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__14130244
CC(=O)NC(CCC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130246
C=CCCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__14130248
CC1(C)CCCCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130256
Cc1[nH]cnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130258
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCOCC1 s275592__15865378__15841170__14130264
CC(C)Oc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14130272
O=C(NCC(F)=C1CN(C(=O)C2CC23CCOCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130274
CC1(C)CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__14130276
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCOCC1 s275592__15865378__15841170__14130278
Cc1ccc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130280
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(=O)N1 s275592__15865378__15841170__14130282
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C(C)C s275592__15865378__15841170__14130284
Cc1oc2ccccc2c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130286
O=C(NCC(F)=C1CN(C(=O)c2cccc3[nH]c(=O)oc23)C1)c1cc(O)no1 s275592__15865378__15841170__14130292
CC1(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(=O)N1 s275592__15865378__15841170__14130294
CCOc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130296
CC(C)Oc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130298
O=C(NCC(F)=C1CN(C(=O)c2cc3n(c2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14130300
NC(=O)c1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14130302
CC(C)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__14130306
Cc1cccc2c1OC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__14130308
CCC(CC)C(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130310
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2CCC1C2 s275592__15865378__15841170__14130314
O=C(NCC(F)=C1CN(C(=O)C2(CCc3ccccc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14130316
CC(F)(F)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14130318
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCc2ccccc2C1 s275592__15865378__15841170__14130320
CC1C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1c1ccccc1 s275592__15865378__15841170__14130322
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCCC1 s275592__15865378__15841170__14130324
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3=CCCC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14130326
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1CC s275592__15865378__15841170__14130332
COCc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130334
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCS1(=O)=O s275592__15865378__15841170__14130338
O=C1NC(=O)C2(CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C2)N1 s275592__15865378__15841170__14130340
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__14130342
CC(=O)NCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130350
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C(C)(C)C s275592__15865378__15841170__14130352
CC(Cc1ccco1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14130354
CC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133416
Cc1cnn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133420
CC(C)C(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133422
CCCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14133424
C=CC(C)C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133426
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__14133428
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__14133430
CC#CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133432
O=C(NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3COC[C@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__14133434
O=C(NCC(F)=C1CN(C(=O)CCCC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133436
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__14133438
CCCC(OCC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133440
CC1(C)CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133442
Cc1coc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14133444
O=C(NCC(F)=C1CN(C(=O)c2csc(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14133446
C=CC(CC)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133450
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__14133452
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3C[C@@H]3C2)C1)c1cc(O)no1 s275592__15865378__15841170__14133454
Cc1noc(C)c1C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133458
CCCc1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133460
CC(C)c1[nH]ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133462
Cc1nc[nH]c(=O)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133464
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(=O)NC1 s275592__15865378__15841170__14133466
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1C(C)C s275592__15865378__15841170__14133470
CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14133476
O=C(NCC(F)=C1CN(C(=O)C2CCCc3cccnc32)C1)c1cc(O)no1 s275592__15865378__15841170__14133478
CCCN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133480
O=C(NCC(F)=C1CN(C(=O)C2(c3cccnc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133482
CCOC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133484
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)s1 s275592__15865378__15841170__14133488
O=C(NCC(F)=C1CN(C(=O)Cc2cnoc2)C1)c1cc(O)no1 s275592__15865378__15841170__14133490
CN1C(=O)CC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133492
Cc1cc(C)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__14133494
CC1(C)CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133496
O=C(NCC(F)=C1CN(C(=O)c2cn[nH]c2C2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__14133498
CC(C)c1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133502
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)CC(F)(F)F s275592__15865378__15841170__14133504
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14133508
O=C(NCC(F)=C1CN(C(=O)c2cncc3sccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133510
CC(C)N1C(=O)CC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133512
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133516
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133518
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cncnc1 s275592__15865378__15841170__14133520
CC1Cc2cn[nH]c2C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133524
CC(=O)N[C@H](CC1CCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133526
Cc1ccc2ncn(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__14133528
Cc1cc(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2)on1 s275592__15865378__15841170__14133530
O=C(NCC(F)=C1CN(C(=O)Cc2c[nH]c3cnccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14133532
CC(C)N1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__14133534
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(=O)[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133536
O=C(NCC(F)=C1CN(C(=O)C2C3C4CC5C6C4CC3C6C52)C1)c1cc(O)no1 s275592__15865378__15841170__14133540
O=C(NCC(F)=C1CN(C(=O)C2(F)CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133542
COc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__14133544
O=C(NCC(F)=C1CN(C(=O)c2nc(Cl)cs2)C1)c1cc(O)no1 s275592__15865378__15841170__14133546
O=C(NCC(F)=C1CN(C(=O)CC2CCCC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14133548
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccncc1 s275592__15865378__15841170__14133550
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1C s275592__15865378__15841170__14133554
Cn1ncc2c1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__14133556
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__14133564
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccc(F)cc32)C1)c1cc(O)no1 s275592__15865378__15841170__14133568
Cn1nnc2c1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__14133570
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]c(=O)[nH]c3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14133572
Cn1cc2c(n1)CCCC2C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14133574
CCCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15841170__14133576
O=C(NCC(F)=C1CN(C(=O)c2ccoc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__14133578
O=C(NCC(F)=C1CN(C(=O)c2coc(C(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__14133580
CC1CCn2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nc2C1 s275592__15865378__15841170__14135018
CC(C)(CN1CCOCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135020
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CS(=O)(=O)C3)C1)c1cc(O)no1 s275592__15865378__15841170__14135022
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)F)ncn2)C1)c1cc(O)no1 s275592__15865378__15841170__14135024
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccsc2)C1)c1cc(O)no1 s275592__15865378__15841170__14135026
Cc1nc2sccn2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135028
Cc1cn2c(n1)CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__14135030
COc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__14135032
O=C(NCC(F)=C1CN(C(=O)Cc2cccc3cnccc23)C1)c1cc(O)no1 s275592__15865378__15841170__14135034
O=C(NCC(F)=C1CN(C(=O)c2cn3c(n2)COCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135036
NC(=O)c1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14135038
COCc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135042
CCC1CCCC1(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135044
O=C(NCC(F)=C1CN(C(=O)c2cc3cnccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__14135046
Cc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)s1 s275592__15865378__15841170__14135052
Cn1nnc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc21 s275592__15865378__15841170__14135054
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__14135056
O=C(NCC(F)=C1CN(C(=O)C2CCCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__14135058
O=C(NCC(F)=C1CN(C(=O)c2cc3sccc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__14135060
COc1cc(OC)nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__14135062
O=C(NCC(F)=C1CN(C(=O)C23CCC(CC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__14135064
CN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135066
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__14135068
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3cnco3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__14135070
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__14135072
O=C(NCC(F)=C1CN(C(=O)c2ccnn2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__14135074
O=C(NCC(F)=C1CN(C(=O)C2(C(F)(F)F)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135076
O=C(NCC(F)=C1CN(C(=O)c2ncc(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__14135078
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)S(C)(=O)=O s275592__15865378__15841170__14135080
CS(=O)(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135082
COCCS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135086
CC(C)CS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135088
O=C(NCC(F)=C1CN(C(=O)Cc2cn3ccccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__14135092
O=C(NCC(F)=C1CN(C(=O)Cc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__14135094
O=C(NCC(F)=C1CN(C(=O)c2cnc3ccccn3c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14135096
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__14135100
NC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__14135102
CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__14135104
C=CCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__14135106
C=CCOc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135108
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15841170__14135110
CC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__14135112
CC(=O)NCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135114
Cc1[nH]c2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc2c1C s275592__15865378__15841170__14135116
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc2ccccc12 s275592__15865378__15841170__14135118
CC(F)(F)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135120
O=C(NCC(F)=C1CN(C(=O)COC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__14135126
O=C(NCC(F)=C1CN(C(=O)CCOCC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__14135128
O=C(NCC(F)=C1CN(C(=O)CCOCC2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__14135132
O=C(NCC(F)=C1CN(C(=O)CCc2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__14135138
CC(C)(C)n1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14135140
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15841170__14135142
CC(C)CN1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135146
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__14135148
CN(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__14135150
CCCc1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135154
CCc1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135156
CC(C)c1[nH]ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__14135158
CC(C)(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__14135160
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ccccc3c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14135162
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135164
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccccc3)no2)C1)c1cc(O)no1 s275592__15865378__15841170__14135166
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__14135168
O=C(NCC(F)=C1CN(C(=O)c2cn(-c3ccccc3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14135170
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nn2)C1)c1cc(O)no1 s275592__15865378__15841170__14135174
O=C(NCC(F)=C1CN(C(=O)CCc2n[nH]c(=O)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__14135176
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__15278136
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1 s275592__15865378__15841170__15585620
NC(=O)NC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15855920
Cc1sc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__15855922
Cc1nc([N+](=O)[O-])cn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855924
N#CCOc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855926
Cc1cccc2[nH]cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c12 s275592__15865378__15841170__15855928
O=C(NCC(F)=C1CN(C(=O)CN2CCC(CO)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855930
O=C(NCC(F)=C1CN(C(=O)c2ccccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15855932
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c([N+](=O)[O-])c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855934
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cccc1[N+](=O)[O-] s275592__15865378__15841170__15855936
O=C(NCC(F)=C1CN(C(=O)c2ccc(NC3CC3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855938
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15855940
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1Cl s275592__15865378__15841170__15855944
O=C(NCC(F)=C1CN(C(=O)CSc2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855950
CC(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15855952
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__15855954
O=C(NCC(F)=C1CN(C(=O)c2nc3ccccc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__15855956
O=C(NCC(F)=C1CN(C(=O)CSc2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855958
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]cnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855960
O=C(NCC(F)=C1CN(C(=O)C2CSCCS2)C1)c1cc(O)no1 s275592__15865378__15841170__15855966
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)ccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15855968
O=C(NCC(F)=C1CN(C(=O)c2cccc(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855974
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)ccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15855976
CCOC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855978
O=C(NCC(F)=C1CN(C(=O)COc2ccccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15855980
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15855984
NC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855986
Nc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855988
Nc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__15855990
O=C(NCC(F)=C1CN(C(=O)c2ccc[n+]([O-])c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855992
CNc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855994
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15855996
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cc(Cl)cn1 s275592__15865378__15841170__15855998
C=CCCCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856002
COC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856004
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ncn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856006
C#CCSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856008
O=C(NCC(F)=C1CN(C(=O)CSCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856012
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2NCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15857750
CCn1cc(C(F)(F)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15857754
CSC=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857758
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2OCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15857760
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1Cl s275592__15865378__15841170__15857762
CN1C2CCC1CC(=CC(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15857770
O=C(NCC(F)=C1CN(C(=O)c2cnccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857774
CC1=NC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CS1 s275592__15865378__15841170__15857776
O=C(NCC(F)=C1CN(C(=O)C(=O)C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15857778
CCC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857780
Cc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__15857782
O=C(NCC(F)=C1CN(C(=O)C2(CO)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857784
Cc1ccc(C#N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857788
Nc1ccn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857790
O=C(CCc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857792
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc1N s275592__15865378__15841170__15857794
N#Cc1cc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857796
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857798
Cn1ccnc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857800
CC(C)(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)[N+](=O)[O-] s275592__15865378__15841170__15857802
CN1C(=O)CSC1=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857804
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CC(F)(F)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15857806
Nc1c(F)cc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857808
COC1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857810
CC1C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCN1C s275592__15865378__15841170__15857814
O=C(NCC(F)=C1CN(C(=O)c2cncc(O)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15857816
N#CC(CCc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857818
CN1CCCCC1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857822
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)s2)C1)c1cc(O)no1 s275592__15865378__15841170__15857824
CCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15857826
NC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857828
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857832
O=C(NCC(F)=C1CN(C(=O)COC(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15857834
COc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1O s275592__15865378__15841170__15857836
O=C(NCC(F)=C1CN(C(=O)CC2COc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15857842
Cc1c(C#N)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857844
COC(=Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857846
Cc1nc(=O)[nH]c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857850
CC(C)(C)OC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15857852
Cc1nc2cccnn2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857856
[N-]=[N+]=NCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15857862
CCC(CC)(CC(=O)OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857864
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(=O)N1 s275592__15865378__15841170__15857868
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1Cl s275592__15865378__15841170__15857870
O=C(NCC(F)=C1CN(C(=O)C(=O)c2ccc(Cl)s2)C1)c1cc(O)no1 s275592__15865378__15841170__15857872
Cc1csc(NCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859740
CCOC(=O)NCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859742
O=C(NCC(F)=C1CN(C(=O)CSCc2ncc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15859744
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCSCC1 s275592__15865378__15841170__15859748
O=C(NCC(F)=C1CN(C(=O)C2=CCCS2)C1)c1cc(O)no1 s275592__15865378__15841170__15859750
CC1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859752
O=C(NC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859754
CC(C)Nc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859756
CCn1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859758
O=C(NCC(F)=C1CN(C(=O)c2ncc(Cl)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15859760
CCC1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859762
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccoc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859766
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__15859768
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)(c2ccccc2)C1 s275592__15865378__15841170__15859770
Cc1noc(COCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859772
O=C(NCC(F)=C1CN(C(=O)C2CCSC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859774
O=C(NCC(F)=C1CN(C(=O)C2CCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15859778
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1C s275592__15865378__15841170__15859780
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(Cl)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15859782
CCNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15859784
Nc1nc2c(cc1C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CCC2 s275592__15865378__15841170__15859786
O=C(NCC(F)=C1CN(C(=O)C=CC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859790
CC(O)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(F)c1 s275592__15865378__15841170__15859792
CCCC(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859794
Cn1ncc([N+](=O)[O-])c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859798
O=C(NCC(F)=C1CN(C(=O)CC2CNc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15859800
O=C(NCC(F)=C1CN(C(=O)C2CSc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15859802
CC(O)(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859804
CC(C)(CC#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859806
O=C(NCC(F)=C1CN(C(=O)C2(Cl)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859808
O=C(NCC(F)=C1CN(C(=O)C2=CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15859810
O=C(NCC(F)=C1CN(C(=O)C2(O)Cc3ccccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15859812
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)o2)C1)c1cc(O)no1 s275592__15865378__15841170__15859816
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1O s275592__15865378__15841170__15859822
O=C(NCC(F)=C1CN(C(=O)C2CCC(C3CCCO3)O2)C1)c1cc(O)no1 s275592__15865378__15841170__15859824
COc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859828
O=C(NCC(F)=C1CN(C(=O)C2(CO)COC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859830
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15859832
CC1CC(C#N)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859834
CC(C)=CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859836
CC=C(C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CC s275592__15865378__15841170__15859838
O=C(NCC(F)=C1CN(C(=O)C2COC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859842
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)n1 s275592__15865378__15841170__15859846
O=C(NCC(F)=C1CN(C(=O)C=CC2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859850
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859852
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859854
O=C(NCC(F)=C1CN(C(=O)C23CCC(F)(CC2)CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15859856
N#CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15859858
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(C3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15859860
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15859862
CNc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15859864
Cc1nccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861706
O=C(NCC(F)=C1CN(C(=O)c2cnc(F)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15861708
O=C(NCC(F)=C1CN(C(=O)c2ccnc(F)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15861710
O=C(NCC(F)=C1CN(C(=O)[C@H](O)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861712
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccc3c2OCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15861714
Cc1ccc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15861716
Nc1nc2ccccc2cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861718
Nc1c[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861720
COC(=O)c1ccn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861722
COc1c(F)ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15861724
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1O s275592__15865378__15841170__15861728
O=C(NCC(F)=C1CN(C(=O)c2cccc([N+](=O)[O-])c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15861734
O=C(NCC(F)=C1CN(C(=O)COc2ccc(O)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861736
CC1(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15861738
O=C(NCC(F)=C1CN(C(=O)C2CCOC3(CCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15861746
CC(C)(C)OC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861748
O=C(NCC(F)=C1CN(C(=O)c2cc([N+](=O)[O-])[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__15861750
O=C(NCC(F)=C1CN(C(=O)c2cc3ccsc3s2)C1)c1cc(O)no1 s275592__15865378__15841170__15861752
O=C(NCC(F)=C1CN(C(=O)C=CCO)C1)c1cc(O)no1 s275592__15865378__15841170__15861754
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n2c1CCCC2 s275592__15865378__15841170__15861756
CCC(O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861758
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(N)c1N s275592__15865378__15841170__15861760
O=C(NCC(F)=C1CN(C(=O)C2CCCc3ncnn32)C1)c1cc(O)no1 s275592__15865378__15841170__15861762
O=C(NCC(F)=C1CN(C(=O)C2(CO)CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15861764
O=C(NCC(F)=C1CN(C(=O)c2cnc(O)c3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861768
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3nc[nH]c(=O)c23)C1)c1cc(O)no1 s275592__15865378__15841170__15861770
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cc(F)cc(F)c1 s275592__15865378__15841170__15861776
CC(C)(OCC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861780
COc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861782
Cn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1=O s275592__15865378__15841170__15861786
C=CC1(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CCC2)CCC1 s275592__15865378__15841170__15861788
COc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15861794
CC(C)(C)c1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15861796
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15861798
[N-]=[N+]=NCC(F)(F)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861800
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(F)(F)C1 s275592__15865378__15841170__15861802
CCc1c[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861804
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCC[C@H]2CF)C1)c1cc(O)no1 s275592__15865378__15841170__15861806
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CCC3)on2)C1)c1cc(O)no1 s275592__15865378__15841170__15861810
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCC[C@H]2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15861812
CC(C)[C@@H](O)[C@@H](C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861816
O=C(NCC(F)=C1CN(C(=O)C2(F)C3CCCCC32)C1)c1cc(O)no1 s275592__15865378__15841170__15861818
O=C(NCC(F)=C1CN(C(=O)c2onc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861820
CC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CC1)CO2 s275592__15865378__15841170__15861822
CCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__15861824
O=C(NCC(F)=C1CN(C(=O)Cn2cc(C3CCC3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15861826
O=C(C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15863540
CC(C)(Cc1cnn[nH]1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863542
O=C(NCC(F)=C1CN(C(=O)C2(C(=O)C3CC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863548
O=CN1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863550
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__15863554
CC(C)(C)N1CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863556
O=C(NCC(F)=C1CN(C(=O)CCC2CC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863560
O=C(NCC(F)=C1CN(C(=O)CCCC(=O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863562
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cnc(C#N)n1 s275592__15865378__15841170__15863564
Cc1c(F)ccc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863566
Nc1ccn(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863568
Cc1nnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15863572
C[C@@H](Oc1ccc(O)cc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863574
Cc1cnnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863576
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__15863578
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cccc1 s275592__15865378__15841170__15863580
CSCC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15863582
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__15863584
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863586
O=C(NCC(F)=C1CN(C(=O)c2ncccc2OC(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863588
O=C(NCC(F)=C1CN(C(=O)c2nc3c(s2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863590
CC(C)(C)OC(=O)COCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863592
CCn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc1O s275592__15865378__15841170__15863594
O=C(NCC(F)=C1CN(C(=O)c2coc(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15863596
CC=CC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863598
O=C(NCC(F)=C1CN(C(=O)c2cc3cccnc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15863602
CCCC[C@H](C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863606
N#Cc1ccn2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc2n1 s275592__15865378__15841170__15863608
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15863610
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__15863612
O=C(NCC(F)=C1CN(C(=O)c2noc3cc(F)ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863614
COC(=O)c1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863616
CCC=C(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863618
O=C(NCC(F)=C1CN(C(=O)C2C3(CC3)C23CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863620
CCC=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863622
Cn1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15863624
CCC(F)(F)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863628
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15863630
[N-]=[N+]=NCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863632
O=C(NCC(F)=C1CN(C(=O)c2noc3ccc(F)cc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863634
Cc1nocc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863636
Cc1nc2cncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2[nH]1 s275592__15865378__15841170__15863638
O=C(NCC(F)=C1CN(C(=O)Cc2csnn2)C1)c1cc(O)no1 s275592__15865378__15841170__15863642
CC(=Cc1cccnc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863644
O=C(NCC(F)=C1CN(C(=O)CC(F)(F)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15863646
CC(C)c1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15863650
O=C(NCC(F)=C1CN(C(=O)C2(c3ncccc3F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863654
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15863656
COCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__15863658
CN(C)Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15863660
O=C1N[C@@H](CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15863662
CC(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15864230
COc1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1OC s275592__15865378__15841170__15864232
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc1C#N s275592__15865378__15841170__15864234
CCc1cn2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc2n1 s275592__15865378__15841170__15864236
C=CCC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__15864238
CC1CCOC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864240
O=C(NCC(F)=C1CN(C(=O)c2cncc3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15864242
O=C(NCC(F)=C1CN(C(=O)C2=C(Cl)CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864244
Nc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856020
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15841170__15856024
CC1CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15856026
CC(Sc1ncccn1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856030
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(=O)OC1(C)C s275592__15865378__15841170__15856034
CC(SCC1CCCO1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856036
CCCCSC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856038
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc2cccnc12 s275592__15865378__15841170__15856040
NS(=O)(=O)c1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856042
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15856044
CC(=O)CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856046
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3N2)C1)c1cc(O)no1 s275592__15865378__15841170__15856050
Nc1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856052
COC(=O)NC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856054
CCc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856058
Nc1nonc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856062
O=C(NCC(F)=C1CN(C(=O)c2cn(CCO)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856064
O=C(NCC(F)=C1CN(C(=O)COC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15856066
Cc1ccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c[nH]c2c1 s275592__15865378__15841170__15856068
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3cc(F)ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15856070
O=C1NC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15856072
CC(C)Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856074
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1F s275592__15865378__15841170__15856076
O=C(NCC(F)=C1CN(C(=O)c2cncs2)C1)c1cc(O)no1 s275592__15865378__15841170__15856078
O=C(NCC(F)=C1CN(C(=O)CNc2cccc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856080
O=C(NCC(F)=C1CN(C(=O)CNc2ccccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15856082
Nc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856084
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc2ccccc12 s275592__15865378__15841170__15856090
Cc1nc(N)[nH]c(=O)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856092
COC(=O)C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856094
Cc1nn(CCO)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856096
O=C(NCC(F)=C1CN(C(=O)CCN2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856100
CCCC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856102
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1C#N s275592__15865378__15841170__15856104
Cc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856106
O=C(NCC(F)=C1CN(C(=O)c2c(O)cc(O)cc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856108
[N-]=[N+]=NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856110
O=C(NCC(F)=C1CN(C(=O)Cn2cc(CO)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856114
C#CCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856116
O=C(NCC(F)=C1CN(C(=O)Cc2nnco2)C1)c1cc(O)no1 s275592__15865378__15841170__15856118
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)SCCO1 s275592__15865378__15841170__15856120
CN(CCO)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856124
O=C(NCC(F)=C1CN(C(=O)c2cnc(Cl)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856126
O=C(NCC(F)=C1CN(C(=O)C2CCCS2)C1)c1cc(O)no1 s275592__15865378__15841170__15856128
CCCC(O)(CCC)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856130
COC(=O)CC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856132
O=C(NCC(F)=C1CN(C(=O)c2cccc(O)c2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15856134
COC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857874
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2nccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15857878
Cc1cc(F)c(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857880
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3ncccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857882
O=C(NCC(F)=C1CN(C(=O)CC2CCCC(O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15857884
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857886
CC(O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857888
CC1(C)CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__15857894
N#Cc1ccn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__15857896
Cn1cccc1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857900
CCS(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857902
Cc1n[nH]c(C)c1SCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857904
CC(=O)c1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857906
NC(=O)NCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857908
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857910
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1[N+](=O)[O-] s275592__15865378__15841170__15857912
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15857914
O=C(NCC(F)=C1CN(C(=O)CNC(=O)C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15857916
NC1=NC(=O)C(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)S1 s275592__15865378__15841170__15857920
O=C(NCC(F)=C1CN(C(=O)C2=NN(CCO)C(=O)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857926
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15857932
O=C(NCC(F)=C1CN(C(=O)COCC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15857934
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15841170__15857936
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15841170__15857938
NC(=O)CSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857940
CCCCSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857942
Nc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857944
Cc1ccc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15857946
O=C(NCC(F)=C1CN(C(=O)C2CC(=O)c3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15857948
O=C(NCC(F)=C1CN(C(=O)c2c(F)cc(O)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857950
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15857952
CC(C)CSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857954
CC(=O)N1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857958
O=C(NCC(F)=C1CN(C(=O)c2cc(=O)[nH]c(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15857960
Nc1nc(C2CC2)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15857962
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccnc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857964
O=C(NCC(F)=C1CN(C(=O)c2coc3cccc(O)c23)C1)c1cc(O)no1 s275592__15865378__15841170__15857966
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)cc1N s275592__15865378__15841170__15857968
O=C(NCC(F)=C1CN(C(=O)c2cnc(Cl)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857970
O=C(NCC(F)=C1CN(C(=O)C2CN3CCCN2CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15857974
COC(=O)c1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857976
O=C(NCC(F)=C1CN(C(=O)CC(O)c2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857978
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__15857980
O=C(NCC(F)=C1CN(C(=O)Cn2cccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857988
CCC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(C)cc1 s275592__15865378__15841170__15857990
O=C(NCC(F)=C1CN(C(=O)c2c(Cl)ccnc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857996
O=C(NCC(F)=C1CN(C(=O)C2CCCCS2)C1)c1cc(O)no1 s275592__15865378__15841170__15859866
O=C(NCC(F)=C1CN(C(=O)C2SCCS2)C1)c1cc(O)no1 s275592__15865378__15841170__15859868
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15859870
CC1=NOC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859874
O=C(NCC(F)=C1CN(C(=O)c2csc(NC3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15859876
Nc1c(F)ccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859880
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15859884
O=C(NCC(F)=C1CN(C(=O)c2ccn(CO)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15859886
Nc1nc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15859890
O=C(NCC(F)=C1CN(C(=O)c2cccc3ncoc23)C1)c1cc(O)no1 s275592__15865378__15841170__15859896
O=C(NCC(F)=C1CN(C(=O)CSCc2cscn2)C1)c1cc(O)no1 s275592__15865378__15841170__15859898
C#CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859904
CC(=NO)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__15859906
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__15859912
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1CO s275592__15865378__15841170__15859914
O=C(NCC(F)=C1CN(C(=O)c2cc(O)cc(=O)o2)C1)c1cc(O)no1 s275592__15865378__15841170__15859916
COC(=O)c1cn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__15859920
Nc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15859924
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)B(O)OC3)C1)c1cc(O)no1 s275592__15865378__15841170__15859926
CC(Cc1ccc(N)cc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859928
Cc1c(F)ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15859932
COc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859934
O=C(NCC(F)=C1CN(C(=O)C(O)CC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859936
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15859938
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCSCC1 s275592__15865378__15841170__15859942
CC(C)(C#N)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15859944
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15859946
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCC(C3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15859952
N#Cc1c(F)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859954
O=C(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccnc1 s275592__15865378__15841170__15859958
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)ncc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15859960
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15859962
CC(C)(C)SCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859964
Nc1cccc([N+](=O)[O-])c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859966
Cc1nc(N)nc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859970
O=C(NCC(F)=C1CN(C(=O)C2(O)CCSCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859972
O=C(NCC(F)=C1CN(C(=O)c2coc3c2C(=O)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15859974
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)[nH]c1=O s275592__15865378__15841170__15859980
O=C(NCC(F)=C1CN(C(=O)Cn2cnc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15859986
CC(C)OC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859988
COc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861828
O=C(NCC(F)=C1CN(C(=O)C2C[C@H]3[C@@H](C2)C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15861830
CC1(C)CC(O)(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15861832
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1C(F)(F)F s275592__15865378__15841170__15861834
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ncnc(O)c23)C1)c1cc(O)no1 s275592__15865378__15841170__15861836
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@H]3C[C@@H]2CO3)C1)c1cc(O)no1 s275592__15865378__15841170__15861838
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2n1CCCC2 s275592__15865378__15841170__15861840
COC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15861842
O=C(NCC(F)=C1CN(C(=O)C2CNc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15861846
Cc1cc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2o1 s275592__15865378__15841170__15861848
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC12CCC2 s275592__15865378__15841170__15861850
CNc1c(N)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861852
Cn1ncc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861854
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCCO3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861858
O=C(NCC(F)=C1CN(C(=O)Cn2ncc(=O)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15861860
C#Cc1cccc(NC(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861862
O=C(NCC(F)=C1CN(C(=O)CC2CC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15861866
O=C(NCC(F)=C1CN(C(=O)CC2C=CS(=O)(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15861868
COc1cnnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861870
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)nc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15861874
CC(Cn1ccnc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861876
O=C(NCC(F)=C1CN(C(=O)CSCCC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15861878
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccc3[nH]ncc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861880
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1CCO s275592__15865378__15841170__15861884
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ncn2)C1)c1cc(O)no1 s275592__15865378__15841170__15861886
CC(C)(C)OCCOCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861888
CCCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861890
O=C(NCC(F)=C1CN(C(=O)c2coc3ccc(O)cc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861892
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1F s275592__15865378__15841170__15861896
Cc1cccn2c(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc12 s275592__15865378__15841170__15861900
COc1c(Cl)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861902
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15861904
CN1CC=C(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15861906
CC[C@H](C)[C@H](O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861908
Cc1ncn(C)c(=O)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861912
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15841170__15861914
CC(C)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841170__15861920
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCO[C@H]2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15861922
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(F)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861926
CC(C)CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15861928
O=C(NCC(F)=C1CN(C(=O)CCC(O)C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15861930
O=C(NCC(F)=C1CN(C(=O)CCc2n[nH]c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861932
Cn1cnc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861936
Cc1cc(C2CC2)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861938
O=C(NCC(F)=C1CN(C(=O)Cc2n[nH]c(C3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15861940
CC1(C)CC1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861942
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15861944
O=C(NCC(F)=C1CN(C(=O)C2CCS2(=O)=O)C1)c1cc(O)no1 s275592__15865378__15841170__15861946
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CC(C)(C)C(O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864254
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O=C(NCC(F)=C1CN(C(=O)C(O)c2c[nH]cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15864266
O=C(NCC(F)=C1CN(C(=O)C=CC=C(Cl)Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15864272
CCC(C)(C)C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864274
CCC(C)(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864276
Nc1ncc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864278
O=C(NCC(F)=C1CN(C(=O)CN2CCn3ccnc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864280
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O=C(NCC(F)=C1CN(C(=O)CC2CCC3(CCC3)O2)C1)c1cc(O)no1 s275592__15865378__15841170__15864286
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Nc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15864294
C#CC1CC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15864296
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(CO)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15864298
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CSc1ccc(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864304
CSc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15864306
COc1cnnc(OC)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864308
CC=CC=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864312
CN1CC(O)CC1(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864316
COCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15864318
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCCC3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15864320
C[C@@H]1[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[C@@H](O)C(=O)N1C s275592__15865378__15841170__15864324
O=C(NCC(F)=C1CN(C(=O)C=CSc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15864326
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CS(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864332
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864334
O=C(NCC(F)=C1CN(C(=O)c2ccc(CC3CCC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15864336
O=C(NCC(F)=C1CN(C(=O)c2cc3c(=O)[nH]ccn3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15864338
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(C)(C)O1 s275592__15865378__15841170__15864340
Cn1c(Cl)cnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864342
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC=CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864344
COCC=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864348
Cc1cc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2s1 s275592__15865378__15841170__15864352
CN1CCN(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15864354
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCCC(O)C1 s275592__15865378__15841170__15864356
O=C(NCC(F)=C1CN(C(=O)c2cccc3nonc23)C1)c1cc(O)no1 s275592__15865378__15841170__15864358
O=C(NCC(F)=C1CN(C(=O)CCOC2COC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864360
[N-]=[N+]=N[C@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15864362
CC(=O)C(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864364
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccncc3)no2)C1)c1cc(O)no1 s275592__15865378__15841170__15864366
Cc1ccc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856136
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15856138
O=C(NCC(F)=C1CN(C(=O)C2CC3CC3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15856140
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCC3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15856148
CCC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856150
O=C(NCC(F)=C1CN(C(=O)CSc2ccc(O)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856152
Cc1cc([N+](=O)[O-])cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15856156
O=C(NCC(F)=C1CN(C(=O)Cc2cncnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856158
Cc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15856160
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)cc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15856162
CCOC(=O)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856166
O=C(NCC(F)=C1CN(C(=O)CCc2nc(=O)[nH][nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15856168
O=C1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856170
O=C(NCC(F)=C1CN(C(=O)C2C3CCC(=O)C32)C1)c1cc(O)no1 s275592__15865378__15841170__15856176
COC(=O)C12CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(C1)C2 s275592__15865378__15841170__15856182
O=C(NCC(F)=C1CN(C(=O)c2cc3[nH]nnc3cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15856184
Cc1ccncc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856186
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15856188
CNc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15856190
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(Cl)n1 s275592__15865378__15841170__15856192
CS(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856194
O=C(NCC(F)=C1CN(C(=O)C(=O)C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856196
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)n1 s275592__15865378__15841170__15856198
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cnn(C)c1 s275592__15865378__15841170__15856202
CCOC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15856204
Nc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15856208
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15856210
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc2ccnn12 s275592__15865378__15841170__15856212
Nc1ncc2c(c1C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CCC2 s275592__15865378__15841170__15856214
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)C(=O)OC3)C1)c1cc(O)no1 s275592__15865378__15841170__15856216
O=C(NCC(F)=C1CN(C(=O)C2=C(c3ccccc3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856220
O=NN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856224
O=C(NCC(F)=C1CN(C(=O)C=C(Cl)Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15856226
CSc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15856230
O=C(NCC(F)=C1CN(C(=O)c2cnncc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856232
CN1CCCC(O)(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15856236
Cc1[nH]c(C#N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856238
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__15856240
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1C s275592__15865378__15841170__15856242
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(C)(C)C1 s275592__15865378__15841170__15856244
O=C(NCC(F)=C1CN(C(=O)C2(c3ccc(O)cc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856246
CC(F)(F)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15856248
CC1CN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15856250
Nc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__15856252
O=C(NCC(F)=C1CN(C(=O)c2nc3cc(O)ccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15856256
CCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857998
COc1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858000
Cc1cccc(O)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858002
O=C(NCC(F)=C1CN(C(=O)c2cccc(F)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858004
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858006
CCN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15858008
O=C(Cc1ccc(F)cc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858012
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3cccc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15858018
O=C(NCC(F)=C1CN(C(=O)CNc2ccc(Cl)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15858020
Cc1nn(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1[N+](=O)[O-] s275592__15865378__15841170__15858026
CC1CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15858032
CC(OC1CCCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858036
CN(C)C(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858038
C#CCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858040
O=C(NCC(F)=C1CN(C(=O)c2cncc(Cl)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858042
Nc1ncccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858044
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC12CCCC2 s275592__15865378__15841170__15858046
O=C(NCC(F)=C1CN(C(=O)c2ccc(OC3CC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858050
O=C(NCC(F)=C1CN(C(=O)c2cc(O)cc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858052
O=C(NCC(F)=C1CN(C(=O)Cn2ncc3ncccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15858054
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)S(C)(=O)=O s275592__15865378__15841170__15858056
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15858058
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC(O)CC1 s275592__15865378__15841170__15858060
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC(C)(O)CC1 s275592__15865378__15841170__15858062
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15858064
C=CC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858068
[N-]=[N+]=NCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858070
Cc1ccc(C)n1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858072
Cc1cccnc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858074
CC(O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858076
O=C(NCC(F)=C1CN(C(=O)C2CCCN2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858078
CC1(C)COC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858080
CSCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858082
Cc1c(N)ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__15858084
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(Cl)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15858086
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15858088
Cn1nncc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858092
O=C(NCC(F)=C1CN(C(=O)Cc2cnccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858096
O=C(NCC(F)=C1CN(C(=O)CCCc2cncs2)C1)c1cc(O)no1 s275592__15865378__15841170__15858098
[N-]=[N+]=Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858100
[N-]=[N+]=Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858102
[N-]=[N+]=Nc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858104
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__15858106
O=C(NCC(F)=C1CN(C(=O)c2cc3[nH]cnc3cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15858108
COC(=O)COCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858110
O=C(NCC(F)=C1CN(C(=O)CC2CCCCC2F)C1)c1cc(O)no1 s275592__15865378__15841170__15858112
N#Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15858114
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15858116
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)COB3O)C1)c1cc(O)no1 s275592__15865378__15841170__15858118
O=C(NCC(F)=C1CN(C(=O)c2cccc3ccc(O)nc23)C1)c1cc(O)no1 s275592__15865378__15841170__15858120
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCO1 s275592__15865378__15841170__15859990
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15859994
O=C(NCC(F)=C1CN(C(=O)c2ccc(N3CCC3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15859996
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__15859998
CCC(CC)(CO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860000
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15860002
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15860004
CSc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860006
Cc1ccc(NCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15860008
Cc1ccc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860010
O=C(NCC(F)=C1CN(C(=O)C2CCC3CC3CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860022
O=C(NCC(F)=C1CN(C(=O)c2cccn3ncnc23)C1)c1cc(O)no1 s275592__15865378__15841170__15860024
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860026
COc1cc(N)c(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860030
[N-]=[N+]=NCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860032
CC1(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N=N1 s275592__15865378__15841170__15860034
Nc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860038
O=C(NCC(F)=C1CN(C(=O)C2CC3CC2C2C3C2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860040
O=C(NCC(F)=C1CN(C(=O)C23CCC2C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860044
CCCC(C)=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860050
O=C(NCC(F)=C1CN(C(=O)c2cccc(C#CCO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860052
Cc1cc(C)c(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1 s275592__15865378__15841170__15860054
O=C(NCC(F)=C1CN(C(=O)c2nc(C3CC3)cs2)C1)c1cc(O)no1 s275592__15865378__15841170__15860056
O=C(NCC(F)=C1CN(C(=O)C(=O)C2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860058
C=C[C@H](C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860060
COC(=O)[C@@H]1CCCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860062
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CCC3)[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__15860064
O=C(NCC(F)=C1CN(C(=O)c2noc3c(F)cccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15860066
CCc1nn(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__15860068
O=C(NCC(F)=C1CN(C(=O)C2CCc3ccccc3N2)C1)c1cc(O)no1 s275592__15865378__15841170__15860072
CS(=O)(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860076
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)NCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860080
O=C(NCC(F)=C1CN(C(=O)c2ccn3nccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15860082
O=C(NCC(F)=C1CN(C(=O)C=CCN2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860084
O=C(NCC(F)=C1CN(C(=O)c2nocc2-c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15860086
Cn1cc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15860088
O=C(NCC(F)=C1CN(C(=O)C=CC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860092
CCOC(=O)N(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860094
O=C(NCC(F)=C1CN(C(=O)C23CCC(CC2)O3)C1)c1cc(O)no1 s275592__15865378__15841170__15860096
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3ncncc23)C1)c1cc(O)no1 s275592__15865378__15841170__15860100
O=C(NCC(F)=C1CN(C(=O)CCc2cccc(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860102
Cc1cc(C#N)cc(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860104
O=C(NCC(F)=C1CN(C(=O)c2cc3cc(O)ccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15860106
CC(C)(C)c1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860108
N#Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15860110
O=C(NCC(F)=C1CN(C(=O)C=CC2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15861948
O=C(NCC(F)=C1CN(C(=O)C#CC2CCCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15861950
Cc1ccc2cccnc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861952
O=C(NCC(F)=C1CN(C(=O)Cn2cnc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15861958
Cc1oncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861960
O=C(NCC(F)=C1CN(C(=O)C2=Cc3ccccc3OC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861962
COC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15861964
CC(C)CC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861966
O=C(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861968
CCC(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861972
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15861974
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15861976
O=C(NCC(F)=C1CN(C(=O)CCNc2nccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15861980
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)N=S=N3)C1)c1cc(O)no1 s275592__15865378__15841170__15861982
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15861986
CC1CC1(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861988
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1(Cl)Cl s275592__15865378__15841170__15861990
O=C(NCC(F)=C1CN(C(=O)C2CCN(C3CC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861992
CCC(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861996
O=C(NCC(F)=C1CN(C(=O)C2(CO)CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861998
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)S(N)(=O)=O s275592__15865378__15841170__15862000
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15862002
CS(=O)(=O)N1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15862006
NS(=O)(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15862012
O=C(NCC(F)=C1CN(C(=O)c2coc(CO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862014
CC(C)[C@H]1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15862018
O=C1NC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15862020
Cn1cc(NCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15862022
Cn1nnc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15841170__15862024
Cc1onc(CO)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862026
COCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862028
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862030
COc1nscc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862032
Cc1ccc2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2c1 s275592__15865378__15841170__15862036
O=C(NCC(F)=C1CN(C(=O)C23CC2(c2ccccc2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15862038
O=C(NCC(F)=C1CN(C(=O)c2cccc(O)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15862040
CCOCCOCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862046
Nc1nn2ccccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862048
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCC[C@H]2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862050
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(N)c1O s275592__15865378__15841170__15862052
O=C(NCC(F)=C1CN(C(=O)c2cccnc2CO)C1)c1cc(O)no1 s275592__15865378__15841170__15862054
CC1(C)CC2(CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C2)C1 s275592__15865378__15841170__15862056
C=CCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15862060
Cn1ccc(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15862066
O=C(NCC(F)=C1CN(C(=O)C2(n3ccnn3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862070
O=C(NCC(F)=C1CN(C(=O)c2csc3nnsc23)C1)c1cc(O)no1 s275592__15865378__15841170__15864370
[N-]=[N+]=NC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15864374
O=C(NCC(F)=C1CN(C(=O)C23CCC(CO2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15864376
O=C(NCC(F)=C1CN(C(=O)C2C3CCC32)C1)c1cc(O)no1 s275592__15865378__15841170__15864378
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc(Cl)c1O s275592__15865378__15841170__15864380
CC1(C)CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15864382
COC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1C s275592__15865378__15841170__15864384
CC(C)(C)C(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864386
C=C1CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864388
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@H]3CC[C@H]2O3)C1)c1cc(O)no1 s275592__15865378__15841170__15864390
C[C@@H]1C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[C@@H]1C s275592__15865378__15841170__15864392
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15841170__15864394
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CCCC3)n[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15864396
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CCC3)OC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864398
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(F)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15864400
Cc1cn2c(n1)CCC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15864402
O=C(NCC(F)=C1CN(C(=O)c2ccc(CC3CC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15864406
Cc1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15864408
O=C(NCC(F)=C1CN(C(=O)c2ncc(C(F)F)s2)C1)c1cc(O)no1 s275592__15865378__15841170__15864410
Cc1nnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15864412
COc1ccc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15864414
CC(C)n1cncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864416
Cc1cn2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2n1 s275592__15865378__15841170__15864418
C=CCOCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__15864420
Cc1nnc2n1C(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__15864422
CCN(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864424
Nc1cc(O)nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864426
O=C(NCC(F)=C1CN(C(=O)c2ccn3c(=O)[nH]nc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864428
O=C(NCC(F)=C1CN(C(=O)C2CCCC(F)(F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864430
O=C(NCC(F)=C1CN(C(=O)c2cccn3cnnc23)C1)c1cc(O)no1 s275592__15865378__15841170__15864432
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2C=CC1C2 s275592__15865378__15841170__15864434
COC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__15864436
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1nc[nH]n1 s275592__15865378__15841170__15864442
CCOc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15864444
Cc1cc2c(c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c1)OCC2 s275592__15865378__15841170__15864446
O=C(NCC(F)=C1CN(C(=O)c2[nH]ncc2C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864448
O=C(NCC(F)=C1CN(C(=O)C2CCC3C2C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15864450
Cc1nn(C2CCC2)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864454
O=C(NCC(F)=C1CN(C(=O)C(F)OC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15864456
C=C1CC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15864458
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc2ncnn12 s275592__15865378__15841170__15864460
O=C(NCC(F)=C1CN(C(=O)CC2CCn3cncc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864462
Cc1ncc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__15864464
Cn1nncc1C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864466
COc1n[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__15864468
O=C(NCC(F)=C1CN(C(=O)C2=Cc3ccccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864472
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccnc1 s275592__15865378__15841170__15864474
CCC1(C#CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841170__15864476
COc1ccc(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864478
O=C(NCC(F)=C1CN(C(=O)C2=C[C@@H]3CCCC[C@H]23)C1)c1cc(O)no1 s275592__15865378__15841170__15864482
CC1(C)CC1(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864484
CC(C)c1c[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864486
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccc3occc23)C1)c1cc(O)no1 s275592__15865378__15841170__15856262
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)N=N3)C1)c1cc(O)no1 s275592__15865378__15841170__15856264
O=C(NCC(F)=C1CN(C(=O)c2ccnc(-c3ncc[nH]3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856272
O=C(NCC(F)=C1CN(C(=O)Cc2cncc(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856274
NC(=O)CCNC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856276
O=C(NCC(F)=C1CN(C(=O)C2CC23CCC(F)(F)CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15856278
Nc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856282
O=C(NCC(F)=C1CN(C(=O)c2cnc3ccnn3c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856284
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1C(F)(F)F s275592__15865378__15841170__15856286
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sn1 s275592__15865378__15841170__15856288
CC1(C)C(=O)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856290
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__15856292
O=C(NCC(F)=C1CN(C(=O)c2cccc3sccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15856294
O=C(NCC(F)=C1CN(C(=O)c2cccnc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15856296
Nc1cc(N)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856298
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc3[nH]cnc23)C1)c1cc(O)no1 s275592__15865378__15841170__15856302
O=C(NCC(F)=C1CN(C(=O)Cc2cn3ccsc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15856304
Nc1cc2ccccc2cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856306
O=C(NCC(F)=C1CN(C(=O)c2cc(O)nc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15856308
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])c(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856314
O=C(NCC(F)=C1CN(C(=O)c2cc(O)c(O)c(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856316
O=C(NCC(F)=C1CN(C(=O)C(O)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856318
CCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856320
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856328
Cc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856330
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15856332
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856334
COC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856336
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15856338
Nc1cc(F)c(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856340
CC(=O)c1c(C)[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__15856344
O=C(NCC(F)=C1CN(C(=O)Cc2ccc([N+](=O)[O-])cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856346
CCCCOC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856348
Cc1ccc(OCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856352
Nc1n[nH]cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856354
CC(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856356
N#Cc1ccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856362
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])s2)C1)c1cc(O)no1 s275592__15865378__15841170__15856364
CCCn1cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856370
CCOC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856372
O=C(NCC(F)=C1CN(C(=O)CN2CC3C=CC2C3)C1)c1cc(O)no1 s275592__15865378__15841170__15856374
O=C(NCC(F)=C1CN(C(=O)CSC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15856376
O=C(NCC(F)=C1CN(C(=O)CCSC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15856378
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15856380
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15856382
O=C(NCC(F)=C1CN(C(=O)C2CCCC23OCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15858122
CCCCCC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858124
O=C(NCC(F)=C1CN(C(=O)C2CC2(F)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858126
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(=O)CC1 s275592__15865378__15841170__15858128
O=C(NCC(F)=C1CN(C(=O)c2c[nH]cc2Br)C1)c1cc(O)no1 s275592__15865378__15841170__15858130
O=C(NCC(F)=C1CN(C(=O)c2c(F)cc(F)nc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15858132
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ncccc1F s275592__15865378__15841170__15858134
CCc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858136
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C#N s275592__15865378__15841170__15858138
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1ccnc1 s275592__15865378__15841170__15858144
O=C(NCC(F)=C1CN(C(=O)CSc2ncn[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15858148
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c(=O)[nH]c1=O s275592__15865378__15841170__15858150
O=C(NCC(F)=C1CN(C(=O)c2cccnc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858152
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15858154
Cc1oncc1C(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858156
O=C(CC(F)(F)F)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858158
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)c1 s275592__15865378__15841170__15858160
CC(C)CSCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858164
O=C(NCC(F)=C1CN(C(=O)CCSC2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858166
Nc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858168
Cc1ccc(NCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15858170
Nc1c(F)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858172
Cc1ccc(SCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858174
O=C(NCC(F)=C1CN(C(=O)CSC(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15858176
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15858178
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(O)n1 s275592__15865378__15841170__15858180
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15841170__15858182
Cc1nc(O)nc(C)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858184
Cc1ncc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858186
Cc1noc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858188
CS(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858194
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(O)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858196
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15858198
O=C(NCC(F)=C1CN(C(=O)c2cccc[n+]2[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15858200
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15858204
Cc1ccc(C)n1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858206
N#Cc1cccc(NCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858208
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cc2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15858210
CCc1ncc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15858214
Cc1nn2ccccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858218
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)=NN1 s275592__15865378__15841170__15858220
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__15858222
Cc1csc(NC(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15858224
O=C1CCC(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15858226
COCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858228
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15858230
CC(=O)c1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858232
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__15858234
CP(C)(=O)C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858236
N#CCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858238
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15858240
C=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15858242
CC1(C)CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15858244
CN1N=C(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1=O s275592__15865378__15841170__15858246
CN(C)C(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860112
CSc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860114
CC(C)c1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860116
CC(C)(C)C(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)F s275592__15865378__15841170__15860120
CC(C)(C)n1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15860126
CC(=O)NC(COC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860128
O=C(NCC(F)=C1CN(C(=O)[C@@]23C[C@@H](O)[C@@H]2C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860130
COCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15860132
O=C(NCC(F)=C1CN(C(=O)C23CCCCC2C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860134
O=C(Cc1ccsc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860136
CCCOCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860140
O=C(NCC(F)=C1CN(C(=O)C(F)C2(O)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860142
COc1cccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15860144
CC1(C)COCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860146
C=C1CCC1(C(=O)OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860148
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(C)n1 s275592__15865378__15841170__15860150
Cn1ccn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c12 s275592__15865378__15841170__15860152
O=C(NCC(F)=C1CN(C(=O)C=Cc2cnc[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15860154
C=CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15860156
CC1OC2(CO)CC1(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15860160
Cc1n[nH]c2cnc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__15860162
O=C(NCC(F)=C1CN(C(=O)C2CCCC3C2C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860164
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]c1C s275592__15865378__15841170__15860166
CC1CC1c1nocc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860172
O=C(NCC(F)=C1CN(C(=O)C2CC=Cc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15860174
N#C[C@]1(O)C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860176
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15860180
CCCc1ncoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860182
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2O)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860184
O=C(NCC(F)=C1CN(C(=O)C2COc3ccc(F)cc32)C1)c1cc(O)no1 s275592__15865378__15841170__15860186
O=C(NCC(F)=C1CN(C(=O)C2CCc3ccnn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860188
O=C(NCC(F)=C1CN(C(=O)CCCCCF)C1)c1cc(O)no1 s275592__15865378__15841170__15860190
N#CC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860192
CC1(C)CCCOC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860194
O=C(NCC(F)=C1CN(C(=O)C2CCCCC23CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860196
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3nc[nH]n3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15860198
Cc1cccn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c12 s275592__15865378__15841170__15860202
CC(C)(C)C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)=NO1 s275592__15865378__15841170__15860204
CCC(C)(C)C(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860206
O=C(NCC(F)=C1CN(C(=O)C2(F)CCCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860208
O=C(NCC(F)=C1CN(C(=O)C=CCOCC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860210
C#CC[C@]1(O)C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860212
O=C(NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3CCCC(=O)[C@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__15860214
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CC3F)C1)c1cc(O)no1 s275592__15865378__15841170__15860216
O=C(NCC(F)=C1CN(C(=O)C2CN3CCN2CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860220
O=C(NCC(F)=C1CN(C(=O)C2CCCc3nncn32)C1)c1cc(O)no1 s275592__15865378__15841170__15860222
C=CCCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860224
O=C(NCC(F)=C1CN(C(=O)C2CCCC3(C2)CC3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860226
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCOCC1 s275592__15865378__15841170__15860228
O=C(NCC(F)=C1CN(C(=O)C23CC(CO2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860230
O=C(NCC(F)=C1CN(C(=O)C2CCCc3ccnn32)C1)c1cc(O)no1 s275592__15865378__15841170__15860232
CC12COC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(C1)C2 s275592__15865378__15841170__15862074
O=C(NCC(F)=C1CN(C(=O)c2cc3n(c2)CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862080
CC(=O)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862082
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c(O)c1F s275592__15865378__15841170__15862090
C#CC1(O)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15862092
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccc3[nH]cnc23)C1)c1cc(O)no1 s275592__15865378__15841170__15862100
COC(=O)c1sccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862102
C[C@@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(C)(C)C1 s275592__15865378__15841170__15862106
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c1C s275592__15865378__15841170__15862108
Cc1cnc2ccccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862110
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)n[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15862112
COCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__15862114
O=C(NCC(F)=C1CN(C(=O)C2CCCc3[nH]cnc32)C1)c1cc(O)no1 s275592__15865378__15841170__15862116
CC1(C)C(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__15862118
NC(=O)c1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15862120
Cc1oc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)[nH]c2c1C s275592__15865378__15841170__15862122
O=C(NCC(F)=C1CN(C(=O)C2(C3(O)CCOCC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862124
CCOC(=O)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862126
O=C(NCC(F)=C1CN(C(=O)CC(O)C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862132
CC1(C)COCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15862138
O=C(NCC(F)=C1CN(C(=O)CCC2CC(F)(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862140
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862142
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccc3ccoc23)C1)c1cc(O)no1 s275592__15865378__15841170__15862144
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCC32)C1)c1cc(O)no1 s275592__15865378__15841170__15862146
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)COCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862148
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15862150
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc2cccnc12 s275592__15865378__15841170__15862152
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15862154
CCN1C(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862156
CC1(C)CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15862166
O=C(NCC(F)=C1CN(C(=O)[C@@]2(F)C[C@@H]2c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15862168
Cn1nccc1C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862170
Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15862172
COCc1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862174
O=C(NCC(F)=C1CN(C(=O)C2=CS(=O)(=O)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862176
O=C(NCC(F)=C1CN(C(=O)c2cc3cn[nH]c3s2)C1)c1cc(O)no1 s275592__15865378__15841170__15862178
CC(=O)N1CSC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862180
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15862182
O=C(NCC(F)=C1CN(C(=O)c2ccc(-n3ccnc3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15862184
CC1CCSC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862188
O=C1CC2CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2C1 s275592__15865378__15841170__15862190
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc(F)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15862192
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2nc[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__15864490
O=C(NCC(F)=C1CN(C(=O)c2cnoc2C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864492
CC(C)(F)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864494
COC1CC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15864496
Cc1ncccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864500
Cc1ccc(C=CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15864502
O=C(NCC(F)=C1CN(C(=O)C23CCCCN2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15864504
O=C(NCC(F)=C1CN(C(=O)CC2CC(C(F)F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864506
Cc1c(N)cc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864508
Cc1c(C(N)=O)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864510
O=C(NCC(F)=C1CN(C(=O)c2cncc3[nH]ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15864512
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2C[C@H]2C[C@@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__15864514
Cc1cccc([C@@H](C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864516
CC1(C)OC[C@@H]([C@@H](O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15864518
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc2sccc21 s275592__15865378__15841170__15864522
Cc1nn(C(C)C)c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864524
O=C(NCC(F)=C1CN(C(=O)c2cccc3cnsc23)C1)c1cc(O)no1 s275592__15865378__15841170__15864526
O=C(NCC(F)=C1CN(C(=O)C23CC=CCN2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15864528
CC(C)C(C)C(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864532
Cn1nccc1C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864534
O=C(NCC(F)=C1CN(C(=O)c2cnc3ncnn3c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15864538
CC[C@H](CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15864540
CS(=O)(=O)c1coc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864542
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCCO3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864544
CCC=CC=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864546
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N=[N+]=[N-])c1 s275592__15865378__15841170__15864550
O=C(NCC(F)=C1CN(C(=O)CC2CC3(CCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864552
CNC(=O)N[C@H](C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864554
COc1ncnc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864558
CC(OCCN(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864560
O=C(NCC(F)=C1CN(C(=O)c2ccn(O)c(=O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864562
O=C(NCC(F)=C1CN(C(=O)c2cccc3sncc23)C1)c1cc(O)no1 s275592__15865378__15841170__15864564
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15841170__15864566
Cc1ncn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864570
CC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CO1)C2 s275592__15865378__15841170__15864572
CCn1c(C)nn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15841170__15864574
Cc1nc(C#N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864576
O=C(NCC(F)=C1CN(C(=O)C=Cc2c[nH]c(=O)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15864578
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CC(F)(F)F s275592__15865378__15841170__15864580
O=C(NCC(F)=C1CN(C(=O)Cc2nncs2)C1)c1cc(O)no1 s275592__15865378__15841170__15864586
O=C(NCC(F)=C1CN(C(=O)C2(C3CCC3)CC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15864588
CN(C)CCOCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864590
Cc1cc(N)cnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864592
COCCN(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864594
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CC(F)(F)F s275592__15865378__15841170__15864596
O=C(NCC(F)=C1CN(C(=O)C2CN(C3CCOC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864600
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]cnc3c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15864602
COc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__15864604
O=C(NCC(F)=C1CN(C(=O)CCCc2c[nH]nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15864606
CC(=C(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__15864610
CC(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__15864612
O=C(NCC(F)=C1CN(C(=O)c2ccccc2OC(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15856384
Cc1ccc(NCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856386
O=C(NCC(F)=C1CN(C(=O)CCCN2CCOC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15856390
CC1=NOC(=O)C1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856392
CC(=O)Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15856394
O=C(NCC(F)=C1CN(C(=O)CNc2ccc(Cl)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856396
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15856398
Cn1cc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856400
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc2ncnn12 s275592__15865378__15841170__15856402
Nc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856406
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(N)=O s275592__15865378__15841170__15856410
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15856412
CC1=NOC(=O)C1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856418
O=C(NCC(F)=C1CN(C(=O)CSc2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15856422
O=C(NCC(F)=C1CN(C(=O)c2nc(=O)[nH][nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15856424
O=C(NCC(F)=C1CN(C(=O)CSc2nccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15856426
CC(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856432
O=C(NCC(F)=C1CN(C(=O)C2(F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856434
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc([N+](=O)[O-])c1 s275592__15865378__15841170__15856436
O=C(NCC(F)=C1CN(C(=O)c2c(O)cccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15856438
CC(C)CCSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856444
CC(C)CCCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856446
COc1cc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15856450
CCCCC(ON=C(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856452
CN1CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856454
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)cc1F s275592__15865378__15841170__15856456
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856460
O=C(NCC(F)=C1CN(C(=O)c2cccn(O)c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15856462
Nc1ncncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856466
Nc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15856468
Cc1nc(N)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856474
Cc1ccc(F)cc1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856476
N#Cc1ccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858248
CC(C)n1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15858252
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858256
CCN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__15858258
O=C(NCC(F)=C1CN(C(=O)c2cc(O)c3ccccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858260
CCOC(=O)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858262
O=C(NCC(F)=C1CN(C(=O)C=C(C2CC2)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858264
CC(O)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__15858266
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCSC1 s275592__15865378__15841170__15858268
O=C(NCC(F)=C1CN(C(=O)CSCC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15858270
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15858272
CC1(C)OCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15858274
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C2(O)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858276
O=C(NCC(F)=C1CN(C(=O)c2[nH]ncc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15858278
O=C(NCC(F)=C1CN(C(=O)C(O)c2ccc(Cl)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858280
Cc1scnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858282
Nc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15858284
Nc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15858286
O=C(NCC(F)=C1CN(C(=O)c2cccc(F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15858288
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858290
COC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858294
O=C(NCC(F)=C1CN(C(=O)c2nccnc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15858296
CCOC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15858298
CC1CN2CCN1C(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15858300
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)F s275592__15865378__15841170__15858302
O=C(NCC(F)=C1CN(C(=O)C(F)=CC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858304
Cc1cccnc1C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858306
CC(CC#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858308
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccccn3)n[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15858314
CC1C(=O)CCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858316
O=C(NCC(F)=C1CN(C(=O)c2ccnn2CC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858318
CS(=O)(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15858322
Nc1cc(F)cc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858328
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccc(O)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15858334
O=C(NCC(F)=C1CN(C(=O)C[C@H]2CCCC[C@@H]2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858336
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__15858338
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cnnn1 s275592__15865378__15841170__15858340
O=C(NCC(F)=C1CN(C(=O)c2cnnc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858342
O=C(NCC(F)=C1CN(C(=O)C23C4C(=O)C5C6CC(C52)C3C64)C1)c1cc(O)no1 s275592__15865378__15841170__15858348
Cn1cc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15858350
COC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CC1)CC2 s275592__15865378__15841170__15858352
O=NN1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858354
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)c(Cl)n1 s275592__15865378__15841170__15858356
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15858358
O=C(NCC(F)=C1CN(C(=O)CCCc2nccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15858360
Cc1csc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15858362
Nc1cccc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858364
CCC1CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858366
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3ccncc3)[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__15858368
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCNC3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15858370
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]3C[C@@H]2CC3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15860234
O=C(NCC(F)=C1CN(C(=O)CC2CCC(O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860236
Cc1c(O)c(=O)ccn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860238
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)O s275592__15865378__15841170__15860240
CC(C)N(C)C(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860242
CN1c2ccccc2CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860244
Cc1scc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15860246
O=C(CF)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15860248
CN1CC2CC1(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15860250
Cn1ncc(C(F)F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860252
Cc1cc(=O)[nH]nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860254
O=C1OCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15860258
CC1(C)CCCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15860264
O=C(NCC(F)=C1CN(C(=O)CC23CNC(=O)C(C2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860266
Cc1cnccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860268
COc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15860270
Cn1nncc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860272
Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15860276
Cc1nc(N)ccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860278
Cc1nnc2n1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15860280
CCc1ccc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15860282
O=C(NCC(F)=C1CN(C(=O)C23COC(C2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860284
CC(O)C1CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860286
O=C(NCC(F)=C1CN(C(=O)C2C3CC4C(C3=O)C42)C1)c1cc(O)no1 s275592__15865378__15841170__15860288
O=C(NCC(F)=C1CN(C(=O)c2cc[nH]c2C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860290
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccnc(O)c3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15860294
CCCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__15860296
O=C(NCC(F)=C1CN(C(=O)CN2CC3CCC2C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860298
Nc1sc2c(c1C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CCC2 s275592__15865378__15841170__15860302
O=C1C[C@@H]2OCC[C@]2(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15841170__15860304
O=C(NCC(F)=C1CN(C(=O)c2cncc(-n3cccc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860306
O=C(NCC(F)=C1CN(C(=O)c2cccc(CF)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860310
COCC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860312
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15860314
O=C(NCC(F)=C1CN(C(=O)C2CCc3[nH]c(O)nc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860316
CC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(C1)OC2 s275592__15865378__15841170__15860318
O=C(NCC(F)=C1CN(C(=O)c2cncc(-n3ccnc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15860320
CCC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15860322
O=C(NCC(F)=C1CN(C(=O)C#CC2(C(F)(F)F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860324
N#Cc1c[nH]c2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__15860326
Cc1nc(=O)c(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__15860328
C[C@@H]1C[C@@]2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C[C@@H]12 s275592__15865378__15841170__15860334
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15860338
CC(C)N1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860344
O=C(NCC(F)=C1CN(C(=O)Cn2cncn2)C1)c1cc(O)no1 s275592__15865378__15841170__15860346
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2CCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15860350
O=C(NCC(F)=C1CN(C(=O)c2cccc(=O)o2)C1)c1cc(O)no1 s275592__15865378__15841170__15860352
Cc1cc(O)ccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860354
O=C(NCC(F)=C1CN(C(=O)COc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862196
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1ccnc1 s275592__15865378__15841170__15862200
O=C(NCC(F)=C1CN(C(=O)c2cn3cc[nH]c(=O)c3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15862202
O=C(NCC(F)=C1CN(C(=O)c2nc(C3CC3)n[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15862204
O=C(NCC(F)=C1CN(C(=O)COc2ccc(F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862206
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CC2)N=N3)C1)c1cc(O)no1 s275592__15865378__15841170__15862208
CC1CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(C)O1 s275592__15865378__15841170__15862210
O=C(NCC(F)=C1CN(C(=O)c2ccnc(OC3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862212
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCCC1 s275592__15865378__15841170__15862214
CC(CN(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862216
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCO1 s275592__15865378__15841170__15862220
COC(=O)c1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]c1C s275592__15865378__15841170__15862222
O=C(NCC(F)=C1CN(C(=O)C2CCCc3cn[nH]c32)C1)c1cc(O)no1 s275592__15865378__15841170__15862224
CNc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15862226
COc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccnc1F s275592__15865378__15841170__15862230
O=C(NCC(F)=C1CN(C(=O)CC2CCCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862232
O=C(NCC(F)=C1CN(C(=O)Cn2nnc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15862234
Cn1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__15862236
CC1(C)C(C#N)C1(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862238
O=C(NCC(F)=C1CN(C(=O)C2Cc3cccnc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862240
COc1cnc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862242
C=CC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862244
O=C(NCC(F)=C1CN(C(=O)CCC2(O)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862246
CCc1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15862248
CC(C)(C)c1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862250
CCC(C)(CO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862252
Cn1c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc2ccccc21 s275592__15865378__15841170__15862256
CC[C@H](C)[C@H](NC(=O)OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862258
Nc1nc(Cl)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15862260
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15862262
O=C(NCC(F)=C1CN(C(=O)CS(=O)(=O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862266
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccsc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862270
Cn1nc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862272
CCc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15862276
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1(F)Cl s275592__15865378__15841170__15862280
Cc1cccc2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)n12 s275592__15865378__15841170__15862284
CCCC=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862286
CC=C(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862288
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc2ccccc12 s275592__15865378__15841170__15862290
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__15862292
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOC1 s275592__15865378__15841170__15862294
O=C(NCC(F)=C1CN(C(=O)C(=O)C2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862296
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CC3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15862298
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15862300
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15862302
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)n(C3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862304
CC(C)Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__15862306
Cc1nc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2n1C s275592__15865378__15841170__15862308
O=C(NCC(F)=C1CN(C(=O)c2cccc(-n3cncn3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862310
CCS(=O)(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862312
CC(O)CCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862314
O=C(NCC(F)=C1CN(C(=O)c2ncn3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15862316
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__15864614
CCNc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864616
O=C(NCC(F)=C1CN(C(=O)c2cncc(F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15864618
O=C(NCC(F)=C1CN(C(=O)c2cnn(C3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864620
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__15864622
O=C(NCC(F)=C1CN(C(=O)c2ccccc2-n2cncn2)C1)c1cc(O)no1 s275592__15865378__15841170__15864624
Nc1cc(O)nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15864626
C[C@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__15864628
Cc1cccc(COCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864632
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccc(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864634
O=C(NCC(F)=C1CN(C(=O)CCc2nnc(C3CC3)o2)C1)c1cc(O)no1 s275592__15865378__15841170__15864636
CC(C)C(CO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864638
CCOC=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864642
Nc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15864644
O=C(NCC(F)=C1CN(C(=O)Cc2cc(F)ccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15864646
CC1c2cn[nH]c2CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864648
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)c1Cl s275592__15865378__15841170__15864650
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc2[nH]ncc12 s275592__15865378__15841170__15864654
CCN1CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864656
Cc1nc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15864662
CSc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15864664
O=C(CO)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864668
CCC(O)Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__15864670
CS(=O)(=O)SCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864678
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(O)c1 s275592__15865378__15841170__15864680
O=C(NCC(F)=C1CN(C(=O)c2cn3cnnc3cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15864684
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccs1 s275592__15865378__15841170__15864686
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCS1(=O)=O s275592__15865378__15841170__15864688
O=C(NCC(F)=C1CN(C(=O)C=CCCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15864692
Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)o1 s275592__15865378__15841170__15864694
O=C1CCC(C#CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15864696
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2CCC1C2 s275592__15865378__15841170__15864698
CC(C)N1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15864700
COc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15864706
Cc1ccc2c(c1)C(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15864710
O=C(NCC(F)=C1CN(C(=O)C2CCCc3scnc32)C1)c1cc(O)no1 s275592__15865378__15841170__15864712
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__15864716
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@H]2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15864718
O=C(NCC(F)=C1CN(C(=O)[C@H]2CCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15864720
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)Cc2ccccc2N1 s275592__15865378__15841170__15864722
Nc1cc(F)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15864728
O=C(NCC(F)=C1CN(C(=O)C2(C3CC3)CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15864730
Cc1ncc2ccccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864734
Cn1cc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2n1 s275592__15865378__15841170__15864736
O=C(NCC(F)=C1CN(C(=O)c2ccc(OC(F)F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856480
Cc1nn(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__15856484
Cc1c([N+](=O)[O-])c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__15856486
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)cc1F s275592__15865378__15841170__15856492
CCc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15856494
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c([N+](=O)[O-])c1 s275592__15865378__15841170__15856498
CC(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(O)n1 s275592__15865378__15841170__15856500
N#Cc1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856502
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1Cl s275592__15865378__15841170__15856504
COC(=O)CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856506
CCC(C)(C)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856508
CSSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856512
CCOC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856516
NC(=O)C(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856518
CCC(C)=C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856520
Nc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15856522
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2NCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15856526
CSC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__15856528
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15856530
CSc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856532
O=C(NCC(F)=C1CN(C(=O)c2coc(Cl)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15856534
O=C(NCC(F)=C1CN(C(=O)C=CC(=O)N2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856538
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(O)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856540
CCC(C)C(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856542
CCC(Oc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856544
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)=NN1 s275592__15865378__15841170__15856546
NC(=O)N1CC(O)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856548
COC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856550
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15856552
CC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856554
N#Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856556
O=C(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15856558
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856560
Nc1cc([N+](=O)[O-])ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856562
O=C(NCC(F)=C1CN(C(=O)CNc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856566
O=C(NCC(F)=C1CN(C(=O)c2ccccc2NCCO)C1)c1cc(O)no1 s275592__15865378__15841170__15856568
Nc1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856572
Nc1ccc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856576
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__15856578
O=C(NCC(F)=C1CN(C(=O)c2cc(F)ccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856580
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15856582
O=C(NCC(F)=C1CN(C(=O)CSc2cccc[n+]2[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15856584
NC(=O)NCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856586
O=C(NCC(F)=C1CN(C(=O)CNc2ccc(O)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856588
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856592
O=C(NCC(F)=C1CN(C(=O)CSc2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856594
Cc1ccnc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnn12 s275592__15865378__15841170__15856596
Nc1cc2c(cc1C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)OCO2 s275592__15865378__15841170__15856598
O=C(NCC(F)=C1CN(C(=O)c2ccccc2OCCO)C1)c1cc(O)no1 s275592__15865378__15841170__15856600
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CCc1ccccc1 s275592__15865378__15841170__15856602
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__15856604
CS(C)(=O)=NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858372
Cc1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15858374
[N-]=[N+]=NCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858376
C=CCCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858382
CC(C)C(=O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858384
Nc1nc2ncccc2cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858386
CC(O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858388
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15858392
CC(C)(C)OCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858396
CC(C)Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__15858404
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1CCO s275592__15865378__15841170__15858406
CC(=O)OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858408
O=C(NCC(F)=C1CN(C(=O)C(O)CCc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858410
C#CCN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858412
O=C(NCC(F)=C1CN(C(=O)c2cccc(OC(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858414
O=C(Cc1cccc(F)c1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858416
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1[N+](=O)[O-] s275592__15865378__15841170__15858418
CNc1nc(C)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858420
Nc1ccncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858424
CC(Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858426
Nc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858428
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)c1 s275592__15865378__15841170__15858430
O=C(NCC(F)=C1CN(C(=O)Cn2cccnc2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15858432
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15858434
CC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858440
O=C(NCC(F)=C1CN(C(=O)C2CCCN2C(=O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858442
O=C(NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)NC1CC1 s275592__15865378__15841170__15858444
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc([N+](=O)[O-])c1 s275592__15865378__15841170__15858446
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15858448
Cc1nc2ccccc2cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858452
CCCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__15858458
O=C(NCC(F)=C1CN(C(=O)C=CC2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858460
Nc1ccc(Cl)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858462
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15841170__15858466
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15858468
Cn1cc([N+](=O)[O-])c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15858472
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15858474
Cc1onc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C#N s275592__15865378__15841170__15858476
CN(C)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858478
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(-c3ccccc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858480
O=C(NCC(F)=C1CN(C(=O)C(F)(F)CO)C1)c1cc(O)no1 s275592__15865378__15841170__15858486
Cc1nc(O)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858488
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c3cccc(F)c23)C1)c1cc(O)no1 s275592__15865378__15841170__15858492
Cc1cc(F)ccc1C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860356
N#CCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860358
O=C(NCC(F)=C1CN(C(=O)C=Cc2nccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15860360
CC1(C#CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860362
O=C(NCC(F)=C1CN(C(=O)C2(F)CCS(=O)(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860364
O=C(NCC(F)=C1CN(C(=O)C2OCCn3ccnc32)C1)c1cc(O)no1 s275592__15865378__15841170__15860366
CCc1nc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__15860370
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc3[nH]ccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860374
COc1ccc(OC)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15860376
C=CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15860378
CC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860380
Cc1ncsc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860382
[N-]=[N+]=N[C@@H]1C=CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860386
O=C(NCC(F)=C1CN(C(=O)COC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860388
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CCCC3O)C1)c1cc(O)no1 s275592__15865378__15841170__15860390
Nc1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15860392
O=C(NCC(F)=C1CN(C(=O)c2ncc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15860394
O=C(NCC(F)=C1CN(C(=O)C=CC2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860398
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1nccs1 s275592__15865378__15841170__15860400
O=C(NCC(F)=C1CN(C(=O)C=CBr)C1)c1cc(O)no1 s275592__15865378__15841170__15860402
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15860404
CC(CCN(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860406
O=C1CC(C#CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860408
CSc1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860410
CC(C)Nc1nnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860412
CC1(C)OC[C@H](C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15860414
O=C(NCC(F)=C1CN(C(=O)C2=Cc3ccccc3C2O)C1)c1cc(O)no1 s275592__15865378__15841170__15860416
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(-c3ccncc3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15860418
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15860420
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15860424
NC(=O)c1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860426
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15860430
O=C(NCC(F)=C1CN(C(=O)C2CC(C3CC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860432
O=C(NCC(F)=C1CN(C(=O)c2cn(C3CC3)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15860434
CC1CNc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnn2C1 s275592__15865378__15841170__15860438
Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15860440
CC(C)[C@H](NC=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860442
Cc1cc(C)c(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__15860444
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15860448
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__15860450
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc1C(F)F s275592__15865378__15841170__15860452
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cncnc1 s275592__15865378__15841170__15860458
O=C(NCC(F)=C1CN(C(=O)C23OC4C5COCC4C2C53)C1)c1cc(O)no1 s275592__15865378__15841170__15860460
O=C(NCC(F)=C1CN(C(=O)c2ccn3c2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860462
O=C(NCC(F)=C1CN(C(=O)C=C2CCCCCC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860464
C=C(C)[C@@H]1OCCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860466
O=C(NCC(F)=C1CN(C(=O)C2CCCc3ncccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15860468
[N-]=[N+]=NC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CC1)C2 s275592__15865378__15841170__15860470
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc2nn[nH]c12 s275592__15865378__15841170__15860472
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nnc1C s275592__15865378__15841170__15860474
CC1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860476
CN(C)c1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860478
O=C(NCC(F)=C1CN(C(=O)C2CCC3C(C2)C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15862318
Cc1cc(Cl)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15862322
O=C(NCC(F)=C1CN(C(=O)C2CCOC2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15862324
Cn1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15841170__15862326
CSC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862328
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(N)cn1 s275592__15865378__15841170__15862330
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862332
N#Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15862334
Cc1c(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__15862338
Nc1cccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15862342
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccc(CO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862344
CC(C)c1nnc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15862346
CCn1nccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862348
Cc1coc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15862350
Cc1cc(C)cc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15862352
O=C(NCC(F)=C1CN(C(=O)c2nncs2)C1)c1cc(O)no1 s275592__15865378__15841170__15862356
CC(=O)N[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__15862358
O=C(NCC(F)=C1CN(C(=O)C#CC2CCCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862360
O=C(NCC(F)=C1CN(C(=O)CC2CCC=CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862364
Cc1cc(C)n2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2n1 s275592__15865378__15841170__15862370
O=C(NCC(F)=C1CN(C(=O)c2c3c(n[nH]c2=O)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862372
O=C(NCC(F)=C1CN(C(=O)[C@@H]2[C@H]3CCCO[C@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__15862374
CCCCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15862376
O=C(NCC(F)=C1CN(C(=O)C2(c3cccs3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862378
CCC(C)(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862380
O=C(NCC(F)=C1CN(C(=O)CC(C(F)F)n2ccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15862384
O=C(NCC(F)=C1CN(C(=O)COC2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862388
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCO3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862390
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__15862392
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCCN3CCCC[C@H]23)C1)c1cc(O)no1 s275592__15865378__15841170__15862394
CC(C)COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15862396
O=C(NCC(F)=C1CN(C(=O)[C@@]23CCCCC[C@H]2OCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862398
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3ocnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862400
CC1(C)CC(=O)NCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862402
CN(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cscn1 s275592__15865378__15841170__15862404
O=C(NCC(F)=C1CN(C(=O)c2cnn(CCO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862406
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@@H](OC(F)F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862408
CCc1[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1Cl s275592__15865378__15841170__15862410
O=C(NCC(F)=C1CN(C(=O)c2cccn3nncc23)C1)c1cc(O)no1 s275592__15865378__15841170__15862412
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2cnccc2c1 s275592__15865378__15841170__15862414
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__15862416
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1(O)CCCCC1 s275592__15865378__15841170__15862418
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2cscn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862422
O=C(NCC(F)=C1CN(C(=O)c2csc3cncn23)C1)c1cc(O)no1 s275592__15865378__15841170__15862424
CC(C)(C)c1noc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15862426
C=C(F)C1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15862428
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)c(F)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15862430
Cc1cccc(NC(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15862432
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(=O)[nH][nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862434
O=C1COC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15862436
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2CCC(C1)S2 s275592__15865378__15841170__15862438
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1Cl s275592__15865378__15841170__15863664
Cc1ccc2occ(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__15863668
CC12CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(C1)C(C)(C)O2 s275592__15865378__15841170__15863670
O=C(NCC(F)=C1CN(C(=O)c2coc(C(F)F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863672
O=C(C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)NC1CC1 s275592__15865378__15841170__15863674
O=C(NCC(F)=C1CN(C(=O)Cc2nc3c([nH]2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863676
CN1Cc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2C1 s275592__15865378__15841170__15863678
CC(C)NC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863680
Nc1ccc2nccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__15863684
C=C(Cl)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863686
CC(C)(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__15863690
CCC(CCOC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863692
O=C(NCC(F)=C1CN(C(=O)C2CC3C=CCC(C3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863694
Cc1nc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc1C s275592__15865378__15841170__15863696
Cc1coc(C)c1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863698
O=C(NCC(F)=C1CN(C(=O)C23CC(CN2C2CC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15863700
Cc1cn2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)sc2n1 s275592__15865378__15841170__15863702
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__15863704
O=C(NCC(F)=C1CN(C(=O)CCn2ccc3cccnc32)C1)c1cc(O)no1 s275592__15865378__15841170__15863706
COCC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15863712
C=Cn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863714
Cc1coc(C(C)C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863716
O=C(NCC(F)=C1CN(C(=O)c2ccc3ncc(=O)[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863718
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863720
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CNC3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15863722
Cn1ccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863724
O=C(NCC(F)=C1CN(C(=O)c2coc3c(F)cccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863726
O=C(NCC(F)=C1CN(C(=O)c2coc3c2C(=O)NCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863730
CC(=O)OCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863732
Cc1nc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c1C s275592__15865378__15841170__15863736
CCc1oc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863738
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC=CC1 s275592__15865378__15841170__15863740
CCc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__15863742
O=C(NCC(F)=C1CN(C(=O)CCNc2cncnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15864740
O=C(NCC(F)=C1CN(C(=O)C2CCN(CCO)C(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864744
CCc1cscc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864748
O=C(NCC(F)=C1CN(C(=O)CC2CCCC(F)(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864756
Cc1n[nH]c2c1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__15864758
O=C1CSC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15864760
O=C(NCC(F)=C1CN(C(=O)c2ccnn2C2CC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15864762
Nc1cc2[nH]cnc2cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864764
O=C(NCC(F)=C1CN(C(=O)C2=CC3CCC=CCCC23)C1)c1cc(O)no1 s275592__15865378__15841170__15864766
CC1(C)OC2(CO)CC1(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15864768
O=C(NCC(F)=C1CN(C(=O)c2cnn(C(F)(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864770
C=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)(C(F)F)C1 s275592__15865378__15841170__15864772
C#Cc1ccc(C2CC2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15864774
CO[C@@H]1C[C@@]2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C[C@@H]12 s275592__15865378__15841170__15864778
O=C(NCC(F)=C1CN(C(=O)c2cc3cncnc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15864780
Cc1ccc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15864782
CC1OC2(C)CC1(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15864784
Cn1cnnc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864786
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc1C(F)F s275592__15865378__15841170__15864788
CCc1nonc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864792
O=C(NCC(F)=C1CN(C(=O)CC2(CO)CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864796
O=C(NCC(F)=C1CN(C(=O)Cc2cnsn2)C1)c1cc(O)no1 s275592__15865378__15841170__15864798
C=CCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864800
Nc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15864802
O=C(NCC(F)=C1CN(C(=O)C2CCC(=O)N(C3CC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864804
O=C(NCC(F)=C1CN(C(=O)c2ccc(C#CC3CC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15864806
O=C(NCC(F)=C1CN(C(=O)c2cccc(C#CC3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864808
COCCCCN(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864810
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc1N s275592__15865378__15841170__15864814
O=C(NCC(F)=C1CN(C(=O)C2CC(c3ccccc3)O2)C1)c1cc(O)no1 s275592__15865378__15841170__15864816
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15864818
O=C(NCC(F)=C1CN(C(=O)C2CC(OC(F)(F)F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864820
CC(C)(C)O[C@H]1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15864826
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1(O)CCOC1 s275592__15865378__15841170__15864828
CCSC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15864830
CCC(C)CC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864832
O=C(NCC(F)=C1CN(C(=O)CC2CCCC3(CCC3)O2)C1)c1cc(O)no1 s275592__15865378__15841170__15864834
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOC1 s275592__15865378__15841170__15864836
COc1cncc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864838
CN1CC(C)(C)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864842
Cc1c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc2ccccc12 s275592__15865378__15841170__15864844
O=C(NCC(F)=C1CN(C(=O)C(F)n2cccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15864846
O=C(NCC(F)=C1CN(C(=O)CC2(CO)CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864848
COC(=O)[C@@]1(Cl)C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864850
Cc1ccn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2n1 s275592__15865378__15841170__15864852
CN(C)CCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864854
COc1ccnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15864856
CC1(C)CC(=O)N(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15864858
O=C(NCC(F)=C1CN(C(=O)CCN2CCOC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15856606
CCSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15856610
O=C(NCC(F)=C1CN(C(=O)CCN2CCC(O)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856612
Cc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856614
Cn1ccnc1SCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856616
COc1ccccc1NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856618
O=C(NCC(F)=C1CN(C(=O)CCOc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856620
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15856622
CCCN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856624
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)c1 s275592__15865378__15841170__15856628
Cc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856632
CC(C)CCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856634
Cc1c(Cl)ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856636
O=C(NCC(F)=C1CN(C(=O)COCc2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__15856638
CC(CO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856640
O=C(NCC(F)=C1CN(C(=O)c2cc3sccc3cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856642
O=C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc2c(c1)CCC2 s275592__15865378__15841170__15856644
Cc1ccc(F)c(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856646
CCN1CCN(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856648
O=C(NCC(F)=C1CN(C(=O)c2cnoc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856650
Nc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15856652
O=C(NCC(F)=C1CN(C(=O)CSCC2CCCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15856654
CN1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856658
COC(=O)N1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15856660
Cn1cc(C(F)(F)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15858496
Nc1c(F)cc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858498
O=C(NCC(F)=C1CN(C(=O)CCCCO)C1)c1cc(O)no1 s275592__15865378__15841170__15858500
CCOC(=O)C(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858502
O=C(NCC(F)=C1CN(C(=O)C(=O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858504
Cc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__15858508
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c([N+](=O)[O-])c1 s275592__15865378__15841170__15858510
CCCCCCCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858514
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__15858516
O=C1N[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15858518
O=C(NCC(F)=C1CN(C(=O)Cc2c(F)cncc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15858520
O=C(NCC(F)=C1CN(C(=O)c2cncc(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858522
COc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858524
O=C(NCC(F)=C1CN(C(=O)Cc2cnccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15858526
O=C(NCC(F)=C1CN(C(=O)CC2(O)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858528
CCOC(=O)C(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858532
O=C(NCC(F)=C1CN(C(=O)CCCCC(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15858536
O=C(NCC(F)=C1CN(C(=O)Cc2ccn[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15858540
CNc1ccc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858542
Cc1oc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858544
COC(=O)c1cscc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858546
COC(=O)CC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858548
Cc1cc(=O)n(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15858552
Cc1nc(CO)sc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858554
O=C(NCC(F)=C1CN(C(=O)c2cccc(=S)n2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858556
O=C(NCC(F)=C1CN(C(=O)Cc2cc(Cl)ccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858558
CC1COc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15841170__15858560
NC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15858562
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15841170__15858564
CNc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15858566
Cc1ncsc1COCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858568
O=C(NCC(F)=C1CN(C(=O)COc2ccc(CO)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858570
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CC3)ccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15858572
O=C(NCC(F)=C1CN(C(=O)C2CCC2F)C1)c1cc(O)no1 s275592__15865378__15841170__15858574
N#CCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858576
CCOC(=O)C(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)=O s275592__15865378__15841170__15858578
O=C(NCC(F)=C1CN(C(=O)C2C(F)(F)C23CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15858582
N#Cc1ccc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858584
CC(C)C(=O)N[C@@H](CO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858586
O=C(NCC(F)=C1CN(C(=O)c2cc3c([nH]2)CCCC3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15858588
CC1C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)=Cc2ccccc21 s275592__15865378__15841170__15858590
O=C(NCC(F)=C1CN(C(=O)c2ccccc2OC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858592
CN(C)c1nc(N)nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15858594
O=C(NCC(F)=C1CN(C(=O)c2ccn3nccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858596
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(C)n1 s275592__15865378__15841170__15858598
O=C(NCC(F)=C1CN(C(=O)C(CO)c2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858600
Nc1c(F)ccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858602
CCSc1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858604
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)(F)F)on2)C1)c1cc(O)no1 s275592__15865378__15841170__15858606
CC(C)(C)c1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15858608
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cnc(C#N)n1 s275592__15865378__15841170__15858610
Nc1ccccc1CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858612
CCOC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858618
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CCC3)O2)C1)c1cc(O)no1 s275592__15865378__15841170__15860482
O=C(NCC(F)=C1CN(C(=O)C[C@H]2Cc3ccccc3N2)C1)c1cc(O)no1 s275592__15865378__15841170__15860484
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2cnccc12 s275592__15865378__15841170__15860486
O=C(NCC(F)=C1CN(C(=O)C2CC(n3ccnc3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860488
O=C(NCC(F)=C1CN(C(=O)C(F)C2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860490
O=C(NCC(F)=C1CN(C(=O)C2CCCC23CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860492
NC(=O)c1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860494
Cc1oc(Cl)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860498
Cc1cnsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860502
O=C(NCC(F)=C1CN(C(=O)C2=CC3CCCCCCC23)C1)c1cc(O)no1 s275592__15865378__15841170__15860504
O=C(NCC(F)=C1CN(C(=O)c2cnc3[nH]ccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15860506
O=C(NCC(F)=C1CN(C(=O)[C@@H](O)Cc2c[nH]cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15860508
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1CC1CC1 s275592__15865378__15841170__15860510
CCc1onc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__15860512
Cn1cc(SCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15860514
CC(C)CC(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860516
O=C(NCC(F)=C1CN(C(=O)C(F)C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860518
CC(OC(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860520
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15860522
O=C(NCC(F)=C1CN(C(=O)COc2ccc(Cl)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15860524
O=C(NCC(F)=C1CN(C(=O)c2ccn3nncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860526
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCNC1=O s275592__15865378__15841170__15860528
CC1CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__15860530
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCCC3)CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15860532
O=C(NCC(F)=C1CN(C(=O)CC2CC3(CC3)CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15860534
O=C(NCC(F)=C1CN(C(=O)c2cc3oc(Cl)cc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15860536
Cn1cnc2c1CCCC2C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860538
Cn1ncc2c1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CN2 s275592__15865378__15841170__15860540
CC(C)(F)C(C)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860542
O=C(NCC(F)=C1CN(C(=O)[C@]23COC[C@H]2C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860544
O=C1CCC(F)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860546
Cc1cn(C(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860550
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCS1 s275592__15865378__15841170__15860552
CC12CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CCO1)C2 s275592__15865378__15841170__15860554
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CC2)CC(O)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860556
CC(C)(CCC#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860558
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]3CCCCC[C@@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__15860560
CC1=NOC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15860562
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)nc1C s275592__15865378__15841170__15860568
C#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15860570
O=C(NCC(F)=C1CN(C(=O)c2cncc3c(=O)[nH]ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15860572
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CC2(CC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860576
O=C(NCC(F)=C1CN(C(=O)c2nnc3n2CCCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860580
O=C(NCC(F)=C1CN(C(=O)c2cccc(-c3cc[nH]n3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860582
O=C(NCC(F)=C1CN(C(=O)c2ccccc2-c2ncn[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15860586
CC1(C)CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15860588
CC(C)C[C@H](CNC=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860590
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(N)c1 s275592__15865378__15841170__15860596
O=C(NCC(F)=C1CN(C(=O)CC2CCCCC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860598
O=C1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(=O)N1 s275592__15865378__15841170__15860600
CC1(c2cccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2)CC1 s275592__15865378__15841170__15862440
O=C(NCC(F)=C1CN(C(=O)CC2CCC3CC3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862442
Cn1ncc2ccnc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c21 s275592__15865378__15841170__15862444
CC1(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15862446
CC(C)n1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15841170__15862448
Cc1ccsc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862452
Cc1ccccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862454
Cn1cccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862458
CCc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15862460
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc3c(c2)CCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15862462
O=C(NCC(F)=C1CN(C(=O)C=Cc2c[nH]cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862464
Cc1csc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15862468
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(F)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862472
O=C(NCC(F)=C1CN(C(=O)C=Cc2cncs2)C1)c1cc(O)no1 s275592__15865378__15841170__15862474
Nc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15862476
Cc1cc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15841170__15862480
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(C3CC3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15862482
O=C(NCC(F)=C1CN(C(=O)C=Cc2ncc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15862484
Cn1cc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__15862486
O=C(NCC(F)=C1CN(C(=O)[C@]23C[C@H]2COC32CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862490
CCC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841170__15862492
Cn1nccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862498
O=C(NCC(F)=C1CN(C(=O)C=Cc2cn[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862500
CCc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15862504
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__15862508
O=C(NCC(F)=C1CN(C(=O)C=Cc2nc3ccccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__15862512
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CS(=O)(=O)C1 s275592__15865378__15841170__15862516
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)s1 s275592__15865378__15841170__15862518
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2CF)C1)c1cc(O)no1 s275592__15865378__15841170__15862520
CC(C)CN1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15862522
O=C(NCC(F)=C1CN(C(=O)c2cnc3n2CCS3)C1)c1cc(O)no1 s275592__15865378__15841170__15862524
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15862526
CC1CN(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15862530
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccncc1 s275592__15865378__15841170__15862534
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)ncc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15862538
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CON1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15862560
O=C(NCC(F)=C1CN(C(=O)c2cn(C3COC3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15863744
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Cn1ccc2ccnc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c21 s275592__15865378__15841170__15863754
Cc1c(O)ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__15863760
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CC2)CC3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863762
O=C(NCC(F)=C1CN(C(=O)COC2CCCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863764
COC1(C(F)(F)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15863766
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCOC1 s275592__15865378__15841170__15863768
CC(C)CC(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863770
CC1(C#CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841170__15863772
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15841170__15863774
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15863776
Nc1cccc2c1ccn2CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863784
CC(=CC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863786
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1nc[nH]n1 s275592__15865378__15841170__15863788
O=C1CC2(CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C2)N1 s275592__15865378__15841170__15863790
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15841170__15863792
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(CO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863794
CC1(C)C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(F)F s275592__15865378__15841170__15863800
N#C[C@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863804
CC(=O)c1cn(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863810
O=C(NCC(F)=C1CN(C(=O)C2(O)CC3CCC2C3)C1)c1cc(O)no1 s275592__15865378__15841170__15863812
CCC1CCCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863814
O=C(NCC(F)=C1CN(C(=O)C=Cc2cocn2)C1)c1cc(O)no1 s275592__15865378__15841170__15863816
N#Cc1cnn2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc12 s275592__15865378__15841170__15863818
CC(=Cn1ccnn1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863820
CC(C)n1cnnc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863824
O=C(NCC(F)=C1CN(C(=O)c2cc(O)nc3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863826
CCC(O)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15863828
O=C(NCC(F)=C1CN(C(=O)CC2(CO)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863830
O=C(NCC(F)=C1CN(C(=O)c2coc3c2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863832
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCO3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863834
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(N)c1O s275592__15865378__15841170__15863836
CN(C)Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15863838
CC(C)(C)c1nocc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863842
O=C(NCC(F)=C1CN(C(=O)CC2(CO)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863844
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(O)c1Cl s275592__15865378__15841170__15863846
CCCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__15863848
Cc1sc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C#N s275592__15865378__15841170__15863850
Cn1nnc2c1C(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CCC2 s275592__15865378__15841170__15863852
CON=C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccco1 s275592__15865378__15841170__15863854
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(Cl)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863856
O=C(NCC(F)=C1CN(C(=O)C2CCn3ncnc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863858
CC1(C)NC(=O)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863860
O=C1C[C@@H]2CCC[C@]2(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863862
O=C(NCC(F)=C1CN(C(=O)c2cccnc2-n2nccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15863864
CNC(=O)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15864860
O=C1CC2(CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2)C1 s275592__15865378__15841170__15864862
O=C(NCC(F)=C1CN(C(=O)C2=NNC(C(F)(F)F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864864
Nc1ccc2c(c1)CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)N2 s275592__15865378__15841170__15864866
Nc1nc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2o1 s275592__15865378__15841170__15864868
O=C(NCC(F)=C1CN(C(=O)Cc2cnco2)C1)c1cc(O)no1 s275592__15865378__15841170__15864872
O=C(NCC(F)=C1CN(C(=O)CC23CCC(CC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15864874
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2CC=CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864876
CC(=Cc1cccs1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864878
COCCOCC=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864882
O=C(NCC(F)=C1CN(C(=O)CN2CC3CC3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864884
CCCc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nnn1CC s275592__15865378__15841170__15864888
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)n1cccn1 s275592__15865378__15841170__15864890
Cn1nc2c(c1C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)COCC2 s275592__15865378__15841170__15864892
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@H](n3ccnn3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864894
CC1CNc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc21 s275592__15865378__15841170__15864896
CC(C)(C)[C@@H]1CCCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864898
O=C(NCC(F)=C1CN(C(=O)CC2CC3CC3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864900
O=C(NCC(F)=C1CN(C(=O)c2cc(CF)on2)C1)c1cc(O)no1 s275592__15865378__15841170__15864906
CC(F)(F)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864908
O=C(NCC(F)=C1CN(C(=O)c2cn(C3CCOC3)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15864914
O=C(NCC(F)=C1CN(C(=O)c2ccc3cnnn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864916
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccccc3c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15864918
O=C(NCC(F)=C1CN(C(=O)C2CCC(=C(F)F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864920
O=C(NCC(F)=C1CN(C(=O)C2Cc3nccnc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864926
O=C(NCC(F)=C1CN(C(=O)C2CNc3ccnn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864928
O=C(NCC(F)=C1CN(C(=O)C23CC=CC(C2)OC3)C1)c1cc(O)no1 s275592__15865378__15841170__15864930
O=C(NCC(F)=C1CN(C(=O)CCCC(F)(F)CO)C1)c1cc(O)no1 s275592__15865378__15841170__15864936
O=C(NCC(F)=C1CN(C(=O)C(C2CC2)C2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15864938
O=C(NCC(F)=C1CN(C(=O)CC2(N3CCCC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864940
CC1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1C s275592__15865378__15841170__15864944
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15864946
O=C(NCC(F)=C1CN(C(=O)c2ccn3cccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__15864948
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C2CCC2)n1 s275592__15865378__15841170__15864950
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C(F)F)nn1C s275592__15865378__15841170__15864952
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)cc1N s275592__15865378__15841170__15864958
O=C(NCC(F)=C1CN(C(=O)Cc2coc(C(F)F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15864960
COC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856662
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O=C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(Cl)cc1 s275592__15865378__15841170__15856672
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)OCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15856674
CSc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856676
Nc1ccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c[nH]c2c1 s275592__15865378__15841170__15856678
Nc1nc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15856684
O=C(NCC(F)=C1CN(C(=O)c2nc(Cl)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15856686
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(N)cc1 s275592__15865378__15841170__15856688
O=C(NCC(F)=C1CN(C(=O)c2cnc3cccnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856690
CC(NC1(CO)CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856692
O=C(NCC(F)=C1CN(C(=O)c2cnc(Cl)s2)C1)c1cc(O)no1 s275592__15865378__15841170__15856694
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCCCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15856696
CC(C)(O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856700
COCCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856702
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(O)cc1 s275592__15865378__15841170__15856704
CCOC(=O)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__15856706
COc1cc(C)c(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856708
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CCC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856710
CCOc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856714
COC(OC)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15856716
CC(C)(C)C(CO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856718
CS(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856724
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)cc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15856726
COC(=O)N1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856728
Cc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__15856730
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)cc1N s275592__15865378__15841170__15856732
O=C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__15856734
N#Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856736
CN(C)c1nc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15856740
CN(C)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15856746
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__15856748
CC1CCC(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2)CC1 s275592__15865378__15841170__15856752
O=C(NCC(F)=C1CN(C(=O)C=CCN2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856754
CCC(C#N)(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856756
O=C(NCC(F)=C1CN(C(=O)c2noc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15856758
CCOC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)OCC s275592__15865378__15841170__15856760
O=C(NCC(F)=C1CN(C(=O)C(F)(F)CC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856762
O=C1CSC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)=N1 s275592__15865378__15841170__15856764
N#Cc1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856766
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1CCO s275592__15865378__15841170__15856768
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15856770
O=C(NCC(F)=C1CN(C(=O)C2(Br)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856772
CN1CCCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856776
Nc1ccc(OCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856780
O=C(NCC(F)=C1CN(C(=O)c2ccnnc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15856782
CCOC(=O)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858620
CCOC(=O)NC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15858622
CSCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858624
O=C(NCC(F)=C1CN(C(=O)C2(O)CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858626
O=C(C=Cc1cccs1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858628
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1O s275592__15865378__15841170__15858634
O=C(NCC(F)=C1CN(C(=O)CNc2ncccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15858636
O=C(NCC(F)=C1CN(C(=O)CSCc2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858638
O=C(NCC(F)=C1CN(C(=O)c2cnccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15858640
O=C(NCC(F)=C1CN(C(=O)Cn2cc([N+](=O)[O-])cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15858642
CC(C)CN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15858644
O=C(NCC(F)=C1CN(C(=O)c2c(F)cccc2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15858646
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15858650
CS(=O)(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858654
O=C(NCC(F)=C1CN(C(=O)c2c(O)cccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15858656
CC(C)CC(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858660
O=C(NCC(F)=C1CN(C(=O)CC2CC(F)(F)C2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15858662
O=C(NCC(F)=C1CN(C(=O)Cn2[nH]c(=O)ccc2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15858666
Cc1ccc(NCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858670
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)cc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858678
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15858680
O=C(NCC(F)=C1CN(C(=O)C2(O)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858682
O=C(Cc1cccs1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858688
COC(=O)N(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858692
C=CCn1ccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858694
CC(Sc1nncn1C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858696
O=C(NCC(F)=C1CN(C(=O)CSc2nncs2)C1)c1cc(O)no1 s275592__15865378__15841170__15858698
N#Cc1ccccc1OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858702
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ncccn1 s275592__15865378__15841170__15858704
Cc1c(N)cc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858710
N#Cc1ccc(C(O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858712
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1Cl s275592__15865378__15841170__15858714
CNc1c(F)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858716
Nc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1[N+](=O)[O-] s275592__15865378__15841170__15858718
O=C(NCC(F)=C1CN(C(=O)C2=CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858720
C=CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__15858722
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2C(=O)NC3)C1)c1cc(O)no1 s275592__15865378__15841170__15858724
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15858726
Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15858732
COc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15858734
O=C(NCC(F)=C1CN(C(=O)c2ccnc(OC(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858738
O=C(NCC(F)=C1CN(C(=O)C(O)Cc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858740
Cc1ccnc(O)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858742
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCC3)CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15860602
O=C(NCC(F)=C1CN(C(=O)c2cc(CC3CCC3)c[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15860604
Cc1csc2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)n12 s275592__15865378__15841170__15860608
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc2nc[nH]c12 s275592__15865378__15841170__15860610
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@@](F)(CO)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860612
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)=NO1 s275592__15865378__15841170__15860614
O=C(NCC(F)=C1CN(C(=O)c2snc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15860616
CC(C)C1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860618
C=CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15860620
Cc1cccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nn12 s275592__15865378__15841170__15860624
O=C(NCC(F)=C1CN(C(=O)CC2CC3(CCC3)CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15860626
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2Cc3ccccc3N2)C1)c1cc(O)no1 s275592__15865378__15841170__15860628
O=C(NCC(F)=C1CN(C(=O)C2=CC3CCCCCC23)C1)c1cc(O)no1 s275592__15865378__15841170__15860630
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2C(=O)NCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860632
COC(=O)[C@@H]1C[C@@]1(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15860636
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccc(F)cc3N2)C1)c1cc(O)no1 s275592__15865378__15841170__15860638
O=C(NCC(F)=C1CN(C(=O)c2nnc3n2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860640
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCCC[C@H]2O)C1)c1cc(O)no1 s275592__15865378__15841170__15860642
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C=CCCC1 s275592__15865378__15841170__15860644
O=C(NCC(F)=C1CN(C(=O)C2=CNc3ncnn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860646
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(F)cccn23)C1)c1cc(O)no1 s275592__15865378__15841170__15860648
O=C(NCC(F)=C1CN(C(=O)c2ccn3ccnc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15860650
O=C(NCC(F)=C1CN(C(=O)CC2CC3(CC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860654
CCCN1C(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860662
Cc1ccc(F)c(O)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860664
O=C(NCC(F)=C1CN(C(=O)c2cnccc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860666
CC1CCCC(O)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860668
O=C(NCC(F)=C1CN(C(=O)CSC2CCCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15860670
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1C s275592__15865378__15841170__15860672
CC12CC(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CO1)C2 s275592__15865378__15841170__15860676
O=C(NCC(F)=C1CN(C(=O)C2(F)CC3(CCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860678
O=C(NCC(F)=C1CN(C(=O)C2CCn3nccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860684
CC1CCCc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nn21 s275592__15865378__15841170__15860686
CN(C)C1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860688
O=C(NCC(F)=C1CN(C(=O)c2ccc3sncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860690
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c2c1CCCC2 s275592__15865378__15841170__15860694
CCc1[nH]c(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860696
O=C(NCC(F)=C1CN(C(=O)C2CC3(CC(O)C3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860698
O=C(NCC(F)=C1CN(C(=O)c2ccc(CCF)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15860700
O=C(NCC(F)=C1CN(C(=O)C23COC(CF)(C2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860702
CN1C(=O)OCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860704
O=C(NCC(F)=C1CN(C(=O)C2CCCCC23OCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15860708
CCSC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860710
CCn1ccnc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860712
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cncn1 s275592__15865378__15841170__15860714
Cc1[nH]c(C(C)(C)C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860716
Nc1nnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15860718
COc1ncc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15860720
CC(CF)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862566
CC1(C)CCCC(O)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15862570
CC(=CC1CCC(C)CC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862572
CC(Cl)=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862574
O=C(NCC(F)=C1CN(C(=O)C=Cc2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15862576
Nc1cc(Cl)cc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862578
O=C(NCC(F)=C1CN(C(=O)C2(N3CCOCC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862580
O=C(NCC(F)=C1CN(C(=O)C2(Oc3ccccc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862582
CC1(c2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)no2)CC1 s275592__15865378__15841170__15862584
CN1C(=O)NCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862588
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15862590
CCC(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862594
O=C(NCC(F)=C1CN(C(=O)C2CCCCC2F)C1)c1cc(O)no1 s275592__15865378__15841170__15862596
CC(C(=O)OC(C)(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862598
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1F s275592__15865378__15841170__15862600
O=C(NCC(F)=C1CN(C(=O)C2CCNc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15862602
CSCCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862604
CCC(F)(F)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862606
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCOC1 s275592__15865378__15841170__15862610
CC(C)(C)OC(=O)C(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862618
CC(=Cc1ccncc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862620
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CC2)CC3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15862622
Cc1ccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2c1 s275592__15865378__15841170__15862626
COc1ccccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862628
O=C(NCC(F)=C1CN(C(=O)C=Cc2cc(F)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15862630
N#CC(=Cc1ccoc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862632
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CO[C@@H]3CCCC[C@H]23)C1)c1cc(O)no1 s275592__15865378__15841170__15862634
O=C(NCC(F)=C1CN(C(=O)C=Cc2cc3ccccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__15862640
Cn1ncc(Cl)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862644
Cc1cc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc2o1 s275592__15865378__15841170__15862646
O=C(NCC(F)=C1CN(C(=O)C=Cc2cscn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862648
N#CC(=Cc1ccco1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862650
O=C1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15862656
Cn1nnc2c1NCCC2C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862658
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2COC[C@H]2O)C1)c1cc(O)no1 s275592__15865378__15841170__15862660
O=C(NCC(F)=C1CN(C(=O)CSc2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862662
Cc1cc(F)sc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862664
Cc1ccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15862668
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@H]3[C@@H](C2)C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15862670
CCOC(=O)c1conc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862674
O=C(NCC(F)=C1CN(C(=O)C2=CC3(CCOCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862676
O=C(NCC(F)=C1CN(C(=O)c2cnc3occc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862680
O=C1CCCC(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15862682
CCOC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__15862684
C=CCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863866
COC1C[C@@H]2CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C[C@H]12 s275592__15865378__15841170__15863868
O=C(NCC(F)=C1CN(C(=O)C2C3CCOCC32)C1)c1cc(O)no1 s275592__15865378__15841170__15863872
Cc1cnn(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863874
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cnnc1 s275592__15865378__15841170__15863876
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(F)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15863878
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2CC2C1 s275592__15865378__15841170__15863882
O=C(NCC(F)=C1CN(C(=O)C=CCF)C1)c1cc(O)no1 s275592__15865378__15841170__15863884
O=C(NCC(F)=C1CN(C(=O)C2(CC(F)F)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863888
O=C(NCC(F)=C1CN(C(=O)C(F)CC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863892
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__15863894
Cc1c(O)cc(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863896
Cc1cnn2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nc12 s275592__15865378__15841170__15863898
CC(C)CCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863902
O=C(NCC(F)=C1CN(C(=O)C2(c3cccnc3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863904
CN1CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863906
O=C(NCC(F)=C1CN(C(=O)c2ccnc3c2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863910
O=C(NCC(F)=C1CN(C(=O)C=CCn2cncn2)C1)c1cc(O)no1 s275592__15865378__15841170__15863914
CC1CCC(C(C)C)C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863916
O=C(NCC(F)=C1CN(C(=O)C=CC2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863918
CSc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863920
O=C(NCC(F)=C1CN(C(=O)CNc2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__15863922
O=C(NCC(F)=C1CN(C(=O)Cc2sc(O)nc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15863924
N#Cc1ccccc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863926
Cc1nnc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15863928
CC(C)(C)O[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863930
N#Cc1cccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863932
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)n(CCF)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863934
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863936
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(N)c1 s275592__15865378__15841170__15863938
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c1C s275592__15865378__15841170__15863940
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CN1CCOCC1 s275592__15865378__15841170__15863942
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__15863944
O=C(NCC(F)=C1CN(C(=O)c2ncc3c(F)cccn23)C1)c1cc(O)no1 s275592__15865378__15841170__15863946
CCOC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15863948
CCOC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15863954
Cc1cc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__15863956
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sn1 s275592__15865378__15841170__15863960
O=C(NCC(F)=C1CN(C(=O)c2ncoc2C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863962
O=C1N[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15863964
COC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863966
CC(O)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863968
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccco1 s275592__15865378__15841170__15863970
Cc1nn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)o1 s275592__15865378__15841170__15863972
O=C(NCC(F)=C1CN(C(=O)c2cccc3cccc(O)c23)C1)c1cc(O)no1 s275592__15865378__15841170__15863974
N#CCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863976
O=C(NCC(F)=C1CN(C(=O)c2cnn3ccsc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863978
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cnc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15863982
O=C(NCC(F)=C1CN(C(=O)C(O)c2cccc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856784
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]n1 s275592__15865378__15841170__15856786
Cn1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C#N s275592__15865378__15841170__15856788
O=C(NCC(F)=C1CN(C(=O)c2cc3ncccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15856790
O=C(NCC(F)=C1CN(C(=O)C2(CO)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856792
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15856796
O=C(NCC(F)=C1CN(C(=O)c2ccc(CO)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856800
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(F)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15856804
CSc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__15856806
CCC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15841170__15856808
O=C(NCC(F)=C1CN(C(=O)c2cc([N+](=O)[O-])cnc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856812
O=C(NCC(F)=C1CN(C(=O)[C@H](O)c2ccccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15856814
O=C(NCC(F)=C1CN(C(=O)c2csc([N+](=O)[O-])c2)C1)c1cc(O)no1 s275592__15865378__15841170__15856816
O=C1Cc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2N1 s275592__15865378__15841170__15856818
O=C(NCC(F)=C1CN(C(=O)c2cc([N+](=O)[O-])c[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15856822
Cc1cc(C)c(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856824
O=C(NCC(F)=C1CN(C(=O)c2cccc(Cl)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856826
O=C(NCC(F)=C1CN(C(=O)CCSc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15856828
O=C(NCC(F)=C1CN(C(=O)c2ccno2)C1)c1cc(O)no1 s275592__15865378__15841170__15856830
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15856834
O=C(NCC(F)=C1CN(C(=O)[C@@H]2Cc3ccccc3N2)C1)c1cc(O)no1 s275592__15865378__15841170__15856836
CNc1snc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856838
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15856842
O=C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15856844
Nc1c(Cl)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856846
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1N s275592__15865378__15841170__15856850
Nc1cc(F)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856854
Cc1nsc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856856
O=C(NCC(F)=C1CN(C(=O)C2CNc3ccccc3O2)C1)c1cc(O)no1 s275592__15865378__15841170__15856858
O=C(NCC(F)=C1CN(C(=O)CC2C=CS(=O)(=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15856860
CC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856862
O=C(NCC(F)=C1CN(C(=O)CSc2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15856864
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15856868
COc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856870
O=C(NCC(F)=C1CN(C(=O)c2c(O)cccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856872
[N-]=[N+]=NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856874
Cc1c(N)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856876
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15856878
Cc1nn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1[N+](=O)[O-] s275592__15865378__15841170__15856880
CN(C)c1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856882
O=C(NCC(F)=C1CN(C(=O)C2=CCCSC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856886
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__15856890
Cc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sc1C s275592__15865378__15841170__15856894
CCN1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15856896
C[C@@](O)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15856898
O=C(NCC(F)=C1CN(C(=O)C2(O)CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856902
O=C(NCC(F)=C1CN(C(=O)C=C2CN3CCC2CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15858744
CCCC(CCC)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858748
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15858750
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)o2)C1)c1cc(O)no1 s275592__15865378__15841170__15858752
CCCC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CCC s275592__15865378__15841170__15858754
O=C(NCC(F)=C1CN(C(=O)c2cccc3nc(O)ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15858756
Cc1cc(=O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__15858758
O=C(NCC(F)=C1CN(C(=O)C=C2CCSCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858760
CON=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858762
N#CC1(c2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2)CC1 s275592__15865378__15841170__15858764
C#CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858766
Nc1ncc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858768
O=C(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(O)cc1 s275592__15865378__15841170__15858770
CCSc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858772
O=C(NCC(F)=C1CN(C(=O)C[C@@H](O)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15858774
Nc1c(Cl)cc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858776
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1[N+](=O)[O-] s275592__15865378__15841170__15858780
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc1Cl s275592__15865378__15841170__15858782
Cc1ncnc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858784
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15841170__15858790
CC(C)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N=[N+]=[N-] s275592__15865378__15841170__15858792
COC(=O)c1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15858794
COC(=O)CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858796
CC1(F)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15858798
Cn1ncc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858800
Nc1nc(O)c(Cl)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858802
CCSc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858804
CCC(C)(OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858808
Nc1cc(F)cc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858810
CC(C)(C)CCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858812
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(CO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858816
CCOC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15858818
CCCC(CCCO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858820
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15858822
COC(=O)[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15858824
CC(O)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15858826
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCN1 s275592__15865378__15841170__15858828
CC(C)[C@H](O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858830
CSC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15858832
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(O)c1 s275592__15865378__15841170__15858834
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15841170__15858840
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1C s275592__15865378__15841170__15858842
O=C(NCC(F)=C1CN(C(=O)C(O)c2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15858844
CC(O)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15841170__15858846
O=C(NCC(F)=C1CN(C(=O)c2cccc(=O)n2O)C1)c1cc(O)no1 s275592__15865378__15841170__15858848
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(O)cc1 s275592__15865378__15841170__15858850
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15858852
O=C(NCC(F)=C1CN(C(=O)CCCCCn2cnnn2)C1)c1cc(O)no1 s275592__15865378__15841170__15858856
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15858858
Nc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1[N+](=O)[O-] s275592__15865378__15841170__15858860
COc1cccnc1C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858862
Cn1ccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc21 s275592__15865378__15841170__15858864
CN(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15858866
CCCCCCC(O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860724
O=C(NCC(F)=C1CN(C(=O)c2ccnn2CCF)C1)c1cc(O)no1 s275592__15865378__15841170__15860726
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(C)c1C#N s275592__15865378__15841170__15860728
COC(=O)[C@@H]1O[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C[C@H]1C s275592__15865378__15841170__15860732
O=C(NCC(F)=C1CN(C(=O)c2cc(F)c(CO)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860734
O=C(NCC(F)=C1CN(C(=O)c2cccc3nc[nH]c(=O)c23)C1)c1cc(O)no1 s275592__15865378__15841170__15860738
N#Cc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860740
O=C(NCC(F)=C1CN(C(=O)c2cnc(F)c(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860742
CC1=NS(=O)(=O)NC=C1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860744
N#Cc1ccnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860746
O=C(NCC(F)=C1CN(C(=O)CC=C(Cl)Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15860748
CN(C)C(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860752
Cc1cc(C#N)cc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860754
C#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860756
O=C(NCC(F)=C1CN(C(=O)c2ccnc(CO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860758
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(OC)n1 s275592__15865378__15841170__15860760
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)[C@@H]1CCC[C@H]1O s275592__15865378__15841170__15860762
O=C(NCC(F)=C1CN(C(=O)C2(F)C(F)(F)C2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860764
O=C(NCC(F)=C1CN(C(=O)c2cnc3cc(O)ccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860766
Cc1ccc(C(=O)C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15860768
CC(C)(C)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15860770
N#Cc1cncc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860772
C[C@H]1c2cn[nH]c2CC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860774
CC(=O)Nc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860776
CCC1CN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860778
Nc1ccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15860780
O=C1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15860782
Cc1cn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860784
O=C(NCC(F)=C1CN(C(=O)C2CN(C3CCOCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860786
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(Cl)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15860790
O=C(NCC(F)=C1CN(C(=O)C2(N3CCCC3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860792
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15860798
CC(=O)CCC(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860800
C=CC=CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860802
COC(=O)[C@@H]1C[C@]1(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860804
C=CCC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860806
O=C(NCC(F)=C1CN(C(=O)COCc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15860808
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__15860810
O=C(NCC(F)=C1CN(C(=O)COc2nc(=O)[nH]c(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15860812
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC(C2)S3)C1)c1cc(O)no1 s275592__15865378__15841170__15860814
O=C(C=CCl)NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860816
Cn1ncc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ncnc21 s275592__15865378__15841170__15860818
CCc1ccc(C(C)=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15860820
O=C(NCC(F)=C1CN(C(=O)C=Cc2cncc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860822
COC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15860824
C#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15860826
CN1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860828
CCCC=CC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860832
CC1(C)OCC(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15860834
O=C(NCC(F)=C1CN(C(=O)C2CCOC3(CCCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860836
COC(=O)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15860838
O=C(NCC(F)=C1CN(C(=O)Cc2nc(C3CC3)cs2)C1)c1cc(O)no1 s275592__15865378__15841170__15860840
O=C(NCC(F)=C1CN(C(=O)C2CC=CCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15860842
O=C(NCC(F)=C1CN(C(=O)C23CCOC2CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__15860844
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(C#N)cc1 s275592__15865378__15841170__15860846
O=C(NCC(F)=C1CN(C(=O)C2CCCNS2(=O)=O)C1)c1cc(O)no1 s275592__15865378__15841170__15862686
CC(C)(C)c1nnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15862690
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(c2)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862692
O=C(NCC(F)=C1CN(C(=O)C=CCCCCCCCO)C1)c1cc(O)no1 s275592__15865378__15841170__15862694
O=C(NCC(F)=C1CN(C(=O)Cc2c[nH]c3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15862696
CCCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15862698
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC(C3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862700
Cn1ccnc1C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862702
O=C(NCC(F)=C1CN(C(=O)C=Cc2ncco2)C1)c1cc(O)no1 s275592__15865378__15841170__15862704
Cc1nc(C2CC2)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862706
COC(=O)C(OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862708
CC(=O)N[C@H]1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15862710
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(C)(C)O1 s275592__15865378__15841170__15862712
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ccc2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15862714
O=C(NCC(F)=C1CN(C(=O)C2(F)C#CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862716
CC(CC1CCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862718
Cc1nsc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15862722
O=C(NCC(F)=C1CN(C(=O)C2CCC3(C2)N=N3)C1)c1cc(O)no1 s275592__15865378__15841170__15862724
CC1(C)C=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15862726
O=C(NCC(F)=C1CN(C(=O)CCC=CBr)C1)c1cc(O)no1 s275592__15865378__15841170__15862728
O=C(NCC(F)=C1CN(C(=O)CCc2ccn[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15862730
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n2ncnc2n1 s275592__15865378__15841170__15862732
CC12CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(C1)C1(CCC1)O2 s275592__15865378__15841170__15862734
O=C(NCC(F)=C1CN(C(=O)c2cnnn2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862736
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCCO1 s275592__15865378__15841170__15862738
COC(=O)[C@@H]1[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(F)F s275592__15865378__15841170__15862742
CC1CCC(F)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15862744
O=C(NCC(F)=C1CN(C(=O)C2CCC3(C2)CC3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15862746
O=C(NCC(F)=C1CN(C(=O)C(F)=Cc2c[nH]cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862748
O=C(NCC(F)=C1CN(C(=O)Cc2ccncc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15862750
CS(C)(=O)=NC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862754
CCN1CCOCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862758
O=C(NCC(F)=C1CN(C(=O)Cc2nnc3n2CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862760
O=C(NCC(F)=C1CN(C(=O)Cc2nnc3n2CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862762
CC1(C)CCOC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862764
O=C(NCC(F)=C1CN(C(=O)c2nc3ccccn3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15862766
O=C(NCC(F)=C1CN(C(=O)C2(Cc3cnn[nH]3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862768
CC12CC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(C1)C1(COC1)O2 s275592__15865378__15841170__15862770
CC1(C)CC(O)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15862772
COC(=O)CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15862774
O=C(NCC(F)=C1CN(C(=O)c2ccc3cccc(O)c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862778
CC(=Cc1c[nH]cn1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862782
Cc1cc(O)c(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862784
O=C(NCC(F)=C1CN(C(=O)Cn2nnnc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862786
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc(O)c1Cl s275592__15865378__15841170__15862788
Cc1ccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc2c1 s275592__15865378__15841170__15862790
CC1(C)OC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15862796
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__15862798
COc1cc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sn1 s275592__15865378__15841170__15862800
CN(C)C(=O)C#CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862802
CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1(F)Cl s275592__15865378__15841170__15863986
CC(=O)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15863988
CC1(C)OCC2CC21C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863990
C#C[C@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863992
CCN1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1=O s275592__15865378__15841170__15863994
CC(C)CCCC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863996
O=C(NCC(F)=C1CN(C(=O)C23CCC(CC2=O)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15863998
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1O s275592__15865378__15841170__15864000
O=C(NCC(F)=C1CN(C(=O)[C@H]2Cc3ccccc3N2)C1)c1cc(O)no1 s275592__15865378__15841170__15864002
O=C(NCC(F)=C1CN(C(=O)C2CN(C3CCCCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864010
[N-]=[N+]=NC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15864012
CON1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15864014
O=C(NCC(F)=C1CN(C(=O)CN2CCN(C3CC3)C2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15864016
[N-]=[N+]=N[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15864020
Cn1nccc1C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864022
CC12CCCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CO1)C2 s275592__15865378__15841170__15864024
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2c1CCOC2 s275592__15865378__15841170__15864026
Cc1cccnc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864032
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC1 s275592__15865378__15841170__15864034
Cc1ccc2c(C)c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)[nH]c2c1 s275592__15865378__15841170__15864040
COCc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__15864042
Cc1nc(CO)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864044
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(C2CC2)=NO1 s275592__15865378__15841170__15864046
CC(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15864048
CC(C)(C)c1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864050
N#CCCSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864052
COC1CN2CCCC2(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15864054
O=C(NCC(F)=C1CN(C(=O)C=Cc2ncc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15864060
O=C(NCC(F)=C1CN(C(=O)c2cncc(-c3ccoc3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864062
CC(=Cc1ccc(F)cc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864064
O=C(NCC(F)=C1CN(C(=O)c2cccc3cnnn23)C1)c1cc(O)no1 s275592__15865378__15841170__15864066
CC(=O)NC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15864068
CNC(=O)N[C@@H](C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864072
O=C(NCC(F)=C1CN(C(=O)C2CC(C3CC3)=NO2)C1)c1cc(O)no1 s275592__15865378__15841170__15864074
O=C(NCC(F)=C1CN(C(=O)C23CCC(F)(CC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15864076
CNc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864080
O=C(NCC(F)=C1CN(C(=O)C2CC(C3CCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15864082
Nc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15864084
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(c2)CCCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15864086
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C1CC1 s275592__15865378__15841170__15864088
Cc1ccc2ncccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864090
O=C(NCC(F)=C1CN(C(=O)C=Cc2nc3ccccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15864092
[N-]=[N+]=Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1O s275592__15865378__15841170__15864094
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)OC s275592__15865378__15841170__15864096
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C1CCC1 s275592__15865378__15841170__15864098
O=C(NCC(F)=C1CN(C(=O)Cc2ccn3cncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15864100
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC=CCC1 s275592__15865378__15841170__15864102
CC(=O)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15864104
O=C(NCC(F)=C1CN(C(=O)C2(C(=O)NC3CC3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856906
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cccn1 s275592__15865378__15841170__15856910
COC(=O)N[C@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15856912
COC(=O)NC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15856914
O=C(NCC(F)=C1CN(C(=O)CSCC2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15856916
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15856920
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856922
CCC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15856924
CCSC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15856926
COC(=O)N1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856928
Cc1cc(C)c(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15856930
CCSc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15856932
CCCC(NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856936
COc1ccc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15856938
O=C(NCC(F)=C1CN(C(=O)c2cscn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856940
CCCCc1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15856942
Nc1nc(Cl)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856944
CC(c1ccccc1)C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856946
CCC(Nc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856948
O=C(NCC(F)=C1CN(C(=O)CNc2nccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15856954
CNC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15856956
Cc1cc([N+](=O)[O-])ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856958
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccnc1F s275592__15865378__15841170__15856960
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__15856962
CC1OC(=O)NC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856964
O=C(NCC(F)=C1CN(C(=O)CN2CCOC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15856968
CC=C(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856970
O=C(NCC(F)=C1CN(C(=O)C23CCCC2CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15856974
Cc1[nH]nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15856978
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C2=CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15856980
O=C(NCC(F)=C1CN(C(=O)CC23CC(C2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15856982
CC1(Br)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856986
O=C(NCC(F)=C1CN(C(=O)C=C2CCOc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15856988
O=C(NCC(F)=C1CN(C(=O)c2cncc(F)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856990
Cc1cccn2nc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__15856992
C#CCC(CC#C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15856994
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2cnccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15856996
O=C(NCC(F)=C1CN(C(=O)c2c(F)ccc(O)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15856998
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15857000
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)O s275592__15865378__15841170__15857002
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCCC3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15857008
COc1ccnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858870
COC(=O)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858872
CC(CS(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858874
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C#N s275592__15865378__15841170__15858876
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ccc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15858878
COC(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858882
CC(C)(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15858886
N#Cc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858888
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc(Cl)c1F s275592__15865378__15841170__15858890
Nc1nc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc2[nH]1 s275592__15865378__15841170__15858892
O=C(NCC(F)=C1CN(C(=O)COC2C#CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858894
N#CC(=CC1CC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858896
COc1cccc(O)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858898
CCc1cnoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858900
O=C(NCC(F)=C1CN(C(=O)C2CN(CC(F)F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15858904
NS(=O)(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858910
NS(=O)(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858912
O=C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)c(F)c1 s275592__15865378__15841170__15858916
COc1ccc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15858918
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15858920
COC(=O)NCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858924
Cc1ccc(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858926
COC(=O)NC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15858928
COC(=O)NC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858930
CC(C)Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15858936
COc1cccc(C(O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858942
CC(C)c1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858946
Nc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858948
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15858950
COc1cc(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__15858952
N#Cc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858958
CSc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15858964
CC(=O)c1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858966
O=C(NCC(F)=C1CN(C(=O)C=C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15858972
COC(=O)c1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858976
CC(C)(C#N)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858978
Cc1cnc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15858980
CSC(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858982
O=C(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)NC1CC1 s275592__15865378__15841170__15858984
CC(O)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15858986
CC(=O)OCC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858988
COCC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858990
CC(C)(CCCO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860848
Cn1nnc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15841170__15860850
CCCc1nsc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860852
Cn1ncc(C#N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860854
NC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15860860
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15860862
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCOC1 s275592__15865378__15841170__15860864
O=C(NCC(F)=C1CN(C(=O)c2ccc3nc[nH]c(=O)c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860866
Cc1cn2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc2s1 s275592__15865378__15841170__15860868
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc1F s275592__15865378__15841170__15860870
O=C(NCC(F)=C1CN(C(=O)C2(c3ccncc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860872
O=C(NCC(F)=C1CN(C(=O)c2coc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860876
O=C(NCC(F)=C1CN(C(=O)C2CCc3cnnn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860880
CCOc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc(=O)c1 s275592__15865378__15841170__15860882
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2cc[nH]c2n1 s275592__15865378__15841170__15860884
O=C(NCC(F)=C1CN(C(=O)Cc2c[nH]c3cccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__15860886
CN(C)[C@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860888
CSc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15860890
O=C(NCC(F)=C1CN(C(=O)C2CCCCNC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15860894
O=C(NCC(F)=C1CN(C(=O)c2nncn2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860896
CC1(C)[C@@H](C(F)F)[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860900
O=C(NCC(F)=C1CN(C(=O)C2CCC(OC(F)F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860902
O=C(NCC(F)=C1CN(C(=O)C23CC4CC(CC(C4)O2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860904
O=C(NCC(F)=C1CN(C(=O)CC2(C3CC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860906
CC(C)[C@@H](NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860908
Cc1cccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnn12 s275592__15865378__15841170__15860910
O=C(NCC(F)=C1CN(C(=O)c2cc(C3CCC3)no2)C1)c1cc(O)no1 s275592__15865378__15841170__15860912
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15860916
Cc1c[nH]c2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__15860918
CN(C)CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15860920
COC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CC1)C2 s275592__15865378__15841170__15860922
CC1CCCC(C)N1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860924
O=C(NCC(F)=C1CN(C(=O)C(F)C2CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860926
O=C(NCC(F)=C1CN(C(=O)c2nn[nH]c2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860928
CN(C)C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860930
CN(C)CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860932
O=C(NCC(F)=C1CN(C(=O)c2cncc(-n3cccn3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15860934
C#Cc1ccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15860936
Cc1ccc(C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C2CC2)cc1 s275592__15865378__15841170__15860938
CCOC(=O)[C@H]1C[C@](F)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15860940
CN(C)[C@H]1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860942
CN1CC=CCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860944
CCc1nc2ccccn2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860948
O=C(NCC(F)=C1CN(C(=O)C2CNc3ncnn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860950
O=C(NCC(F)=C1CN(C(=O)CCC23CCC(CC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15860952
Cc1cc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__15860954
COc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(F)c1F s275592__15865378__15841170__15860958
Cc1ccc2ncnc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c2c1 s275592__15865378__15841170__15860960
O=C(NCC(F)=C1CN(C(=O)C(O)CCn2cncn2)C1)c1cc(O)no1 s275592__15865378__15841170__15860962
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@](F)(CO)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860964
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCCCCC32)C1)c1cc(O)no1 s275592__15865378__15841170__15860966
CC1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(C)O1 s275592__15865378__15841170__15860968
N#C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862806
CCCC(CC)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862808
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862812
C=C(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862818
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)OCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15862822
Cc1nn2c(c1C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)NCCC2 s275592__15865378__15841170__15862824
CC1(C)C(O)CC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862826
O=C(NCC(F)=C1CN(C(=O)c2conc2C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862828
CCc1nc(N)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862830
O=C(NCC(F)=C1CN(C(=O)C=Cc2cnccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862832
N#Cc1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15862834
CCC(=O)N1CSC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862836
O=C(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccncc1 s275592__15865378__15841170__15862838
CCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1 s275592__15865378__15841170__15862840
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(n2)CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862842
CCOC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC=CC1 s275592__15865378__15841170__15862844
CC(F)(F)C(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862848
O=C(NCC(F)=C1CN(C(=O)C2CCCC3(CCC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862850
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__15862852
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@H](C(F)(F)F)O2)C1)c1cc(O)no1 s275592__15865378__15841170__15862854
O=C(NCC(F)=C1CN(C(=O)C2(n3cnnn3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862856
CNc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15862858
O=C(NCC(F)=C1CN(C(=O)C2CCc3nnnn3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862860
O=C(NCC(F)=C1CN(C(=O)CSc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15862862
O=C(NCC(F)=C1CN(C(=O)CC2CCC(F)(F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862864
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3[nH]nnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862866
O=C1Cc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2N1 s275592__15865378__15841170__15862868
O=C(NCC(F)=C1CN(C(=O)C2CC3CC(O)CC(C3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862870
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc(N)n1 s275592__15865378__15841170__15862872
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@@H](O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15862874
CC(=Cc1ccco1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862876
O=C(NCC(F)=C1CN(C(=O)CCC2CC2(Cl)Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15862878
COC(=O)C1CCOC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862880
CC1(C)CC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862884
O=C(NCC(F)=C1CN(C(=O)c2ccn3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15862890
O=C(NCC(F)=C1CN(C(=O)CCc2cccnc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15862898
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15841170__15862900
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2C(=O)CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862902
O=C(NCC(F)=C1CN(C(=O)c2cnc(S)n2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862904
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__15862906
Cc1sc(O)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862908
O=C(NCC(F)=C1CN(C(=O)C2(c3ccncc3)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862912
CSc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862914
O=C(NCC(F)=C1CN(C(=O)C2CCC23CCOCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862916
CC1(c2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)[nH]n2)CC1 s275592__15865378__15841170__15862920
O=C(NCC(F)=C1CN(C(=O)c2cn(O)c(=O)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15862922
O=C(NCC(F)=C1CN(C(=O)c2noc3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15862924
O=C(NCC(F)=C1CN(C(=O)c2cccc(C(=O)C3CC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862926
Nc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__15864112
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(F)F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15864118
O=C(NCC(F)=C1CN(C(=O)C2=C(Cl)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864120
CCCc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15864122
Cc1cc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc1N s275592__15865378__15841170__15864124
COc1cccc(NCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864126
Cc1nnnn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864128
O=C(NCC(F)=C1CN(C(=O)c2cccc3nncn23)C1)c1cc(O)no1 s275592__15865378__15841170__15864130
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__15864132
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]2c2nc[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__15864134
O=C(NCC(F)=C1CN(C(=O)C2COC3COCC32)C1)c1cc(O)no1 s275592__15865378__15841170__15864136
O=C(NCC(F)=C1CN(C(=O)[C@@]23C[C@@H](F)[C@@H]2C3)C1)c1cc(O)no1 s275592__15865378__15841170__15864138
CC(C)(C)c1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864140
O=C(NCC(F)=C1CN(C(=O)CCc2cccc(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15864142
CC(F)(F)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]n1 s275592__15865378__15841170__15864146
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)o2)C1)c1cc(O)no1 s275592__15865378__15841170__15864148
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1CC(F)F s275592__15865378__15841170__15864150
CC12CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(CC1)OC2 s275592__15865378__15841170__15864152
CC(C)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864156
CN(C)CCOCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864158
Cc1nn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1C s275592__15865378__15841170__15864160
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CCCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15864170
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CCCCCN(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864174
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccncc1 s275592__15865378__15841170__15864176
CN1CSCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864178
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COCc1noc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15864190
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)c(F)cc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15864192
O=C(NCC(F)=C1CN(C(=O)CC2CC(O)C23CCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15864194
[N-]=[N+]=N[C@@H]1C[C@@]2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C[C@@H]12 s275592__15865378__15841170__15864196
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O=C(NCC(F)=C1CN(C(=O)C2(n3cccc3)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15864206
CN(C)C[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15864208
C[C@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__15864210
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Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ncccc2c1 s275592__15865378__15841170__15864214
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Cc1cc(N)c(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15864220
Cn1cnc(CC(O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15864224
O=C(NCC(F)=C1CN(C(=O)C23CCCC2C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15864226
Nc1cc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1Cl s275592__15865378__15841170__15864228
CCOC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15857012
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__15857014
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857016
CC(=O)OC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857018
CCOc1oc(C)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857022
N#Cc1ccc(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2)cc1 s275592__15865378__15841170__15857024
CCCCC[C@H](O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857028
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(c2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15857030
CC(=O)OC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15841170__15857036
O=C(NCC(F)=C1CN(C(=O)COCCO)C1)c1cc(O)no1 s275592__15865378__15841170__15857042
CC(=O)c1cn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__15857044
CC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)=NO1 s275592__15865378__15841170__15857048
O=C(NCC(F)=C1CN(C(=O)c2ncc(F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15857050
CC(C)(CF)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857052
CC(C)[C@@H](O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857054
O=C(NCC(F)=C1CN(C(=O)c2cnc3sccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857056
O=C(NCC(F)=C1CN(C(=O)c2n[nH]cc2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15857058
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857060
O=C(NCC(F)=C1CN(C(=O)C2CC(=O)N(C3CC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15857062
C=CCNc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15857064
CC(C)(CO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857066
O=C(NCC(F)=C1CN(C(=O)CSCc2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15857068
N=c1sccn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857070
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3c(c2)OCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15857072
O=C(NCC(F)=C1CN(C(=O)CN2CSCC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15857074
O=C(NCC(F)=C1CN(C(=O)c2cccc(CO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857078
O=C(NCC(F)=C1CN(C(=O)c2ccc3cccnc3c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857080
C=CCC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857082
Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15857086
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])cc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857088
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15857090
CSCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15857094
O=C(NCC(F)=C1CN(C(=O)c2cc([N+](=O)[O-])ccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857096
Cc1cccc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857098
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15857100
CCSc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857102
COc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857104
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1C s275592__15865378__15841170__15857106
CC(NC(=O)c1ccco1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857110
NC(=O)NC(CO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857112
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)cc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857114
O=C(NCC(F)=C1CN(C(=O)CSc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857116
O=C(NCC(F)=C1CN(C(=O)C2CC2(Cl)Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15857118
CC(C)(C)SCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857120
Cc1ccc(C=C(C#N)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15857122
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)cc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857124
CC1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)S1 s275592__15865378__15841170__15858992
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N#CCc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15858996
CC(O)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__15858998
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CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__15859004
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CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC(=O)OC1 s275592__15865378__15841170__15859010
CSc1ccccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859014
COc1ccc(F)c(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859016
Nc1cccc(C(O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859018
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Cc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)c1 s275592__15865378__15841170__15859022
CNC(=O)N1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859026
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O=C(NCC(F)=C1CN(C(=O)c2ccc3nsnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859032
O=C(NCC(F)=C1CN(C(=O)CC(O)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15859036
N#Cc1ncn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859038
CC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1=O s275592__15865378__15841170__15859040
O=C(NCC(F)=C1CN(C(=O)C2(O)CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859044
O=C(NCC(F)=C1CN(C(=O)c2cc(O)cc([N+](=O)[O-])c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859046
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccnc1Cl s275592__15865378__15841170__15859050
COC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15859052
CNC(=O)N1CCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859054
Cc1nc(N)c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(=O)[nH]1 s275592__15865378__15841170__15859056
N#CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15859058
CC1CCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859060
CC1CCC(O)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15859062
CC1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859064
Cc1cc(O)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859066
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)sc2cncn12 s275592__15865378__15841170__15859068
CC1(C)CCC(O)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15859070
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)c(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859072
O=C(NCC(F)=C1CN(C(=O)c2cc(O)cc(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859074
Nc1cc(F)c(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859076
O=C(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc[nH]1 s275592__15865378__15841170__15859082
CCOC(=O)C(CC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859084
Cn1cncc1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859088
Cc1ccsc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859094
O=C(NCC(F)=C1CN(C(=O)C(F)(F)Cc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15859096
CNc1nc(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859100
Cc1cc(Cl)nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859102
Cc1oc(C#N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859104
CCC(C)CCC(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859106
O=C(NCC(F)=C1CN(C(=O)c2cccc3cc(F)ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15859108
CN(C)c1cc(C#N)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859110
O=C(NCC(F)=C1CN(C(=O)c2cnc3ncnn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15860970
O=C(NCC(F)=C1CN(C(=O)C2Cc3cscc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15860972
CCNc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15860974
CCOc1sccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860978
O=C(NCC(F)=C1CN(C(=O)C2C3CC4C(C3)C42)C1)c1cc(O)no1 s275592__15865378__15841170__15860980
CC(C)(C)c1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860982
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)noc1C1CC1 s275592__15865378__15841170__15860984
Cn1c([N+](=O)[O-])cnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860986
O=C(NCC(F)=C1CN(C(=O)[C@@H](O)C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15860990
CC1(C)CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15860992
Cc1nn2c(C)cccc2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860994
COC(=O)[C@@H]1[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__15860996
COCC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15860998
CC1(C)CCCC(O)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15861000
C[C@]1(C(F)(F)F)C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861002
CC(Cc1ccncc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861004
CCOC(=O)[C@H]1C[C@@](F)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861008
COC1CC(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861010
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(c2)CCOC3)C1)c1cc(O)no1 s275592__15865378__15841170__15861012
CC(F)(F)[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861014
O=C(NCC(F)=C1CN(C(=O)c2nnc3ccccn23)C1)c1cc(O)no1 s275592__15865378__15841170__15861018
N#Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861020
O=C(NCC(F)=C1CN(C(=O)[C@]23C[C@@H]4C[C@@H]2C3[C@H]4O)C1)c1cc(O)no1 s275592__15865378__15841170__15861022
Nc1nccn2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c12 s275592__15865378__15841170__15861028
C[C@@H](OCCN(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861032
O=C(NCC(F)=C1CN(C(=O)c2ccc3oc(=O)oc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15861034
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCOCC3)CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15861038
CNC(=O)NC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861040
O=C(NCC(F)=C1CN(C(=O)C23COC(CCO2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15861048
CCn1cnnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861050
CCC(=Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861056
O=C(NCC(F)=C1CN(C(=O)C2(C3CCC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861058
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(=O)[nH]ncc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15861062
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@@H]3C[C@@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__15861066
CC1(C)C(C)(C)C1(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861068
C[C@@H]1C(=O)N(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(=O)[C@@H]1C s275592__15865378__15841170__15861070
CC(C)[C@@H]1CCC[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861072
COC(=O)c1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861074
CC(C)Cc1nccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861076
CCOC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__15861080
O=C(NCC(F)=C1CN(C(=O)CC2CC3(CCCC3)CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15861082
O=C(NCC(F)=C1CN(C(=O)C2CCC3(CCOCC3)O2)C1)c1cc(O)no1 s275592__15865378__15841170__15861084
O=C(NCC(F)=C1CN(C(=O)c2ccn(CCF)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15861086
COC(=O)c1oc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__15861088
O=C(NCC(F)=C1CN(C(=O)c2cnc3cn[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862930
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3ncc[nH]3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15862934
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc2ccccc12 s275592__15865378__15841170__15862938
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@H]2c2cccc(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862940
O=C(NCC(F)=C1CN(C(=O)C2(Nc3ccccc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15862942
COc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15862944
CC(=Cc1ccccn1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862946
O=C(NCC(F)=C1CN(C(=O)c2ccccc2-c2ncc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15862948
CC(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__15862950
O=C(NCC(F)=C1CN(C(=O)c2conc2C2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15862952
O=C(NCC(F)=C1CN(C(=O)Cc2csc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15862954
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(F)C1 s275592__15865378__15841170__15862956
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15862958
O=C(NCC(F)=C1CN(C(=O)c2nc(=O)[nH]c(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15862962
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(N)c1Cl s275592__15865378__15841170__15862966
CCc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15862970
Cc1cccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nccc12 s275592__15865378__15841170__15862972
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C1CCCCC1 s275592__15865378__15841170__15862978
CC(C)C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C(=O)N1 s275592__15865378__15841170__15862982
O=C(NCC(F)=C1CN(C(=O)C#CC2CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15862984
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CC[C@H]3[C@@H](C2)C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15862986
C=CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC=CC1 s275592__15865378__15841170__15862988
O=C(NCC(F)=C1CN(C(=O)C23CCCC(C2)OC3)C1)c1cc(O)no1 s275592__15865378__15841170__15862990
CC1OCCC1(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862992
O=C(C=Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862994
CC(C)(Nc1ccccn1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15862996
CC1(C)OCc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)n[nH]c21 s275592__15865378__15841170__15862998
Cc1ncc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15863006
CCc1scnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863008
Cn1ncc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)sc21 s275592__15865378__15841170__15863010
Cc1cccc(SCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863016
Cc1cccc(C(O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863018
O=C(NCC(F)=C1CN(C(=O)Cn2cc3ncccc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863022
O=C(NCC(F)=C1CN(C(=O)COCCc2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15863026
O=C1CC2CCC(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2N1 s275592__15865378__15841170__15863030
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1ncc(N)n1 s275592__15865378__15841170__15863032
C[C@@H]1C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863036
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2cncs2)C1)c1cc(O)no1 s275592__15865378__15841170__15863038
CC1(C)C2CCC1(CC(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__15863044
CC(F)(F)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863046
Cc1ccc([N+](=O)[O-])c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857136
CC(=O)NC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15857138
Nc1ccc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857140
O=C(NCC(F)=C1CN(C(=O)CCc2ccccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857146
CC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857148
Cc1ccccc1NCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857150
Cc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857154
O=C(NCC(F)=C1CN(C(=O)c2ccc3nnn(O)c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857160
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15857162
O=C(NCC(F)=C1CN(C(=O)CCN2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857164
Cc1nc(C)n(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857168
Nc1ccc2oc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2c1 s275592__15865378__15841170__15857170
N#CCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857172
O=C(NCC(F)=C1CN(C(=O)CN2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857176
O=C(NCC(F)=C1CN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1)c1cc(O)no1 s275592__15865378__15841170__15857178
CN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15857180
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)c([N+](=O)[O-])[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15857182
O=C(NCC(F)=C1CN(C(=O)CN2CCC(CO)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857184
O=C(NCC(F)=C1CN(C(=O)CCn2cc([N+](=O)[O-])cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15857186
CSc1cc(F)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857188
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1CCC#N s275592__15865378__15841170__15857190
CC(C)=C(Br)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857192
COC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857194
O=C(NCC(F)=C1CN(C(=O)CN2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857196
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCOCC1 s275592__15865378__15841170__15857200
COC(=O)C1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15857202
O=C(NCC(F)=C1CN(C(=O)CCNc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15857204
Cc1cnc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857206
CCCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15857208
CCc1n[nH]c(CC)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857210
Cn1cc[n+](CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857214
COC(=O)[C@H]1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15857216
O=C(NCC(F)=C1CN(C(=O)C=CSCc2ccco2)C1)c1cc(O)no1 s275592__15865378__15841170__15857220
CNc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15857224
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15857226
Cc1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857228
O=C(NCC(F)=C1CN(C(=O)CCCc2ccc(O)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857230
CSC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857232
Cc1cc(Cl)cc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857236
Cc1cccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cnc12 s275592__15865378__15841170__15857238
Cn1cc(C=C(C#N)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15857240
O=C(NCC(F)=C1CN(C(=O)c2cc(C(F)F)no2)C1)c1cc(O)no1 s275592__15865378__15841170__15857242
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)co1 s275592__15865378__15841170__15857244
COC(=O)c1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857246
O=C(NCC(F)=C1CN(C(=O)C2=NOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857252
O=C(NCC(F)=C1CN(C(=O)C2(C(=O)c3ccccc3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857256
COc1cccc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859116
O=C(NCC(F)=C1CN(C(=O)c2cn(C3CC3)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15859120
O=C(NCC(F)=C1CN(C(=O)COc2ccon2)C1)c1cc(O)no1 s275592__15865378__15841170__15859122
CN1CCCC(C(C)(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859126
O=C(NCC(F)=C1CN(C(=O)c2ncc3ccccc3c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15859128
O=C(NCC(F)=C1CN(C(=O)c2snc(O)c2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15859130
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(O)CC1 s275592__15865378__15841170__15859132
Cc1coc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__15859134
Cc1csc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859136
CN(C)Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15859138
CCOC(=O)CC(C)(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859140
COc1cc(C)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15859144
N#Cc1cccc(F)c1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859148
O=C(NCC(F)=C1CN(C(=O)c2occc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859150
Cn1cnc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc21 s275592__15865378__15841170__15859152
O=C(NCC(F)=C1CN(C(=O)CC2CC2(Cl)Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15859156
O=C(NCC(F)=C1CN(C(=O)Cc2cnccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15859158
CN(C)Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15859160
CC(C#N)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859162
CC(C)c1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15859164
COC(=O)c1ccoc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859166
COC(=O)Cc1occc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859170
CSc1cccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859174
Nc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859176
Cn1cc(C(O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15859178
CCC1OCCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859182
O=C(NCC(F)=C1CN(C(=O)C2CCC(=O)c3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15859184
COc1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15859186
O=C(NCC(F)=C1CN(C(=O)C23CCC(CO)(CC2)CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15859188
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)n1 s275592__15865378__15841170__15859190
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15841170__15859194
O=C(NCC(F)=C1CN(C(=O)c2cccc(-c3nnco3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859196
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2OCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15859198
CC(C)(Oc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859202
CCCc1ccc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859204
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15859208
O=C(NCC(F)=C1CN(C(=O)CN2CCC(O)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859210
O=C(NCC(F)=C1CN(C(=O)c2cc3c(cc2O)OCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15859212
CCc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__15859214
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1O s275592__15865378__15841170__15859216
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)c1 s275592__15865378__15841170__15859218
N#Cc1ccc(NCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15859220
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__15859226
Cn1cccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859228
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCN(C)CC1 s275592__15865378__15841170__15859230
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__15859236
O=C(NCC(F)=C1CN(C(=O)COc2ccsn2)C1)c1cc(O)no1 s275592__15865378__15841170__15861094
CC1(C)[C@@H]2CC[C@@]1(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C(=O)C2 s275592__15865378__15841170__15861096
O=C(NCC(F)=C1CN(C(=O)CCN2CCC(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15861098
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(=O)[nH]1 s275592__15865378__15841170__15861100
CCOC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861102
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2(CC2)C1 s275592__15865378__15841170__15861106
CN1CCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__15861108
O=C(NCC(F)=C1CN(C(=O)CCOC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861110
CC(C)(Nc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861112
CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)c1 s275592__15865378__15841170__15861114
Cn1cncc1C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861118
Cc1cccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861120
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cnccn1 s275592__15865378__15841170__15861122
CCCCC(O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861126
O=C1CCCCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__15861128
Cc1cc(C#N)c(=O)[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861130
CC1(C)Cc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2C1 s275592__15865378__15841170__15861132
COC(=O)c1cc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15861134
COC1CN(C)C(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861136
O=C(NCC(F)=C1CN(C(=O)CCCCCO)C1)c1cc(O)no1 s275592__15865378__15841170__15861138
Cc1n[nH]c2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc12 s275592__15865378__15841170__15861140
O=C(NCC(F)=C1CN(C(=O)C2=CS(=O)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861142
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2CCC1CC2 s275592__15865378__15841170__15861144
NS(=O)(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861146
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCSC1 s275592__15865378__15841170__15861148
O=C(NCC(F)=C1CN(C(=O)c2csnc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15861150
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861154
CCn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc2ccccc21 s275592__15865378__15841170__15861156
Cc1ncc([N+](=O)[O-])n1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861162
O=C(NCC(F)=C1CN(C(=O)c2ccnnc2NC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861164
COC(=O)[C@@H]1C[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861166
N#Cc1c[nH]c2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc12 s275592__15865378__15841170__15861170
Cc1conc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861172
CCOCC(N=[N+]=[N-])C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861174
O=C(NCC(F)=C1CN(C(=O)C2CCC(F)(F)CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15861176
C#Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861178
CCOC(=O)[C@@H]1CC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861180
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)c(O)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15861188
N#Cc1cccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861190
Cc1cc(C#N)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861192
CCc1noc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861194
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CN(C)C s275592__15865378__15841170__15861196
CCOCn1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15861198
COc1cccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861200
Cc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15861202
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(Cl)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861204
N#CCc1ccsc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861206
CCNc1ccc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861208
O=C(NCC(F)=C1CN(C(=O)c2cc3ccc(O)cc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15861210
O=C(NCC(F)=C1CN(C(=O)[C@@H]2CCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15861212
Nc1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863050
O=C(NCC(F)=C1CN(C(=O)CN2Cc3ccccc3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863052
CC(CCO)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863056
O=C(NCC(F)=C1CN(C(=O)C(F)=CC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863058
O=C(NCC(F)=C1CN(C(=O)[C@@H]2COC[C@H]2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863060
O=C(NCC(F)=C1CN(C(=O)c2nc3c(s2)COCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863062
CC(C)N1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1=O s275592__15865378__15841170__15863066
CC(C)(C)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15863072
COC(=O)c1nn(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863074
O=C(NCC(F)=C1CN(C(=O)CC2CC(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863076
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc(C)n1 s275592__15865378__15841170__15863078
O=C(NCC(F)=C1CN(C(=O)C(F)CC2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863080
COc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc1F s275592__15865378__15841170__15863082
O=C(NCC(F)=C1CN(C(=O)C2CCN3CCOCC23)C1)c1cc(O)no1 s275592__15865378__15841170__15863086
COC(=O)C12CC(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)(C1)C2 s275592__15865378__15841170__15863088
O=C(NCC(F)=C1CN(C(=O)C(F)CC2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863090
O=C(NCC(F)=C1CN(C(=O)C2CCC3C(CC2)C3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863092
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CC3(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863094
O=C(NCC(F)=C1CN(C(=O)c2ncccc2CO)C1)c1cc(O)no1 s275592__15865378__15841170__15863096
O=C(NCC(F)=C1CN(C(=O)C(F)=Cc2cnc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15863098
O=C(NCC(F)=C1CN(C(=O)c2cc3ccncc3c(O)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863100
O=C(NCC(F)=C1CN(C(=O)C(F)(F)CCn2cccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15863102
Cc1ncc2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cn12 s275592__15865378__15841170__15863106
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ccsc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863108
CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cccn1 s275592__15865378__15841170__15863110
O=C1CCC2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CCCC2C1 s275592__15865378__15841170__15863118
O=C1CCC(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15841170__15863120
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(n2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863122
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2CCC[C@H](C3CC3)O2)C1)c1cc(O)no1 s275592__15865378__15841170__15863128
O=C(NCC(F)=C1CN(C(=O)[C@H](O)CF)C1)c1cc(O)no1 s275592__15865378__15841170__15863130
O=C(NCC(F)=C1CN(C(=O)C2=CC3(CCOC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863132
CCC1(C)C=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863134
CCC1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863136
Cc1nnc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1C s275592__15865378__15841170__15863138
O=C(NCC(F)=C1CN(C(=O)Cn2nc3c(n2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863142
O=C(NCC(F)=C1CN(C(=O)c2cc3ccoc3cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15863144
O=C(NCC(F)=C1CN(C(=O)c2coc3c2COC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863146
O=C(NCC(F)=C1CN(C(=O)[C@H]2C[C@H](n3cnnc3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863148
CC(C(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15841170__15863150
O=C(NCC(F)=C1CN(C(=O)c2cc3n(n2)CC(F)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15863152
CCn1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863154
O=C(NCC(F)=C1CN(C(=O)C2CC3(C2)CC2(CCC2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15863156
CN1CCOCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863160
C=CCCCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15863162
CCCC(C)(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863166
COC(=O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857258
O=C(NCC(F)=C1CN(C(=O)c2cc(F)c(O)c(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857262
COCc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)n1 s275592__15865378__15841170__15857264
O=C(NCC(F)=C1CN(C(=O)C2(CCO)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857266
Nc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1O s275592__15865378__15841170__15857270
CCOC(=O)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15857272
CC(C)C(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857276
O=C(NCC(F)=C1CN(C(=O)c2cnc(O)c([N+](=O)[O-])c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857280
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)cc1N s275592__15865378__15841170__15857282
O=C(NCC(F)=C1CN(C(=O)Cc2cccc(O)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857284
CCN1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857286
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn(C)c1=O s275592__15865378__15841170__15857288
CCSCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)no1 s275592__15865378__15841170__15857290
COc1nc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857294
Cc1sc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__15857296
O=C(NCC(F)=C1CN(C(=O)C(=O)c2cc(F)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857298
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]nnc3c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857300
COC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857302
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15857304
CC(C)(O)C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857306
O=C(NCC(F)=C1CN(C(=O)C(O)c2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857308
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15857310
CC(C)(OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15841170__15857312
Cc1cc(Cl)cc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857314
Cc1c(N)cnn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857316
CC1(c2ccccc2)CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857318
CNc1nnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15857320
CC(=O)[C@@H]1C[C@H](CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__15857322
COC(=O)CSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857326
O=C(NCC(F)=C1CN(C(=O)c2nccc(Cl)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857328
N#CC1CC2(C1)CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15857330
CC(Sc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857334
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ccc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857336
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCC(C2)C3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15857338
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)c1 s275592__15865378__15841170__15857340
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)c(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857342
Nc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857346
Nc1ccc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857348
COC(=O)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857352
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1N s275592__15865378__15841170__15857354
Cc1oc(CO)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857358
O=C(NCC(F)=C1CN(C(=O)c2ccnc3ncnn23)C1)c1cc(O)no1 s275592__15865378__15841170__15857362
CC(O)(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)(F)F s275592__15865378__15841170__15857366
Cc1csc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857370
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857372
O=C(NCC(F)=C1CN(C(=O)Cc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15857374
CC(=O)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857376
O=C(NCC(F)=C1CN(C(=O)c2ccnc(Cl)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857378
O=C(NCC(F)=C1CN(C(=O)C2(O)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859240
O=C(NCC(F)=C1CN(C(=O)CSCc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15859244
O=C(NCC(F)=C1CN(C(=O)C(O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859246
O=C(NCC(F)=C1CN(C(=O)c2ccccc2CO)C1)c1cc(O)no1 s275592__15865378__15841170__15859248
O=C(NCC(F)=C1CN(C(=O)c2nc3n(n2)CCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15859254
NC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15859256
O=C(NCC(F)=C1CN(C(=O)Cn2cnnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15859258
O=C(NCC(F)=C1CN(C(=O)C2CCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15859260
Nc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cccc1[N+](=O)[O-] s275592__15865378__15841170__15859262
CSc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15859266
O=C(NCC(F)=C1CN(C(=O)C2(C(=O)NC3CC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859268
CCc1[nH]nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1[N+](=O)[O-] s275592__15865378__15841170__15859270
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2OCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15859276
CC(=O)CCCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859278
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1O s275592__15865378__15841170__15859280
C=C(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859282
Cc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1Cl s275592__15865378__15841170__15859284
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15859286
CC(C)(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859288
O=C(NCC(F)=C1CN(C(=O)c2cccc(O)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15859290
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1CC s275592__15865378__15841170__15859292
CCCn1nc(C)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859296
CC1=CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15859298
CCSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859302
CC(=O)OCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859304
CC(C)=C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859306
Cc1c(O)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859308
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1O s275592__15865378__15841170__15859310
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)c(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859314
O=C(NCC(F)=C1CN(C(=O)c2ccnc(F)c2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15859320
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15859322
Cc1cc(N)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859324
CC(C)C(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1ccnc1 s275592__15865378__15841170__15859326
COc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859328
Nc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15859330
Nc1c(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15859332
Cc1nn2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)nc2s1 s275592__15865378__15841170__15859334
O=C(NCC(F)=C1CN(C(=O)c2ccc3cnsc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859336
Cc1sncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859338
O=C(NCC(F)=C1CN(C(=O)c2ccncc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15859340
CC(=O)CSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859342
O=C(NCC(F)=C1CN(C(=O)CCSc2ccccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15859344
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15859346
CC(C)c1nnc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15859348
Cc1ccccc1C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859350
CCNc1scnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859352
N#Cc1csc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859354
CC1(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N=N1 s275592__15865378__15841170__15859356
Cc1ccc(Cl)c(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859358
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(O)no1 s275592__15865378__15841170__15859360
NC(=O)c1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15861218
CC(Oc1cccc(N)c1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861222
O=C(NCC(F)=C1CN(C(=O)COC2COC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861226
C[C@@H]1C[C@]2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C[C@H]12 s275592__15865378__15841170__15861228
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1CCO s275592__15865378__15841170__15861230
Cc1ccnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861234
O=C(NCC(F)=C1CN(C(=O)[C@@H]2NC(=O)[C@H]3CC[C@H]32)C1)c1cc(O)no1 s275592__15865378__15841170__15861236
CCc1nsc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861238
CNC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861240
CC(OC1COC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861248
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(c2)COCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15861250
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1(F)F s275592__15865378__15841170__15861252
C#Cc1cccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861254
Cn1cc([N+](=O)[O-])c(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861256
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCOC1 s275592__15865378__15841170__15861260
O=C(NCC(F)=C1CN(C(=O)[C@]23C[C@H]2[C@H](c2ccccc2)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15861266
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2COC3)C1)c1cc(O)no1 s275592__15865378__15841170__15861268
O=C(NCC(F)=C1CN(C(=O)c2nnn3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861270
CS(=O)(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15861272
N#Cc1cccc2[nH]cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c12 s275592__15865378__15841170__15861274
CN1CCOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__15861276
N#Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c2ccccc12 s275592__15865378__15841170__15861282
Cc1ccnc(N)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861284
CN1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1=O s275592__15865378__15841170__15861286
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(F)c1O s275592__15865378__15841170__15861288
O=C(NCC(F)=C1CN(C(=O)C=Cc2c(F)cccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15861290
O=C(NCC(F)=C1CN(C(=O)C=CCOC2CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861292
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__15861294
O=C(NCC(F)=C1CN(C(=O)c2cccc(C(F)F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15861296
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccsc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861298
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccncn2)C1)c1cc(O)no1 s275592__15865378__15841170__15861300
CC(=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)F s275592__15865378__15841170__15861304
CN1[C@H](C(N)=O)CC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861306
Cc1cc(F)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861310
Cc1sc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1O s275592__15865378__15841170__15861312
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC2(CC2)C1 s275592__15865378__15841170__15861316
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2CCSC3)C1)c1cc(O)no1 s275592__15865378__15841170__15861318
O=C(NCC(F)=C1CN(C(=O)C2CC3(CSC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15861320
CCOC(=O)C=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861322
O=C(NCC(F)=C1CN(C(=O)c2cccc3cc(O)ncc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861324
COC(C(=O)OC(C)(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861326
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccnn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15861328
CC1(O)CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861330
C=CCOC(=O)NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863174
O=C(NCC(F)=C1CN(C(=O)C2CCCSS2)C1)c1cc(O)no1 s275592__15865378__15841170__15863176
Cc1ccc(C(C)CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15863178
Cn1cnnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863182
O=C(NCC(F)=C1CN(C(=O)CC2C[C@@H]3COC[C@H]23)C1)c1cc(O)no1 s275592__15865378__15841170__15863184
N#Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__15863186
N#CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863188
CN(C)CCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863190
CC(Cc1ccc(C#N)cc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863192
O=C(NCC(F)=C1CN(C(=O)c2ccccc2C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863194
O=C(NCC(F)=C1CN(C(=O)c2nn[nH]c2C(F)(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863196
Cc1cc(N)n(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863198
Nc1ncn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863202
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(n2)CCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15863206
CC(=O)[C@@H]1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__15863208
CC(=O)NC(CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863210
O=C(NCC(F)=C1CN(C(=O)C2=CCCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863212
C[C@@H]1OCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863214
O=C(NCC(F)=C1CN(C(=O)c2nccc3ncccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863216
Cn1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863218
O=C(NCC(F)=C1CN(C(=O)C2CC(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863220
CCON1CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15863224
CCC(=O)N[C@@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863226
O=C(NCC(F)=C1CN(C(=O)C2C[C@H]3CC(=O)[C@@H]2C3)C1)c1cc(O)no1 s275592__15865378__15841170__15863228
COC(=O)c1nccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863230
CCC(O)C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863232
O=C(NCC(F)=C1CN(C(=O)c2ncnc3nc[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__15863234
CN(C)c1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863236
O=C(NCC(F)=C1CN(C(=O)c2ncn3cccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863240
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ncc1C#N s275592__15865378__15841170__15863244
Cc1cnc(F)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863246
O=C(NCC(F)=C1CN(C(=O)c2csc(CO)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863250
CCC(C)(C)OCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863252
CC(=O)c1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15863254
CC(C)C(=O)c1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863256
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15863258
Cn1ccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863260
Cc1ncc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15863262
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863264
O=C1NC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCO1 s275592__15865378__15841170__15863266
CCSc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863268
CCC1(CC)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863270
O=C(NCC(F)=C1CN(C(=O)c2c(O)ccc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863274
CN1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863276
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__15863278
O=C(NCC(F)=C1CN(C(=O)c2cccc3nnoc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863280
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc1F s275592__15865378__15841170__15863282
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3c(c2)NCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863284
Cc1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15863286
O=C(NCC(F)=C1CN(C(=O)C2CCN2C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863288
CC1(O)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863290
COC(=O)N[C@@H](CC(C)C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863292
CCCCCC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863294
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15855626
O=C(NCC(F)=C1CN(C(=O)C=Cc2cc3ccccc3o2)C1)c1cc(O)no1 s275592__15865378__15841170__15855628
COC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15855630
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855632
O=C(NCC(F)=C1CN(C(=O)c2cc(=O)[nH]c(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15855636
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)OCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15855638
CN(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855640
Nc1ccc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855642
Nc1cc(Cl)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855644
O=C(NCC(F)=C1CN(C(=O)c2ccc3ccccc3c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15855646
Nc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15855648
O=C(NCC(F)=C1CN(C(=O)c2ccc(Cl)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855650
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15855654
Cc1ccc(SCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15855656
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15855660
O=C(NCC(F)=C1CN(C(=O)CCC(=O)c2cccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15855662
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1[N+](=O)[O-] s275592__15865378__15841170__15855664
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3cc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15855666
CC(SC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857380
O=C(NCC(F)=C1CN(C(=O)c2cccnc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857384
O=C(NCC(F)=C1CN(C(=O)c2ccc3cc(O)ccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857392
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)n[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15857394
N#Cc1ccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15857396
CS(=O)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857402
N#CCc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857404
O=C1NC(=O)C(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15857406
O=C(NCC(F)=C1CN(C(=O)CCNc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857410
Cc1c(N)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15857412
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c2c(C)cccc12 s275592__15865378__15841170__15857416
O=C(NCC(F)=C1CN(C(=O)c2cnn(CC(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857418
CCOC1C(C)C1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857420
O=C(NCC(F)=C1CN(C(=O)C2CCCn3ccnc32)C1)c1cc(O)no1 s275592__15865378__15841170__15857422
Cc1nc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)[nH]c2s1 s275592__15865378__15841170__15857426
CC(C)[C@H](NC(N)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857428
CC1=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)Cc2ccccc2O1 s275592__15865378__15841170__15857430
Cc1cccc(C)c1NCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857436
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(C#N)c1 s275592__15865378__15841170__15857438
O=C(NCC(F)=C1CN(C(=O)C2CC2C2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857440
CNc1cc(Cl)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857444
O=C(NCC(F)=C1CN(C(=O)c2cnc(NC3CC3)s2)C1)c1cc(O)no1 s275592__15865378__15841170__15857446
O=C(NCC(F)=C1CN(C(=O)Cc2c(O)ncnc2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857448
O=C(NCC(F)=C1CN(C(=O)c2cc(-c3cccnc3)no2)C1)c1cc(O)no1 s275592__15865378__15841170__15857450
O=CNc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15857452
O=C(NCC(F)=C1CN(C(=O)C2CC2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857454
COC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15857456
N#Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1 s275592__15865378__15841170__15857458
N#CC(=Cc1ccc(O)cc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857460
O=C(NCC(F)=C1CN(C(=O)c2ccccc2C(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15857462
O=C(NCC(F)=C1CN(C(=O)c2ccnc(OCCO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857464
CC1(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15857466
COC(=O)C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15857468
CN(CCO)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857470
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__15857472
O=C(NCC(F)=C1CN(C(=O)c2ccc3ocnc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857474
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15857478
O=C(NCC(F)=C1CN(C(=O)CCF)C1)c1cc(O)no1 s275592__15865378__15841170__15857480
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15857484
O=C(NCC(F)=C1CN(C(=O)c2cc(F)n[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15857486
CC1(C)CC=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857490
O=C(NCC(F)=C1CN(C(=O)C2C=CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857492
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1N s275592__15865378__15841170__15857494
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC(=O)C1 s275592__15865378__15841170__15857496
CC(C)(C)c1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857498
O=C(NCC(F)=C1CN(C(=O)C2CCCC(O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15857500
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(=O)C1 s275592__15865378__15841170__15857502
CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841170__15859370
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Cc1cc(O)nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859430
COC(C)C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859432
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N#Cc1cscc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859436
O=C1NC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15859438
CC(C)(CS(N)(=O)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859440
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1O s275592__15865378__15841170__15859442
Cc1cc(N)c(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15859444
Nc1ncnc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc12 s275592__15865378__15841170__15859448
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CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1O s275592__15865378__15841170__15859454
O=C(NCC(F)=C1CN(C(=O)c2cnc(C=NO)s2)C1)c1cc(O)no1 s275592__15865378__15841170__15859458
CCSC(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859462
CCSc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859464
Cc1ncn2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__15859466
CC1CN(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859468
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CC(=O)NCCNC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859472
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15859476
Nc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15859478
CSCc1cccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859480
CC1CCN1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859482
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COC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC1 s275592__15865378__15841170__15859488
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Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15861338
CC(C)OC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15861340
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(Cl)s2)C1)c1cc(O)no1 s275592__15865378__15841170__15861342
Cc1ccc(N)c(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861344
CC1(C)CC2(CC2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861346
Cc1cccc2c1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)N2 s275592__15865378__15841170__15861348
O=C(NCC(F)=C1CN(C(=O)c2cn([C@@H]3CC[C@H]3O)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15861350
COC(=O)[C@@H]1CC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861354
CO[C@]12CCC[C@@]1(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CCO2 s275592__15865378__15841170__15861356
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CCc1cccc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__15861364
Cc1ncc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15861366
CCSc1cnccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861368
COc1nsc(OC)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861370
O=C(NCC(F)=C1CN(C(=O)Cc2cc(C3CC3)on2)C1)c1cc(O)no1 s275592__15865378__15841170__15861372
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Cc1cc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1F s275592__15865378__15841170__15861378
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CCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15841170__15861382
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CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(C#N)C1 s275592__15865378__15841170__15861388
COC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15861390
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CC(C)(C)C(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861394
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15861396
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CCCCOCCNC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861402
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CC1(C)CN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861410
Cn1cnnc1SCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861412
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)cc1F s275592__15865378__15841170__15861416
CS(=O)(=O)NCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861418
Cc1ccc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861422
O=C(NCC(F)=C1CN(C(=O)CCn2cccnc2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15861424
CCc1ccc(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861426
CC(=O)c1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15861428
N#Cc1cccc(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861430
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CC(C)(C)n1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15861438
O=C(NCC(F)=C1CN(C(=O)c2coc3cc(O)ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861440
Nc1nc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15861442
O=C(NCC(F)=C1CN(C(=O)CCCCN2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861444
CCn1cc([N+](=O)[O-])c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15861448
CSc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)n1 s275592__15865378__15841170__15861452
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc([N+](=O)[O-])c2)C1)c1cc(O)no1 s275592__15865378__15841170__15861454
Nc1cc(F)c(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861456
O=C(NCC(F)=C1CN(C(=O)C2(n3cncn3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863296
Cn1cccc1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863298
N#Cc1ccc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863300
Cn1c(C#N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863302
Nc1ccnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863304
O=C(NCC(F)=C1CN(C(=O)c2cc(O)nc(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863308
CO[C@H](C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863310
Cc1cc(F)cc(C(C)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15863312
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863314
Cc1nc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]c1C s275592__15865378__15841170__15863316
O=C(NCC(F)=C1CN(C(=O)c2cnn(C3CC3(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863320
Cc1cc(C)c2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2c1 s275592__15865378__15841170__15863322
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCO3)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863324
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1cnnn1 s275592__15865378__15841170__15863326
O=C(NCC(F)=C1CN(C(=O)C2CCn3c(n[nH]c3=O)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863328
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc2n1C s275592__15865378__15841170__15863330
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O=C(NCC(F)=C1CN(C(=O)C23CCC(C2)OC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863334
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__15863336
O=C1CC2(CCC2)C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15841170__15863338
O=C(NCC(F)=C1CN(C(=O)C2CC23CC(O)C3)C1)c1cc(O)no1 s275592__15865378__15841170__15863340
O=C(NCC(F)=C1CN(C(=O)Cc2cnc3ccccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863344
CN1CCC(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2)CC1 s275592__15865378__15841170__15863346
Cn1ccc([C@@H]2C[C@H]2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863348
O=C(NCC(F)=C1CN(C(=O)C=Cc2cc[nH]n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863350
Cc1c[nH]c(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863352
O=C(NCC(F)=C1CN(C(=O)c2cccc3ccnn23)C1)c1cc(O)no1 s275592__15865378__15841170__15863354
COCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15863358
O=C(NCC(F)=C1CN(C(=O)C(F)(F)Oc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15863360
O=C(NCC(F)=C1CN(C(=O)c2ccn(C3CC3(F)F)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863362
Cc1cccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)n[nH]c12 s275592__15865378__15841170__15863364
CC1(c2nocc2C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841170__15863366
Cc1ncn2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15841170__15863368
Cc1cc2nccnc2cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863370
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)Cc2ccccc2C1 s275592__15865378__15841170__15863372
CC1(C#CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15841170__15863376
O=C(NCC(F)=C1CN(C(=O)C2(F)CCC(F)(F)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863378
CC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(F)F s275592__15865378__15841170__15863380
CC(C)(C)C1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15863382
Cc1cc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__15863388
O=C(NCC(F)=C1CN(C(=O)Cn2nnc(C3CC3)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15863390
O=C(NCC(F)=C1CN(C(=O)c2cnc3c(c2)OCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15863394
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2CCC[C@H]2O)C1)c1cc(O)no1 s275592__15865378__15841170__15863396
CCCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__15863398
CN(C)CCSCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863400
[N-]=[N+]=N[C@H]1CC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15863402
Nc1ccc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2c1 s275592__15865378__15841170__15863404
COC(=O)[C@@H]1CCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863406
O=C(Nc1ncc[nH]1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863410
C[C@@H](C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1cccc(Cl)c1 s275592__15865378__15841170__15863412
O=C(NCC(F)=C1CN(C(=O)C2C(F)(F)C23CC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863414
O=C(NCC(F)=C1CN(C(=O)CCC2=CCc3ccccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15863416
N#CC(=Cc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855668
O=C(NCC(F)=C1CN(C(=O)c2c[nH]c(=O)[nH]c2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15855670
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15855672
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)oc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855674
O=C(NCC(F)=C1CN(C(=O)c2ccc([N+](=O)[O-])o2)C1)c1cc(O)no1 s275592__15865378__15841170__15855676
CCOC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855678
CC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855680
CON=Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15855682
CCCCCC(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855684
O=C(NCC(F)=C1CN(C(=O)c2c[nH]nc2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15855686
CSCCCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855690
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc(O)n1 s275592__15865378__15841170__15855692
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855696
O=C(NCC(F)=C1CN(C(=O)C2CCCC2O)C1)c1cc(O)no1 s275592__15865378__15841170__15855698
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855700
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cnc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15855704
Cc1cc(Cl)c(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15855708
CC(C)c1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__15855710
CCc1nc(C)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855714
O=C(NCC(F)=C1CN(C(=O)CNc2cccc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855716
Cc1[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)c1C s275592__15865378__15841170__15855718
O=C(NCC(F)=C1CN(C(=O)CN2CCCC2CO)C1)c1cc(O)no1 s275592__15865378__15841170__15855720
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccn3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15855724
CCCCSCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855726
CCN(CC)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855728
Cc1n[nH]c(SCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15855730
CC1CCC(=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15855732
CC(OC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855734
CNc1ncccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855738
CCc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)csc1C s275592__15865378__15841170__15855742
Cc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15855744
CC(OCc1ccccc1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855746
CCOC=C(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855752
CC(C)(C#N)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855756
CCn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15855758
CN(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCSC1 s275592__15865378__15841170__15855762
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15855764
O=C(NCC(F)=C1CN(C(=O)CN2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855766
CC(C)C(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855768
Nc1cc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15855770
COc1noc(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855772
CC(C)(C)OC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855776
COc1cc(C#N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855778
O=C(NCC(F)=C1CN(C(=O)C2=C(Cl)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855780
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)SC s275592__15865378__15841170__15855784
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CO1 s275592__15865378__15841170__15855790
CC(=O)CCC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855792
CC1CC=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857504
CC(O)C(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857506
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCOCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857508
Cc1ccnc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857510
Cc1cc(CO)oc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857514
O=C(NCC(F)=C1CN(C(=O)C2(O)CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857516
O=C(CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccn1 s275592__15865378__15841170__15857518
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)C(=O)NC3)C1)c1cc(O)no1 s275592__15865378__15841170__15857520
CCC(C)(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857522
Cn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15857524
COc1ccc(O)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857526
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)n1 s275592__15865378__15841170__15857528
O=C(NCC(F)=C1CN(C(=O)c2cc(Cl)on2)C1)c1cc(O)no1 s275592__15865378__15841170__15857530
O=C(NCC(F)=C1CN(C(=O)C2SCCCS2)C1)c1cc(O)no1 s275592__15865378__15841170__15857532
O=C(NCC(F)=C1CN(C(=O)C2CC23CCSCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15857534
C=C1CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857536
Nc1nc(C2CC2)ncc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857538
O=C(NCC(F)=C1CN(C(=O)COc2cncc(Cl)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15857540
CC1C(=O)CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1(C)C s275592__15865378__15841170__15857544
O=C(NCC(F)=C1CN(C(=O)CC2CC=CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857548
O=C(NCC(F)=C1CN(C(=O)c2cnoc2-c2ccoc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857550
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CC3)o2)C1)c1cc(O)no1 s275592__15865378__15841170__15857552
COc1cc(CO)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857554
O=C(NCC(F)=C1CN(C(=O)Cc2ccccc2CO)C1)c1cc(O)no1 s275592__15865378__15841170__15857558
CC(=O)OC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857560
CN(C)c1noc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857564
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15857566
O=C(NCC(F)=C1CN(C(=O)CC2OCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15857568
Cc1[nH]c(=O)nc(S)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857570
COC(OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857572
Cn1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc1S s275592__15865378__15841170__15857574
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(O)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857576
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC=CC1 s275592__15865378__15841170__15857578
O=C(NCC(F)=C1CN(C(=O)C(O)c2ccc(F)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857580
O=C(NCC(F)=C1CN(C(=O)CCC[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15857582
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2cccnc2)C1)c1cc(O)no1 s275592__15865378__15841170__15857584
N#CC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15857586
[N-]=[N+]=Nc1cncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857588
Cn1ccc2cccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c21 s275592__15865378__15841170__15857590
C#CCNc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857596
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(Cl)n1 s275592__15865378__15841170__15857600
Nc1cccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857602
COC(=O)c1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857604
O=C(NCC(F)=C1CN(C(=O)c2cc3c(F)cccc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15857606
CSc1ccc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15857608
O=C(NCC(F)=C1CN(C(=O)c2cccc(Cl)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15857612
COC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857614
Cc1nc2ccccn2c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857616
Cc1cccc([N+](=O)[O-])c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857618
O=C(NCC(F)=C1CN(C(=O)c2cccc([N+](=O)[O-])c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857622
CCN(CC)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857624
COC(=O)C1=NOC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859490
NC(=O)Nc1ccccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859492
CNc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(Cl)n1 s275592__15865378__15841170__15859496
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2ccccc2c1 s275592__15865378__15841170__15859498
O=C(NCC(F)=C1CN(C(=O)Cc2ccc(Cl)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15859500
O=C(NCC(F)=C1CN(C(=O)C2=CCCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859502
N#Cc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15859504
COC(=O)CSCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859506
CCn1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__15859508
COc1ccc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15859510
O=C(NCC(F)=C1CN(C(=O)C2CC3CCC(C2)C3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15859512
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1(F)F s275592__15865378__15841170__15859514
Nc1nnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859516
Cc1c(Cl)cnn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859518
CCc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15859520
CC(C)(C)C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859522
O=CNc1nc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15859526
CCCCn1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859528
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCOCC1 s275592__15865378__15841170__15859530
O=C(NCC(F)=C1CN(C(=O)C2CCSCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859532
Nc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__15859534
COCn1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859536
CCCn1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15859538
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)NCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15859540
NC(=O)C1CCN(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15859542
O=C(NCC(F)=C1CN(C(=O)C(O)C2CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859546
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841170__15859548
Cc1nc(Cl)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859550
Cc1cc(O)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859552
Cc1cccc2cc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)[nH]c12 s275592__15865378__15841170__15859554
Cn1nc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859556
O=C(NCC(F)=C1CN(C(=O)C2=CCCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15859558
Cn1cc(C#N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859560
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15841170__15859562
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15859564
O=C(NCC(F)=C1CN(C(=O)c2cnn(C3CCCC3)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859566
O=C(NCC(F)=C1CN(C(=O)C2CC2Cc2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15859568
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(c2)COCO3)C1)c1cc(O)no1 s275592__15865378__15841170__15859570
O=C(NCC(F)=C1CN(C(=O)c2cc(CO)on2)C1)c1cc(O)no1 s275592__15865378__15841170__15859574
CCNc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15859576
CC1CC(=O)NCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859578
CSCCC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859580
O=C1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15859582
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2COCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15859586
CCNc1nc(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15859588
CCNc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15859592
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)c1F s275592__15865378__15841170__15859594
O=C(NCC(F)=C1CN(C(=O)c2ccc3[nH]ncc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15859596
O=C(NCC(F)=C1CN(C(=O)c2c(O)cnc3ccccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15859600
Cc1cc(O)cc(=O)n1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859602
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCS1 s275592__15865378__15841170__15859604
O=C(NCC(F)=C1CN(C(=O)C2=CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859608
Cn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(N)n1 s275592__15865378__15841170__15859612
CC(F)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(F)cc1 s275592__15865378__15841170__15861460
Cc1csc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861462
CCC[C@H](O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861464
O=C(NCC(F)=C1CN(C(=O)C2CCCn3cnnc32)C1)c1cc(O)no1 s275592__15865378__15841170__15861466
CC(=O)N1CSC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861468
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC=CCC1 s275592__15865378__15841170__15861470
O=C(NCC(F)=C1CN(C(=O)c2csc3nccn23)C1)c1cc(O)no1 s275592__15865378__15841170__15861472
O=C1CC(c2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2)C1 s275592__15865378__15841170__15861474
Cn1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861476
CC(C)(C)n1nccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861480
CC1(C)C2CCC(C2)C1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861482
CC1(C)C2CCC1(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)CC2 s275592__15865378__15841170__15861486
C#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15861488
Cn1ncc2ncc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc21 s275592__15865378__15841170__15861490
O=C(NCC(F)=C1CN(C(=O)C2(C3CCOCC3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861492
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc3cc[nH]c23)C1)c1cc(O)no1 s275592__15865378__15841170__15861496
O=C(NCC(F)=C1CN(C(=O)CC2COCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15861498
CC(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841170__15861502
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CC(F)(F)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15861504
Cn1ncc(N)c1CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861508
O=C(NCC(F)=C1CN(C(=O)C2(n3cccn3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861510
Nc1ccnn1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861512
CC1(C)CCC=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861514
CCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c[nH]1 s275592__15865378__15841170__15861516
O=C(NCC(F)=C1CN(C(=O)c2cn3ccncc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15861518
CN(C)Cc1c[nH]c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861522
NC(=O)c1cccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861524
CC(C)(C)C1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861526
CCc1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15861528
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C(O)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861530
C#CCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCO1 s275592__15865378__15841170__15861532
O=C(NCC(F)=C1CN(C(=O)CC2(O)CCOC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861534
CCOc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15861536
CSC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)C s275592__15865378__15841170__15861540
Cn1nc(C2CCC2)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861544
C#CCCC1(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N=N1 s275592__15865378__15841170__15861546
Nc1cc(O)c(O)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861548
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CC1(O)CCC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15861552
COC1(C#N)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861554
CC1CC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861556
[N-]=[N+]=NCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15861558
Cn1ncnc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861562
O=C(NCC(F)=C1CN(C(=O)CCc2ccc(Cl)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861564
O=C1CSC[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15861570
C[C@H]1C[C@@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C[C@@H](C)O1 s275592__15865378__15841170__15861572
CC(C)n1ccnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861574
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCC(O)CC1 s275592__15865378__15841170__15861576
CC1(OCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15861580
O=C(NCC(F)=C1CN(C(=O)C(O)c2cc(F)cc(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863418
O=C(NCC(F)=C1CN(C(=O)c2coc3c2CSC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863420
CCc1occ(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863422
O=C1C[C@]2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CCCC[C@@H]2N1 s275592__15865378__15841170__15863424
Cn1nnc2cccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)c21 s275592__15865378__15841170__15863426
O=C(NCC(F)=C1CN(C(=O)c2ccnc3nccnc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863428
O=C(NCC(F)=C1CN(C(=O)C2CC3COCCN3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863430
N#Cc1c[nH]c2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cccc12 s275592__15865378__15841170__15863432
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)cn1 s275592__15865378__15841170__15863434
O=C(NCC(F)=C1CN(C(=O)C2(C(F)F)CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15863436
CC(=O)N1C[C@H](O)C[C@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863438
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3c[nH]nn3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15863440
O=C(NCC(F)=C1CN(C(=O)c2cncc3ccsc23)C1)c1cc(O)no1 s275592__15865378__15841170__15863442
CC(C)(C)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15863444
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2NCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863446
Cc1c[nH]c(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15863448
Cc1ccc2c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)coc2c1 s275592__15865378__15841170__15863452
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__15863454
O=C(NCC(F)=C1CN(C(=O)c2ccc3c(n2)CCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15863456
CC(=O)N[C@H]1CC[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15863460
Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n(C)n1 s275592__15865378__15841170__15863462
COc1ccnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15863464
O=C(NCC(F)=C1CN(C(=O)C2(C3CCCO3)CCCO2)C1)c1cc(O)no1 s275592__15865378__15841170__15863466
CC1(C)[C@H]2C[C@H](C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)C[C@H]21 s275592__15865378__15841170__15863468
NC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]1 s275592__15865378__15841170__15863472
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N1CCC1 s275592__15865378__15841170__15863476
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15863478
O=C(NCC(F)=C1CN(C(=O)c2ccn(CCO)c(=O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863480
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC12CCOCC2 s275592__15865378__15841170__15863482
O=C(NCC(F)=C1CN(C(=O)[C@H](O)Cc2c[nH]cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15863486
O=C(NCC(F)=C1CN(C(=O)C#CC2CCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863488
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CNC3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15863492
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)n(CCO)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863494
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CC(F)(F)C1 s275592__15865378__15841170__15863496
CCOCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15863500
O=C(NCC(F)=C1CN(C(=O)C2CC3(CCOC3)C2)C1)c1cc(O)no1 s275592__15865378__15841170__15863502
CCC(CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)CN(C)C s275592__15865378__15841170__15863504
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n[nH]c1=O s275592__15865378__15841170__15863506
O=C(NCC(F)=C1CN(C(=O)[C@H]2CC2(F)F)C1)c1cc(O)no1 s275592__15865378__15841170__15863508
CC(C)c1cnn(C)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863512
CCCCc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cs1 s275592__15865378__15841170__15863514
COCC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C=CCC1 s275592__15865378__15841170__15863516
O=C(NCC(F)=C1CN(C(=O)Cc2cn[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__15863518
COCC1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCC1 s275592__15865378__15841170__15863520
Nc1ccc(C=CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15863522
CN(C)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15863524
O=C(NCC(F)=C1CN(C(=O)CON=C2CCCCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15863528
O=C(NCC(F)=C1CN(C(=O)C(F)c2ccc(F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15863532
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CS(=O)(=O)C1 s275592__15865378__15841170__15863534
O=C(NCC(F)=C1CN(C(=O)c2cccc3c2CCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15863536
O=C(NCC(F)=C1CN(C(=O)c2cn(CCCF)nn2)C1)c1cc(O)no1 s275592__15865378__15841170__15863538
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15855796
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)=NN1 s275592__15865378__15841170__15855798
CCc1csc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15855800
CC(C)(C)CC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855802
CC(=O)C(C)(C)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855804
O=C(NCC(F)=C1CN(C(=O)C2CCCc3sccc32)C1)c1cc(O)no1 s275592__15865378__15841170__15855806
O=C(NCC(F)=C1CN(C(=O)c2cnc(F)cc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15855810
O=C(NCC(F)=C1CN(C(=O)c2ccc(O)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855812
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(=O)C1 s275592__15865378__15841170__15855814
O=C(NCC(F)=C1CN(C(=O)Cc2cc[nH]c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855816
O=C(NCC(F)=C1CN(C(=O)CSC2CCOC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15855818
O=C(NCC(F)=C1CN(C(=O)Cc2ccc3[nH]ccc3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855820
O=C(NCC(F)=C1CN(C(=O)CC2CSCCS2)C1)c1cc(O)no1 s275592__15865378__15841170__15855822
CCc1nc(N)sc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855828
O=C(NCC(F)=C1CN(C(=O)C(F)(F)C2(O)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855830
O=C(NCC(F)=C1CN(C(=O)c2cc3ccncc3[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15855832
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc2ccccc12 s275592__15865378__15841170__15855834
CCCC(C)(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855836
CCOC(C)(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855838
O=C(NCC(F)=C1CN(C(=O)Cc2cccnc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15855842
Cc1nc(Cl)ccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855844
O=C(NCC(F)=C1CN(C(=O)c2cc3ccccc3cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15855846
O=C(NCC(F)=C1CN(C(=O)CSCc2cscn2)C1)c1cc(O)no1 s275592__15865378__15841170__15855848
O=C(NCC(F)=C1CN(C(=O)c2ccnc(Cl)c2F)C1)c1cc(O)no1 s275592__15865378__15841170__15855850
COC(=O)C(C)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855852
O=C(NCC(F)=C1CN(C(=O)CC2CCSCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855854
O=C(NCC(F)=C1CN(C(=O)C(CO)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855856
Cc1cc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15855858
Nc1ccc(CCCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15855860
O=C(NCC(F)=C1CN(C(=O)[C@@H]2C[C@@H]2c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855862
CC(O)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C1CCC1 s275592__15865378__15841170__15855864
N#CCCCn1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__15855866
CC1(C)CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)O1 s275592__15865378__15841170__15855868
Nc1cccn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1=O s275592__15865378__15841170__15855870
CC(=O)CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15855876
CC(O)c1cn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1 s275592__15865378__15841170__15855878
Cn1nccc1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855880
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15855882
O=C(NCC(F)=C1CN(C(=O)CC2CSC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855884
Cc1[nH]nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1[N+](=O)[O-] s275592__15865378__15841170__15855886
O=C(NCC(F)=C1CN(C(=O)c2cnc3ncccn23)C1)c1cc(O)no1 s275592__15865378__15841170__15855888
CSc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)oc1C s275592__15865378__15841170__15855890
COCCNC(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855892
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)n1ccc(C2CC2)n1 s275592__15865378__15841170__15855894
O=C(NCC(F)=C1CN(C(=O)C2(F)CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855898
Cn1cc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15855902
CC(C)c1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnn1C s275592__15865378__15841170__15855904
N#CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCCCC1 s275592__15865378__15841170__15855906
Nc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc(Cl)n1 s275592__15865378__15841170__15855908
O=C(NCC(F)=C1CN(C(=O)c2ccc3nccnc3n2)C1)c1cc(O)no1 s275592__15865378__15841170__15855910
CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1Br s275592__15865378__15841170__15855914
O=C(NCC(F)=C1CN(C(=O)CSCc2ccncc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855916
Cn1nnnc1SCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855918
CN1N=C(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1=O s275592__15865378__15841170__15857632
COC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nc1 s275592__15865378__15841170__15857634
O=C(NCC(F)=C1CN(C(=O)c2cnc[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15857636
O=C(NCC(F)=C1CN(C(=O)C2Cc3ccccc3S2)C1)c1cc(O)no1 s275592__15865378__15841170__15857638
O=C(NCC(F)=C1CN(C(=O)c2ccc3cn[nH]c3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857640
Cc1noc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857642
CCOC(=O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857644
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1[N+](=O)[O-] s275592__15865378__15841170__15857646
CCc1noc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857652
O=C1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15857654
CSc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15857656
Cc1nn(C)c(C)c1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857660
Cc1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)n1C1CC1 s275592__15865378__15841170__15857666
O=C(NCC(F)=C1CN(C(=O)Cn2ccnn2)C1)c1cc(O)no1 s275592__15865378__15841170__15857670
CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1N s275592__15865378__15841170__15857672
CN1CCCC[C@@H]1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857674
O=C(NCC(F)=C1CN(C(=O)c2cc(F)c(O)c(F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15857676
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__15857678
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3ccc(F)cc23)C1)c1cc(O)no1 s275592__15865378__15841170__15857680
O=C(NCC(F)=C1CN(C(=O)CCc2ncc(F)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15857682
C=CC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15857684
N#Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15857686
O=C(NCC(F)=C1CN(C(=O)c2ccnc(Cl)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15857688
O=C(NCC(F)=C1CN(C(=O)C2(O)COC2)C1)c1cc(O)no1 s275592__15865378__15841170__15857690
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__15857692
O=C(NCC(F)=C1CN(C(=O)c2ccc(F)nc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857694
CCC(C)C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857696
CCOC(=O)C1(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15857698
COc1ccccc1C(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857700
O=C(NCC(F)=C1CN(C(=O)c2ncncc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15857702
COc1cc(N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857704
CC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)=C1CC1 s275592__15865378__15841170__15857712
CC1CN2CCN1CC2C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857714
O=C(NCC(F)=C1CN(C(=O)C(F)(F)c2ccccc2F)C1)c1cc(O)no1 s275592__15865378__15841170__15857716
N#Cc1nc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccc1Cl s275592__15865378__15841170__15857718
CNc1cnc(Cl)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857720
Cc1ccc(C(F)(F)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15857722
Cc1cc(N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857726
CC1CC(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857728
CCn1cc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15857730
COC(=O)N[C@@H](C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857732
Cc1c(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15841170__15857734
N#CCc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1 s275592__15865378__15841170__15857738
CC1=NN(C)C(=O)C1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857742
N#Cc1cccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15857744
CC1=CC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857746
CN(C)C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15857748
CC(O)C(NC(=O)C1CC1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859616
O=C(NCC(F)=C1CN(C(=O)CN2CCCOC2=O)C1)c1cc(O)no1 s275592__15865378__15841170__15859618
O=C(NCC(F)=C1CN(C(=O)c2cncc(F)c2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15859622
O=C(NCC(F)=C1CN(C(=O)c2cccc3occc23)C1)c1cc(O)no1 s275592__15865378__15841170__15859624
CC(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15859626
CC(Sc1ccccn1)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859628
N#Cc1cc(F)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1 s275592__15865378__15841170__15859630
CC(CSC(F)(F)F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859634
Cc1cnc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15859640
Nc1cnc(Cl)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859642
CCc1cc(N)ccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859644
CCc1sc(N)nc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859646
C=CCNc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)s1 s275592__15865378__15841170__15859648
Cn1ccc2[nH]c(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc21 s275592__15865378__15841170__15859656
O=C1CCCCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859658
CN(C)CC(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859662
O=C1CCCCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15859666
O=C(NCC(F)=C1CN(C(=O)c2ccc3nc(O)cn3c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859668
CN1C2CCC1CC(C(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15859670
CCCC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859672
CC(=O)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15841170__15859674
CCCCC(O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859676
O=C(NCC(F)=C1CN(C(=O)Cc2ncncc2Cl)C1)c1cc(O)no1 s275592__15865378__15841170__15859678
CC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)[nH]1 s275592__15865378__15841170__15859680
O=C(NCC(F)=C1CN(C(=O)CC(c2ccccc2)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859682
CC(C)(O)C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15859684
Cc1cc(C#N)cnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859686
O=C1CC(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC(=O)N1 s275592__15865378__15841170__15859688
COC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)C(C)O s275592__15865378__15841170__15859690
COC(=O)c1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1C s275592__15865378__15841170__15859692
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)ccn1C1CC1 s275592__15865378__15841170__15859694
CC(C)(C)OC(=O)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859696
O=C(NCC(F)=C1CN(C(=O)CSC2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859698
O=C(NCC(F)=C1CN(C(=O)CCCC2CCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859702
CC(C)(C)c1cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)on1 s275592__15865378__15841170__15859704
COC(=O)CC(NC(C)=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859706
O=C(NCC(F)=C1CN(C(=O)c2cncc(C(F)F)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15859708
CCC(O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859710
N#Cc1c(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1F s275592__15865378__15841170__15859712
CCCCC[C@@H](O)CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859716
Cc1cc(N)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15859718
CN1C(=O)CCC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15859720
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(N)cc1 s275592__15865378__15841170__15859722
O=C(NCC(F)=C1CN(C(=O)c2ccn3ccsc23)C1)c1cc(O)no1 s275592__15865378__15841170__15859726
O=C(NCC(F)=C1CN(C(=O)C2(c3ccc(F)cn3)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15859728
O=C(NCC(F)=C1CN(C(=O)C[C@@H]2CCCC[C@H]2O)C1)c1cc(O)no1 s275592__15865378__15841170__15859730
Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(O)c1 s275592__15865378__15841170__15859732
Nc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1F s275592__15865378__15841170__15859734
CCn1nnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1C s275592__15865378__15841170__15859736
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c2cccnc12 s275592__15865378__15841170__15859738
O=C(NCC(F)=C1CN(C(=O)c2ccc(C3CCC3)nc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861582
N#Cc1cn[nH]c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861586
O=C(NCC(F)=C1CN(C(=O)C(Cc2ccccc2)C2CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15861588
O=C(NCC(F)=C1CN(C(=O)C2CCc3cn[nH]c32)C1)c1cc(O)no1 s275592__15865378__15841170__15861590
CNC(=O)CCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861592
CC1(c2ccc(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)cc2)CC1 s275592__15865378__15841170__15861594
COC(=O)C1(C)CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861598
O=C(NCC(F)=C1CN(C(=O)c2ccc(CC3CC3)s2)C1)c1cc(O)no1 s275592__15865378__15841170__15861600
O=C(NCC(F)=C1CN(C(=O)CCc2cnoc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861604
COc1cn(C)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1=O s275592__15865378__15841170__15861606
O=C(NCC(F)=C1CN(C(=O)Cc2cnsc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861610
O=C(NCC(F)=C1CN(C(=O)c2c(O)ccc(Cl)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15861612
O=C(NCC(F)=C1CN(C(=O)CC(C(F)F)n2cccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15861614
O=C(NCC(F)=C1CN(C(=O)C2CCCC23CCOCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15861616
O=C(NCC(F)=C1CN(C(=O)C=Cc2ccc(C(F)F)o2)C1)c1cc(O)no1 s275592__15865378__15841170__15861618
O=C(NCC(F)=C1CN(C(=O)c2n[nH]c3c2CCCN3)C1)c1cc(O)no1 s275592__15865378__15841170__15861620
CCc1nn(C)c(CC)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861624
C=CCC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)N(C)C s275592__15865378__15841170__15861626
O=C(NCC(F)=C1CN(C(=O)[C@]2(F)C[C@H]2c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861630
CC1OC(C)(C)OC1(C)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861632
O=C(NCC(F)=C1CN(C(=O)c2ccc(C(O)CF)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861638
COc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(F)c1N s275592__15865378__15841170__15861642
CCCC(C(=O)OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861644
O=C(NCC(F)=C1CN(C(=O)CCCCF)C1)c1cc(O)no1 s275592__15865378__15841170__15861646
CC1(C)CCCCC1=CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861648
NS(=O)(=O)C1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15841170__15861650
CCC1CC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CCC1=O s275592__15865378__15841170__15861652
COC(=O)N(C)CCCC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861658
O=C(NCC(F)=C1CN(C(=O)c2ccnc3[nH]ccc23)C1)c1cc(O)no1 s275592__15865378__15841170__15861660
O=C(NCC(F)=C1CN(C(=O)C2CC3CCCCN3C2)C1)c1cc(O)no1 s275592__15865378__15841170__15861664
O=C(NCC(F)=C1CN(C(=O)[C@@H](O)c2ccccc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861666
O=C(NCC(F)=C1CN(C(=O)c2cc(O)ccn2)C1)c1cc(O)no1 s275592__15865378__15841170__15861668
O=C(NCC(F)=C1CN(C(=O)c2cc(O)cs2)C1)c1cc(O)no1 s275592__15865378__15841170__15861670
Cc1cc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1C s275592__15865378__15841170__15861672
CC1CC(=O)NC1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861676
COc1ccc(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15861680
O=C(NCC(F)=C1CN(C(=O)c2cnsc2)C1)c1cc(O)no1 s275592__15865378__15841170__15861686
Nc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1Cl s275592__15865378__15841170__15861688
O=C(NCC(F)=C1CN(C(=O)c2cncc(Cl)n2)C1)c1cc(O)no1 s275592__15865378__15841170__15861692
Cn1nc(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15861694
COC(=O)c1cnn(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15861696
O=C1CCC(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)C1 s275592__15865378__15841170__15861700
O=C(NCC(F)=C1CN(C(=O)c2cccnc2OCCO)C1)c1cc(O)no1 s275592__15865378__15841170__15861702
CN1CCC(C)(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15861704
O=C(NCC(F)=C1CN(C(=O)c2ccccc2[N+](=O)[O-])C1)c1cc(O)no1 s275592__15865378__15841170__15855502
O=C(NCC(F)=C1CN(C(=O)c2ccc(OC(F)F)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855506
CCOc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1O s275592__15865378__15841170__15855510
COc1cc(F)cc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1N s275592__15865378__15841170__15855512
CN1CCC(O)(CC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15855514
O=C(NCC(F)=C1CN(C(=O)C2CCCSC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855516
O=C1C[C@H](C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841170__15855518
Cc1cccc(C(=O)C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15855522
Cc1ncc(N)cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855524
Cn1cc(N)c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)n1 s275592__15865378__15841170__15855526
O=C(NCC(F)=C1CN(C(=O)c2ccc(=O)n(O)c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855528
O=C(NCC(F)=C1CN(C(=O)C2CC3COCC(C2)C3=O)C1)c1cc(O)no1 s275592__15865378__15841170__15855532
CC(C)C=C(C#N)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855536
Nc1csnc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855538
COc1ccccc1C(=O)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855540
O=C(NCC(F)=C1CN(C(=O)Cn2cncn2)C1)c1cc(O)no1 s275592__15865378__15841170__15855544
O=C(NCC(F)=C1CN(C(=O)c2cc(F)cc(Cl)c2O)C1)c1cc(O)no1 s275592__15865378__15841170__15855546
COC1(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15841170__15855548
CCC(C(=O)OC)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855550
O=C(NCC(F)=C1CN(C(=O)C2CSC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855552
COCCN1CCCC1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855554
O=C(NCC(F)=C1CN(C(=O)c2cnc3sccn23)C1)c1cc(O)no1 s275592__15865378__15841170__15855556
Nc1ncc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)o1 s275592__15865378__15841170__15855558
O=C(NCC(F)=C1CN(C(=O)CC2(CO)CC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855560
N#Cc1cccc(C2(C(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)CC2)c1 s275592__15865378__15841170__15855562
CC(C)(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccc(C#N)cc1 s275592__15865378__15841170__15855564
N#Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c(Cl)c1 s275592__15865378__15841170__15855566
Nc1c(O)ccc(Cl)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855568
N#Cc1cnc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cn1 s275592__15865378__15841170__15855572
CSC(C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1)c1ccccc1 s275592__15865378__15841170__15855574
Cn1ncc2cc(CC(=O)N3CC(=C(F)CNC(=O)c4cc(O)no4)C3)ccc21 s275592__15865378__15841170__15855576
O=C(NCC(F)=C1CN(C(=O)c2ccnc3[nH]c(O)nc23)C1)c1cc(O)no1 s275592__15865378__15841170__15855580
O=C(NCC(F)=C1CN(C(=O)Cc2nccs2)C1)c1cc(O)no1 s275592__15865378__15841170__15855582
Cc1cccnc1C(F)(F)C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855584
CN1C2CCC1CC(CC(=O)N1CC(=C(F)CNC(=O)c3cc(O)no3)C1)C2 s275592__15865378__15841170__15855588
CSc1c(F)cccc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855590
CNc1cccc(CCC(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841170__15855592
O=C(NCC(F)=C1CN(C(=O)C2CCC=CO2)C1)c1cc(O)no1 s275592__15865378__15841170__15855594
O=C(NCC(F)=C1CN(C(=O)c2cn(-c3ncccn3)cn2)C1)c1cc(O)no1 s275592__15865378__15841170__15855596
Cc1nc2ccccc2n1CC(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855602
O=C(NCC(F)=C1CN(C(=O)c2cnn3c2NCCC3)C1)c1cc(O)no1 s275592__15865378__15841170__15855604
O=C(NCC(F)=C1CN(C(=O)c2ccc(-c3nnco3)cc2)C1)c1cc(O)no1 s275592__15865378__15841170__15855606
O=C(NCC(F)=C1CN(C(=O)Cc2cc(=O)[nH]c(=O)[nH]2)C1)c1cc(O)no1 s275592__15865378__15841170__15855608
O=C(NCC(F)=C1CN(C(=O)C23CCC(=O)N2CCS3)C1)c1cc(O)no1 s275592__15865378__15841170__15855610
O=C(NCC(F)=C1CN(C(=O)Cc2cccc([N+](=O)[O-])c2)C1)c1cc(O)no1 s275592__15865378__15841170__15855614
Nc1ccc([N+](=O)[O-])cc1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855616
Cc1c(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cnc2nncn12 s275592__15865378__15841170__15855618
Cc1ccc(C(=O)N2CC(=C(F)CNC(=O)c3cc(O)no3)C2)cc1[N+](=O)[O-] s275592__15865378__15841170__15855620
O=C(NCC(F)=C1CN(C(=O)C2(O)CCCC2)C1)c1cc(O)no1 s275592__15865378__15841170__15855622
Nc1cccc(F)c1C(=O)N1CC(=C(F)CNC(=O)c2cc(O)no2)C1 s275592__15865378__15841170__15855624
CCC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)COC1 s275592__15865378__15841178__15862300
CCC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15841178__15859360
CCC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)COC1 s275592__15865378__15841178__15857566
Cc1cccc(C(F)(F)C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c1 s275592__15865378__15841180__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15841182__15862300
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15841182__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CCCO1 s275592__15865378__15841182__15857566
O=C1CC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)N1 s275592__15865378__15841184__15862300
O=C1CC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)N1 s275592__15865378__15841184__15859360
O=C1CC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)N1 s275592__15865378__15841184__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnn(C2CCCC2)c1 s275592__15865378__15841186__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC1Cc1ccccc1 s275592__15865378__15841188__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc(CO)on1 s275592__15865378__15841192__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(CO)on1 s275592__15865378__15841192__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1cc(CO)on1 s275592__15865378__15841192__15857566
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)S(C)(=O)=O s275592__15865378__15842942__15859360
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC(O)CC1 s275592__15865378__15842944__15859360
CC(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC(C)(O)CC1 s275592__15865378__15842946__15859360
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(C)(C)C s275592__15865378__15842948__15862300
CC(=CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(C)(C)C s275592__15865378__15842948__15859360
CC(=CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(C)(C)C s275592__15865378__15842948__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc(S)n1C1CC1 s275592__15865378__15842950__15859360
CSc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)co1 s275592__15865378__15842952__15862300
CSc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)co1 s275592__15865378__15842952__15859360
Cc1sc(O)nc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842954__15862300
Cc1sc(O)nc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842954__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(c3ccncc3)CCC2)C1 s275592__15865378__15842956__15859360
CSc1cccnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842958__15862300
CSc1cccnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842958__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CCC12CCOCC2 s275592__15865378__15842960__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCC12CCOCC2 s275592__15865378__15842960__15859360
CC1(c2cc(C(=O)NCC(F)=C3CN(C(=O)c4nsnc4O)C3)[nH]n2)CC1 s275592__15865378__15842962__15862300
CC1(c2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)[nH]n2)CC1 s275592__15865378__15842962__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cn(O)c(=O)[nH]c1=O s275592__15865378__15842964__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cn(O)c(=O)[nH]c1=O s275592__15865378__15842964__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1noc2ncccc12 s275592__15865378__15842966__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1noc2ncccc12 s275592__15865378__15842966__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cnc2cn[nH]c2c1 s275592__15865378__15842970__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnc2cn[nH]c2c1 s275592__15865378__15842970__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(-c2ncc[nH]2)nc1 s275592__15865378__15842974__15859360
CC(=Cc1ccccn1)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842976__15862300
CC(=Cc1ccccn1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842976__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1-c1ncc[nH]1 s275592__15865378__15842978__15859360
CN(C)CCn1nccc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842980__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccccc1C1CC1 s275592__15865378__15842982__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccccc1C1CC1 s275592__15865378__15842982__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nn[nH]c1C(F)(F)F s275592__15865378__15842984__15859360
CC(=O)NC(CC(C)C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842986__15862300
CC(=O)NC(CC(C)C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842986__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1=CCCOCC1 s275592__15865378__15842988__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1=CCCOCC1 s275592__15865378__15842988__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1=CCCOCC1 s275592__15865378__15842988__15857566
C[C@@H]1OCC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15842990__15862300
C[C@@H]1OCC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15842990__15859360
C[C@@H]1OCC[C@@H]1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15842990__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1nccc2ncccc12 s275592__15865378__15842992__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC(F)C1 s275592__15865378__15842994__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC(F)C1 s275592__15865378__15842994__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC(F)C1 s275592__15865378__15842994__15857566
CCON1CCC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15842998__15859360
CCC(=O)N[C@@H]1CC[C@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15843000__15859360
CCC(O)C(C)C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843002__15862300
CCC(O)C(C)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843002__15859360
CCC(O)C(C)C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15843002__15857566
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ncnc2nc[nH]c12 s275592__15865378__15843004__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ncnc2nc[nH]c12 s275592__15865378__15843004__15859360
CN(C)c1cccnc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843006__15862300
CN(C)c1cccnc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843006__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ncn2cccnc12 s275592__15865378__15843010__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ncn2cccnc12 s275592__15865378__15843010__15859360
Cc1cnc(F)cc1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843014__15862300
Cc1cnc(F)cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843014__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1csc(CO)n1 s275592__15865378__15843018__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1csc(CO)n1 s275592__15865378__15843018__15859360
CCC(C)(C)OCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843020__15862300
CCC(C)(C)OCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843020__15859360
O=C(CC1CC(=O)N1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843022__15862300
O=C(CC1CC(=O)N1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843022__15859360
O=C(CC1CC(=O)N1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15843022__15857566
Cc1ncc(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)s1 s275592__15865378__15843024__15862300
Cc1ncc(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)s1 s275592__15865378__15843024__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(O)C1CCC1 s275592__15865378__15843026__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)C1CCC1 s275592__15865378__15843026__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(O)C1CCC1 s275592__15865378__15843026__15857566
CCC(C)C(NC(N)=O)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843028__15859360
CCC(Oc1ccccc1)C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843030__15859360
O=C1CCC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)=NN1 s275592__15865378__15843032__15862300
O=C1CCC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)=NN1 s275592__15865378__15843032__15859360
O=C1CCC(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)=NN1 s275592__15865378__15843032__15857566
NC(=O)N1CC(O)CC1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843034__15859360
CC1CCC(CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15843036__15862300
CC1CCC(CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15843036__15859360
O=C(CSc1cccc[n+]1[O-])NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843040__15859360
NC(=O)NCCCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15843042__15862300
NC(=O)NCCCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843042__15859360
O=C(CSc1ccc(F)cc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843044__15859360
Cc1ccnc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cnn12 s275592__15865378__15843046__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc([N+](=O)[O-])cnc1O s275592__15865378__15843048__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)[C@H](O)c1ccccc1Cl s275592__15865378__15843050__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1csc([N+](=O)[O-])c1 s275592__15865378__15843052__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1csc([N+](=O)[O-])c1 s275592__15865378__15843052__15859360
O=C1Cc2cc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)ccc2N1 s275592__15865378__15843054__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cc([N+](=O)[O-])c[nH]1 s275592__15865378__15843058__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc([N+](=O)[O-])c[nH]1 s275592__15865378__15843058__15859360
O=C(CCSc1ccccc1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15843060__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1ccno1 s275592__15865378__15843062__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccno1 s275592__15865378__15843062__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)c1ccno1 s275592__15865378__15843062__15857566
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cc(Cl)c([N+](=O)[O-])[nH]1 s275592__15865378__15843064__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C3CCCO3)CCCC2)C1 s275592__15865378__15844798__15859360
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)n1cnnn1 s275592__15865378__15844800__15862300
CC(C)(C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)n1cnnn1 s275592__15865378__15844800__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CCn2c(n[nH]c2=O)C1 s275592__15865378__15844802__15859360
Cc1c(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c2ccccc2n1C s275592__15865378__15844804__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1coc2c1C(O)CCC2 s275592__15865378__15844806__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C23CCC(C2)OC3)C1 s275592__15865378__15844808__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C23CCC(C2)OC3)C1 s275592__15865378__15844808__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CC(=C(F)CNC(=O)C23CCC(C2)OC3)C1 s275592__15865378__15844808__15857566
CCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15844810__15862300
CCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15844810__15859360
O=C1CC2(CCC2)C(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CN1 s275592__15865378__15844812__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC12CC(O)C2 s275592__15865378__15844814__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC12CC(O)C2 s275592__15865378__15844814__15859360
O=C(NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C1CC12CC(O)C2 s275592__15865378__15844814__15857566
O=C(Cc1cnc2ccccc2c1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844818__15859360
CN1CCC(C2(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)CC2)CC1 s275592__15865378__15844820__15859360
Cn1ccc([C@@H]2C[C@H]2C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844822__15862300
Cn1ccc([C@@H]2C[C@H]2C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844822__15859360
O=C(C=Cc1cc[nH]n1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844824__15862300
O=C(C=Cc1cc[nH]n1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844824__15859360
O=C(C=Cc1cc[nH]n1)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844824__15857566
Cc1c[nH]c(C=CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844826__15862300
Cc1c[nH]c(C=CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844826__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1cccc2ccnn12 s275592__15865378__15844828__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc2ccnn12 s275592__15865378__15844828__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cnn(C2CC2(F)F)c1 s275592__15865378__15844830__15859360
Cc1cc(C)c2[nH]c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc2c1 s275592__15865378__15844832__15859360
COCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)on1 s275592__15865378__15844836__15862300
COCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)on1 s275592__15865378__15844836__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C(F)(F)Oc2ccccc2)C1 s275592__15865378__15844838__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccn(C2CC2(F)F)n1 s275592__15865378__15844840__15859360
Cc1cccc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)n[nH]c12 s275592__15865378__15844842__15859360
CC1(c2nocc2C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)COC1 s275592__15865378__15844844__15859360
Cc1ncn2ccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)cc12 s275592__15865378__15844846__15859360
Cc1cc2nccnc2cc1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844848__15859360
CC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)Cc2ccccc2C1 s275592__15865378__15844850__15859360
CC1(C#CC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCCO1 s275592__15865378__15844854__15862300
CC1(C#CC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCCO1 s275592__15865378__15844854__15859360
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(F)CCC(F)(F)CC2)C1 s275592__15865378__15844856__15859360
CC(CC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(F)F s275592__15865378__15844858__15862300
CC(CC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(F)F s275592__15865378__15844858__15859360
CC(CC(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1)C(F)F s275592__15865378__15844858__15857566
CC(C)(C)C1=NOC(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)C1 s275592__15865378__15844860__15862300
CC(C)(C)C1=NOC(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)C1 s275592__15865378__15844860__15859360
Cc1cc(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)nn1C s275592__15865378__15844866__15862300
Cc1cc(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)nn1C s275592__15865378__15844866__15859360
O=C(Cn1nnc(C2CC2)n1)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844868__15862300
O=C(Cn1nnc(C2CC2)n1)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844868__15859360
O=C(C[C@@H]1CCC[C@H]1O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844872__15862300
O=C(C[C@@H]1CCC[C@H]1O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844872__15859360
O=C(C[C@@H]1CCC[C@H]1O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15844872__15857566
CCCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(C)o1 s275592__15865378__15844874__15862300
CCCc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)o1 s275592__15865378__15844874__15859360
CN(C)CCSCC(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844876__15862300
CN(C)CCSCC(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844876__15859360
[N-]=[N+]=N[C@H]1CC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__15844878__15862300
[N-]=[N+]=N[C@H]1CC[C@@H](C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__15844878__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C(=O)Nc1ncc[nH]1 s275592__15865378__15844880__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(=O)Nc1ncc[nH]1 s275592__15865378__15844880__15859360
C[C@@H](C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cccc(Cl)c1 s275592__15865378__15844882__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1C(F)(F)C12CC2 s275592__15865378__15844884__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1C(F)(F)C12CC2 s275592__15865378__15844884__15859360
O=C(CCC1=CCc2ccccc21)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844886__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C(O)c1cc(F)cc(F)c1 s275592__15865378__15844888__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)c1coc2c1CSC2 s275592__15865378__15844890__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1coc2c1CSC2 s275592__15865378__15844890__15859360
CCc1occ(C)c1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844892__15862300
CCc1occ(C)c1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844892__15859360
O=C1C[C@]2(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)CCCC[C@@H]2N1 s275592__15865378__15844894__15859360
Cn1nnc2cccc(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)c21 s275592__15865378__15844896__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccnc2nccnc12 s275592__15865378__15844898__15859360
O=C(NCC(F)=C1CN(C(=O)c2nsnc2O)C1)C1CC2COCCN2C1 s275592__15865378__15844900__15862300
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)C1CC2COCCN2C1 s275592__15865378__15844900__15859360
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)c(C)cn1 s275592__15865378__15844902__15862300
Cc1cc(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)c(C)cn1 s275592__15865378__15844902__15859360
O=C(c1nsnc1O)N1CC(=C(F)CNC(=O)C2(C(F)F)CCCO2)C1 s275592__15865378__15844904__15862300
O=C(c1cc(O)no1)N1CC(=C(F)CNC(=O)C2(C(F)F)CCCO2)C1 s275592__15865378__15844904__15859360
CC(=O)N1C[C@H](O)C[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15844906__15862300
CC(=O)N1C[C@H](O)C[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15844906__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1ccc(-c2c[nH]nn2)cc1 s275592__15865378__15844908__15859360
O=C(NCC(F)=C1CN(C(=O)c2cc(O)no2)C1)c1cncc2ccsc12 s275592__15865378__15844910__15859360
CC(C)(C)C1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CCC1 s275592__15865378__15844912__15862300
CC(C)(C)C1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CCC1 s275592__15865378__15844912__15859360
Cc1c[nH]c(CCC(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)n1 s275592__15865378__15844914__15862300
Cc1c[nH]c(CCC(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)n1 s275592__15865378__15844914__15859360
Cc1ccc2c(C(=O)NCC(F)=C3CN(C(=O)c4cc(O)no4)C3)coc2c1 s275592__15865378__15844916__15859360
C[C@@H]1CC=CC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2nsnc2O)C1 s275592__15865378__15909372__15862300
C[C@@H]1CC=CC[C@H]1C(=O)NCC(F)=C1CN(C(=O)c2cc(O)no2)C1 s275592__15865378__15909372__15859360
C[C@@H]1CC=CC[C@H]1C(=O)NCC(F)=C1CN(C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865378__15909372__15857566
NC(=O)NC1(C(=O)NCC(F)=C2CN(C(=O)c3nsnc3O)C2)CC1 s275592__15865378__16147560__15862300
NC(=O)NC1(C(=O)NCC(F)=C2CN(C(=O)c3cc(O)no3)C2)CC1 s275592__15865378__16147560__15859360
NC(=O)NC1(C(=O)NCC(F)=C2CN(C(=O)CSc3n[nH]c(=O)[nH]3)C2)CC1 s275592__15865378__16147560__15857566
CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186874__15862300
CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186874__15857566
COCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186876__15862300
COCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186876__15859360
COCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186876__15857566
CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186878__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__13186882__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__13186882__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC1 s275592__15865748__13186882__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC1 s275592__15865748__13186884__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC1 s275592__15865748__13186884__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCC1 s275592__15865748__13186884__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCC1 s275592__15865748__13186886__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC1 s275592__15865748__13186886__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCCC1 s275592__15865748__13186886__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCOCC1 s275592__15865748__13186888__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCOCC1 s275592__15865748__13186888__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCOCC1 s275592__15865748__13186888__15857566
O=C(CC1CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186890__15862300
O=C(CC1CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186890__15859360
O=C(CC1CC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186890__15857566
CC(C)(F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186892__15862300
CC(C)(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186892__15859360
CC(C)(F)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186892__15857566
CC(F)(F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186894__15862300
CC(F)(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186894__15859360
CC(F)(F)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186894__15857566
COCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186896__15862300
COCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186896__15859360
COCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186896__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccn1 s275592__15865748__13186898__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccn1 s275592__15865748__13186898__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ccccn1 s275592__15865748__13186898__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccncc1 s275592__15865748__13186900__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccncc1 s275592__15865748__13186900__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ccncc1 s275592__15865748__13186900__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(F)cc1 s275592__15865748__13186902__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)cc1 s275592__15865748__13186902__15859360
CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186904__15862300
CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186904__15859360
CCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186904__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccnc1 s275592__15865748__13186906__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnc1 s275592__15865748__13186906__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1cccnc1 s275592__15865748__13186906__15857566
O=C(Cc1cccs1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186908__15862300
O=C(Cc1cccs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186908__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccco1 s275592__15865748__13186910__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccco1 s275592__15865748__13186910__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ccco1 s275592__15865748__13186910__15857566
CC(=O)NCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186912__15862300
CC(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186912__15859360
CC(=O)NCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186912__15857566
Cc1ccsc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186914__15862300
Cc1ccsc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186914__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)s1 s275592__15865748__13186916__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__13186916__15859360
O=C(C=Cc1ccco1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186918__15862300
O=C(C=Cc1ccco1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186918__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccc1F s275592__15865748__13186920__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1F s275592__15865748__13186920__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccc1 s275592__15865748__13186922__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__13186922__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ccccc1 s275592__15865748__13186922__15857566
CC(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186924__15862300
CC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186924__15859360
CC(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186924__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCCC1 s275592__15865748__13186926__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCC1 s275592__15865748__13186926__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCCCC1 s275592__15865748__13186926__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnccn1 s275592__15865748__13186928__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnccn1 s275592__15865748__13186928__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1cnccn1 s275592__15865748__13186928__15857566
Cc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186930__15862300
Cc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186930__15859360
O=C(CC1CCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186932__15862300
O=C(CC1CCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186932__15859360
O=C(CC1CCCC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186932__15857566
O=C(CCC1CCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186934__15862300
O=C(CCC1CCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186934__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc(F)c1 s275592__15865748__13186936__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(F)c1 s275592__15865748__13186936__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccs1 s275592__15865748__13186938__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccs1 s275592__15865748__13186938__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1cccs1 s275592__15865748__13186938__15857566
Cc1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__13186940__15862300
Cc1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__13186940__15859360
O=C(Cc1ccsc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186942__15862300
O=C(Cc1ccsc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186942__15859360
CC1CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186944__15862300
CC1CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186944__15859360
CC1CC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186944__15857566
Cc1cccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__13186946__15862300
Cc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__13186946__15859360
CCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186948__15862300
CCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186948__15859360
CCOCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186948__15857566
CC(C)=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186950__15862300
CC(C)=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186950__15859360
CC(C)=CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186950__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=COCCO1 s275592__15865748__13186952__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=COCCO1 s275592__15865748__13186952__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1=COCCO1 s275592__15865748__13186952__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc[n+]([O-])cc1 s275592__15865748__13186954__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc[n+]([O-])cc1 s275592__15865748__13186954__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC2C=CC1C2 s275592__15865748__13186956__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2C=CC1C2 s275592__15865748__13186956__15859360
CC(=O)NC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186958__15862300
CC(=O)NC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186958__15859360
CC(=O)NC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186958__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(=O)[nH]n1 s275592__15865748__13186960__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(=O)[nH]n1 s275592__15865748__13186960__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__13186962__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__13186962__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)o1 s275592__15865748__13186962__15857566
O=C(CC1CCCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186964__15862300
O=C(CC1CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186964__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCO1 s275592__15865748__13186966__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCO1 s275592__15865748__13186966__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCCO1 s275592__15865748__13186966__15857566
CSCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186968__15862300
CSCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186968__15859360
CSCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186968__15857566
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)no1 s275592__15865748__13186970__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__13186970__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)no1 s275592__15865748__13186970__15857566
CSCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186972__15862300
CSCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186972__15859360
CSCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186972__15857566
CC(C)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186974__15862300
CC(C)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186974__15859360
CC(C)CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186974__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccsc1 s275592__15865748__13186978__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccsc1 s275592__15865748__13186978__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ccsc1 s275592__15865748__13186978__15857566
Cc1occc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186980__15862300
Cc1occc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186980__15859360
Cc1occc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186980__15857566
O=C(CC1C=CCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186982__15862300
O=C(CC1C=CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186982__15859360
O=C(CC1C=CCC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186982__15857566
O=C(Cn1cnnn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186984__15862300
O=C(Cn1cnnn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186984__15859360
O=C(Cn1cnnn1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13186984__15857566
O=C(CN1CCCC1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186986__15862300
O=C(CN1CCCC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186986__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__13186988__15862300
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__13186988__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)cn1 s275592__15865748__13186988__15857566
Cc1noc(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186990__15862300
Cc1noc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186990__15859360
Cc1nnsc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13186992__15862300
Cc1nnsc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13186992__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)o1 s275592__15865748__13186994__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)o1 s275592__15865748__13186994__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC=CCC1 s275592__15865748__13186996__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC=CCC1 s275592__15865748__13186996__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC=CCC1 s275592__15865748__13186996__15857566
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)on1 s275592__15865748__13187000__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__13187000__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)on1 s275592__15865748__13187000__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc[nH]1 s275592__15865748__13187002__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc[nH]1 s275592__15865748__13187002__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ccc[nH]1 s275592__15865748__13187002__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(Cl)c[nH]1 s275592__15865748__13187004__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(Cl)c[nH]1 s275592__15865748__13187004__15859360
CC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187006__15862300
CC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187006__15859360
CC(=O)CCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187006__15857566
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1C s275592__15865748__13187008__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1C s275592__15865748__13187008__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccoc1 s275592__15865748__13187010__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccoc1 s275592__15865748__13187010__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ccoc1 s275592__15865748__13187010__15857566
O=C(Cn1cccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187012__15862300
O=C(Cn1cccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187012__15859360
O=C(Cn1cccn1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187012__15857566
Cc1ccoc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187014__15862300
Cc1ccoc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187014__15859360
Cc1ccoc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187014__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC2CCC1C2 s275592__15865748__13187016__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2CCC1C2 s275592__15865748__13187016__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(Cl)o1 s275592__15865748__13187018__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(Cl)o1 s275592__15865748__13187018__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cnn1C s275592__15865748__13187020__15862300
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1C s275592__15865748__13187020__15859360
CCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187022__15862300
CCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187022__15859360
CCCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187022__15857566
CC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187024__15862300
CC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187024__15859360
CC(C)(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187024__15857566
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__13187026__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__13187026__15859360
Cn1cccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187028__15862300
Cn1cccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187028__15859360
Cn1cccc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187028__15857566
O=C(CCn1cncn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187030__15862300
O=C(CCn1cncn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187030__15859360
CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187034__15862300
CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187034__15859360
CCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187034__15857566
Cc1cccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__13187036__15862300
Cc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__13187036__15859360
CC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187038__15862300
CC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187038__15859360
CC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187038__15857566
O=C(CCn1cccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187040__15862300
O=C(CCn1cccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187040__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccc1O s275592__15865748__13187042__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1O s275592__15865748__13187042__15859360
CCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187044__15862300
CCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187044__15859360
CCC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187044__15857566
CC(C)SCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187046__15862300
CC(C)SCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187046__15859360
CC(=O)N(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187050__15862300
CC(=O)N(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187050__15859360
CC(=O)N(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187050__15857566
CCC(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187052__15862300
CCC(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187052__15859360
CCC(CC)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187052__15857566
CC(C)OCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187054__15862300
CC(C)OCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187054__15859360
CC(C)OCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187054__15857566
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)[nH]n1 s275592__15865748__13187056__15862300
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)[nH]n1 s275592__15865748__13187056__15859360
O=C(CCC1CCCO1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187058__15862300
O=C(CCC1CCCO1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187058__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1COCCO1 s275592__15865748__13187060__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1COCCO1 s275592__15865748__13187060__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1COCCO1 s275592__15865748__13187060__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc[nH]n1 s275592__15865748__13187062__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc[nH]n1 s275592__15865748__13187062__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1cc[nH]n1 s275592__15865748__13187062__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)n1cccn1 s275592__15865748__13187064__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)n1cccn1 s275592__15865748__13187064__15859360
CCCCC(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187066__15862300
CCCCC(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187066__15859360
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CSC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187068__15859360
CSC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187068__15857566
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CCOC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187070__15859360
CCOC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187070__15857566
CC(C)COCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187072__15862300
CC(C)COCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187072__15859360
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Cc1cc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)[nH]n1 s275592__15865748__13187108__15857566
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Cc1ocnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187130__15862300
Cc1ocnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187130__15859360
Cc1ocnc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187130__15857566
CCOC(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187132__15862300
CCOC(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187132__15859360
CCOC(CC)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187132__15857566
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COC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187136__15862300
COC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187136__15859360
COC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187136__15857566
CC(C)OCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187138__15862300
CC(C)OCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187138__15859360
CC(C)OCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187138__15857566
CC(OCC1CC1)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187140__15862300
CC(OCC1CC1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187140__15859360
CCCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187142__15862300
CCCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187142__15859360
CCCOCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187142__15857566
CCCCOC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187144__15862300
CCCCOC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187144__15859360
C=CCCOC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187146__15862300
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Cc1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)s1 s275592__15865748__13187152__15862300
Cc1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__13187152__15859360
Cn1nccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187154__15862300
Cn1nccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187154__15859360
Cn1nccc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187154__15857566
CCC(OC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187156__15862300
CCC(OC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187156__15859360
CCC(OC)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187156__15857566
COCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187158__15862300
COCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187158__15859360
COCCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187158__15857566
CCCC(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187160__15862300
CCCC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187160__15859360
CCCC(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187160__15857566
COC(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187162__15862300
COC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187162__15859360
COC(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187162__15857566
Cn1cc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__13187164__15862300
Cn1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__13187164__15859360
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C=CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187168__15862300
C=CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187168__15859360
C=CCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187168__15857566
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COC(=O)C1CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187172__15859360
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CCOCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187178__15857566
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CCNC(=O)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187180__15859360
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COCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187184__15862300
COCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187184__15859360
COCC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187184__15857566
CC(C)(C)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187186__15862300
CC(C)(C)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187186__15859360
C=CCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187188__15862300
C=CCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187188__15859360
C=CCOCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187188__15857566
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O=C(CC1=CCCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187194__15862300
O=C(CC1=CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187194__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c[nH]1 s275592__15865748__13187196__15862300
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c[nH]1 s275592__15865748__13187196__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)c[nH]1 s275592__15865748__13187196__15857566
CSCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187198__15862300
CSCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187198__15859360
CN1CCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187200__15862300
CN1CCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187200__15859360
CN1CCCC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187200__15857566
CCC(=O)NCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187202__15862300
CCC(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187202__15859360
CCC(=O)NCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187202__15857566
CC(C)(C)/C=C/C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187204__15862300
CC(C)(C)/C=C/C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187204__15859360
CC(C)(C)/C=C/C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187204__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(F)nc1 s275592__15865748__13187206__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)nc1 s275592__15865748__13187206__15859360
COCCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187210__15862300
COCCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187210__15859360
CCCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187212__15862300
CCCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187212__15859360
CCCC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187212__15857566
Cc1nn(C)cc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187214__15862300
Cc1nn(C)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187214__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC2CCC1O2 s275592__15865748__13187218__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2CCC1O2 s275592__15865748__13187218__15859360
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)no1 s275592__15865748__13187220__15862300
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__13187220__15859360
CCn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__13187222__15862300
CCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__13187222__15859360
Nc1nccnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187224__15862300
Nc1nccnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187224__15859360
O=C(CCC1CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187226__15862300
O=C(CCC1CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187226__15859360
O=C(CCC1CC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187226__15857566
Cc1[nH]nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1C s275592__15865748__13187228__15862300
Cc1[nH]nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__13187228__15859360
O=C(CC1CCOCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187230__15862300
O=C(CC1CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187230__15859360
CCCCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187232__15862300
CCCCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187232__15859360
CCCCOCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187232__15857566
O=C(Cc1ccon1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187234__15862300
O=C(Cc1ccon1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187234__15859360
O=C(Cc1ccon1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187234__15857566
CCc1ocnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187238__15862300
CCc1ocnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187238__15859360
O=C(CC1CCOC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187240__15862300
O=C(CC1CCOC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187240__15859360
O=C(CC1CCOC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187240__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC=CC1 s275592__15865748__13187242__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC=CC1 s275592__15865748__13187242__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC=CC1 s275592__15865748__13187242__15857566
O=C(Cc1ccn[nH]1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187244__15862300
O=C(Cc1ccn[nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187244__15859360
O=C(Cc1ccn[nH]1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187244__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccncc1F s275592__15865748__13187246__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccncc1F s275592__15865748__13187246__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nnn1C s275592__15865748__13187248__15862300
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nnn1C s275592__15865748__13187248__15859360
Cc1ccncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187250__15862300
Cc1ccncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187250__15859360
Cc1cncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__13187252__15862300
Cc1cncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__13187252__15859360
CN1CCOC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__13187254__15862300
CN1CCOC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__13187254__15859360
Cc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__13187256__15862300
Cc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__13187256__15859360
O=C(CCC(F)(F)F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187258__15862300
O=C(CCC(F)(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187258__15859360
C=CCOCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187260__15862300
C=CCOCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187260__15859360
O=C(CC1CCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187264__15862300
O=C(CC1CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187264__15859360
O=C(CC1CCC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187264__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc(=O)[nH]1 s275592__15865748__13187268__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(=O)[nH]1 s275592__15865748__13187268__15859360
CC1(C)C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1(C)C s275592__15865748__13187270__15862300
CC1(C)C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1(C)C s275592__15865748__13187270__15859360
Cc1ncoc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187272__15862300
Cc1ncoc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187272__15859360
Cc1ncoc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187272__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__13187274__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__13187274__15859360
CC(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC1 s275592__15865748__13187274__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1C2CCCC21 s275592__15865748__13187276__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1C2CCCC21 s275592__15865748__13187276__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1C2CCCC21 s275592__15865748__13187276__15857566
N#Cc1c[nH]c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__13187278__15862300
N#Cc1c[nH]c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__13187278__15859360
Cc1cscc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187280__15862300
Cc1cscc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187280__15859360
O=C(CCC1CCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187282__15862300
O=C(CCC1CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187282__15859360
O=C(CCC1CCC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187282__15857566
Cc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__13187284__15862300
Cc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__13187284__15859360
O=C(CCc1nnc[nH]1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187286__15862300
O=C(CCc1nnc[nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187286__15859360
Cc1cccnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187288__15862300
Cc1cccnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187288__15859360
CC=C(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187292__15862300
CC=C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187292__15859360
CC=C(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187292__15857566
O=C(CCC1CCOC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187294__15862300
O=C(CCC1CCOC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187294__15859360
O=C(CCc1ccoc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187296__15862300
O=C(CCc1ccoc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187296__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC(F)(F)C1 s275592__15865748__13187298__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC(F)(F)C1 s275592__15865748__13187298__15859360
CC1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__13187300__15862300
CC1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__13187300__15859360
CC1CC(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865748__13187300__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)=C1CCCC1 s275592__15865748__13187302__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)=C1CCCC1 s275592__15865748__13187302__15859360
O=C(CC1CCCCO1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187304__15862300
O=C(CC1CCCCO1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187304__15859360
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n[nH]1 s275592__15865748__13187306__15862300
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n[nH]1 s275592__15865748__13187306__15859360
O=C(C=C1CCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187308__15862300
O=C(C=C1CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187308__15859360
O=C(C=C1CCC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187308__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cncc(F)c1 s275592__15865748__13187310__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cncc(F)c1 s275592__15865748__13187310__15859360
CCC(=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)CC s275592__15865748__13187312__15862300
CCC(=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC s275592__15865748__13187312__15859360
CCC(=CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)CC s275592__15865748__13187312__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc[nH]c(=O)c1 s275592__15865748__13187314__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc[nH]c(=O)c1 s275592__15865748__13187314__15859360
CC(C)=C(F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187316__15862300
CC(C)=C(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187316__15859360
CC(C)=C(F)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187316__15857566
O=C1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCN1 s275592__15865748__13187318__15862300
O=C1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCN1 s275592__15865748__13187318__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=CCCC1 s275592__15865748__13187320__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CCCC1 s275592__15865748__13187320__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1=CCCC1 s275592__15865748__13187320__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(F)=C1CCCC1 s275592__15865748__13187322__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)=C1CCCC1 s275592__15865748__13187322__15859360
Cn1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__13187324__15862300
Cn1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__13187324__15859360
Cn1ccc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)c1 s275592__15865748__13187324__15857566
Cn1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__13187326__15862300
Cn1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__13187326__15859360
Cn1cnc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)c1 s275592__15865748__13187326__15857566
O=C(CC1COC(=O)C1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187328__15862300
O=C(CC1COC(=O)C1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187328__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)oc1C s275592__15865748__13187330__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)oc1C s275592__15865748__13187330__15859360
O=C(Cc1cccnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187332__15862300
O=C(Cc1cccnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187332__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCCO1 s275592__15865748__13187334__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCO1 s275592__15865748__13187334__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCCCO1 s275592__15865748__13187334__15857566
Cc1n[nH]c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1O s275592__15865748__13187336__15862300
Cc1n[nH]c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1O s275592__15865748__13187336__15859360
CCC(SC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187338__15862300
CCC(SC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187338__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ncn1 s275592__15865748__13187342__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ncn1 s275592__15865748__13187342__15859360
CC1(C)CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187344__15862300
CC1(C)CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187344__15859360
CC1(C)CC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187344__15857566
CCC(C)OCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187348__15862300
CCC(C)OCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187348__15859360
CCC(C)OCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187348__15857566
CC1(C)C[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187350__15862300
CC1(C)C[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187350__15859360
CC1(C)C[C@@H]1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187350__15857566
CC(O)(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__13187354__15862300
CC(O)(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__13187354__15859360
CSC(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187358__15862300
CSC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187358__15859360
O=C(CN1CCOCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187360__15862300
O=C(CN1CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187360__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1CCCO1 s275592__15865748__13187362__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1CCCO1 s275592__15865748__13187362__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)[C@@H]1CCCO1 s275592__15865748__13187362__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)n1cncn1 s275592__15865748__13187364__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)n1cncn1 s275592__15865748__13187364__15859360
CN1CCOCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187368__15862300
CN1CCOCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187368__15859360
Cc1nscc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187370__15862300
Cc1nscc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187370__15859360
C#CCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187372__15862300
C#CCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187372__15859360
C#CCCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187372__15857566
C#CCNC(=O)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187378__15862300
C#CCNC(=O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187378__15859360
CCNC(=O)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187380__15862300
CCNC(=O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187380__15859360
CCNC(=O)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187380__15857566
CNC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187382__15862300
CNC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187382__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)on1 s275592__15865748__13187386__15862300
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__13187386__15859360
COC(C)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187388__15862300
COC(C)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187388__15859360
COC(C)CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187388__15857566
CCc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)co1 s275592__15865748__13187390__15862300
CCc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)co1 s275592__15865748__13187390__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(F)cn1 s275592__15865748__13187392__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)cn1 s275592__15865748__13187392__15859360
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1N s275592__15865748__13187394__15862300
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1N s275592__15865748__13187394__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cncnc1 s275592__15865748__13187396__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cncnc1 s275592__15865748__13187396__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1cncnc1 s275592__15865748__13187396__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=CCOCC1 s275592__15865748__13187402__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CCOCC1 s275592__15865748__13187402__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1=CCOCC1 s275592__15865748__13187402__15857566
O=C(Cc1ccoc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187404__15862300
O=C(Cc1ccoc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187404__15859360
O=C(Cc1ccoc1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187404__15857566
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)co1 s275592__15865748__13187408__15862300
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)co1 s275592__15865748__13187408__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)co1 s275592__15865748__13187408__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=CCCCCC1 s275592__15865748__13187412__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CCCCCC1 s275592__15865748__13187412__15859360
C[C@H](NC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187414__15862300
C[C@H](NC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187414__15859360
C[C@H](NC(N)=O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187414__15857566
O=C(CC1OCCCO1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187416__15862300
O=C(CC1OCCCO1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187416__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)co1 s275592__15865748__13187418__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)co1 s275592__15865748__13187418__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)co1 s275592__15865748__13187418__15857566
Cc1ccn(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187422__15862300
Cc1ccn(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187422__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cnn1 s275592__15865748__13187424__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1 s275592__15865748__13187424__15859360
O=C(CCn1ccnn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187426__15862300
O=C(CCn1ccnn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187426__15859360
CC(=O)N1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__13187428__15862300
CC(=O)N1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__13187428__15859360
Cn1oc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1=O s275592__15865748__13187430__15862300
Cn1oc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1=O s275592__15865748__13187430__15859360
CCC(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187432__15862300
CCC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187432__15859360
CCC(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187432__15857566
COC1(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__13187434__15862300
COC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__13187434__15859360
CC1OCCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187436__15862300
CC1OCCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187436__15859360
C#CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187438__15862300
C#CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187438__15859360
C#CCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187438__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccoc1Cl s275592__15865748__13187440__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccoc1Cl s275592__15865748__13187440__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ns1 s275592__15865748__13187444__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ns1 s275592__15865748__13187444__15859360
CCn1ccnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187450__15862300
CCn1ccnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187450__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCOCC1 s275592__15865748__13187452__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCOCC1 s275592__15865748__13187452__15859360
O=C(CCc1ncc[nH]1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187454__15862300
O=C(CCc1ncc[nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187454__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC(O)CC1 s275592__15865748__13187456__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC(O)CC1 s275592__15865748__13187456__15859360
CC(C)(O)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187458__15862300
CC(C)(O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187458__15859360
CC(C)(O)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187458__15857566
Cc1ccnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__13187460__15862300
Cc1ccnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__13187460__15859360
COC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__13187462__15862300
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__13187462__15859360
COC(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC1 s275592__15865748__13187462__15857566
CCc1occc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187464__15862300
CCc1occc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187464__15859360
Cn1nncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187468__15862300
Cn1nncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187468__15859360
Cn1nncc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187468__15857566
CCCCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187472__15862300
CCCCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187472__15859360
CCCCC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187472__15857566
CC1CC(C)C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)O1 s275592__15865748__13187474__15862300
CC1CC(C)C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)O1 s275592__15865748__13187474__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@H]1C[C@@H]1C(F)F s275592__15865748__13187476__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@H]1C[C@@H]1C(F)F s275592__15865748__13187476__15859360
Cc1coc(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187478__15862300
Cc1coc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187478__15859360
CC1(C)CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__13187482__15862300
CC1(C)CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__13187482__15859360
CC1(C)CC(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865748__13187482__15857566
CC(C)[C@@H](O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187486__15862300
CC(C)[C@@H](O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187486__15859360
CC(C)[C@@H](O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187486__15857566
CCOC1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__13187488__15862300
CCOC1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__13187488__15859360
CC1(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCC1 s275592__15865748__13187490__15862300
CC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__13187490__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__13187492__15862300
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__13187492__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)nn1 s275592__15865748__13187492__15857566
Cc1nnc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__13187494__15862300
Cc1nnc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__13187494__15859360
Cn1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__13187496__15862300
Cn1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__13187496__15859360
Cn1cnc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)n1 s275592__15865748__13187496__15857566
CNC(=O)NCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187498__15862300
CNC(=O)NCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187498__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1sccc1F s275592__15865748__13187500__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1sccc1F s275592__15865748__13187500__15859360
CCn1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__13187502__15862300
CCn1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__13187502__15859360
CC(C)(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__13187504__15862300
CC(C)(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__13187504__15859360
CCn1nncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187506__15862300
CCn1nncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187506__15859360
Cc1csc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__13187508__15862300
Cc1csc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__13187508__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1(F)F s275592__15865748__13187510__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1(F)F s275592__15865748__13187510__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC1(F)F s275592__15865748__13187510__15857566
CCC(C)=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187512__15862300
CCC(C)=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187512__15859360
CCC(C)=CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187512__15857566
Cc1cnccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187514__15862300
Cc1cnccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187514__15859360
CC(C)C#CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187518__15862300
CC(C)C#CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187518__15859360
CC(C)C#CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187518__15857566
Cc1sccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187520__15862300
Cc1sccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187520__15859360
O=C(CC1(O)CCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187522__15862300
O=C(CC1(O)CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187522__15859360
O=C(CC1(O)CCC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187522__15857566
Cc1c[nH]nc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187524__15862300
Cc1c[nH]nc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187524__15859360
Cc1c[nH]nc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187524__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)=C1CCC1 s275592__15865748__13187526__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)=C1CCC1 s275592__15865748__13187526__15859360
CC(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)=C1CCC1 s275592__15865748__13187526__15857566
O=C(C#CC1CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187528__15862300
O=C(C#CC1CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187528__15859360
O=C(C#CC1CC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187528__15857566
CC(C)(C)C#CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187530__15862300
CC(C)(C)C#CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187530__15859360
CC(C)(C)C#CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__13187530__15857566
Cc1n[nH]c(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__13187532__15862300
Cc1n[nH]c(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__13187532__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__13187534__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__13187534__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@H]1[N+](=O)[O-] s275592__15865748__13187536__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]1[N+](=O)[O-] s275592__15865748__13187536__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)[C@@H]1C[C@H]1[N+](=O)[O-] s275592__15865748__13187536__15857566
Cc1cn(C)nc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__13187538__15862300
Cc1cn(C)nc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__13187538__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCC(F)C1 s275592__15865748__13187540__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC(F)C1 s275592__15865748__13187540__15859360
Cn1ccc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__13187542__15862300
Cn1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__13187542__15859360
COCC1(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__13187544__15862300
COCC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__13187544__15859360
Cc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)s1 s275592__15865748__14135846__15862300
Cc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14135846__15859360
O=C(CCC1NC(=O)NC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135850__15859360
NC(=O)NCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135854__15862300
NC(=O)NCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135854__15859360
NC(=O)NCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14135854__15857566
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14135856__15859360
NC(=O)c1nccnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135858__15859360
O=C(CN1C(=O)CCC1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135872__15862300
O=C(CN1C(=O)CCC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135872__15859360
NC(=O)N1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14135878__15859360
CC(=O)N1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14135880__15859360
Cc1cccc2nc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cn12 s275592__15865748__14135884__15859360
Cc1ccccc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135886__15862300
Cc1ccccc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135886__15859360
O=C(CCc1cccs1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135896__15862300
O=C(CCc1cccs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135896__15859360
CC(C)Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135898__15859360
O=C(Cn1ccccc1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135900__15862300
O=C(Cn1ccccc1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135900__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(c1)CCC2 s275592__15865748__14135904__15859360
Cc1noc(C)c1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135906__15859360
COCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135908__15859360
CCc1onc(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135920__15862300
CCc1onc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135920__15859360
O=C(COc1ccc(F)cc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135930__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2[nH]nnc2c1 s275592__15865748__14135934__15859360
Cc1n[nH]c(C)c1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135944__15859360
O=C(COCc1ccccc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135948__15859360
NC(=O)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135952__15859360
O=C(Cc1ccc2c(c1)CCC2)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135954__15859360
O=C(CCc1ccccc1F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135958__15859360
Cc1csc(=O)n1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135960__15859360
Cc1noc(C)c1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135968__15862300
Cc1noc(C)c1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135968__15859360
Cc1n[nH]c(C)c1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135970__15862300
Cc1n[nH]c(C)c1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135970__15859360
CCc1ccc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135972__15859360
CC(C)(C)C(=O)NCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135974__15862300
CC(C)(C)C(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135974__15859360
CCc1noc(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135976__15862300
CCc1noc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135976__15859360
Cc1cccc(OCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14135988__15859360
O=C(COc1cccc(F)c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135994__15859360
O=C(CCOc1ccccc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136002__15859360
O=C(COc1ccccc1F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136008__15859360
Cc1ccccc1C(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138336__15859360
O=C(CCC1CCOCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138340__15862300
O=C(CCC1CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138340__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnc1 s275592__15865748__14138342__15859360
CC1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14138346__15862300
CC1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14138346__15859360
CC1CCC(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865748__14138346__15857566
COc1cc(C)sc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138352__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCCCCC1 s275592__15865748__14138354__15859360
CC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)on1 s275592__15865748__14138356__15862300
CC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__14138356__15859360
CC(C)N1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138360__15859360
CCn1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14138362__15862300
CCn1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14138362__15859360
C[C@H]1CC[C@@](C)(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1(C)C s275592__15865748__14138368__15859360
CC(C)CCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138372__15862300
CC(C)CCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138372__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(Cl)cs1 s275592__15865748__14138376__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1csc(Cl)c1 s275592__15865748__14138378__15859360
CC(CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14138380__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccsc1Cl s275592__15865748__14138384__15859360
C=C(C)CC(NC(C)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138388__15859360
CCCCCC(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138392__15862300
CCCCCC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138392__15859360
Cc1ncc(Cl)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14138394__15859360
COc1cncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14138398__15862300
COc1cncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14138398__15859360
CC(=O)N[C@@H](CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(N)=O s275592__15865748__14138400__15859360
Cc1sccc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138404__15862300
Cc1sccc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138404__15859360
CC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1C s275592__15865748__14138412__15859360
CCOC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)C s275592__15865748__14138416__15862300
CCOC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__14138416__15859360
CC(C)CC(C)OCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138422__15859360
O=C(CNC(=O)N1CCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138426__15859360
C#CCOCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138428__15862300
C#CCOCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138428__15859360
C#CCOCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138428__15857566
COCCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14138430__15859360
C#CCOC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138432__15862300
C#CCOC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138432__15859360
C#CCOC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138432__15857566
CC(C)N1CCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138436__15862300
CC(C)N1CCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138436__15859360
O=C(CCOCC1CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138440__15862300
O=C(CCOCC1CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138440__15859360
CNS(=O)(=O)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138444__15859360
CC1CC1c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__14138448__15859360
CCCc1onc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138450__15859360
CCCCCCOC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138454__15859360
C=CCCOCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138456__15859360
O=C(COC1CCOC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138460__15862300
O=C(COC1CCOC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138460__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)NC(N)=O s275592__15865748__14138464__15862300
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)NC(N)=O s275592__15865748__14138464__15859360
CC(C)(C)c1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)co1 s275592__15865748__14138468__15859360
Cc1oc(C(C)C)nc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138470__15859360
Cc1cccn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1=O s275592__15865748__14138472__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(C(F)F)CC1 s275592__15865748__14138488__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C(F)F)CC1 s275592__15865748__14138488__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCC2(CC2)C1 s275592__15865748__14138490__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC2(CC2)C1 s275592__15865748__14138490__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(c2ccccn2)CC1 s275592__15865748__14138492__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn(C2CCC2)c1 s275592__15865748__14138494__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2CCCCN2C1 s275592__15865748__14138498__15859360
CC(C)C(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14140834__15859360
C=CCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140840__15862300
C=CCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140840__15859360
C=CCC(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140840__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(F)c1ccccc1 s275592__15865748__14140846__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)c1ccccc1 s275592__15865748__14140846__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC12CCC2 s275592__15865748__14140850__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC12CCC2 s275592__15865748__14140850__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC12CCC2 s275592__15865748__14140850__15857566
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Cc1cccc(C(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140866__15859360
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CCc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14140882__15859360
CCCN1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1=O s275592__15865748__14140884__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)n1ccnc1 s275592__15865748__14140886__15862300
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)n1ccnc1 s275592__15865748__14140886__15859360
CCn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)n1 s275592__15865748__14140888__15862300
CCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)n1 s275592__15865748__14140888__15859360
Cc1c(Cl)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1C s275592__15865748__14140890__15859360
Cc1ccnn1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140892__15862300
Cc1ccnn1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140892__15859360
CCCn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__14140898__15862300
CCCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14140898__15859360
Cc1cnc2c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cnn2c1 s275592__15865748__14140900__15859360
Cc1ccn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(=O)c1 s275592__15865748__14140902__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(C2CC2)no1 s275592__15865748__14140906__15862300
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CCc1oncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140908__15862300
CCc1oncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140908__15859360
CC(Cc1cccs1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140910__15859360
CC(C)c1nccn1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140912__15859360
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O=C(Cc1cscn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140922__15862300
O=C(Cc1cscn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140922__15859360
CC1CCN(C(=O)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140926__15859360
CC1CCCN(C(=O)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140928__15859360
COc1nc(C)ccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140930__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1coc(C2CC2)n1 s275592__15865748__14140932__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1coc(C2CC2)n1 s275592__15865748__14140932__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@H]1C[C@@H]1c1ccccc1 s275592__15865748__14140934__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1C2Cc3ccccc3C21 s275592__15865748__14140940__15859360
COCc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)no1 s275592__15865748__14140942__15862300
COCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__14140942__15859360
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O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2cccnn12 s275592__15865748__14140960__15859360
CN(C)C(=O)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140962__15862300
CN(C)C(=O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140962__15859360
CN(C)C(=O)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140962__15857566
C#CCOc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14140966__15859360
O=C(Cc1ccc(Cl)s1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140968__15859360
CCC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__14140976__15859360
CC1(C)C2CCC1(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC2 s275592__15865748__14140984__15859360
C=CCn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__14140988__15862300
C=CCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14140988__15859360
CC(C)c1ncsc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140992__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1scnc1C1CC1 s275592__15865748__14140996__15859360
Cc1noc(CCCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14136014__15859360
Cc1cc(NC(=O)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__14136020__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(=O)[nH]c1=O s275592__15865748__14136024__15859360
CC(C)c1nn(C)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136030__15859360
CN(C)c1ncccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136040__15859360
O=C(Cc1nc2ncccn2n1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136044__15859360
Cn1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14136050__15862300
Cn1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14136050__15859360
Cn1ccc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)n1 s275592__15865748__14136050__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2cnccc12 s275592__15865748__14136052__15859360
Cc1[nH]nc2ncc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc12 s275592__15865748__14136054__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(-c2ccoc2)n[nH]1 s275592__15865748__14136058__15859360
Cc1nccn1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136066__15862300
Cc1nccn1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136066__15859360
CC(CN1CCOCC1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136070__15859360
Cc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__14136072__15862300
Cc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14136072__15859360
NC(=O)c1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c[nH]1 s275592__15865748__14136078__15862300
NC(=O)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c[nH]1 s275592__15865748__14136078__15859360
CCn1cccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136082__15862300
CCn1cccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136082__15859360
CC(C)n1cccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136084__15862300
CC(C)n1cccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136084__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1scnc1Cl s275592__15865748__14136092__15859360
CCn1cc(Cl)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136096__15859360
CCc1ncncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136098__15862300
CCc1ncncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136098__15859360
CC(C)c1ncncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136100__15859360
O=C(CC1CCCOC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136104__15862300
O=C(CC1CCCOC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136104__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC=CCC1 s275592__15865748__14136106__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC=CCC1 s275592__15865748__14136106__15859360
NC(=O)c1cncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14136108__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCS(=O)(=O)N1 s275592__15865748__14136110__15859360
Cc1nccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14136112__15862300
Cc1nccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14136112__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc(C)c1F s275592__15865748__14136114__15859360
Cc1nn2cccnc2c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136116__15859360
O=C(CCCN1CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136118__15859360
CCC(C)C(=O)NCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136120__15862300
CCC(C)C(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136120__15859360
O=C(CCN1CCCC1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136122__15862300
O=C(CCN1CCCC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136122__15859360
CNS(=O)(=O)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136126__15862300
CNS(=O)(=O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136126__15859360
CCCS(=O)(=O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136130__15859360
CC(C)S(=O)(=O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136132__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c[nH]c2ncccc12 s275592__15865748__14136134__15859360
O=C(CN1CCc2ccccc21)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136140__15859360
O=C(CCCn1cccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136144__15862300
O=C(CCCn1cccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136144__15859360
CC(C)(C)CC(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136156__15859360
O=C(Cn1ccc2ccccc21)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136158__15859360
O=C(CCc1nccs1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136162__15862300
O=C(CCc1nccs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136162__15859360
COCCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136172__15862300
COCCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136172__15859360
COCCC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14136172__15857566
CCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCCC1=O s275592__15865748__14136176__15859360
CC(C)Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c[nH]1 s275592__15865748__14138506__15859360
CN(C)c1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14138510__15859360
Cc1cnc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccn12 s275592__15865748__14138514__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnn1CC(F)F s275592__15865748__14138522__15859360
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCCCC1 s275592__15865748__14138526__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCc2[nH]ncc21 s275592__15865748__14138530__15859360
CCOCCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14138548__15859360
CCOC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__14138560__15862300
CCOC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__14138560__15859360
O=C(CCOCC(F)F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138566__15862300
O=C(CCOCC(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138566__15859360
O=C(Cn1ncnn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138568__15862300
O=C(Cn1ncnn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138568__15859360
O=C(Cn1ncnn1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138568__15857566
Cn1ncc(Cl)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138570__15862300
Cn1ncc(Cl)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138570__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ncn1 s275592__15865748__14138572__15862300
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ncn1 s275592__15865748__14138572__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CN2CCC1CC2 s275592__15865748__14138574__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CN2CCC1CC2 s275592__15865748__14138574__15859360
CCCC[C@@H](C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138576__15862300
CCCC[C@@H](C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138576__15859360
CCCC[C@@H](C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138576__15857566
CCc1ccnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14138578__15862300
CCc1ccnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14138578__15859360
O=C(CC1Cc2ccccc2O1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138580__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2nn[nH]c12 s275592__15865748__14138582__15859360
CC1=C(C)CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14138584__15862300
CC1=C(C)CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14138584__15859360
CC(C)(C)CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138586__15862300
CC(C)(C)CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138586__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2c1CCCC2 s275592__15865748__14138590__15859360
Cc1oc2ccccc2c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138594__15859360
Cc1csc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1Cl s275592__15865748__14138596__15859360
C=CCC(CC=C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138600__15862300
C=CCC(CC=C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138600__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC=CCC1 s275592__15865748__14138604__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC=CCC1 s275592__15865748__14138604__15859360
Cn1cc(Cl)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14138606__15862300
Cn1cc(Cl)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14138606__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CS(=O)(=O)C1 s275592__15865748__14138608__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CS(=O)(=O)C1 s275592__15865748__14138608__15859360
Cc1scc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1C s275592__15865748__14138610__15862300
Cc1scc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14138610__15859360
CCn1ncc(Cl)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138612__15859360
CCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138616__15862300
CCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138616__15859360
CCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138616__15857566
CCCC(C)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138618__15862300
CCCC(C)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138618__15859360
CCC(C)CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138620__15862300
CCC(C)CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138620__15859360
CC(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138622__15862300
CC(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138622__15859360
CC(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138622__15857566
Cc1ccn(CC(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14138630__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccn2nnnc12 s275592__15865748__14138636__15859360
C=C(Cl)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138638__15862300
C=C(Cl)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138638__15859360
CC(C)n1nccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138640__15862300
CC(C)n1nccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138640__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccn(C(F)F)n1 s275592__15865748__14138644__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnn1C(F)F s275592__15865748__14138646__15859360
C=CC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138648__15862300
C=CC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138648__15859360
C=CC(C)(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138648__15857566
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc(C)n1 s275592__15865748__14138654__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc(C)n1 s275592__15865748__14138654__15859360
O=C(Cn1nccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138660__15862300
O=C(Cn1nccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138660__15859360
O=C(Cn1nccn1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138660__15857566
Cc1nc(Cl)sc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138662__15859360
Cc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)s1 s275592__15865748__14138664__15862300
Cc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14138664__15859360
COCc1ncsc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140998__15859360
CC(C)c1nnnn1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141000__15859360
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCC1 s275592__15865748__14141002__15859360
Cc1nc(C2CC2)oc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141010__15859360
Cc1nc(C(C)C)oc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141012__15859360
O=C(CCc1cn[nH]c1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141032__15862300
O=C(CCc1cn[nH]c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141032__15859360
CC(Cc1cnc[nH]1)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141040__15862300
CC(Cc1cnc[nH]1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141040__15859360
C=CCCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14141042__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@H]1C1CC1 s275592__15865748__14141044__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]1C1CC1 s275592__15865748__14141044__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)[C@@H]1C[C@H]1C1CC1 s275592__15865748__14141044__15857566
C[C@]1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C[C@@H]1c1ccccc1 s275592__15865748__14141046__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC2CCCN21 s275592__15865748__14141048__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@H]1C1CCC1 s275592__15865748__14141052__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]1C1CCC1 s275592__15865748__14141052__15859360
Cc1cccc([C@@H]2C[C@H]2C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14141062__15859360
Cc1ccccc1[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141064__15859360
C=C(C)[C@@H]1OCC[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141074__15862300
C=C(C)[C@@H]1OCC[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141074__15859360
O=C(C[C@@H]1C[C@H]1c1ccccc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141078__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cn(C2CCC2)nn1 s275592__15865748__14141084__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cscc1C(F)F s275592__15865748__14141086__15859360
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCO1 s275592__15865748__14141092__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnn1C1CCC1 s275592__15865748__14141094__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccnn1C s275592__15865748__14141112__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnn1C s275592__15865748__14141112__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)sn1 s275592__15865748__14141122__15862300
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)sn1 s275592__15865748__14141122__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cn2c(n1)CCC2 s275592__15865748__14141126__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cn2c(n1)CCC2 s275592__15865748__14141126__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]1c1ccncc1 s275592__15865748__14141128__15859360
C[C@@H]1[C@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCN1C s275592__15865748__14141130__15862300
C[C@@H]1[C@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCN1C s275592__15865748__14141130__15859360
CC(C)(C)c1nc[nH]c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141132__15859360
CC(C)(C)C[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141136__15862300
CC(C)(C)C[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141136__15859360
NC(=O)c1ncn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14141142__15859360
CC[C@@H]1[C@@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCN1C s275592__15865748__14141144__15862300
CC[C@@H]1[C@@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCN1C s275592__15865748__14141144__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@@H]2C=C[C@H]1CC2 s275592__15865748__14141148__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@@H]2C=C[C@H]1CC2 s275592__15865748__14141148__15859360
CCn1ccc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14141150__15862300
CCn1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14141150__15859360
CC1OC(C)C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1C s275592__15865748__14136182__15862300
CC1OC(C)C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1C s275592__15865748__14136182__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cn[nH]c1-c1ccco1 s275592__15865748__14136190__15859360
CCC(C)(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136200__15862300
CCC(C)(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136200__15859360
CCC(C)(CC)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14136200__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(F)c1 s275592__15865748__14136210__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCS1(=O)=O s275592__15865748__14136222__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1noc2c1COCC2 s275592__15865748__14136224__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCc2cn[nH]c2C1 s275592__15865748__14136228__15859360
CCN1CCOC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14136238__15862300
CCN1CCOC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14136238__15859360
CC1CCC(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)O1 s275592__15865748__14136244__15862300
CC1CCC(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)O1 s275592__15865748__14136244__15859360
Cc1cc(=O)[nH]c(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136248__15859360
C[C@@H](Cc1ccccc1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136250__15859360
C[C@H](Cc1ccccc1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136252__15859360
C=CCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14136254__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C12CCC(CC1)CC2 s275592__15865748__14136256__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C12CCC(CC1)CC2 s275592__15865748__14136256__15859360
CCCCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136264__15862300
CCCCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136264__15859360
CC[C@H](C)[C@H](NC(C)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136270__15859360
CCCCCC(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136272__15862300
CCCCCC(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136272__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(C2CC2)cc1 s275592__15865748__14136276__15859360
CC1=CCC(C)(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14136280__15862300
CC1=CCC(C)(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14136280__15859360
CC(C)(C)CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136286__15862300
CC(C)(C)CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136286__15859360
C=CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14136292__15859360
CCN(CC)C(=O)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136300__15859360
C=CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14136304__15859360
C=CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCCC1 s275592__15865748__14136308__15859360
Cc1ccccc1C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136314__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)Cc1ccccc1 s275592__15865748__14136320__15859360
CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCCC1 s275592__15865748__14136324__15862300
CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCCC1 s275592__15865748__14136324__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)n1 s275592__15865748__14136334__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)n1 s275592__15865748__14136334__15859360
CCCn1nccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138672__15862300
CCCn1nccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138672__15859360
CCCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14138674__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C2CC2)n1 s275592__15865748__14138676__15859360
Cc1c(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1C s275592__15865748__14138680__15859360
COc1cc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__14138686__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc2[nH]cnc12 s275592__15865748__14138690__15859360
Cc1cccc(C)c1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138692__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1C=CC=CC=C1 s275592__15865748__14138694__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1C=CC=CC=C1 s275592__15865748__14138694__15859360
C=C(C)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138696__15862300
C=C(C)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138696__15859360
C=C(C)CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138696__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2[nH]cnc2c1 s275592__15865748__14138698__15859360
O=C(CCc1ccncn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138702__15862300
O=C(CCc1ccncn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138702__15859360
CC(C)Cn1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14138704__15859360
CCC(C)n1nccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138708__15859360
CC(C)Cn1nccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138710__15859360
Cn1ccc(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14138714__15862300
Cn1ccc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14138714__15859360
Cn1nccc1CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138716__15862300
Cn1nccc1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138716__15859360
Cn1nc(C2CC2)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138718__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc2occc2[nH]1 s275592__15865748__14138720__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2occc2[nH]1 s275592__15865748__14138720__15859360
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O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccns1 s275592__15865748__14138722__15859360
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CC1CCC(C)(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14136590__15859360
CC(C)Cc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136596__15859360
CC(C)(C)C12CC(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)(C1)C2 s275592__15865748__14136606__15859360
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C#CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCCC1 s275592__15865748__14136618__15859360
CC(CC1CCCO1)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136620__15862300
CC(CC1CCCO1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136620__15859360
CC(C)c1occc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136622__15862300
CC(C)c1occc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136622__15859360
CCOCCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136628__15862300
CCOCCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136628__15859360
CNC(=O)CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136630__15862300
CNC(=O)CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136630__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCc2ccccc21 s275592__15865748__14136634__15859360
CC(C)(C)C1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14136638__15862300
CC(C)(C)C1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14136638__15859360
CC1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1C s275592__15865748__14136640__15862300
CC1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1C s275592__15865748__14136640__15859360
COC1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136642__15862300
COC1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136642__15859360
CC1CCC(C)N1C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136650__15859360
C=CCCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136652__15862300
C=CCCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136652__15859360
C=CCCOCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14136652__15857566
C=CCOC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136654__15862300
C=CCOC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136654__15859360
C=CCOC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14136654__15857566
CC(C)CCOC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136656__15862300
CC(C)CCOC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136656__15859360
CC(OCC1CCCO1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136660__15859360
CCc1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)s1 s275592__15865748__14136670__15862300
CCc1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14136670__15859360
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CC(C)(C)c1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139006__15859360
COCCn1nccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139024__15859360
Cc1cnc2nc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)nn2c1 s275592__15865748__14139028__15859360
Cc1cnccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139032__15862300
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Cc1nc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc2o1 s275592__15865748__14139036__15859360
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C[C@@H]1OCCO[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141518__15862300
C[C@@H]1OCCO[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141518__15859360
Cn1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1=O s275592__15865748__14141520__15862300
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CCc1cnc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)[nH]1 s275592__15865748__14141522__15862300
CCc1cnc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)[nH]1 s275592__15865748__14141522__15859360
Cn1cnc2cncc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c21 s275592__15865748__14141534__15859360
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CN1CCCC1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141536__15859360
CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCNC1=O s275592__15865748__14141544__15862300
CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCNC1=O s275592__15865748__14141544__15859360
CC[C@@H]1CCO[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141550__15862300
CC[C@@H]1CCO[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141550__15859360
O=C(CC=CCc1ccccc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141552__15859360
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CC1C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1C1CC1 s275592__15865748__14141590__15862300
CC1C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1C1CC1 s275592__15865748__14141590__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC2CCCCN21 s275592__15865748__14141594__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccncc1 s275592__15865748__14141598__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCNC(=O)C1 s275592__15865748__14141602__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCNC(=O)C1 s275592__15865748__14141602__15859360
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COc1cncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14141636__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cn2c(n1)COCC2 s275592__15865748__14141640__15859360
COCc1sccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141646__15859360
CCC1CCCC1(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141648__15862300
CCC1CCCC1(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141648__15859360
COCCOCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136676__15862300
COCCOCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136676__15859360
CC1CCCCC1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136680__15862300
CC1CCCCC1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136680__15859360
O=C(CCc1ccccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136686__15862300
O=C(CCc1ccccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136686__15859360
O=C(CCc1cscn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136690__15862300
O=C(CCc1cscn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136690__15859360
Cc1cc(C)n(C(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14136692__15859360
O=C(CCCCN1CCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136694__15859360
CN(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14136696__15859360
CCCCC(NC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136702__15859360
CN(C)c1ccnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14136704__15859360
O=C(CCCn1ccnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136706__15862300
O=C(CCCn1ccnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136706__15859360
COCc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cs1 s275592__15865748__14136712__15859360
NC(=O)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc1 s275592__15865748__14136714__15859360
CC1CCC(OCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14136720__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1csc(C2CC2)n1 s275592__15865748__14136724__15859360
CC(C)OCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136736__15862300
CC(C)OCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136736__15859360
NC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136738__15862300
NC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136738__15859360
NC(=O)CCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14136738__15857566
CN1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14136742__15862300
CN1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14136742__15859360
NC(=O)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14136748__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1COc2ccccc21 s275592__15865748__14136750__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1coc2ccccc12 s275592__15865748__14136752__15859360
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C1CC1 s275592__15865748__14136754__15859360
Cc1ccccc1C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14136762__15859360
NC(=O)N1CCC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136766__15862300
NC(=O)N1CCC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136766__15859360
CC(C)CC(=O)NCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136774__15859360
Cc1cccc(F)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136780__15862300
Cc1cccc(F)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136780__15859360
Cc1ccccc1C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136792__15859360
O=C(COCC1CCCO1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136804__15862300
O=C(COCC1CCCO1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136804__15859360
CC(NC(=O)C1CCC1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136808__15859360
CC(=O)N[C@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)(C)C s275592__15865748__14136816__15859360
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1C s275592__15865748__14136820__15862300
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1C s275592__15865748__14136820__15859360
CCOc1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14136824__15859360
CCn1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14136826__15862300
CCn1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14136826__15859360
O=C(CCc1cncc(F)c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136830__15859360
Cn1cc(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__14136832__15862300
Cn1cc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14136832__15859360
COCc1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14136834__15859360
Cc1ccc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14136836__15859360
CC(C)CC(C(N)=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136838__15862300
CC(C)CC(C(N)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136838__15859360
O=C(CC(F)(F)C(F)(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136840__15859360
CCCC1CCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139168__15862300
CCCC1CCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139168__15859360
CCC(CC)C(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139174__15862300
CCC(CC)C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139174__15859360
O=C(CC1CS(=O)(=O)C1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139176__15859360
Cn1cnn(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1=O s275592__15865748__14139182__15862300
Cn1cnn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1=O s275592__15865748__14139182__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2ccccn12 s275592__15865748__14139186__15859360
Cc1ccn2cnc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c2c1 s275592__15865748__14139190__15859360
Cc1ccc2[nH]ncc2c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139192__15859360
CCc1cnccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139202__15862300
CCc1cnccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139202__15859360
CCN1CCOCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139204__15862300
CCN1CCOCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139204__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(F)CCCC1 s275592__15865748__14139208__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(F)CCCC1 s275592__15865748__14139208__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(F)CCCC1 s275592__15865748__14139208__15857566
CCc1cccnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139210__15862300
CCc1cccnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139210__15859360
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnc1 s275592__15865748__14139214__15859360
Cc1nnc2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cn12 s275592__15865748__14139216__15859360
CN(C)Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__14139224__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc2cncn12 s275592__15865748__14139228__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(=O)NCC(F)F s275592__15865748__14139232__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(=O)NCC(F)F s275592__15865748__14139232__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnn(CCF)c1 s275592__15865748__14139238__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn(CCF)c1 s275592__15865748__14139238__15859360
Cc1cc(C)nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14139240__15862300
Cc1cc(C)nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139240__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2ncnn12 s275592__15865748__14139246__15859360
Cn1cncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139248__15862300
Cn1cncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139248__15859360
Cn1cncc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139248__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2cccnc12 s275592__15865748__14139250__15859360
O=C(CCc1ccc(F)cc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139254__15859360
O=C(CCc1cccnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139258__15862300
O=C(CCc1cccnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139258__15859360
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(F)c1 s275592__15865748__14139260__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ccccc2s1 s275592__15865748__14139262__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1c[nH]c2ccccc12 s275592__15865748__14139270__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c[nH]c2ccccc12 s275592__15865748__14139270__15859360
Cc1ccn2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)nc2c1 s275592__15865748__14139276__15859360
O=C(Cn1ccc(=O)[nH]c1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139282__15859360
COCc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139284__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c2ccccc21 s275592__15865748__14139290__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)s1 s275592__15865748__14139292__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)s1 s275592__15865748__14139292__15859360
NC(=O)NCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139298__15862300
NC(=O)NCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139298__15859360
CCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)s1 s275592__15865748__14139302__15862300
CCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14139302__15859360
Cc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1 s275592__15865748__14139308__15862300
Cc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14139308__15859360
CCc1nnsc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139310__15862300
CCc1nnsc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139310__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc2ccccc12 s275592__15865748__14139312__15859360
COc1ccc(C)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139316__15859360
O=C(CC1CCS(=O)(=O)C1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139322__15859360
O=C(Cc1noc2ccccc12)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139330__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2cnccc2[nH]1 s275592__15865748__14141650__15859360
Cc1nc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)s1 s275592__15865748__14141656__15859360
Cn1nnc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc21 s275592__15865748__14141658__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)(C)C s275592__15865748__14141660__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)(C)C s275592__15865748__14141660__15859360
CC(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C(C)(C)C s275592__15865748__14141660__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCc2ccccc21 s275592__15865748__14141662__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C12CCC(CC1)C2 s275592__15865748__14141668__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C12CCC(CC1)C2 s275592__15865748__14141668__15859360
CN1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141670__15862300
CN1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141670__15859360
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1Cl s275592__15865748__14141672__15862300
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1Cl s275592__15865748__14141672__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C(F)(F)F)CCC1 s275592__15865748__14141680__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ncc(F)cc1F s275592__15865748__14141682__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncc(F)cc1F s275592__15865748__14141682__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)S(C)(=O)=O s275592__15865748__14141684__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)S(C)(=O)=O s275592__15865748__14141684__15859360
CS(=O)(=O)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141686__15862300
CS(=O)(=O)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141686__15859360
O=C(Cc1cn2ccccc2n1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141696__15859360
O=C(Cc1cccnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141698__15862300
O=C(Cc1cccnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141698__15859360
CCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__14141704__15862300
CCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__14141704__15859360
NC(=O)c1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14141706__15859360
CN1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1=O s275592__15865748__14141708__15862300
CN1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1=O s275592__15865748__14141708__15859360
C=CCOc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14141710__15859360
C=CCOc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141712__15859360
Cn1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1=O s275592__15865748__14141714__15862300
Cn1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1=O s275592__15865748__14141714__15859360
CC(=O)NCC(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141718__15859360
CC(F)(F)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141724__15862300
CC(F)(F)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141724__15859360
O=C(COC1CCCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141730__15862300
O=C(COC1CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141730__15859360
O=C(CCOCC(F)(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141732__15859360
O=C(CCOCC1CCCO1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141736__15859360
O=C(CCc1ccncc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141742__15862300
O=C(CCc1ccncc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141742__15859360
CC(C)(C)n1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14141744__15859360
O=C1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CN1 s275592__15865748__14141746__15862300
O=C1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CN1 s275592__15865748__14141746__15859360
CC(C)CN1CCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141750__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ccn1 s275592__15865748__14141752__15862300
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccn1 s275592__15865748__14141752__15859360
CN(C)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14141754__15859360
CCCc1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141758__15862300
CCCc1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141758__15859360
CCc1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141760__15862300
CCc1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141760__15859360
CC(C)c1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141762__15862300
CC(C)c1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141762__15859360
CC(C)(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)[nH]n1 s275592__15865748__14141764__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1n[nH]c2c1CCC2 s275592__15865748__14141768__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1n[nH]c2c1CCC2 s275592__15865748__14141768__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1n[nH]c2c1CCCC2 s275592__15865748__14141772__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1c[nH]nn1 s275592__15865748__14141778__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c[nH]nn1 s275592__15865748__14141778__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1c[nH]nn1 s275592__15865748__14141778__15857566
O=C(CN1CCCCC1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141784__15862300
O=C(CN1CCCCC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141784__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ccc1=O s275592__15865748__14141788__15862300
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc1=O s275592__15865748__14141788__15859360
COCc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141792__15859360
CCc1c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cnn1C s275592__15865748__14141794__15862300
CCc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1C s275592__15865748__14141794__15859360
CCCc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1C s275592__15865748__14141796__15859360
Cc1ccc2[nH]nc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c2c1 s275592__15865748__14141802__15859360
O=C(CN1CCCNC1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141806__15862300
O=C(CN1CCCNC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141806__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(=O)Nc1ccccc1 s275592__15865748__14141810__15859360
COC1CCC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14136844__15859360
CC1(C)C(C)(C)C1(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136846__15862300
CC1(C)C(C)(C)C1(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136846__15859360
C=CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCC1 s275592__15865748__14136848__15862300
C=CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__14136848__15859360
CC1(C)CCCCC1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136860__15859360
Cc1[nH]cnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136862__15862300
Cc1[nH]cnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136862__15859360
Cc1[nH]cnc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14136862__15857566
C[C@@H](C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N1CCOCC1 s275592__15865748__14136868__15862300
C[C@@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCOCC1 s275592__15865748__14136868__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC12CCOCC2 s275592__15865748__14136878__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC12CCOCC2 s275592__15865748__14136878__15859360
CC1(C)CCC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14136880__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCOCC1 s275592__15865748__14136882__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCOCC1 s275592__15865748__14136882__15859360
O=C(CC1CC(=O)NC1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136886__15862300
O=C(CC1CC(=O)NC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136886__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1C(C)C s275592__15865748__14136888__15859360
CC1(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC(=O)N1 s275592__15865748__14136898__15859360
CCOc1cccnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136900__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2n(c1)CCCC2 s275592__15865748__14136904__15859360
NC(=O)c1ccnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14136906__15859360
CC(C)c1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14136910__15859360
Cc1cccc2c1OC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C2 s275592__15865748__14136912__15859360
CCC(CC)C(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136914__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC2CCC1C2 s275592__15865748__14136918__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC2CCC1C2 s275592__15865748__14136918__15859360
CC1C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1c1ccccc1 s275592__15865748__14136926__15859360
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCC1 s275592__15865748__14136928__15859360
CCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1CC s275592__15865748__14136936__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCS1(=O)=O s275592__15865748__14136942__15859360
CCc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)o1 s275592__15865748__14136946__15862300
CCc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)o1 s275592__15865748__14136946__15859360
CC(=O)NCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136954__15862300
CC(=O)NCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136954__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)C(C)(C)C s275592__15865748__14136956__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C(C)(C)C s275592__15865748__14136956__15859360
CC(Cc1ccco1)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136958__15862300
CC(Cc1ccco1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136958__15859360
C=CC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCCC1 s275592__15865748__14136962__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(c1)C=CCC2 s275592__15865748__14136964__15859360
O=C(CCNC(=O)C1CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136966__15859360
CC(=O)NC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__14136970__15859360
CS(=O)(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136974__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(c1)COC2 s275592__15865748__14136976__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCC1 s275592__15865748__14136980__15859360
O=C(CC1CCC(=O)N1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14136982__15862300
O=C(CC1CCC(=O)N1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14136982__15859360
CCc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14136986__15859360
Cc1nnc2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cn12 s275592__15865748__14136994__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2nncn2c1 s275592__15865748__14136996__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccn2ccnc12 s275592__15865748__14137000__15859360
CNC(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14137002__15862300
CNC(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14137002__15859360
O=C(CCN1C(=O)CCC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139338__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCS(=O)(=O)C1 s275592__15865748__14139340__15859360
CC(=O)N1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14139344__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1Cc2ccccc2O1 s275592__15865748__14139348__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(Cl)cc1F s275592__15865748__14139350__15859360
NC(=O)N1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14139352__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1F s275592__15865748__14139354__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1F s275592__15865748__14139354__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc1C s275592__15865748__14139358__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(Cl)ccc1F s275592__15865748__14139360__15859360
CCCCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14139362__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(c2ccccc2)CCC1 s275592__15865748__14139366__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1COc2ccccc2C1 s275592__15865748__14139370__15859360
Cc1[nH]c2ccccc2c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139372__15859360
Cc1oc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1C s275592__15865748__14139380__15862300
Cc1oc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14139380__15859360
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__14139382__15862300
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14139382__15859360
Cc1cc(C)n(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14139390__15862300
Cc1cc(C)n(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14139390__15859360
COCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__14139396__15862300
COCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__14139396__15859360
Cc1cc(=O)oc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139398__15859360
Cn1cc(Cl)cc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139400__15862300
Cn1cc(Cl)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139400__15859360
CC(C)=CC1C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1(C)C s275592__15865748__14139402__15859360
Cc1ccc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14139410__15859360
O=C(Cc1ccc2[nH]ncc2c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139422__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccn2ccnc2c1 s275592__15865748__14139434__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2nccn12 s275592__15865748__14139436__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2[nH]ccc2n1 s275592__15865748__14139438__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2nnnn2c1 s275592__15865748__14139440__15859360
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n(C)n1 s275592__15865748__14139444__15862300
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n(C)n1 s275592__15865748__14139444__15859360
Cc1ccc2ncc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)n2c1 s275592__15865748__14139448__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncc(Cl)s1 s275592__15865748__14139450__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c2ccccn12 s275592__15865748__14139454__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncc2ccccn12 s275592__15865748__14139456__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1onc2c1CCCC2 s275592__15865748__14139460__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(c1ccccc1)C1CC1 s275592__15865748__14139462__15859360
COCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14139464__15862300
COCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14139464__15859360
COCC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC1 s275592__15865748__14139464__15857566
COCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139466__15862300
COCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139466__15859360
COCC(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139466__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2nccn2c1 s275592__15865748__14139480__15859360
O=C(CCc1ccon1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139482__15862300
O=C(CCc1ccon1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139482__15859360
O=C(CCc1cncnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139484__15862300
O=C(CCc1cncnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139484__15859360
Cn1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1C(F)F s275592__15865748__14139488__15859360
COc1coc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1=O s275592__15865748__14139490__15859360
COc1c[nH]c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1=O s275592__15865748__14139492__15859360
Cc1cc(Cl)cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139494__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2cncn2c1 s275592__15865748__14139498__15859360
CCc1cncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14139500__15862300
CCc1cncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139500__15859360
NC(=O)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14137006__15859360
O=C1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC(=O)N1 s275592__15865748__14137010__15862300
O=C1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC(=O)N1 s275592__15865748__14137010__15859360
Cc1noc(Cl)c1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137012__15859360
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14137016__15862300
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14137016__15859360
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)n1 s275592__15865748__14137016__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cncc(Cl)c1 s275592__15865748__14137024__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cncc(Cl)c1 s275592__15865748__14137024__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c2[nH]ncc2c1 s275592__15865748__14137034__15859360
Cc1nccn1CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137036__15859360
Cc1noc(C)c1C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137038__15859360
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1C s275592__15865748__14137040__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cs1 s275592__15865748__14137046__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cs1 s275592__15865748__14137046__15859360
CC1Cc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc2O1 s275592__15865748__14137054__15859360
O=C(CCN1CCOCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137058__15862300
O=C(CCN1CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137058__15859360
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCOCC1 s275592__15865748__14137062__15859360
O=C(COc1cccnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137066__15862300
O=C(COc1cccnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137066__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCOCC1 s275592__15865748__14137068__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCOCC1 s275592__15865748__14137068__15859360
Cc1cc(C(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)o1 s275592__15865748__14137070__15859360
CCc1ccc(C(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14137072__15859360
CC(C)c1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cs1 s275592__15865748__14137074__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(C(F)F)cc1 s275592__15865748__14137082__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCOc2ccccc21 s275592__15865748__14137086__15859360
Cn1ccc2c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cccc21 s275592__15865748__14137092__15859360
CC(C)CCC(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137096__15859360
CCn1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14137102__15859360
CC(C)CC(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137108__15862300
CC(C)CC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137108__15859360
Cn1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C(F)F s275592__15865748__14137112__15859360
CCCCCCC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137114__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2nccn2c1 s275592__15865748__14137118__15859360
CCC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14137128__15859360
CCC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)(C)C s275592__15865748__14137130__15862300
CCC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)(C)C s275592__15865748__14137130__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC(F)(F)C1 s275592__15865748__14137132__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC(F)(F)C1 s275592__15865748__14137132__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc2c([nH]1)CCC2 s275592__15865748__14137134__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2c([nH]1)CCC2 s275592__15865748__14137134__15859360
CC(C)c1scnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137138__15859360
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(Cl)n1 s275592__15865748__14137140__15862300
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(Cl)n1 s275592__15865748__14137140__15859360
COCc1nocc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137154__15862300
COCc1nocc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137154__15859360
CC(C)n1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__14137156__15862300
CC(C)n1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14137156__15859360
Cc1nn(C(C)C)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137158__15859360
CCc1oc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1C s275592__15865748__14137166__15862300
CCc1oc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1C s275592__15865748__14137166__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCCC1=O s275592__15865748__14137168__15859360
Cc1csc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14139502__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2cnccc2c1 s275592__15865748__14139504__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nc1C s275592__15865748__14139506__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc1C s275592__15865748__14139506__15859360
Cc1cncn1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139508__15862300
Cc1cncn1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139508__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nnc2ccccc2n1 s275592__15865748__14139516__15859360
O=C(CCC(F)F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139520__15862300
O=C(CCC(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139520__15859360
O=C(CCC(F)F)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139520__15857566
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc(=O)[nH]1 s275592__15865748__14139532__15859360
CCOc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)on1 s275592__15865748__14139538__15862300
CCOc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__14139538__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC2(CC1)CC2 s275592__15865748__14139540__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC2(CC1)CC2 s275592__15865748__14139540__15859360
COCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__14139542__15862300
COCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14139542__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2ccncc2n1 s275592__15865748__14139544__15859360
O=C(CCC1CCCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139546__15859360
Cc1onc(C2CC2)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139550__15859360
Cc1noc(C2CC2)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139552__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ncccc2o1 s275592__15865748__14139554__15859360
O=C(Cc1ccc(=O)[nH]c1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139556__15862300
O=C(Cc1ccc(=O)[nH]c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139556__15859360
CC(CC(F)F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139558__15862300
CC(CC(F)F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139558__15859360
Cn1nnc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cnc21 s275592__15865748__14139560__15859360
CC1Cc2cccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c2O1 s275592__15865748__14139566__15859360
CC1(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14139572__15862300
CC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14139572__15859360
CC1(CC(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC1 s275592__15865748__14139572__15857566
CCCCC(CC)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139576__15862300
CCCCC(CC)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139576__15859360
CCC1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC(=O)N1 s275592__15865748__14139578__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CNC(=O)C1 s275592__15865748__14139580__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CNC(=O)C1 s275592__15865748__14139580__15859360
O=C(Cc1cccc(C2CC2)c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139588__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c[nH]nc1-c1ccoc1 s275592__15865748__14139592__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC2CC2C1 s275592__15865748__14139598__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC2CC2C1 s275592__15865748__14139598__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(CCF)CC1 s275592__15865748__14139602__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(CCF)CC1 s275592__15865748__14139602__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(CCF)CC1 s275592__15865748__14139602__15857566
COCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139604__15862300
COCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139604__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn(C)c1 s275592__15865748__14139608__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCC1C1CC1 s275592__15865748__14139610__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c2nccn2c1 s275592__15865748__14139612__15859360
Cc1ccc(C2CC2)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139614__15859360
Cc1nccc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14139624__15859360
Cn1cnn(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1=O s275592__15865748__14139626__15859360
O=C(COCC(F)F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139628__15862300
O=C(COCC(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139628__15859360
O=C(CCCCc1c[nH]nn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139634__15859360
NC(=O)c1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)co1 s275592__15865748__14139636__15862300
NC(=O)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)co1 s275592__15865748__14139636__15859360
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)nn1 s275592__15865748__14139644__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCC1(F)F s275592__15865748__14139650__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C2CC2)CCOCC1 s275592__15865748__14139652__15859360
CC(C)n1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14139654__15862300
CC(C)n1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139654__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cn2cccnc2n1 s275592__15865748__14141818__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C12CCCN1CCC2 s275592__15865748__14141822__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C12CCCN1CCC2 s275592__15865748__14141822__15859360
CCc1ccc(F)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141832__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccn2nccc12 s275592__15865748__14141834__15859360
O=C1Cc2c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccnc2N1 s275592__15865748__14141836__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnc1C1CC1 s275592__15865748__14141842__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn2c1OCCC2 s275592__15865748__14141848__15859360
CCOc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)co1 s275592__15865748__14141852__15862300
CCOc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)co1 s275592__15865748__14141852__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncnc2[nH]ccc12 s275592__15865748__14141856__15859360
Cn1nc2c(c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CCC2 s275592__15865748__14137172__15859360
CN1CCCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1=O s275592__15865748__14137174__15859360
Cc1cccn2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc12 s275592__15865748__14137176__15859360
Cc1nc2nccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)n2n1 s275592__15865748__14137178__15859360
CN1C(=O)CN(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1=O s275592__15865748__14137182__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCc2[nH]ncc2C1 s275592__15865748__14137184__15859360
CCCc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)co1 s275592__15865748__14137192__15862300
CCCc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)co1 s275592__15865748__14137192__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2(CCOCC2)C1 s275592__15865748__14137196__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(C2CC2)s1 s275592__15865748__14137198__15859360
COCc1ccsc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137200__15859360
CCCc1occc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137202__15862300
CCCc1occc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137202__15859360
Cc1ccc(C(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14137204__15859360
CCOCCOCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137206__15859360
CC(C)(C)C(NC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137210__15859360
CC(CCC(C)(C)C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137212__15862300
CC(CCC(C)(C)C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137212__15859360
CCCCCCC(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137214__15859360
CN(C)C1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14137226__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(C2CCC2)c1 s275592__15865748__14137228__15859360
CC1(C)CCCC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14137232__15859360
CN1CCC(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14137242__15862300
CN1CCC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14137242__15859360
Cn1cncc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137244__15862300
Cn1cncc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137244__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c[nH]c2cccnc12 s275592__15865748__14137248__15859360
O=C(COc1ccsc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137250__15862300
O=C(COc1ccsc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137250__15859360
CCCc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__14137252__15859360
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CCc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__14137256__15862300
CCc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__14137256__15859360
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)oc1CC s275592__15865748__14137262__15859360
Cc1cccc2c1CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)O2 s275592__15865748__14137264__15859360
COc1cc[nH]c(=O)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137268__15859360
CC(C)Cc1c[nH]c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14137270__15859360
CCn1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14137272__15862300
CCn1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14137272__15859360
CN(C)c1ccncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137274__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(c1)CCC=C2 s275592__15865748__14137276__15859360
CCC(CC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137278__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccco1 s275592__15865748__14137282__15862300
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccco1 s275592__15865748__14137282__15859360
CC(Oc1ccccn1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137284__15859360
CCC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N(C)C s275592__15865748__14137286__15862300
CCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N(C)C s275592__15865748__14137286__15859360
CCC(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)N(C)C s275592__15865748__14137286__15857566
C[C@H](C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccc1 s275592__15865748__14137290__15862300
C[C@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14137290__15859360
CN(C)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14137292__15859360
Cc1ccn2ncc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c2n1 s275592__15865748__14137296__15859360
CN(C)C(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137310__15862300
CN(C)C(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137310__15859360
CCNC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137312__15862300
CCNC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137312__15859360
CCCNC(=O)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137314__15862300
CCCNC(=O)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137314__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1cccnc1 s275592__15865748__14137318__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnc1 s275592__15865748__14137318__15859360
CCCNC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137320__15859360
CC(C)NC(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137322__15859360
O=C(Cn1cc2ccccc2n1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137326__15859360
Cc1ccc(C(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14137334__15859360
CN(C)C1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__14139670__15859360
CNS(=O)(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139672__15859360
O=C1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCN1 s275592__15865748__14139676__15862300
O=C1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCN1 s275592__15865748__14139676__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc2ccncc12 s275592__15865748__14139678__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1occ2c1CCC2 s275592__15865748__14139680__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1occ2c1CCC2 s275592__15865748__14139680__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1occ2c1CCOC2 s275592__15865748__14139682__15859360
Cc1cncc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14139684__15862300
Cc1cncc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139684__15859360
C=CC(C)(CCOC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139686__15862300
C=CC(C)(CCOC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139686__15859360
O=C(CC1CCCS1(=O)=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139688__15859360
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn(C)c1 s275592__15865748__14139690__15859360
COC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCOC1 s275592__15865748__14139694__15862300
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCOC1 s275592__15865748__14139694__15859360
CCOC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC1 s275592__15865748__14139698__15859360
CCOC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCOC1 s275592__15865748__14139700__15859360
COCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCOC1 s275592__15865748__14139704__15862300
COCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCOC1 s275592__15865748__14139704__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(C2CC2)CCC1 s275592__15865748__14139712__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C2CC2)CCC1 s275592__15865748__14139712__15859360
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC1 s275592__15865748__14139726__15862300
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC1 s275592__15865748__14139726__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(C2CCC2)CCC1 s275592__15865748__14139728__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C2CCC2)CCC1 s275592__15865748__14139728__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C2CC2)n1 s275592__15865748__14139734__15859360
COC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC1 s275592__15865748__14139736__15862300
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC1 s275592__15865748__14139736__15859360
Cc1cccc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139740__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1csnn1 s275592__15865748__14139744__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1csnn1 s275592__15865748__14139744__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1csnn1 s275592__15865748__14139744__15857566
CC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)no1 s275592__15865748__14139748__15862300
CC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__14139748__15859360
Cc1ccc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)[nH]c2c1 s275592__15865748__14139756__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(C2CC2)on1 s275592__15865748__14139760__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(C2CC2)on1 s275592__15865748__14139760__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1csc2ccccc12 s275592__15865748__14139762__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCC1 s275592__15865748__14139764__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__14139764__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CCCC1 s275592__15865748__14139764__15857566
Cc1ccc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)c1 s275592__15865748__14139770__15859360
Cc1ccc(F)cc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139772__15862300
Cc1ccc(F)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139772__15859360
Cc1nn(C)c(C)c1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139776__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnco1 s275592__15865748__14139778__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnco1 s275592__15865748__14139778__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1cnco1 s275592__15865748__14139778__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2ncccc12 s275592__15865748__14139782__15859360
Cc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(=O)[nH]1 s275592__15865748__14139784__15859360
Cc1nn(C)c(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139786__15862300
Cc1nn(C)c(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139786__15859360
Cc1nn(C)c(Cl)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139794__15859360
Cc1cc(C)n(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14139798__15859360
O=C(Cc1ccc2c(c1)CCO2)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139800__15859360
O=C(CCn1ccnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139804__15862300
O=C(CCn1ccnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139804__15859360
COc1ccc(F)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139820__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ccsc2[nH]1 s275592__15865748__14139822__15859360
O=C(Cc1cc2ccccc2o1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139826__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2cnccc2o1 s275592__15865748__14141864__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccn2cncc2c1 s275592__15865748__14141866__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1n[nH]c(=O)[nH]c1=O s275592__15865748__14141868__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1n[nH]c(=O)[nH]c1=O s275592__15865748__14141868__15859360
Cc1nnccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141870__15862300
Cc1nnccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141870__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc(C2CC2)c1 s275592__15865748__14141872__15859360
COCc1csc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14141876__15859360
CC(C)c1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14141878__15859360
Cn1cc(C(N)=O)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141884__15859360
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCOCC1 s275592__15865748__14141892__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2c(cn1)CCCC2 s275592__15865748__14141894__15859360
O=C(CC1CCCC(=O)N1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141896__15862300
O=C(CC1CCCC(=O)N1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141896__15859360
NC(=O)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__14141900__15862300
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Cc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc1C s275592__15865748__14141904__15859360
Cn1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1Cl s275592__15865748__14141906__15862300
Cn1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1Cl s275592__15865748__14141906__15859360
Cc1cc(F)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(F)c1 s275592__15865748__14141910__15859360
CCCc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141912__15859360
COc1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nc1 s275592__15865748__14141914__15862300
COc1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc1 s275592__15865748__14141914__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1C s275592__15865748__14141916__15862300
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1C s275592__15865748__14141916__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnc1C(F)F s275592__15865748__14141920__15859360
Cc1cncc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14141922__15859360
CC1(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCCC1 s275592__15865748__14141924__15862300
CC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCCC1 s275592__15865748__14141924__15859360
CC(C)CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__14141928__15862300
CC(C)CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14141928__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCCCCC1 s275592__15865748__14141932__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCCCCC1 s275592__15865748__14141932__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(-c2ccco2)o1 s275592__15865748__14141938__15859360
COCCn1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14141940__15859360
Cn1ccc(=O)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14141942__15862300
Cn1ccc(=O)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14141942__15859360
Cc1cnc(COCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__14141944__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc2nn[nH]c12 s275592__15865748__14141946__15859360
Cc1sc(Cl)nc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141948__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccn2ccccc12 s275592__15865748__14141950__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccn2ccccc12 s275592__15865748__14141950__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nncc2ccccc12 s275592__15865748__14141952__15859360
Cc1n[nH]c2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc12 s275592__15865748__14141954__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2n(n1)CCCO2 s275592__15865748__14141958__15859360
COc1nccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14141960__15862300
COc1nccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14141960__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2c1CCOC2 s275592__15865748__14141970__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(c1)CCOC2 s275592__15865748__14141972__15859360
CC(C)(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__14141974__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC2CC1C1CC21 s275592__15865748__14141976__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2CC1C1CC21 s275592__15865748__14141976__15859360
CC1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C(C)O1 s275592__15865748__14141978__15862300
CC1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C(C)O1 s275592__15865748__14141978__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C12CCCCC1OCC2 s275592__15865748__14141982__15859360
CC(C)(C)[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141984__15862300
CC(C)(C)[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141984__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)[C@]12CCC[C@H]1OCC2 s275592__15865748__14141986__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)[C@]12CCC[C@H]1OCC2 s275592__15865748__14141986__15859360
CC1CC1C1CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14141988__15862300
CC1CC1C1CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14141988__15859360
CC1(C)COC(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14141992__15862300
CC1(C)COC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14141992__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]1C1CCOCC1 s275592__15865748__14141998__15859360
CC(C)(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC(F)F s275592__15865748__14142006__15859360
O=C(Cn1ncc2cccnc21)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14142008__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1OC[C@@H]2CCC[C@@H]21 s275592__15865748__14142010__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1OC[C@@H]2CCC[C@@H]21 s275592__15865748__14142010__15859360
CC1(C)CCC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)OC1 s275592__15865748__14142012__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@@H]2O[C@H]1[C@H]1C[C@@H]21 s275592__15865748__14142022__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@@H]2O[C@H]1[C@H]1C[C@@H]21 s275592__15865748__14142022__15859360
Cn1cccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1=O s275592__15865748__14137338__15862300
Cn1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1=O s275592__15865748__14137338__15859360
C#CCOc1ncccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137340__15859360
Cc1ccc(C(C)(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14137344__15859360
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)no1 s275592__15865748__14137348__15862300
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__14137348__15859360
CCC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)C s275592__15865748__14137350__15862300
CCC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__14137350__15859360
CN(C)CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137352__15862300
CN(C)CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137352__15859360
C#Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nc1 s275592__15865748__14137354__15862300
C#Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc1 s275592__15865748__14137354__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]1c1ccccc1 s275592__15865748__14137366__15859360
CO[C@@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14137368__15859360
O=C1CC[C@@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)N1 s275592__15865748__14137370__15862300
O=C1CC[C@@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)N1 s275592__15865748__14137370__15859360
O=C1CC[C@@H](C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)N1 s275592__15865748__14137370__15857566
CC(=O)N1CCC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137372__15862300
CC(=O)N1CCC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137372__15859360
COc1cc(C)ccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137374__15859360
CC(=O)N[C@@H](C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)C s275592__15865748__14137376__15862300
CC(=O)N[C@@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__14137376__15859360
Cn1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c2ccccc21 s275592__15865748__14137378__15859360
CC(=O)N[C@@H](CC(C)C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137380__15859360
C[C@@H](C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccc1 s275592__15865748__14137382__15862300
C[C@@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14137382__15859360
CC(=O)N[C@H](CC(C)C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137384__15859360
C[C@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14137386__15862300
C[C@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14137386__15859360
CC[C@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14137388__15862300
CC[C@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14137388__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ncccc1Cl s275592__15865748__14137390__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncccc1Cl s275592__15865748__14137390__15859360
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Cc1cc(F)ccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137394__15859360
Cc1ccc(F)c(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14137398__15859360
Cc1ccc2oc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc2n1 s275592__15865748__14137404__15859360
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CC(C)C(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N(C)C s275592__15865748__14137408__15862300
CC(C)C(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N(C)C s275592__15865748__14137408__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(C(F)F)c1 s275592__15865748__14137410__15859360
CCCN(C)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137412__15862300
CCCN(C)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137412__15859360
O=C(CCCc1ccccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137418__15859360
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COc1ccsc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137426__15862300
COc1ccsc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137426__15859360
CCCN(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137428__15862300
CCCN(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137428__15859360
CCCN(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137428__15857566
CC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)(C)C s275592__15865748__14137436__15862300
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)(C)C s275592__15865748__14137436__15859360
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COc1cccnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137438__15859360
CCCCCCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137440__15862300
CCCCCCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137440__15859360
O=C(Cc1ccc2c(c1)COC2)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137442__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnn2cc[nH]c12 s275592__15865748__14137444__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn2cc[nH]c12 s275592__15865748__14137444__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCO1 s275592__15865748__14137446__15862300
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCO1 s275592__15865748__14137446__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1occ2c1CCCC2 s275592__15865748__14137448__15859360
CC1(C)COC(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14137450__15859360
COCCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__14137454__15862300
COCCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14137454__15859360
CCC[C@@H](NC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137458__15862300
CCC[C@@H](NC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137458__15859360
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C#Cc1ccccc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137464__15862300
C#Cc1ccccc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137464__15859360
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Cc1[nH]cnc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137466__15859360
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Cc1csc(Cl)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137478__15859360
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COc1c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cnn1C s275592__15865748__14137486__15862300
COc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1C s275592__15865748__14137486__15859360
CC(F)(F)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137488__15862300
CC(F)(F)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137488__15859360
Cn1nnc2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc21 s275592__15865748__14137490__15859360
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CC(=O)N(C)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137500__15862300
CC(=O)N(C)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137500__15859360
Cc1noc(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14139834__15862300
Cc1noc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14139834__15859360
CC(NC(=O)C(C)(C)C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139844__15859360
CC(C)(C)C(=O)NCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139846__15859360
Cc1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139854__15862300
Cc1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139854__15859360
Cc1[nH]ncc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139854__15857566
Cc1noc2ncc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc12 s275592__15865748__14139856__15859360
CCCc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)[nH]n1 s275592__15865748__14139872__15862300
CCCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)[nH]n1 s275592__15865748__14139872__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2[nH]ncc12 s275592__15865748__14139876__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2cn[nH]c12 s275592__15865748__14139886__15859360
Cc1ccc2[nH]c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc2c1 s275592__15865748__14139888__15859360
Cc1n[nH]c(=O)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14139890__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1OCCc2ccccc21 s275592__15865748__14139892__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn2cccnc12 s275592__15865748__14139898__15859360
C#Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1 s275592__15865748__14139900__15862300
C#Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14139900__15859360
Cc1n[nH]nc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139906__15862300
Cc1n[nH]nc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139906__15859360
Cc1n[nH]nc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139906__15857566
COc1ccnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14139908__15862300
COc1ccnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139908__15859360
Cc1cc(F)cc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139910__15859360
COc1csc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14139918__15862300
COc1csc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14139918__15859360
CN1C(=O)CCC1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139920__15862300
CN1C(=O)CCC1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139920__15859360
O=C(CCc1ccccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139924__15862300
O=C(CCc1ccccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139924__15859360
Cn1cnc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cnc21 s275592__15865748__14139928__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccn2nnnc2c1 s275592__15865748__14139930__15859360
COc1nn(C)cc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139932__15862300
COc1nn(C)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139932__15859360
CCCC(OC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139940__15862300
CCCC(OC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139940__15859360
CCCC(OC)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139940__15857566
C=C(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139944__15862300
C=C(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139944__15859360
C=C(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139944__15857566
Cc1ccn(C(C)CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14139948__15859360
O=C(CN1CCNC(=O)C1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139952__15862300
O=C(CN1CCNC(=O)C1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139952__15859360
CCCCCCC(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139962__15859360
CC(CC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139970__15862300
CC(CC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139970__15859360
CC(CC(N)=O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139970__15857566
NC(=O)C1CCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139972__15862300
NC(=O)C1CCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139972__15859360
O=C1NCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139978__15862300
O=C1NCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139978__15859360
O=C1NCCC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139978__15857566
Cn1c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c[nH]c1=O s275592__15865748__14139980__15862300
Cn1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c[nH]c1=O s275592__15865748__14139980__15859360
CN1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)NC1=O s275592__15865748__14139982__15862300
CN1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)NC1=O s275592__15865748__14139982__15859360
C=CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139984__15862300
C=CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139984__15859360
C=CC(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139984__15857566
C#CCCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139986__15862300
C#CCCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139986__15859360
CN1CCC[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139990__15862300
CN1CCC[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139990__15859360
CN1CCC[C@@H]1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139990__15857566
C[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139992__15862300
C[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139992__15859360
C[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139992__15857566
O=C(CC1CC=CCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139994__15862300
O=C(CC1CC=CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139994__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__14139996__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14139996__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CCC1 s275592__15865748__14139996__15857566
O=C(C[C@@H]1C[C@H]1C1CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14142026__15862300
O=C(C[C@@H]1C[C@H]1C1CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14142026__15859360
CC1COC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14142028__15862300
CC1COC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14142028__15859360
CC1COC(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865748__14142028__15857566
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ncc1=O s275592__15865748__14142034__15862300
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ncc1=O s275592__15865748__14142034__15859360
Cc1nc(C)c(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14142036__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)[C@@]12CCC[C@@H]1C2 s275592__15865748__14142038__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)[C@@]12CCC[C@@H]1C2 s275592__15865748__14142038__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)[C@@]12CCC[C@@H]1C2 s275592__15865748__14142038__15857566
Cc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)n1 s275592__15865748__14142040__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1CCO[C@H]1C1CC1 s275592__15865748__14142042__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1CCO[C@H]1C1CC1 s275592__15865748__14142042__15859360
CC(C)n1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14142046__15859360
CC[C@@H]1OCC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14142052__15862300
CC[C@@H]1OCC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14142052__15859360
O=C(CC1CCC(C2CC2)O1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14142056__15859360
Cc1nc2c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccnc2[nH]1 s275592__15865748__14142060__15859360
CCc1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n(C)n1 s275592__15865748__14142062__15859360
Cc1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)c1 s275592__15865748__14142064__15862300
Cc1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)c1 s275592__15865748__14142064__15859360
Cc1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1C s275592__15865748__14142066__15862300
Cc1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1C s275592__15865748__14142066__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nccc2occc12 s275592__15865748__14142070__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC[C@H]2C[C@H]2CC1 s275592__15865748__14142074__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC[C@H]2C[C@H]2CC1 s275592__15865748__14142074__15859360
CCn1cc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__14142080__15862300
CCn1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14142080__15859360
Cn1nccc1[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14142082__15859360
CC1CC2CC2CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14142084__15862300
CC1CC2CC2CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14142084__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1OC[C@@H]2COCC[C@@H]21 s275592__15865748__14142090__15859360
Cn1ccnc1CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14142096__15862300
Cn1ccnc1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14142096__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@@H]2CCCC[C@@H]21 s275592__15865748__14142098__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@@H]2CCCC[C@@H]21 s275592__15865748__14142098__15859360
C[C@H](CC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14142102__15862300
C[C@H](CC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14142102__15859360
COC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCC1 s275592__15865748__14137504__15862300
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC1 s275592__15865748__14137504__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(Cl)nn1C s275592__15865748__14137512__15859360
C=CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCOCC1 s275592__15865748__14137514__15859360
COCCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14137522__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1C1CCC1 s275592__15865748__14137526__15859360
O=C(CC1OCc2ccccc21)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137528__15859360
Cc1nn(C)c(F)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137530__15862300
Cc1nn(C)c(F)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137530__15859360
C[C@H](CC1CCCCC1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137532__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccsc1C(F)F s275592__15865748__14137534__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1sccc1C(F)F s275592__15865748__14137536__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(C(F)F)o1 s275592__15865748__14137538__15859360
Cc1cc(C)c(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__14137544__15859360
CC(C)(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)(F)F s275592__15865748__14137546__15859360
CCc1nc[nH]c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137550__15862300
CCc1nc[nH]c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137550__15859360
CN(C)S(=O)(=O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137552__15859360
CN1C(=O)CCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137558__15862300
CN1C(=O)CCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137558__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC(C(F)F)CC1 s275592__15865748__14137564__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC(C2CC2)CC1 s275592__15865748__14137566__15859360
O=C(Cc1ccc2cn[nH]c2c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137570__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(C2CC2)cn1 s275592__15865748__14137572__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cncnc1C1CC1 s275592__15865748__14137574__15859360
Cc1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C2CC2)n1 s275592__15865748__14137576__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1Cc2ccccc2CO1 s275592__15865748__14137578__15859360
CC(=O)N1CCOC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14137580__15859360
CN1CCc2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc21 s275592__15865748__14137582__15859360
Cn1cncc1CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137586__15862300
Cn1cncc1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137586__15859360
Cc1nn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(=O)n1C s275592__15865748__14137588__15859360
CC(C)CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__14137596__15859360
Cc1n[nH]c(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137604__15862300
Cc1n[nH]c(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137604__15859360
Cc1n[nH]c(C)c1C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137606__15859360
CCCCCCN(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137608__15859360
O=C(Cn1ncc2ccccc21)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137612__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn2ccccc12 s275592__15865748__14137618__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nccn2ccnc12 s275592__15865748__14137628__15859360
CCN(CC)C(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__14137636__15859360
CCn1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc1=O s275592__15865748__14137642__15859360
Cc1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)n1 s275592__15865748__14137646__15862300
Cc1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)n1 s275592__15865748__14137646__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1F s275592__15865748__14137652__15859360
Cc1ncccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137654__15862300
Cc1ncccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137654__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2cccnc2c1 s275592__15865748__14137656__15859360
Cc1ccc(Cl)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137658__15859360
CC(C)CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137660__15862300
CC(C)CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137660__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCc2ccccc2O1 s275592__15865748__14137662__15859360
CCN(CC)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137664__15862300
CCN(CC)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137664__15859360
CCN(CC)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137664__15857566
CCC(F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14139998__15862300
CCC(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14139998__15859360
CCC(F)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14139998__15857566
O=C(CCCF)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140002__15862300
O=C(CCCF)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140002__15859360
O=C(CCCF)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140002__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(F)(F)F s275592__15865748__14140004__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)(F)F s275592__15865748__14140004__15859360
Cc1cocc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140006__15862300
Cc1cocc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140006__15859360
Cc1cocc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140006__15857566
C[C@H]1C[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140008__15862300
C[C@H]1C[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140008__15859360
C[C@H]1C[C@@H]1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140008__15857566
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C=CCC1 s275592__15865748__14140010__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C=CCC1 s275592__15865748__14140010__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C=CCC1 s275592__15865748__14140010__15857566
CN1C(=O)CC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140014__15862300
CN1C(=O)CC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140014__15859360
Cn1nnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14140016__15862300
Cn1nnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14140016__15859360
Cn1nnc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)n1 s275592__15865748__14140016__15857566
CC1(C)CCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140018__15862300
CC1(C)CCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140018__15859360
CC1CCC(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140020__15862300
CC1CCC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140020__15859360
Cc1cnn(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140024__15862300
Cc1cnn(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140024__15859360
CC(C)C(F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140026__15862300
CC(C)C(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140026__15859360
CC(C)C(F)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140026__15857566
CCCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__14140028__15862300
CCCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14140028__15859360
C=CC(C)C(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140030__15862300
C=CC(C)C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140030__15859360
C=CC(C)C(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140030__15857566
CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__14140032__15862300
CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14140032__15859360
CCC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CCC1 s275592__15865748__14140032__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC2(CCC2)C1 s275592__15865748__14140034__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2(CCC2)C1 s275592__15865748__14140034__15859360
CC#CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140036__15862300
CC#CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140036__15859360
CC#CCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140036__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1[C@H]2COC[C@H]21 s275592__15865748__14140038__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1[C@H]2COC[C@H]21 s275592__15865748__14140038__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)[C@@H]1[C@H]2COC[C@H]21 s275592__15865748__14140038__15857566
O=C(CCCC1CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140040__15862300
O=C(CCCC1CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140040__15859360
O=C(CCCC1CC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140040__15857566
CN1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1=O s275592__15865748__14140042__15862300
CN1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1=O s275592__15865748__14140042__15859360
CCCC(OCC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140044__15862300
CCCC(OCC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140044__15859360
CC1(C)CCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140046__15862300
CC1(C)CCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140046__15859360
CC1(C)CCC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140046__15857566
Cc1coc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14140048__15862300
Cc1coc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140048__15859360
Cc1coc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)c1 s275592__15865748__14140048__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1csc(=O)[nH]1 s275592__15865748__14140050__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1csc(=O)[nH]1 s275592__15865748__14140050__15859360
C=CC(CC)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140054__15862300
C=CC(CC)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140054__15859360
C=CC(CC)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140054__15857566
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__14140056__15862300
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__14140056__15859360
CC(C)(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC1 s275592__15865748__14140056__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@@H]2C[C@@H]2C1 s275592__15865748__14140058__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@@H]2C[C@@H]2C1 s275592__15865748__14140058__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)[C@@H]1C[C@@H]2C[C@@H]2C1 s275592__15865748__14140058__15857566
Cc1nc[nH]c(=O)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140068__15862300
Cc1nc[nH]c(=O)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140068__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC(=O)NC1 s275592__15865748__14140070__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC(=O)NC1 s275592__15865748__14140070__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccn1C(C)C s275592__15865748__14140074__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCc2cccnc21 s275592__15865748__14140082__15859360
CCCN1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140084__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(c2cccnc2)CC1 s275592__15865748__14140086__15859360
CCOC1CC(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140088__15862300
CCOC1CC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140088__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)s1 s275592__15865748__14140092__15862300
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)s1 s275592__15865748__14140092__15859360
O=C(Cc1cnoc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140094__15862300
O=C(Cc1cnoc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140094__15859360
O=C(Cc1cnoc1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140094__15857566
CN1C(=O)CC[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140096__15862300
CN1C(=O)CC[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140096__15859360
CC1(C)CC(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140100__15862300
CC1(C)CC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140100__15859360
CC(C)c1ccoc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140106__15862300
CC(C)c1ccoc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140106__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2n1CCCC2 s275592__15865748__14140112__15859360
CC(C)N1C(=O)CC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140116__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(C(F)F)CCC1 s275592__15865748__14140120__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C(F)F)CCC1 s275592__15865748__14140120__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C(F)F)CCCC1 s275592__15865748__14140122__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1cncnc1 s275592__15865748__14140124__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cncnc1 s275592__15865748__14140124__15859360
Cc1cc(C2(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)CC2)on1 s275592__15865748__14140134__15859360
O=C(Cc1c[nH]c2cnccc12)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140136__15859360
CC(C)N1CCOC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140138__15859360
O=C(CCc1ccc(=O)[nH]c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140140__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(F)CCOC1 s275592__15865748__14140146__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(F)CCOC1 s275592__15865748__14140146__15859360
COc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc1 s275592__15865748__14140148__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nc(Cl)cs1 s275592__15865748__14140150__15859360
O=C(CC1CCCC1(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140152__15859360
Cc1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1C s275592__15865748__14140158__15862300
Cc1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1C s275592__15865748__14140158__15859360
Cc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1Cl s275592__15865748__14137670__15859360
CC(C)(C)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137672__15862300
CC(C)(C)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137672__15859360
CC(C)(C)CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137672__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccncn1 s275592__15865748__14137674__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccncn1 s275592__15865748__14137674__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ccncn1 s275592__15865748__14137674__15857566
O=C(CC1CCc2ccccc21)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137676__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nc2ncccn2n1 s275592__15865748__14137678__15859360
CCCCCCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137680__15862300
CCCCCCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137680__15859360
O=C(CCc1ncccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137686__15862300
O=C(CCc1ncccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137686__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ccn1 s275592__15865748__14137688__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccn1 s275592__15865748__14137688__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ncccn2n1 s275592__15865748__14137692__15859360
O=C(Cc1ccco1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137696__15862300
O=C(Cc1ccco1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137696__15859360
O=C(Cc1ccco1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137696__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ncccn1 s275592__15865748__14137702__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncccn1 s275592__15865748__14137702__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1ncccn1 s275592__15865748__14137702__15857566
CCC(C)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137704__15862300
CCC(C)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137704__15859360
CCC(C)CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137704__15857566
CC(C)(C)c1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14137706__15859360
CC(C)c1nnsc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137712__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2[nH]cnc12 s275592__15865748__14137714__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccnn1 s275592__15865748__14137716__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnn1 s275592__15865748__14137716__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1cccnn1 s275592__15865748__14137716__15857566
COc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1F s275592__15865748__14137718__15859360
CCn1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1C s275592__15865748__14137724__15862300
CCn1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14137724__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)o1 s275592__15865748__14137734__15862300
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)o1 s275592__15865748__14137734__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2nccnc12 s275592__15865748__14137736__15859360
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n(C)n1 s275592__15865748__14137738__15862300
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n(C)n1 s275592__15865748__14137738__15859360
O=C(CCn1cnnn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137740__15862300
O=C(CCn1cnnn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137740__15859360
CC1CCN(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14137742__15862300
CC1CCN(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14137742__15859360
CCCn1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14137748__15859360
CCCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)n1 s275592__15865748__14137750__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ncccc1F s275592__15865748__14137754__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncccc1F s275592__15865748__14137754__15859360
O=C(Cc1coc2ccccc12)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137758__15859360
CC(C)[C@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14137760__15859360
O=C(COCc1ccncc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137766__15859360
Cn1ncc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cnc21 s275592__15865748__14137776__15859360
CC1OCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137780__15862300
CC1OCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137780__15859360
CC1OCCC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137780__15857566
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCOC1 s275592__15865748__14137782__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCOC1 s275592__15865748__14137782__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CCOC1 s275592__15865748__14137782__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn(C(F)F)c1 s275592__15865748__14137784__15859360
CC(C)Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14137786__15859360
NC(=O)c1c[nH]c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14137794__15862300
NC(=O)c1c[nH]c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14137794__15859360
CCC(CC)(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137796__15862300
CCC(CC)(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137796__15859360
CCCC1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCO1 s275592__15865748__14137800__15859360
CC1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCO1 s275592__15865748__14137802__15862300
CC1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCO1 s275592__15865748__14137802__15859360
CCCC(C)(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137804__15862300
CCCC(C)(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137804__15859360
CCC(CC)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137806__15862300
CCC(CC)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137806__15859360
CCC(CC)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137806__15857566
CCC(C)C(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137808__15862300
CCC(C)C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137808__15859360
CCC(C)C(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137808__15857566
CCCC(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137812__15862300
CCCC(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137812__15859360
CCCC(CC)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137812__15857566
Cc1nc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc2[nH]1 s275592__15865748__14137814__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(=O)NCC1CC1 s275592__15865748__14137820__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(=O)NCC1CC1 s275592__15865748__14137820__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(=O)NCC(F)(F)F s275592__15865748__14137822__15859360
O=C(CCCc1cccnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137828__15859360
CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCOCC1 s275592__15865748__14137832__15862300
CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCOCC1 s275592__15865748__14137832__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCOC1 s275592__15865748__14137834__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCOC1 s275592__15865748__14137834__15859360
CN1CCC(OCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14137836__15859360
O=C(Cc1ccc(F)cn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140168__15862300
O=C(Cc1ccc(F)cn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140168__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1Cc2ccc(F)cc21 s275592__15865748__14140172__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccoc1C1CC1 s275592__15865748__14140182__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccoc1C1CC1 s275592__15865748__14140182__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1coc(C(F)F)c1 s275592__15865748__14140184__15859360
Cn1nnc2c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccnc21 s275592__15865748__14140186__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC(F)C1 s275592__15865748__14140188__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC(F)C1 s275592__15865748__14140188__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCC(F)C1 s275592__15865748__14140188__15857566
NC(=O)Cc1occc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140190__15859360
Cn1cc(OCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__14140194__15862300
Cn1cc(OCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14140194__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(C1CCC1)C1CCC1 s275592__15865748__14140196__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc(C)n1 s275592__15865748__14140198__15859360
CN(C)CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140212__15862300
CN(C)CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140212__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCc2[nH]nnc21 s275592__15865748__14140216__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2[nH]ncc2c1 s275592__15865748__14140218__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1c[nH]c(=O)cn1 s275592__15865748__14140222__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c[nH]c(=O)cn1 s275592__15865748__14140222__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nccc2ccccc12 s275592__15865748__14140224__15859360
Cn1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc2ccccc21 s275592__15865748__14140226__15859360
CCCC(CCC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140230__15862300
CCCC(CCC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140230__15859360
CCc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140232__15862300
CCc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140232__15859360
O=C(Cc1cc(F)ccc1F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140234__15859360
O=C(Cc1ccc(F)c(F)c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140236__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc(F)c1F s275592__15865748__14140238__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(F)c1F s275592__15865748__14140238__15859360
O=C(Cc1c(F)cccc1F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140242__15859360
CC1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140246__15862300
CC1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140246__15859360
CC1CCCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140248__15862300
CC1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140248__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(F)c(F)cc1F s275592__15865748__14140250__15859360
COC1CCCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140252__15862300
COC1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140252__15859360
COC1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140254__15862300
COC1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140254__15859360
CCCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14140256__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)c(F)c1F s275592__15865748__14140258__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)c(Cl)c1 s275592__15865748__14140262__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c(F)ccc(F)c1F s275592__15865748__14140264__15859360
Cc1ncccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140266__15862300
Cc1ncccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140266__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1Cc2ccccc21 s275592__15865748__14140276__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1Cc2ccccc21 s275592__15865748__14140276__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc2[nH]ccc2c1 s275592__15865748__14140280__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2[nH]ccc2c1 s275592__15865748__14140280__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c(F)cc(F)cc1F s275592__15865748__14140284__15859360
C=CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140288__15862300
C=CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140288__15859360
C=CCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140288__15857566
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ccc1F s275592__15865748__14140290__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc1F s275592__15865748__14140290__15859360
NS(=O)(=O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140292__15859360
CCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140294__15862300
CCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140294__15859360
CCC(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140294__15857566
CCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140296__15862300
CCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140296__15859360
CCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140296__15857566
Cc1cccc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14140298__15862300
Cc1cccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140298__15859360
NC(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140300__15862300
NC(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140300__15859360
NC(=O)C1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC1 s275592__15865748__14140300__15857566
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)c1 s275592__15865748__14140302__15859360
O=C(CCCCc1ccccc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140304__15859360
NC(=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140308__15862300
NC(=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140308__15859360
NC(=O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140308__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2nonc2c1 s275592__15865748__14140310__15859360
O=C(Cc1cccc(Cl)c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140312__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(Cl)c1F s275592__15865748__14140318__15859360
O=C(CCCc1ccccc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140320__15859360
Cc1nocc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140324__15862300
Cc1nocc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140324__15859360
Cc1nocc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140324__15857566
Cc1cc(C)c(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)c1 s275592__15865748__14140326__15859360
Cc1cc(C)cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140328__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc1Cl s275592__15865748__14140334__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(Cl)no1 s275592__15865748__14135506__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(Cl)no1 s275592__15865748__14135506__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cn(CC2CC2)nn1 s275592__15865748__14137838__15859360
CCCn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__14137840__15862300
CCCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14137840__15859360
CC(C)n1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__14137842__15862300
CC(C)n1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14137842__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nnn1C(C)C s275592__15865748__14137844__15859360
CCn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__14137850__15862300
CCn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14137850__15859360
CC(Cc1cnn(C)c1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137856__15859360
O=C(CCC1CCCOC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137858__15862300
O=C(CCC1CCCOC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137858__15859360
O=C(CCn1cnccc1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137862__15859360
COCc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)co1 s275592__15865748__14137870__15862300
COCc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)co1 s275592__15865748__14137870__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1coc(CC2CC2)n1 s275592__15865748__14137872__15859360
Cc1oc(C2CC2)nc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137874__15859360
Cc1nc2ccnn2cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137876__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1C1CCCC1 s275592__15865748__14137878__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1C1CCCC1 s275592__15865748__14137878__15859360
CCC1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137886__15862300
CCC1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137886__15859360
CCC1(C(C)C)CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137888__15862300
CCC1(C(C)C)CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137888__15859360
CCC1(C)CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137890__15862300
CCC1(C)CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137890__15859360
CCC1(C)CC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137890__15857566
CC(C)C1(C)CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137894__15862300
CC(C)C1(C)CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137894__15859360
Cn1cc(C(C)(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14137898__15859360
CS(=O)(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14137900__15859360
COCC(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137904__15862300
COCC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137904__15859360
COCC(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137904__15857566
CCc1c[nH]c(=O)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14137908__15859360
COCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137918__15862300
COCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137918__15859360
CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCC1 s275592__15865748__14137922__15862300
CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__14137922__15859360
Cc1nonc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137926__15862300
Cc1nonc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137926__15859360
CCCc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)no1 s275592__15865748__14137934__15862300
CCCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__14137934__15859360
Cc1ncsc1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137936__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2sccc2c1 s275592__15865748__14137942__15859360
Cc1oc(C(C)C)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137950__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2ccncc12 s275592__15865748__14137952__15859360
CC(C)N1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14137956__15859360
COc1cccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14137958__15862300
COc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14137958__15859360
CC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n(C)n1 s275592__15865748__14137964__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnoc1C1CC1 s275592__15865748__14137968__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnoc1C1CC1 s275592__15865748__14137968__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1c[nH]nc1C1CC1 s275592__15865748__14137970__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c[nH]nc1C1CC1 s275592__15865748__14137970__15859360
CC(C)c1oncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137972__15862300
CC(C)c1oncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137972__15859360
Cn1cnc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc21 s275592__15865748__14137974__15859360
CC1(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14137980__15862300
CC1(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14137980__15859360
CC1(CCC(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC1 s275592__15865748__14137980__15857566
Cc1cnoc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14137982__15862300
Cc1cnoc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14137982__15859360
Cc1cnoc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14137982__15857566
COc1ncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__14137992__15862300
COc1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14137992__15859360
Cc1cc(=O)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c[nH]1 s275592__15865748__14137994__15862300
Cc1cc(=O)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c[nH]1 s275592__15865748__14137994__15859360
Cc1cc(Cl)ccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140336__15859360
Cc1ccc(CCCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14140340__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2ncccc2c1 s275592__15865748__14140342__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1Cl s275592__15865748__14140344__15859360
CC(CC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140346__15862300
CC(CC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140346__15859360
COc1ncccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140348__15862300
COc1ncccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140348__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCCC1 s275592__15865748__14140350__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCCC1 s275592__15865748__14140350__15859360
CN1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140354__15862300
CN1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140354__15859360
Cc1ccc(C)c(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140360__15859360
Cc1ccc(F)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1F s275592__15865748__14140368__15859360
Cc1cccc(Cl)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140370__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC=CC1 s275592__15865748__14140376__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC=CC1 s275592__15865748__14140376__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC=CC1 s275592__15865748__14140376__15857566
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)[nH]c1=O s275592__15865748__14140378__15862300
Cn1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)[nH]c1=O s275592__15865748__14140378__15859360
COC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)C s275592__15865748__14140380__15862300
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__14140380__15859360
COC(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C(C)C s275592__15865748__14140380__15857566
CC1CC1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140382__15862300
CC1CC1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140382__15859360
CC1CC1CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140382__15857566
CCCCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140384__15862300
CCCCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140384__15859360
C=C1CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140386__15862300
C=C1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140386__15859360
C=CCCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140388__15862300
C=CCCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140388__15859360
C=CC(C)(CC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140390__15862300
C=CC(C)(CC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140390__15859360
C=CC(C)(CC)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140390__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC(F)CC1 s275592__15865748__14140392__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC(F)CC1 s275592__15865748__14140392__15859360
O=C(C[C@H]1CCOC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140394__15862300
O=C(C[C@H]1CCOC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140394__15859360
O=C(C[C@H]1CCOC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140394__15857566
C=CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__14140396__15862300
C=CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__14140396__15859360
O=C(CC1=CCOCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140398__15862300
O=C(CC1=CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140398__15859360
CCc1ccoc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140400__15862300
CCc1ccoc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140400__15859360
CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140402__15862300
CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140402__15859360
CCC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC1 s275592__15865748__14140402__15857566
CC(C)[C@H](C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N(C)C s275592__15865748__14140404__15862300
CC(C)[C@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N(C)C s275592__15865748__14140404__15859360
CCC1CCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140408__15862300
CCC1CCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140408__15859360
CC1CCCC1(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140410__15862300
CC1CCCC1(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140410__15859360
CC(F)(F)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140412__15862300
CC(F)(F)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140412__15859360
CC(F)(F)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140412__15857566
COC(CC(C)C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140414__15862300
COC(CC(C)C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140414__15859360
CCCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140416__15862300
CCCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140416__15859360
CCCC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC1 s275592__15865748__14140416__15857566
C[C@@]1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC(=O)N1 s275592__15865748__14140418__15862300
C[C@@]1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC(=O)N1 s275592__15865748__14140418__15859360
CCc1nocc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140422__15862300
CCc1nocc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140422__15859360
CC1COCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140424__15862300
CC1COCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140424__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(Cl)[nH]1 s275592__15865748__14140428__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(Cl)[nH]1 s275592__15865748__14140428__15859360
COCC(OC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140430__15862300
COCC(OC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140430__15859360
CC1(C)CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140432__15862300
CC1(C)CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140432__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCO1 s275592__15865748__14140434__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCO1 s275592__15865748__14140434__15859360
CCC[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140436__15862300
CCC[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140436__15859360
CCC[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140436__15857566
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C12CCCCC1C2 s275592__15865748__14140438__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C12CCCCC1C2 s275592__15865748__14140438__15859360
CC(C)C1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140440__15862300
CC(C)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140440__15859360
CC(C)C1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC1 s275592__15865748__14140440__15857566
C=C1CC(C)(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140442__15862300
C=C1CC(C)(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140442__15859360
C=C1CC(C)(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865748__14140442__15857566
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(F)F s275592__15865748__14140444__15862300
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)F s275592__15865748__14140444__15859360
Cc1ccoc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140446__15862300
Cc1ccoc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140446__15859360
CCc1ncoc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140448__15862300
CCc1ncoc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140448__15859360
C#Cc1cncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14140450__15862300
C#Cc1cncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140450__15859360
CCOc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccn1 s275592__15865748__14140456__15859360
CC(Oc1cccnc1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140468__15859360
Cn1c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cccc1=O s275592__15865748__14140474__15862300
Cn1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cccc1=O s275592__15865748__14140474__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(CF)CC1 s275592__15865748__14140476__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(CF)CC1 s275592__15865748__14140476__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(CF)CC1 s275592__15865748__14140476__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC2(CC2)C1 s275592__15865748__14140478__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2(CC2)C1 s275592__15865748__14140478__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC2(CC2)C1 s275592__15865748__14140478__15857566
Cc1cc(=O)[nH]cc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140480__15862300
Cc1cc(=O)[nH]cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140480__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(C(F)F)[nH]n1 s275592__15865748__14140484__15859360
Cc1cc(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)no1 s275592__15865748__14140486__15862300
Cc1cc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__14140486__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1conc1C1CC1 s275592__15865748__14140488__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1conc1C1CC1 s275592__15865748__14140488__15859360
Cn1cnc2c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccnc21 s275592__15865748__14140490__15859360
CCC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N(CC)CC s275592__15865748__14140492__15862300
CCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N(CC)CC s275592__15865748__14140492__15859360
CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135512__15862300
CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135512__15859360
CC(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14135512__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccc1Cl s275592__15865748__14135514__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1Cl s275592__15865748__14135514__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(Cl)cc1 s275592__15865748__14135520__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(Cl)cc1 s275592__15865748__14135520__15859360
CCCCCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135522__15862300
CCCCCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135522__15859360
COc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135524__15862300
COc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135524__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2ccccc2n1 s275592__15865748__14135526__15859360
CC(C)(C)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135528__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c(F)cccc1Cl s275592__15865748__14135530__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc(Cl)c1 s275592__15865748__14135538__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(Cl)c1 s275592__15865748__14135538__15859360
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1 s275592__15865748__14135542__15862300
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135542__15859360
CCCCCCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135552__15859360
O=C(CCc1ccccc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135554__15862300
O=C(CCc1ccccc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135554__15859360
O=C(Cc1c[nH]c2ccccc12)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135556__15859360
CC(C)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135558__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1 s275592__15865748__14135562__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135562__15859360
O=C(COc1ccccc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135564__15862300
O=C(COc1ccccc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135564__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2ccccc2c1 s275592__15865748__14135566__15859360
COc1cccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14135568__15862300
COc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14135568__15859360
COc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135570__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1c(F)cccc1F s275592__15865748__14135586__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c(F)cccc1F s275592__15865748__14135586__15859360
CN(C)c1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14135596__15859360
CN(C)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135598__15859360
Cc1ccc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14135600__15862300
Cc1ccc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14135600__15859360
Cc1cc(C)cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14135602__15862300
Cc1cc(C)cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14135602__15859360
O=C(Cc1ccc(Cl)cc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135606__15859360
CCOc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135610__15859360
CCOc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135612__15859360
O=C(Cc1ccc(F)cc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135614__15862300
O=C(Cc1ccc(F)cc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135614__15859360
CCOc1ncccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135616__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(F)cc1F s275592__15865748__14135618__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)cc1F s275592__15865748__14135618__15859360
Cc1cccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1C s275592__15865748__14135620__15862300
Cc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14135620__15859360
CCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1 s275592__15865748__14135628__15862300
CCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135628__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1n[nH]c2ccccc12 s275592__15865748__14135630__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)c1 s275592__15865748__14135632__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)c1 s275592__15865748__14135632__15859360
O=C(Cc1ccccc1F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135634__15862300
O=C(Cc1ccccc1F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135634__15859360
Cc1ccccc1OCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135636__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2ccccc12 s275592__15865748__14135638__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1C s275592__15865748__14135642__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1C s275592__15865748__14135642__15859360
O=C(CC1CC2CCC1C2)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135648__15862300
O=C(CC1CC2CCC1C2)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135648__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)cc1Cl s275592__15865748__14135650__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(=O)[nH]c1 s275592__15865748__14135652__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(=O)[nH]c1 s275592__15865748__14135652__15859360
CC(Oc1ccccc1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135654__15859360
COc1cccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14135656__15859360
O=C(CCC1CCCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135658__15862300
O=C(CCC1CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135658__15859360
CCCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135662__15862300
CCCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135662__15859360
CCCCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14135662__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2sccc2[nH]1 s275592__15865748__14138010__15859360
Cn1nc2ccccc2c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138014__15859360
CC(C)c1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14138016__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(F)CCCCC1 s275592__15865748__14138020__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(F)CCCCC1 s275592__15865748__14138020__15859360
Cn1ccc2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc21 s275592__15865748__14138022__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2ccsc12 s275592__15865748__14138024__15859360
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1 s275592__15865748__14138030__15862300
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__14138030__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ncoc1C1CC1 s275592__15865748__14138032__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncoc1C1CC1 s275592__15865748__14138032__15859360
CCc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__14138034__15862300
CCc1nc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__14138034__15859360
Cc1nc2c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cccc2[nH]1 s275592__15865748__14138036__15859360
CCN(C)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138038__15862300
CCN(C)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138038__15859360
CCN(C)CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138038__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC12CCCC2 s275592__15865748__14138040__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC12CCCC2 s275592__15865748__14138040__15859360
O=C(CCc1cnccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138044__15862300
O=C(CCc1cnccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138044__15859360
Cc1cc(C)cc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14138048__15859360
CC(C)C1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCO1 s275592__15865748__14138050__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn2c1CCCC2 s275592__15865748__14138052__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2ccncc2c1 s275592__15865748__14138056__15859360
O=C(CCCn1cncn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138058__15862300
O=C(CCCn1cncn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138058__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2cnccc2c1 s275592__15865748__14138060__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1csc(Cl)n1 s275592__15865748__14138062__15859360
CC(C)(CC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138064__15859360
CN1CCc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc21 s275592__15865748__14138066__15859360
Cc1conc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138072__15862300
Cc1conc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138072__15859360
Cc1conc1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138072__15857566
CC(C)c1ocnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138074__15862300
CC(C)c1ocnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138074__15859360
CC(C)(Cc1ccccc1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138076__15859360
O=C(CN1CCC(=O)NC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138078__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2c([nH]1)CCCC2 s275592__15865748__14138082__15859360
CCC(=O)N1CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14138088__15859360
COC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)(F)F s275592__15865748__14138094__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn(CC2CC2)c1 s275592__15865748__14138100__15859360
CCC1CC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCO1 s275592__15865748__14138108__15859360
CCC1CC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCO1 s275592__15865748__14138110__15862300
CCC1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCO1 s275592__15865748__14138110__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCc2[nH]cnc2C1 s275592__15865748__14138112__15859360
CC(=O)N1CCC(C)(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14138114__15859360
Cc1cn2ccnc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c2n1 s275592__15865748__14138116__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC12CCOC2 s275592__15865748__14138122__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC12CCOC2 s275592__15865748__14138122__15859360
CCC1CCCN1C(=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138128__15859360
COCCCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138130__15862300
COCCCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138130__15859360
CCC(CC(C)C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138132__15862300
CCC(CC(C)C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138132__15859360
CCCCCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__14138134__15859360
COCCCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138140__15862300
COCCCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138140__15859360
COCCCOCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138142__15859360
CC(C)CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138144__15862300
CC(C)CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138144__15859360
O=C(CC(=O)NCC1CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138146__15862300
O=C(CC(=O)NCC1CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138146__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)n1cccn1 s275592__15865748__14138150__15862300
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)n1cccn1 s275592__15865748__14138150__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1coc(C2CCC2)n1 s275592__15865748__14138152__15859360
Cc1n[nH]c(C(C)C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138160__15859360
NC(=O)CCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138164__15862300
NC(=O)CCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138164__15859360
NC(=O)c1coc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14140506__15862300
NC(=O)c1coc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140506__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC(F)(F)C1 s275592__15865748__14140508__15859360
CC1(c2ccccc2C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140510__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccsc1 s275592__15865748__14140516__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccsc1 s275592__15865748__14140516__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1cccs1 s275592__15865748__14140518__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccs1 s275592__15865748__14140518__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccco1 s275592__15865748__14140520__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccco1 s275592__15865748__14140520__15859360
CCc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nnn1CC s275592__15865748__14140526__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2occc2s1 s275592__15865748__14140536__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCNC1=O s275592__15865748__14140538__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCNC1=O s275592__15865748__14140538__15859360
NC(=O)[C@@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)O1 s275592__15865748__14140546__15862300
NC(=O)[C@@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)O1 s275592__15865748__14140546__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncsc1C1CC1 s275592__15865748__14140548__15859360
CCOC1CC2(C1)CC2C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140550__15859360
Cn1cnc2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)nc21 s275592__15865748__14140552__15859360
Cc1ncccc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140554__15862300
Cc1ncccc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140554__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ocnc1C1CC1 s275592__15865748__14140556__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ocnc1C1CC1 s275592__15865748__14140556__15859360
Cn1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(Cl)n1 s275592__15865748__14140558__15859360
CC(C)(C)n1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14140562__15859360
Cc1cn2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc2n1 s275592__15865748__14140564__15859360
CC1CCCN1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140568__15862300
CC1CCCN1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140568__15859360
CC(C)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc1 s275592__15865748__14140570__15859360
CC1CCN(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140576__15862300
CC1CCN(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140576__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(CF)CCOCC1 s275592__15865748__14140580__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1Cc2ccncc2C1 s275592__15865748__14140590__15859360
O=C(CC(F)(F)C(F)F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140598__15862300
O=C(CC(F)(F)C(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140598__15859360
CC1(C)CCN(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140600__15862300
CC1(C)CCN(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140600__15859360
CN(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)CC(C)(C)C s275592__15865748__14140602__15862300
CN(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC(C)(C)C s275592__15865748__14140602__15859360
O=C(CCc1cncs1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140606__15862300
O=C(CCc1cncs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140606__15859360
NC(=O)[C@@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14140610__15862300
NC(=O)[C@@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14140610__15859360
NC(=O)[C@@H]1C[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140612__15862300
NC(=O)[C@@H]1C[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140612__15859360
NC(=O)[C@@H]1C[C@@H]1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140612__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ocnc1C(F)F s275592__15865748__14140616__15859360
Cn1ncc(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14140618__15862300
Cn1ncc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14140618__15859360
NC(=O)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)[nH]1 s275592__15865748__14140620__15862300
NC(=O)c1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)[nH]1 s275592__15865748__14140620__15859360
CC(F)(F)C1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14140622__15862300
CC(F)(F)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14140622__15859360
CC[C@@H](C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N(C)C s275592__15865748__14140630__15862300
CC[C@@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N(C)C s275592__15865748__14140630__15859360
CC[C@@H](C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)N(C)C s275592__15865748__14140630__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)(F)F s275592__15865748__14140632__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)(F)F s275592__15865748__14140632__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(C)[nH]1 s275592__15865748__14140638__15862300
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)[nH]1 s275592__15865748__14140638__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nccn2ccnc12 s275592__15865748__14140640__15859360
Cc1nc(C2CC2)ccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140642__15859360
Cc1ccn(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14140644__15862300
Cc1ccn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14140644__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nccc2[nH]ccc12 s275592__15865748__14140646__15859360
COc1cc(=O)[nH]cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140650__15859360
Cn1cncc1[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140656__15859360
O=C(CCc1c[nH]nn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140658__15862300
O=C(CCc1c[nH]nn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140658__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(CF)CCC1 s275592__15865748__14140660__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(CF)CCC1 s275592__15865748__14140660__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(CF)CCC1 s275592__15865748__14140660__15857566
C=C[C@@H]1OCC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140662__15862300
C=C[C@@H]1OCC[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140662__15859360
CC(C)C[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140666__15862300
CC(C)C[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140666__15859360
Cc1ccnc2nc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)nn12 s275592__15865748__14135682__15859360
O=C(CNC(=O)c1ccco1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135692__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cn2ccccc2n1 s275592__15865748__14135694__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(Cl)s1 s275592__15865748__14135710__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ccccc2o1 s275592__15865748__14135718__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(c1)CCCC2 s275592__15865748__14135722__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14135724__15859360
O=C(CCCC1CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135728__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2c(s1)CCC2 s275592__15865748__14135736__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)oc2ccccc12 s275592__15865748__14135738__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1sccc1C1CC1 s275592__15865748__14135744__15859360
CCCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__14135748__15859360
CC(=O)NCCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135758__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(c2ccccc2)CC1 s275592__15865748__14135760__15859360
O=C(Cc1cccc(F)c1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135764__15862300
O=C(Cc1cccc(F)c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135764__15859360
O=C(Cc1ccccc1Cl)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135768__15859360
Cc1ccc(OCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14135776__15859360
Cn1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)ccc1=O s275592__15865748__14135778__15862300
Cn1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc1=O s275592__15865748__14135778__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(F)cc(F)c1 s275592__15865748__14135782__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(F)cc(F)c1 s275592__15865748__14135782__15859360
Cc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)c1 s275592__15865748__14135784__15859360
COc1ccccc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135786__15859360
Cc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1C s275592__15865748__14135806__15859360
O=C(Cn1cncn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135814__15862300
O=C(Cn1cncn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135814__15859360
O=C(Cn1cncn1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14135814__15857566
Cc1nc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cs1 s275592__15865748__14135818__15862300
Cc1nc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cs1 s275592__15865748__14135818__15859360
O=C(CCCc1cccs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135822__15859360
CCc1sc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1C s275592__15865748__14135826__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2nccnc2c1 s275592__15865748__14135828__15859360
O=C(CN1C(=O)CNC1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14135832__15862300
O=C(CN1C(=O)CNC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135832__15859360
CN1CC(=O)N(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1=O s275592__15865748__14135834__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc2ccccc2[nH]1 s275592__15865748__14135836__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ccccc2[nH]1 s275592__15865748__14135836__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)sc1C s275592__15865748__14135838__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)sc1C s275592__15865748__14135838__15859360
O=C(CN1CCCCCC1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14135842__15859360
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)sc1C s275592__15865748__14135844__15859360
CC1CCN(C(=O)C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__14138174__15862300
CC1CCN(C(=O)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14138174__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(C1CC1)C1CC1 s275592__15865748__14138178__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(C1CC1)C1CC1 s275592__15865748__14138178__15859360
O=C(CCOC1CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138196__15859360
O=C(Cc1nc[nH]n1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138206__15862300
O=C(Cc1nc[nH]n1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138206__15859360
O=C(Cc1nc[nH]n1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138206__15857566
CN(C)C(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__14138214__15862300
CN(C)C(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__14138214__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1C(C)C s275592__15865748__14138218__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCC1 s275592__15865748__14138222__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC1 s275592__15865748__14138222__15859360
NC(=O)N1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138226__15859360
CC(C)(C)c1n[nH]cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138228__15859360
CCn1cc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__14138242__15862300
CCn1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14138242__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1cnn(C)c1 s275592__15865748__14138244__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn(C)c1 s275592__15865748__14138244__15859360
CCCC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)C s275592__15865748__14138246__15862300
CCCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__14138246__15859360
O=C(CCC1CCCCO1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138248__15862300
O=C(CCC1CCCCO1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138248__15859360
CCC(Cc1ccccc1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138254__15859360
CCC(OC1CCCC1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138256__15859360
COc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(C)nn1C s275592__15865748__14138260__15859360
CC(C)n1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__14138262__15862300
CC(C)n1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__14138262__15859360
CN(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccn1 s275592__15865748__14138264__15859360
NC(=O)C1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14138270__15859360
CC1CCCC(OCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__14138276__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc(C2CC2)n1 s275592__15865748__14138278__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1csc2cncn12 s275592__15865748__14138282__15859360
CC1CCCCC1OCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138284__15859360
O=C(COC1CCOCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138286__15862300
O=C(COC1CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138286__15859360
O=C(COCC1CCOC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138288__15862300
O=C(COCC1CCOC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138288__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCS(=O)(=O)C1 s275592__15865748__14138290__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCS(=O)(=O)CC1 s275592__15865748__14138292__15859360
CC(C)C(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138294__15862300
CC(C)C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138294__15859360
CC(C)C(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14138294__15857566
CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)S(C)(=O)=O s275592__15865748__14138300__15859360
CC(CC1CCCCC1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138304__15859360
CC(CC1CCCC1)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14138312__15862300
CC(CC1CCCC1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138312__15859360
CCC(CC1CCCC1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138314__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc2ccccn2c1 s275592__15865748__14138322__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ccccn2c1 s275592__15865748__14138322__15859360
CCNC(=O)NC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138326__15859360
Cc1nc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cs1 s275592__15865748__14138330__15859360
Cc1nn(C)cc1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14138332__15859360
CC[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140668__15862300
CC[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140668__15859360
CC[C@@H]1C[C@H]1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140668__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@H]2CC[C@@H]1O2 s275592__15865748__14140680__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]2CC[C@@H]1O2 s275592__15865748__14140680__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC(=O)N1 s275592__15865748__14140686__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC(=O)N1 s275592__15865748__14140686__15859360
Cn1cc([C@@H]2C[C@H]2C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__14140690__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@H]1c1ccco1 s275592__15865748__14140692__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]1c1ccco1 s275592__15865748__14140692__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@H]1c1cccnc1 s275592__15865748__14140694__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc2cc[nH]c12 s275592__15865748__14140700__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2cc[nH]c12 s275592__15865748__14140700__15859360
CC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n[nH]1 s275592__15865748__14140704__15862300
CC(C)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n[nH]1 s275592__15865748__14140704__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(Cl)c1 s275592__15865748__14140708__15859360
CCC(NC(C)=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140712__15862300
CCC(NC(C)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140712__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc1F s275592__15865748__14140716__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc2[nH]ccc12 s275592__15865748__14140718__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2[nH]ccc12 s275592__15865748__14140718__15859360
CC(C)=CCCC(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140720__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(F)c1F s275592__15865748__14140722__15859360
C=Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1 s275592__15865748__14140724__15862300
C=Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__14140724__15859360
CC(C)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140726__15862300
CC(C)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140726__15859360
CC(C)CCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140726__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2c1OCC2 s275592__15865748__14140728__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(c1)CCO2 s275592__15865748__14140730__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(-c2ccco2)[nH]n1 s275592__15865748__14140732__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(C(F)(F)F)CC1 s275592__15865748__14140734__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C(F)(F)F)CC1 s275592__15865748__14140734__15859360
Cc1cccc(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140736__15862300
Cc1cccc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140736__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(C2CC2)[nH]n1 s275592__15865748__14140738__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(C2CC2)[nH]n1 s275592__15865748__14140738__15859360
O=C(CCCC(F)(F)F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140740__15862300
O=C(CCCC(F)(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140740__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(F)c(F)c(F)c1 s275592__15865748__14140742__15859360
Cc1cc(F)cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14140746__15862300
Cc1cc(F)cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140746__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)CC(C)(C)C s275592__15865748__14140750__15862300
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC(C)(C)C s275592__15865748__14140750__15859360
CCn1nc(C)cc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140752__15862300
CCn1nc(C)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140752__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1Cc2ccccc2C1 s275592__15865748__14140754__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(Cl)c(F)c1 s275592__15865748__14140756__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1noc2c1CCCC2 s275592__15865748__14140758__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(F)cc(Cl)c1 s275592__15865748__14140760__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(F)ccc1Cl s275592__15865748__14140762__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccncc1Cl s275592__15865748__14140764__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccncc1Cl s275592__15865748__14140764__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(F)c1 s275592__15865748__14140770__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(F)c1 s275592__15865748__14140770__15859360
Cc1ccccc1CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140772__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1C2CCCCCCC21 s275592__15865748__14140776__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC12CC2 s275592__15865748__14140778__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC12CC2 s275592__15865748__14140778__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC12CC2 s275592__15865748__14140778__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2cnccc2n1 s275592__15865748__14140780__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(F)c1Cl s275592__15865748__14140782__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC(F)(F)CC1 s275592__15865748__14140788__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnnc2ccccc12 s275592__15865748__14140798__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCc2ccccc2C1 s275592__15865748__14140800__15859360
Cc1ccc(F)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__14140802__15862300
Cc1ccc(F)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140802__15859360
CC(NS(C)(=O)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140804__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c(=O)[nH]1 s275592__15865748__14140810__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(=O)[nH]1 s275592__15865748__14140810__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2ccccc2c1 s275592__15865748__14140812__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc2cc[nH]c2c1 s275592__15865748__14140816__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2cc[nH]c2c1 s275592__15865748__14140816__15859360
CCOc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__14140818__15859360
COc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1C s275592__15865748__14140820__15859360
O=C(Cc1cnc[nH]1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140826__15862300
O=C(Cc1cnc[nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140826__15859360
O=C(Cc1cnc[nH]1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__14140826__15857566
O=C(Cc1cccc(F)c1F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140828__15859360
O=C(CC1CCCCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__14140832__15862300
O=C(CC1CCCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__14140832__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nn1C s275592__15865748__15278134__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1C s275592__15865748__15278134__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cnn1 s275592__15865748__15571390__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1 s275592__15865748__15571390__15859360
CC1CC(=O)NCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841194__15862300
CC1CC(=O)NCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841194__15859360
CSCCC(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841196__15862300
CSCCC(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841196__15859360
O=C1C[C@@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)N1 s275592__15865748__15841198__15862300
O=C1C[C@@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)N1 s275592__15865748__15841198__15859360
O=C1C[C@@H](C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)N1 s275592__15865748__15841198__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1n[nH]c2c1COCC2 s275592__15865748__15841202__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2[nH]ncc2n1 s275592__15865748__15841206__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCS1 s275592__15865748__15841212__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCS1 s275592__15865748__15841212__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=CCCCC1 s275592__15865748__15841216__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CCCCC1 s275592__15865748__15841216__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1=CCCCC1 s275592__15865748__15841216__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cncc(F)c1Cl s275592__15865748__15841224__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2occc12 s275592__15865748__15841226__15859360
CC(=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(C)C s275592__15865748__15841228__15862300
CC(=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__15841228__15859360
CC(=CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C(C)C s275592__15865748__15841228__15857566
CC(C)(C)SCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841230__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(O)CCSCC1 s275592__15865748__15841234__15859360
O=C(Cn1cnc2ccccc21)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841242__15859360
CC(C)OC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841244__15862300
CC(C)OC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841244__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCCO1 s275592__15865748__15841246__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCCO1 s275592__15865748__15841246__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(N2CCC2)nc1 s275592__15865748__15841250__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2n(n1)CCOC2 s275592__15865748__15841252__15859360
CCC(CC)(CO)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841254__15862300
CCC(CC)(CO)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841254__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(CO)cc1 s275592__15865748__15841256__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(CO)cc1 s275592__15865748__15841256__15859360
CSc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841258__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1[N+](=O)[O-] s275592__15865748__15841262__15859360
CN1CCC(O)(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__15841270__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCSC1 s275592__15865748__15841272__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCSC1 s275592__15865748__15841272__15859360
O=C1C[C@H](C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)N1 s275592__15865748__15841274__15862300
O=C1C[C@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)N1 s275592__15865748__15841274__15859360
O=C1C[C@H](C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)N1 s275592__15865748__15841274__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(=O)n(O)c1 s275592__15865748__15841276__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(=O)n(O)c1 s275592__15865748__15841276__15859360
O=C(Cn1cncn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841284__15862300
O=C(Cn1cncn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841284__15859360
O=C(Cn1cncn1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841284__15857566
COC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__15841286__15862300
COC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__15841286__15859360
COC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CC1 s275592__15865748__15841286__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CSC1 s275592__15865748__15841288__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CSC1 s275592__15865748__15841288__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CSC1 s275592__15865748__15841288__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2sccn12 s275592__15865748__15841292__15859360
Cc1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnc2nncn12 s275592__15865748__15841296__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(O)CCCC1 s275592__15865748__15841300__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(O)CCCC1 s275592__15865748__15841300__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(O)CCCC1 s275592__15865748__15841300__15857566
C=CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841304__15862300
C=CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841304__15859360
C=CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841304__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(=O)[nH]c(=O)[nH]1 s275592__15865748__15841306__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(=O)[nH]c(=O)[nH]1 s275592__15865748__15841306__15859360
CN(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841308__15862300
CN(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841308__15859360
CN(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841308__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(Cl)nc1 s275592__15865748__15841310__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(Cl)nc1 s275592__15865748__15841310__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1c[nH]c(=O)[nH]c1=O s275592__15865748__15841316__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c[nH]c(=O)[nH]c1=O s275592__15865748__15841316__15859360
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__15841318__15859360
O=C(CN1CCC(CO)CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843066__15859360
O=C(CN1CCCCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843074__15862300
O=C(CN1CCCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843074__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N1CCOCC1 s275592__15865748__15843078__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCOCC1 s275592__15865748__15843078__15859360
Cc1cnc(F)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__15843080__15862300
Cc1cnc(F)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15843080__15859360
CCCc1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__15843082__15859360
Cn1cc[n+](CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__15843086__15862300
Cn1cc[n+](CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15843086__15859360
Cc1nccnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843092__15862300
Cc1nccnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843092__15859360
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CCOC1C(C)C1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843098__15862300
CCOC1C(C)C1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843098__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCn2ccnc21 s275592__15865748__15843100__15859360
CC(C)[C@H](NC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843106__15862300
CC(C)[C@H](NC(N)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843106__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1C1CCCCC1 s275592__15865748__15843112__15859360
CN1CCCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__15843114__15862300
CN1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15843114__15859360
C=CC(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843118__15862300
C=CC(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843118__15859360
C=CC(O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843118__15857566
[N-]=[N+]=NCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843120__15862300
[N-]=[N+]=NCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843120__15859360
[N-]=[N+]=NCCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843120__15857566
Cc1cccnc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843122__15862300
Cc1cccnc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843122__15859360
CC(O)C(F)(F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843124__15862300
CC(O)C(F)(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843124__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCCN1C1CC1 s275592__15865748__15843126__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCN1C1CC1 s275592__15865748__15843126__15859360
CC1(C)COC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843128__15862300
CC1(C)COC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843128__15859360
CC1(C)COC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843128__15857566
CSCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843130__15862300
CSCC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843130__15859360
O=C(Cc1ccc(Cl)cn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843132__15859360
COC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCOCC1 s275592__15865748__15843134__15862300
COC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCOCC1 s275592__15865748__15843134__15859360
Cn1nncc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843138__15862300
Cn1nncc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843138__15859360
O=C(Cc1cnccc1O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843142__15862300
O=C(Cc1cnccc1O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843142__15859360
O=C(CCCc1cncs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843144__15859360
[N-]=[N+]=Nc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15843146__15859360
[N-]=[N+]=Nc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__15843148__15859360
[N-]=[N+]=Nc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843150__15859360
O=C(CC1CCCCC1F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843156__15862300
O=C(CC1CCCCC1F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843156__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(c1)COB2O s275592__15865748__15843158__15859360
CCCCCC(=O)NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843162__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c(F)cc(F)nc1F s275592__15865748__15843168__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncccc1F s275592__15865748__15843170__15859360
CCc1sccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843172__15862300
CCc1sccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843172__15859360
CC(C)(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C(F)F s275592__15865748__15843176__15862300
CC(C)(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)F s275592__15865748__15843176__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)=CC1CCCCC1 s275592__15865748__15843178__15859360
Cc1cccnc1C(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843180__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnn1CC1CC1 s275592__15865748__15843186__15859360
CCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(F)c1 s275592__15865748__15844918__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2c(n1)CCCC2 s275592__15865748__15844920__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n(C)n1 s275592__15865748__15844924__15862300
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n(C)n1 s275592__15865748__15844924__15859360
COc1ccnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1F s275592__15865748__15844926__15859360
CC1(C)[C@H]2C[C@H](C(=O)NCCC3CCCCN3C(=O)c3nsnc3O)C[C@H]21 s275592__15865748__15844930__15862300
CC1(C)[C@H]2C[C@H](C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)C[C@H]21 s275592__15865748__15844930__15859360
NC(=O)c1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n[nH]1 s275592__15865748__15844934__15862300
NC(=O)c1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n[nH]1 s275592__15865748__15844934__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N1CCC1 s275592__15865748__15844938__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCC1 s275592__15865748__15844938__15859360
CC(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)N1CCC1 s275592__15865748__15844938__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@H](O)Cc1c[nH]cn1 s275592__15865748__15844944__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@H](O)Cc1c[nH]cn1 s275592__15865748__15844944__15859360
O=C(C#CC1CCCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15844946__15862300
O=C(C#CC1CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15844946__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2c1CNC2=O s275592__15865748__15844950__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC2(CCOC2)C1 s275592__15865748__15844960__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2(CCOC2)C1 s275592__15865748__15844960__15859360
CCC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)CN(C)C s275592__15865748__15844962__15862300
CCC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CN(C)C s275592__15865748__15844962__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n[nH]c1=O s275592__15865748__15844964__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n[nH]c1=O s275592__15865748__15844964__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@H]1CC1(F)F s275592__15865748__15844966__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@H]1CC1(F)F s275592__15865748__15844966__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)[C@H]1CC1(F)F s275592__15865748__15844966__15857566
CC(C)c1cnn(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15844970__15859360
COCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C=CCC1 s275592__15865748__15844974__15862300
COCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C=CCC1 s275592__15865748__15844974__15859360
O=C(Cc1cn[nH]c1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15844976__15862300
O=C(Cc1cn[nH]c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15844976__15859360
O=C(Cc1cn[nH]c1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15844976__15857566
COCC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__15844978__15859360
CN(C)CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15844980__15862300
CN(C)CC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15844980__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)c1ccc(F)cc1 s275592__15865748__15844988__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CS(=O)(=O)C1 s275592__15865748__15844990__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cn(CCCF)nn1 s275592__15865748__15844992__15859360
CC(C)(Cc1cnn[nH]1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15844994__15859360
Cc1ccc2occ(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c2c1 s275592__15865748__15844998__15859360
CC12CC(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)(C1)C(C)(C)O2 s275592__15865748__15845000__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1coc(C(F)F)n1 s275592__15865748__15845002__15859360
O=C(C=CC(=O)NC1CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845004__15862300
O=C(C=CC(=O)NC1CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845004__15859360
CN1Cc2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc2C1 s275592__15865748__15845008__15859360
CC(C)NC(=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845010__15862300
CC(C)NC(=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845010__15859360
CC(C)NC(=O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15845010__15857566
C=C(Cl)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845014__15862300
C=C(Cl)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845014__15859360
CC(C)(C)c1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c[nH]1 s275592__15865748__15845018__15859360
CCC(CCOC)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845020__15862300
CCC(CCOC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845020__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC2C=CCC(C2)C1 s275592__15865748__15845022__15859360
Cc1nc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)oc1C s275592__15865748__15845024__15859360
Cc1coc(C)c1C=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845026__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C12CC(CN1C1CC1)C2 s275592__15865748__15845028__15859360
CC1=C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCO1 s275592__15865748__15845032__15862300
CC1=C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCO1 s275592__15865748__15845032__15859360
CC1=C(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CCO1 s275592__15865748__15845032__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(=O)oc1 s275592__15865748__15841320__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(=O)oc1 s275592__15865748__15841320__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc([N+](=O)[O-])o1 s275592__15865748__15841322__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc([N+](=O)[O-])o1 s275592__15865748__15841322__15859360
O=C(Cc1cc(=O)[nH]c(=O)[nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841338__15859360
CSc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__15841358__15862300
CSc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__15841358__15859360
O=C(C=C1CCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841364__15862300
O=C(C=C1CCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841364__15859360
O=C(C=C1CCCC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841364__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(Cl)nn1 s275592__15865748__15841370__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(Cl)nn1 s275592__15865748__15841370__15859360
O=C(CN1CCC(O)CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841372__15862300
O=C(CN1CCC(O)CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841372__15859360
CN(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__15841376__15862300
CN(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__15841376__15859360
CN(CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC1 s275592__15865748__15841376__15857566
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N1CCN(C)CC1 s275592__15865748__15841378__15859360
Cc1cnc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)s1 s275592__15865748__15841392__15862300
Cc1cnc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__15841392__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(CO)COC1 s275592__15865748__15841398__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(CO)COC1 s275592__15865748__15841398__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(CO)COC1 s275592__15865748__15841398__15857566
CC(C)=CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841400__15862300
CC(C)=CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841400__15859360
CC(C)=CCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841400__15857566
CC=C(C=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)CC s275592__15865748__15841402__15862300
CC=C(C=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC s275592__15865748__15841402__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1COC1 s275592__15865748__15841406__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1COC1 s275592__15865748__15841406__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1COC1 s275592__15865748__15841406__15857566
O=C(C=CC1CCCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841412__15862300
O=C(C=CC1CCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841412__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(CO)c(F)c1 s275592__15865748__15841414__15859360
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COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCOC1 s275592__15865748__15845090__15859360
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CC1(C)C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1(F)F s275592__15865748__15845112__15859360
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CC(C)n1cnnc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845128__15859360
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CC(C)(C)c1nocc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845144__15859360
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O=C(CC1(CO)CCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845146__15859360
CON=C(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccco1 s275592__15865748__15845152__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCn2ncnc2C1 s275592__15865748__15845154__15859360
CC1(C)NC(=O)CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845156__15862300
CC1(C)NC(=O)CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845156__15859360
C=CCc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845160__15859360
COC1C[C@@H]2CC(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)C[C@H]12 s275592__15865748__15845162__15859360
O=C(Cc1nccs1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841446__15862300
O=C(Cc1nccs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841446__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC=CO1 s275592__15865748__15841456__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC=CO1 s275592__15865748__15841456__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCC=CO1 s275592__15865748__15841456__15857566
CC(O)(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC1 s275592__15865748__15841462__15862300
CC(O)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC1 s275592__15865748__15841462__15859360
CC1(C)CCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)O1 s275592__15865748__15841464__15862300
CC1(C)CCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)O1 s275592__15865748__15841464__15859360
CC(O)c1cn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1 s275592__15865748__15841470__15859360
Cn1nccc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841472__15862300
Cn1nccc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841472__15859360
O=C(CC1CSC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841474__15862300
O=C(CC1CSC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841474__15859360
O=C(CC1CSC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841474__15857566
Cc1[nH]nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1[N+](=O)[O-] s275592__15865748__15841476__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc2ncccn12 s275592__15865748__15841478__15859360
CSc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)oc1C s275592__15865748__15841480__15859360
COCCNC(=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841482__15862300
COCCNC(=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841482__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(F)CCC1 s275592__15865748__15841486__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(F)CCC1 s275592__15865748__15841486__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(F)CCC1 s275592__15865748__15841486__15857566
CC(C)c1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cnn1C s275592__15865748__15841490__15859360
O=C(CSc1ccncc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841492__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2[nH]cnc2c1 s275592__15865748__15841498__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CSCCS1 s275592__15865748__15841502__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(Cl)ccn1 s275592__15865748__15841504__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(Cl)ccn1 s275592__15865748__15841504__15859360
O=C(CO)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841508__15862300
O=C(CO)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841508__15857566
CCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__15841510__15859360
NC(=O)C=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841512__15862300
NC(=O)C=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841512__15859360
NC(=O)C=CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841512__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc[n+]([O-])c1 s275592__15865748__15841514__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc[n+]([O-])c1 s275592__15865748__15841514__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)n1cc(Cl)cn1 s275592__15865748__15841516__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cc(O)ncn1 s275592__15865748__15841522__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(O)ncn1 s275592__15865748__15841522__15859360
C#CCSCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841524__15862300
C#CCSCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841524__15859360
C#CCSCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841524__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccnc1Cl s275592__15865748__15841534__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnc1Cl s275592__15865748__15841534__15859360
CC(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841536__15862300
CC(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841536__15859360
CC(O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841536__15857566
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(O)CCC1 s275592__15865748__15841548__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(O)CCC1 s275592__15865748__15841548__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(O)CCC1 s275592__15865748__15841548__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(O)C1CC1 s275592__15865748__15841554__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(O)C1CC1 s275592__15865748__15841554__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C(O)C1CC1 s275592__15865748__15841554__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccc1CO s275592__15865748__15841556__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1CO s275592__15865748__15841556__15859360
NC(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__15841560__15862300
NC(=O)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__15841560__15859360
O=C(Cn1cnnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841562__15862300
O=C(Cn1cnnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841562__15859360
O=C(Cn1cnnc1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841562__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCc2ccccc21 s275592__15865748__15841564__15859360
CSc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__15841566__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C(=O)NC2CC2)CC1 s275592__15865748__15841568__15859360
N=c1sccn1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843316__15862300
N=c1sccn1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843316__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc(CO)c1 s275592__15865748__15843318__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(CO)c1 s275592__15865748__15843318__15859360
C=CCC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843320__15862300
C=CCC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843320__15859360
C=CCC(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843320__15857566
CSCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__15843322__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C(F)(F)C(F)(F)F s275592__15865748__15843324__15859360
O=C(Cc1c(O)ncnc1O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843330__15859360
O=CNc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__15843334__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1F s275592__15865748__15843336__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1F s275592__15865748__15843336__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC1F s275592__15865748__15843336__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1C(F)F s275592__15865748__15843338__15859360
CC1(OCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__15843342__15862300
CC1(OCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__15843342__15859360
CN(CCO)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843344__15862300
CN(CCO)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843344__15859360
C[C@@H](C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N(C)C s275592__15865748__15843346__15862300
C[C@@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N(C)C s275592__15865748__15843346__15859360
C[C@@H](C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)N(C)C s275592__15865748__15843346__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2ocnc2c1 s275592__15865748__15843348__15859360
O=C(CCF)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843350__15862300
O=C(CCF)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843350__15859360
O=C(CCF)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843350__15857566
O=C(Cn1ccnn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843356__15862300
O=C(Cn1ccnn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843356__15859360
O=C(Cn1ccnn1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843356__15857566
CN1CCCC[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843358__15862300
CN1CCCC[C@@H]1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843358__15859360
O=C(CCc1ncc(F)cn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843362__15859360
C=CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__15843364__15862300
C=CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__15843364__15859360
C=CC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CCC1 s275592__15865748__15843364__15857566
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(O)COC1 s275592__15865748__15843366__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(O)COC1 s275592__15865748__15843366__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C1(O)COC1 s275592__15865748__15843366__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccc(F)nc1F s275592__15865748__15843368__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)nc1F s275592__15865748__15843368__15859360
CCC(C)C(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843370__15862300
CCC(C)C(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843370__15859360
CCC(C)C(O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843370__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ncncc1Cl s275592__15865748__15843374__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncncc1Cl s275592__15865748__15843374__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)=C1CC1 s275592__15865748__15843378__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)=C1CC1 s275592__15865748__15843378__15859360
CC(C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)=C1CC1 s275592__15865748__15843378__15857566
CC1CN2CCN1CC2C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843380__15859360
O=C(C[C@H]1CCCC[C@@H]1O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843386__15862300
O=C(C[C@H]1CCCC[C@@H]1O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843386__15859360
C[C@@H](C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)n1cnnn1 s275592__15865748__15843388__15862300
C[C@@H](C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)n1cnnn1 s275592__15865748__15843388__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnnc(Cl)c1 s275592__15865748__15843390__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnnc(Cl)c1 s275592__15865748__15843390__15859360
Cn1cc(OCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cn1 s275592__15865748__15843394__15862300
Cn1cc(OCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__15843394__15859360
O=NN1CCCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843398__15862300
O=NN1CCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843398__15859360
O=C(CCCc1nccs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843400__15859360
CCC1CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843404__15862300
CCC1CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843404__15859360
CCC1CC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843404__15857566
CS(C)(=O)=NCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843410__15862300
CS(C)(=O)=NCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843410__15859360
[N-]=[N+]=NCCCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843412__15859360
CC(O)CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843418__15862300
CC(O)CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843418__15859360
CC(O)CCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843418__15857566
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)on1 s275592__15865748__15843422__15862300
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__15843422__15859360
O=C(Cc1cnccc1Cl)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843426__15859360
O=C(CC1(O)CC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843428__15862300
O=C(CC1(O)CC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843428__15859360
O=C(CC1(O)CC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843428__15857566
O=C(CCCCC(F)(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843432__15859360
O=C(Cc1ccn[nH]c1=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843434__15862300
O=C(Cc1ccn[nH]c1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843434__15859360
Cc1oc([N+](=O)[O-])cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843436__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1C2CCOCC21 s275592__15865748__15845166__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1C2CCOCC21 s275592__15865748__15845166__15859360
Cc1cnn(C(C)C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__15845168__15862300
Cc1cnn(C(C)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15845168__15859360
CC(C)C(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)n1cnnc1 s275592__15865748__15845170__15859360
O=C(CCc1ccc(F)nc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845172__15859360
O=C(C=CCF)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845174__15862300
O=C(C=CCF)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845174__15859360
O=C(C=CCF)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15845174__15857566
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(CC(F)F)CCC1 s275592__15865748__15845178__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(F)CC1CC1 s275592__15865748__15845182__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)CC1CC1 s275592__15865748__15845182__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C(F)CC1CC1 s275592__15865748__15845182__15857566
CCC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__15845184__15862300
CCC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__15845184__15859360
Cc1cnn2ccc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)nc12 s275592__15865748__15845186__15859360
[N-]=[N+]=N[C@H]1CC[C@H](C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__15845190__15859360
Cn1nccc1C(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845192__15862300
Cn1nccc1C(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845192__15859360
CC12CCCC(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)(CO1)C2 s275592__15865748__15845194__15859360
Cc1cccnc1C=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845202__15859360
CCC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC1 s275592__15865748__15845204__15862300
CCC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC1 s275592__15865748__15845204__15859360
COCc1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)no1 s275592__15865748__15845212__15859360
Cc1nc(CO)ncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845214__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC(C2CC2)=NO1 s275592__15865748__15845216__15859360
O=C(C=Cc1ncc[nH]1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845226__15862300
O=C(C=Cc1ncc[nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845226__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2cnnn12 s275592__15865748__15845232__15859360
CC(=O)NC1(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1 s275592__15865748__15845234__15862300
CC(=O)NC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1 s275592__15865748__15845234__15859360
CNC(=O)N[C@@H](C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845238__15862300
CNC(=O)N[C@@H](C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845238__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC(C2CC2)=NO1 s275592__15865748__15845240__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC(C2CC2)=NO1 s275592__15865748__15845240__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C12CCC(F)(CC1)C2 s275592__15865748__15845242__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C12CCC(F)(CC1)C2 s275592__15865748__15845242__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CC(C2CCC2)C1 s275592__15865748__15845246__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC(C2CCC2)C1 s275592__15865748__15845246__15859360
CCC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)OC s275592__15865748__15845254__15862300
CCC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)OC s275592__15865748__15845254__15859360
CCC(CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)OC s275592__15865748__15845254__15857566
O=C(Cc1ccn2cncc2c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845258__15859360
COCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC=CCC1 s275592__15865748__15845260__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(C(F)F)cn1 s275592__15865748__15845268__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=C(Cl)CC1 s275592__15865748__15845270__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=C(Cl)CC1 s275592__15865748__15845270__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1=C(Cl)CC1 s275592__15865748__15845270__15857566
CCCc1ccc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__15845272__15859360
Cc1nnnn1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845274__15862300
Cc1nnnn1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845274__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2nncn12 s275592__15865748__15845276__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1C[C@@H]1c1nc[nH]n1 s275592__15865748__15845278__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@@H]1c1nc[nH]n1 s275592__15865748__15845278__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1COC2COCC21 s275592__15865748__15845280__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1COC2COCC21 s275592__15865748__15845280__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)[C@@]12C[C@@H](F)[C@@H]1C2 s275592__15865748__15845282__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)[C@@]12C[C@@H](F)[C@@H]1C2 s275592__15865748__15845282__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)[C@@]12C[C@@H](F)[C@@H]1C2 s275592__15865748__15845282__15857566
O=C(CCc1cccc(=O)[nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845286__15859360
O=C(Cc1ccc(Cl)nc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841578__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=CCCOC1 s275592__15865748__15841580__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CCCOC1 s275592__15865748__15841580__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1=CCCOC1 s275592__15865748__15841580__15857566
CCn1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1C s275592__15865748__15841582__15862300
CCn1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1C s275592__15865748__15841582__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CC1(F)F s275592__15865748__15841584__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC1(F)F s275592__15865748__15841584__15859360
Cc1c(Cl)cnn1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841586__15859360
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)on1 s275592__15865748__15841588__15862300
CCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__15841588__15859360
CC(C)(C)C(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841590__15862300
CC(C)(C)C(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841590__15859360
CC(C)(C)C(O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841590__15857566
CCCCn1nccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841596__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCSCC1 s275592__15865748__15841598__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCSCC1 s275592__15865748__15841598__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2ncoc12 s275592__15865748__15841602__15859360
C#CCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841610__15862300
C#CCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841610__15859360
C#CCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841610__15857566
CCn1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1O s275592__15865748__15841616__15862300
CCn1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1O s275592__15865748__15841616__15859360
CN(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCSC1 s275592__15865748__15841620__15859360
O=C(CN1CCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841622__15862300
O=C(CN1CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841622__15859360
O=C(CN1CCC1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841622__15857566
CC(C)C(O)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841624__15862300
CC(C)C(O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841624__15859360
CC(C)C(O)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841624__15857566
COc1noc(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841626__15862300
COc1noc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841626__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=C(Cl)CCC1 s275592__15865748__15841630__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=C(Cl)CCC1 s275592__15865748__15841630__15859360
CCC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)SC s275592__15865748__15841632__15862300
CCC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)SC s275592__15865748__15841632__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nc1 s275592__15865748__15841640__15862300
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc1 s275592__15865748__15841640__15859360
O=C(CC1=NNC(=O)C1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841642__15862300
O=C(CC1=NNC(=O)C1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841642__15859360
CCc1csc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15841644__15859360
CC(C)(C)CC(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841646__15862300
CC(C)(C)CC(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841646__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnc(F)cc1F s275592__15865748__15841652__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc(F)cc1F s275592__15865748__15841652__15859360
O=C(Cc1ccc2[nH]ccc2c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841654__15859360
O=C(CC1CSCCS1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841656__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C(F)(F)C1(O)CCC1 s275592__15865748__15841660__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ccncc2[nH]1 s275592__15865748__15841662__15859360
CCCC(C)(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841664__15862300
CCCC(C)(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841664__15859360
CCCC(C)(O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841664__15857566
CCOC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841666__15862300
CCOC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841666__15859360
CCOC(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841666__15857566
O=C(Cc1cccnc1Cl)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841670__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2ccccc2cn1 s275592__15865748__15841674__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc(Cl)c1F s275592__15865748__15841678__15859360
O=C(CC1CCSCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841680__15862300
O=C(CC1CCSCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841680__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(CO)c1ccccc1 s275592__15865748__15841682__15859360
Cc1cc(Cl)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__15841684__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1C[C@@H]1c1ccccc1 s275592__15865748__15841686__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2nccnc2n1 s275592__15865748__15841688__15859360
Cc1nc(CO)sc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843440__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(=S)n1O s275592__15865748__15843442__15859360
CC(=Cc1cccnc1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843444__15859360
CC1=C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCC1 s275592__15865748__15843456__15862300
CC1=C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__15843456__15859360
COCc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n[nH]1 s275592__15865748__15843458__15862300
COCc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n[nH]1 s275592__15865748__15843458__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(c2cccnc2)CCC1 s275592__15865748__15843462__15859360
CN1CCC(=CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__15843464__15862300
CN1CCC(=CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15843464__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc2c1CCC2 s275592__15865748__15843468__15859360
O=C(C=CCn1cncn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843472__15862300
O=C(C=CCn1cncn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843472__15859360
O=C(C=CC1CCCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843476__15859360
CSc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15843478__15859360
O=C(Cc1sc(O)nc1O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843480__15859360
Cc1nnc(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)o1 s275592__15865748__15843482__15862300
Cc1nnc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__15843482__15859360
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)[nH]c1C s275592__15865748__15843486__15862300
Cc1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)[nH]c1C s275592__15865748__15843486__15859360
CCOC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__15843492__15862300
CCOC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__15843492__15859360
CCOC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCOCC1 s275592__15865748__15843498__15859360
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)sn1 s275592__15865748__15843502__15862300
Cc1cc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)sn1 s275592__15865748__15843502__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ncoc1C1CCC1 s275592__15865748__15843504__15859360
CC(O)c1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843506__15859360
CC(=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccco1 s275592__15865748__15843508__15862300
CC(=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccco1 s275592__15865748__15843508__15859360
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Cc1nn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(=O)o1 s275592__15865748__15843510__15859360
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C[C@@H]1C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)[C@@H]1C s275592__15865748__15845402__15862300
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CC(=C(F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C1CC1 s275592__15865748__15839944__15862300
CC(=C(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1CC1 s275592__15865748__15839944__15859360
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Cc1cccc2[nH]cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c12 s275592__15865748__15841702__15859360
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CS(=O)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841706__15862300
CS(=O)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841706__15859360
COc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(F)n1 s275592__15865748__15841708__15859360
CC(=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnn(C)c1 s275592__15865748__15841712__15859360
Cn1nc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)cc1F s275592__15865748__15841714__15862300
Cn1nc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1F s275592__15865748__15841714__15859360
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O=NN1CCCCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841718__15859360
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O=C(C=C(Cl)Cl)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841720__15859360
CSc1ccnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15841724__15859360
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CN1CCCC(O)(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15841730__15859360
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n[nH]1 s275592__15865748__15841732__15862300
COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n[nH]1 s275592__15865748__15841732__15859360
CC1=C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC(C)(C)C1 s275592__15865748__15841734__15859360
CC1CN(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__15841738__15862300
CC1CN(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15841738__15859360
CC1CN(CC(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865748__15841738__15857566
COCn1ccc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__15841750__15862300
COCn1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15841750__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(O)C1CCCC1 s275592__15865748__15841758__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(O)C1CCCC1 s275592__15865748__15841758__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)COC1 s275592__15865748__15841760__15862300
CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)COC1 s275592__15865748__15841760__15859360
CC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)COC1 s275592__15865748__15841760__15857566
Cc1nc(Cl)ccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841762__15859360
Cc1cccc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)[nH]c12 s275592__15865748__15841764__15859360
Cn1nc([N+](=O)[O-])cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841766__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=CCCCO1 s275592__15865748__15841768__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CCCCO1 s275592__15865748__15841768__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1=CCCCO1 s275592__15865748__15841768__15857566
O=C(CSCc1ncc[nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841770__15859360
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O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CCCS1 s275592__15865748__15841774__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1=CCCS1 s275592__15865748__15841774__15857566
CC1=NOC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__15841776__15862300
CC1=NOC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15841776__15859360
CC1=NOC(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865748__15841776__15857566
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CCn1cc(Cl)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15841780__15859360
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CCC1=NOC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__15841784__15862300
CCC1=NOC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15841784__15859360
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Cc1noc(COCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15841790__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCSC1 s275592__15865748__15841792__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCSC1 s275592__15865748__15841792__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCSC1 s275592__15865748__15841792__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCO1 s275592__15865748__15841796__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCO1 s275592__15865748__15841796__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCO1 s275592__15865748__15841796__15857566
CC(=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1C s275592__15865748__15841798__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(F)c(Cl)n1 s275592__15865748__15841800__15859360
[N-]=[N+]=NCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841802__15862300
[N-]=[N+]=NCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841802__15859360
[N-]=[N+]=NCCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841802__15857566
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O=C(Cn1cc(CO)nn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841804__15859360
C#CCOCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841806__15862300
C#CCOCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841806__15859360
C#CCOCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841806__15857566
O=C(Cc1nnco1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841808__15862300
O=C(Cc1nnco1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841808__15859360
O=C(Cc1nnco1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841808__15857566
CC1=C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)SCCO1 s275592__15865748__15841810__15862300
CC1=C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)SCCO1 s275592__15865748__15841810__15859360
CN(CCO)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841814__15862300
CN(CCO)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841814__15859360
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O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCS1 s275592__15865748__15841818__15859360
O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CCCS1 s275592__15865748__15841818__15857566
CCCC(O)(CCC)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841820__15859360
CC(C)(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843566__15862300
CC(C)(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843566__15859360
CC(C)(O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843566__15857566
Cc1oc(CO)cc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843580__15862300
Cc1oc(CO)cc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843580__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc2ncnn12 s275592__15865748__15843584__15859360
CC(O)(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)(F)F s275592__15865748__15843588__15859360
Cc1csc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__15843592__15862300
Cc1csc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15843592__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C(F)(F)c1ccccc1 s275592__15865748__15843594__15859360
O=C(Cc1ccccn1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843596__15862300
O=C(Cc1ccccn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843596__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1ccnc(Cl)c1 s275592__15865748__15843598__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccnc(Cl)c1 s275592__15865748__15843598__15859360
CC(SC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843600__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccnc1F s275592__15865748__15843604__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccnc1F s275592__15865748__15843604__15859360
CC1=NN(C)C(=O)C1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843616__15859360
CC1=CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843618__15862300
CC1=CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843618__15859360
CC1=CC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843618__15857566
CN(C)C(=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843620__15862300
CN(C)C(=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843620__15859360
CN(C)C(=O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843620__15857566
CSC=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843626__15862300
CSC=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843626__15859360
CSC=CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843626__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnccc1O s275592__15865748__15843636__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnccc1O s275592__15865748__15843636__15859360
CC1=NC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CS1 s275592__15865748__15843638__15862300
CC1=NC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CS1 s275592__15865748__15843638__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1c(F)ccnc1F s275592__15865748__15843640__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c(F)ccnc1F s275592__15865748__15843640__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnc(Cl)c(F)c1 s275592__15865748__15843642__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CN2CCCN1CC2 s275592__15865748__15843644__15859360
Cc1cncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1O s275592__15865748__15843648__15862300
Cc1cncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1O s275592__15865748__15843648__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1c(Cl)ccnc1F s275592__15865748__15843658__15859360
CCC(C)(O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843660__15862300
CCC(C)(O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843660__15859360
CCC(C)(O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843660__15857566
COc1ccncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843662__15862300
COc1ccncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843662__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(O)C1CCOCC1 s275592__15865748__15843664__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(O)C1CCOCC1 s275592__15865748__15843664__15859360
CCN1CCCC(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__15843666__15862300
CCN1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15843666__15859360
CCc1noc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__15843670__15862300
CCc1noc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15843670__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)CN(C)C s275592__15865748__15843672__15862300
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CN(C)C s275592__15865748__15843672__15859360
COc1cccc(C=CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15843674__15859360
Cc1ccc(C=CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__15843676__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1CCc2ccccc21 s275592__15865748__15843680__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2c1COC2 s275592__15865748__15843686__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc(CC2CC2)cc1 s275592__15865748__15845414__15859360
Cc1cc(Cl)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__15845416__15859360
Cc1nnn(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__15845420__15862300
Cc1nnn(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15845420__15859360
CC(C)n1cncc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845424__15862300
CC(C)n1cncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845424__15859360
Cc1cn2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc2n1 s275592__15865748__15845426__15859360
Cc1nnc2n1C(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC2 s275592__15865748__15845428__15859360
CCN(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845430__15862300
CCN(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845430__15859360
CCN(C)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15845430__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCCC(F)(F)CC1 s275592__15865748__15845434__15859360
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CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1nc[nH]n1 s275592__15865748__15845444__15859360
Cc1cc2c(c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c1)OCC2 s275592__15865748__15845446__15859360
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C=C1CC2(C1)CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C2 s275592__15865748__15845456__15859360
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CC(C)c1c[nH]nc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845478__15862300
CC(C)c1c[nH]nc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845478__15859360
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O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cnoc1C1CCC1 s275592__15865748__15845484__15859360
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CC(C)(F)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845486__15859360
COC1CC2(C1)CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C2 s275592__15865748__15845488__15859360
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O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cncc2[nH]ccc12 s275592__15865748__15845502__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1n[nH]c2c1C[C@H]1C[C@@H]21 s275592__15865748__15845504__15859360
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CC[C@H](CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)C s275592__15865748__15845526__15859360
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CCC=CC=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845532__15859360
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Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c[nH]1 s275592__15865748__15840030__15862300
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Cc1cc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)c[nH]1 s275592__15865748__15840030__15857566
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Cc1ncc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)o1 s275592__15865748__15840058__15857566
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O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1[nH]ncc1Cl s275592__15865748__15840062__15859360
Cc1scnc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840066__15862300
Cc1scnc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840066__15859360
CC1COc2c(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cccc21 s275592__15865748__15840068__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(C2CC2)ccn1 s275592__15865748__15840076__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC1F s275592__15865748__15840078__15862300
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Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc(Cl)n1 s275592__15865748__15839960__15859360
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Cc1nc2ccccn2c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15839970__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc([N+](=O)[O-])c1 s275592__15865748__15839974__15859360
CCN(CC)CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15839976__15862300
CCN(CC)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15839976__15859360
CN1N=C(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1=O s275592__15865748__15839984__15862300
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O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cnc[nH]1 s275592__15865748__15839986__15862300
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O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)c1cnc[nH]1 s275592__15865748__15839986__15857566
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2cn[nH]c2c1 s275592__15865748__15839990__15859360
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Cc1noc(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)n1 s275592__15865748__15839992__15857566
COC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__15841822__15859360
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O=C(NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1)C1CC2CC2C1 s275592__15865748__15841824__15857566
O=C(Cc1cncnc1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841834__15862300
O=C(Cc1cncnc1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841834__15859360
O=C(CCc1nc(=O)[nH][nH]1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841838__15862300
O=C(CCc1nc(=O)[nH][nH]1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841838__15859360
Cc1ccncc1C=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841848__15859360
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O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C(F)F)CCCCC1 s275592__15865748__15841858__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccn(O)c1=O s275592__15865748__15841860__15862300
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Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)sn1 s275592__15865748__15841874__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)sn1 s275592__15865748__15841874__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc2sccc12 s275592__15865748__15841876__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CCS(=O)(=O)C1 s275592__15865748__15841878__15859360
Cc1cc(CCC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)on1 s275592__15865748__15841880__15862300
Cc1cc(CCC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)on1 s275592__15865748__15841880__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1=CCSC1 s275592__15865748__15841882__15862300
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O=C(CCCC(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841884__15859360
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Cc1ccc(Cl)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15841900__15859360
O=C(CCn1cccnc1=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841902__15859360
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O=C(C=CC1CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841918__15859360
CCCC(O)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15841922__15862300
CCCC(O)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841922__15859360
CCCC(O)CC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15841922__15857566
Cn1ncc([N+](=O)[O-])c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841926__15859360
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CN1CCC(C)(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1=O s275592__15865748__15843696__15862300
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CC1(O)CCN(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__15843730__15862300
CC1(O)CCN(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15843730__15859360
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CC(C)OC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__15843738__15862300
CC(C)OC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__15843738__15859360
CC1(C)CC2(CC2C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)C1 s275592__15865748__15843742__15862300
CC1(C)CC2(CC2C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15843742__15859360
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Cc1ncc(C=CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__15843754__15859360
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Cc1csc(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)c1 s275592__15865748__15843776__15862300
Cc1csc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15843776__15859360
CCC[C@H](O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843778__15862300
CCC[C@H](O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843778__15859360
CCC[C@H](O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843778__15857566
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C#CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CC=CCC1 s275592__15865748__15843782__15859360
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CC1(C)C2CCC(C2)C1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843790__15859360
CC1(C)C2CCC1(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC2 s275592__15865748__15843794__15859360
C#CC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCC1 s275592__15865748__15843796__15862300
C#CC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__15843796__15859360
Cn1ncc2ncc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)cc21 s275592__15865748__15843798__15859360
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CC(C)C1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)COC1 s275592__15865748__15843808__15862300
CC(C)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)COC1 s275592__15865748__15843808__15859360
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COc1ncnc(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845544__15859360
CC(OCCN(C)C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845546__15862300
CC(OCCN(C)C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845546__15859360
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CC1(CC(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCO1 s275592__15865748__15845552__15862300
CC1(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCO1 s275592__15865748__15845552__15859360
Cc1ncn(C)c1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845556__15862300
Cc1ncn(C)c1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845556__15859360
CC12CCC(C(=O)NCCC3CCCCN3C(=O)c3nsnc3O)(CO1)C2 s275592__15865748__15845558__15862300
CC12CCC(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)(CO1)C2 s275592__15865748__15845558__15859360
CC(CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)CC(F)(F)F s275592__15865748__15845564__15859360
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O=C(Cc1nncs1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845568__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C1(C2CCC2)CC1(F)F s275592__15865748__15845570__15859360
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CN(C)CCOCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845572__15859360
COCCN(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845574__15862300
COCCN(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845574__15859360
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C1(C2CC2)CCCO1 s275592__15865748__15845580__15862300
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Cn1cc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc2n1 s275592__15865748__15845586__15859360
CCc1cscc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845596__15862300
CCc1cscc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845596__15859360
O=C(CC1CCCC(F)(F)C1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845604__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1=CC2CCC=CCCC12 s275592__15865748__15845610__15859360
C=C1CC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)(C(F)F)C1 s275592__15865748__15845616__15859360
CO[C@@H]1C[C@@]2(C(=O)NCCC3CCCCN3C(=O)c3nsnc3O)C[C@@H]12 s275592__15865748__15845622__15862300
CO[C@@H]1C[C@@]2(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)C[C@@H]12 s275592__15865748__15845622__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc2cncnc2[nH]1 s275592__15865748__15845624__15859360
Cc1ccc(C)c(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__15845626__15862300
Cc1ccc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15845626__15859360
CC1OC2(C)CC1(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)C2 s275592__15865748__15845628__15862300
CC1OC2(C)CC1(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C2 s275592__15865748__15845628__15859360
Cn1cnnc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845630__15862300
Cn1cnnc1CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845630__15859360
CCc1nonc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845636__15862300
CCc1nonc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845636__15859360
O=C(CC1(CO)CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845640__15859360
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O=C(Cc1cnsn1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845642__15859360
C=CCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845644__15862300
C=CCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845644__15859360
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CC1C(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)=Cc2ccccc21 s275592__15865748__15840084__15859360
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COc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc(C)n1 s275592__15865748__15840090__15859360
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CCC(C)(OC)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840100__15859360
CCC(C)(OC)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15840100__15857566
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CCCC(CCCO)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840106__15859360
CC(O)c1ncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__15840110__15859360
O=C1CC(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCN1 s275592__15865748__15840112__15859360
CC(C)[C@H](O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840114__15862300
CC(C)[C@H](O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840114__15859360
CC(C)[C@H](O)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15840114__15857566
CSC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCC1 s275592__15865748__15840116__15862300
CSC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCC1 s275592__15865748__15840116__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccn1 s275592__15865748__15840122__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccn1 s275592__15865748__15840122__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(O)c1ccccn1 s275592__15865748__15840124__15862300
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CC(O)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccn1 s275592__15865748__15840126__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc(=O)n1O s275592__15865748__15840128__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(=O)n1O s275592__15865748__15840128__15859360
Cn1ccc2cc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)ccc21 s275592__15865748__15840134__15859360
CN(C)C1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCCC1 s275592__15865748__15840136__15862300
CN(C)C1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCCC1 s275592__15865748__15840136__15859360
COc1ccnc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15840138__15859360
CC(CS(C)=O)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840140__15862300
CC(CS(C)=O)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840140__15859360
CC(CCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N(C)C s275592__15865748__15840142__15862300
CC(CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N(C)C s275592__15865748__15840142__15859360
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CCN1CCC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840164__15862300
CCN1CCC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840164__15859360
CCN1CCC1C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15840164__15857566
Cc1nc(C=CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cs1 s275592__15865748__15840168__15859360
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Cc1cc(C)c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(=O)o1 s275592__15865748__15840196__15859360
CC(C)N1CCCC(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)C1 s275592__15865748__15840198__15859360
COc1ccc(C=CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__15840202__15859360
Cc1ccc2c(c1)C(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C2 s275592__15865748__15840204__15859360
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CSCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841948__15859360
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)nc(O)n1 s275592__15865748__15841950__15862300
Cc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nc(O)n1 s275592__15865748__15841950__15859360
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CCc1nc(C)ncc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15841966__15859360
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CCc1cnc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)s1 s275592__15865748__15841992__15862300
CCc1cnc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)s1 s275592__15865748__15841992__15859360
CSSCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15842002__15862300
CSSCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15842002__15859360
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CCC(C)=C(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15842008__15862300
CCC(C)=C(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15842008__15859360
CCC(C)=C(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15842008__15857566
CSC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)(C)C s275592__15865748__15842010__15859360
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COC1(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)CCC1 s275592__15865748__15842012__15857566
CSc1cccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c1 s275592__15865748__15842014__15859360
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CC(C)(O)CCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15842026__15859360
CC(C)(O)CCC(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15842026__15857566
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COCCC(C)(C)CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15842028__15859360
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CC1CC(=O)NC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15842050__15862300
CC1CC(=O)NC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15842050__15859360
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CC1CC(C)(C(=O)NCCC2CCCCN2C(=O)CSc2n[nH]c(=O)[nH]2)C1 s275592__15865748__15843850__15857566
[N-]=[N+]=NCc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)o1 s275592__15865748__15843852__15859360
Cn1ncnc1CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843856__15862300
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O=C(C=CCO)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15843928__15857566
CCC(O)C(F)(F)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15843930__15862300
CCC(O)C(F)(F)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15843930__15859360
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CC(C)(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C1(O)CCOC1 s275592__15865748__15845662__15859360
CCC(C)CC(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845666__15862300
CCC(C)CC(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845666__15859360
C#CCC1(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)CCOC1 s275592__15865748__15845670__15862300
C#CCC1(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)CCOC1 s275592__15865748__15845670__15859360
CN1CC(C)(C)CC1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845674__15862300
CN1CC(C)(C)CC1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845674__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C(F)n1cccn1 s275592__15865748__15845678__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C(F)n1cccn1 s275592__15865748__15845678__15859360
O=C(CC1(CO)CCCCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845680__15859360
Cc1ccn2ncc(C(=O)NCCC3CCCCN3C(=O)c3cc(O)no3)c2n1 s275592__15865748__15845682__15859360
CN(C)CCCCCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845684__15862300
CN(C)CCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845684__15859360
COc1ccnc(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15845686__15859360
CC1(C)CC(=O)N(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)O1 s275592__15865748__15845688__15859360
O=C(Cc1cnco1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845696__15862300
O=C(Cc1cnco1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845696__15859360
O=C(Cc1cnco1)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15845696__15857566
O=C(CC12CCC(CC1)C2)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845698__15862300
O=C(CC12CCC(CC1)C2)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845698__15859360
O=C(C[C@@H]1CC=CCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845700__15862300
O=C(C[C@@H]1CC=CCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845700__15859360
CC(=Cc1cccs1)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845702__15859360
COCCOCC=CC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845706__15862300
COCCOCC=CC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845706__15859360
O=C(CN1CC2CC2C1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845708__15862300
O=C(CN1CC2CC2C1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15845708__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C(C)n1cccn1 s275592__15865748__15845714__15859360
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)[C@H]1C[C@H](n2ccnn2)C1 s275592__15865748__15845718__15859360
O=C(CC1CC2CC2C1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15845722__15862300
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O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cc(CF)on1 s275592__15865748__15845728__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccc2cnnn2c1 s275592__15865748__15845738__15859360
CCCc1cc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)nn1C s275592__15865748__15840210__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)[C@@H]1CC[C@H]1C(F)F s275592__15865748__15840212__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@@H]1CC[C@H]1C(F)F s275592__15865748__15840212__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)[C@H]1CCc2ccccc21 s275592__15865748__15840214__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)C1CCC2CC2CC1 s275592__15865748__15840224__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)C1CCC2CC2CC1 s275592__15865748__15840224__15859360
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccn2ncnc12 s275592__15865748__15840226__15859360
O=C(C=Cc1cccc(F)c1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840228__15859360
[N-]=[N+]=NCc1ccccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840232__15859360
CSc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cc1 s275592__15865748__15840236__15859360
NC(=O)NCCCCCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840248__15859360
Cn1c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)ccc1[N+](=O)[O-] s275592__15865748__15840250__15859360
CC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)c1ccccc1 s275592__15865748__15840252__15862300
CC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)c1ccccc1 s275592__15865748__15840252__15859360
O=C(CNC(=O)C(F)(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840254__15859360
NC1=NC(=O)C(CC(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)S1 s275592__15865748__15840258__15859360
O=C(COCC(F)(F)F)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840270__15862300
O=C(COCC(F)(F)F)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840270__15859360
Cc1ccc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)c(Cl)n1 s275592__15865748__15840272__15859360
NC(=O)CSCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840274__15862300
NC(=O)CSCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840274__15859360
CCCCSCC(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840276__15862300
CCCCSCC(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840276__15859360
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1cccc(F)n1 s275592__15865748__15840278__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1cccc(F)n1 s275592__15865748__15840278__15859360
COC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840284__15862300
COC(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840284__15859360
COC(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15840284__15857566
O=C(NCCC1CCCCN1C(=O)c1nsnc1O)c1nccnc1Cl s275592__15865748__15840286__15862300
O=C(NCCC1CCCCN1C(=O)c1cc(O)no1)c1nccnc1Cl s275592__15865748__15840286__15859360
CC1CN2CCN1C(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)C2 s275592__15865748__15840288__15859360
CCCC(C(=O)NCCC1CCCCN1C(=O)c1nsnc1O)N(C)C s275592__15865748__15840292__15862300
CCCC(C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1)N(C)C s275592__15865748__15840292__15859360
O=C(C=CC1CCOCC1)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840294__15862300
O=C(C=CC1CCOCC1)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840294__15859360
Cn1cc([N+](=O)[O-])c(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15840300__15859360
Cc1cncc(C(=O)NCCC2CCCCN2C(=O)c2nsnc2O)n1 s275592__15865748__15840302__15862300
Cc1cncc(C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)n1 s275592__15865748__15840302__15859360
CN(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840304__15862300
CN(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840304__15859360
CN(C)C(C)(C)C(=O)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15840304__15857566
O=C(c1nsnc1O)N1CCCCC1CCNC(=O)C(F)(F)CO s275592__15865748__15840310__15862300
O=C(c1cc(O)no1)N1CCCCC1CCNC(=O)C(F)(F)CO s275592__15865748__15840310__15859360
O=C(CSc1n[nH]c(=O)[nH]1)N1CCCCC1CCNC(=O)C(F)(F)CO s275592__15865748__15840310__15857566
Cc1nc(O)ccc1C(=O)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840312__15862300
Cc1nc(O)ccc1C(=O)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840312__15859360
Cn1cc(C(F)(F)C(=O)NCCC2CCCCN2C(=O)c2cc(O)no2)cn1 s275592__15865748__15840318__15859360
O=C(CCCCO)NCCC1CCCCN1C(=O)c1nsnc1O s275592__15865748__15840320__15862300
O=C(CCCCO)NCCC1CCCCN1C(=O)c1cc(O)no1 s275592__15865748__15840320__15859360
O=C(CCCCO)NCCC1CCCCN1C(=O)CSc1n[nH]c(=O)[nH]1 s275592__15865748__15840320__15857566
